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Search Results for " mycobacterium "
Targets Recommended: Antibacterial

166

抑制剂 & 化合物

41

天然产物

41

重组蛋白

4

同位素标记化合物

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Cat. No. Product Name Target Signaling Pathways
T7342 BM212

Antibacterial Microbiology/Virology
BM212 是一种分枝杆菌膜蛋白 MmpL3抑制剂。它抑制结核分枝杆菌和部分非结核分枝杆菌,抗结核杆菌 H37Rv 菌株的 MIC 值为 5 µM。
T38359 Dup-721

Antibacterial Microbiology/Virology
DuP-721 是广谱的口服有效的抗菌剂,可以抑制多种临床敏感和耐药细菌,特别是结核杆菌M. tuberculosis。
T10411 AU1235

Antibacterial Microbiology/Virology
AU1235是金刚烷脲,是一种MmpL3抑制剂。结核分枝杆菌蛋白MmpL3在细胞壁合成中起重要作用,它影响海藻糖单支霉菌酸酯跨内膜转运。
T8694 ML406

Antibacterial; Antibiotic Microbiology/Virology
ML406 是一种小分子探针,通过抑制M.tuberculosisBioA(DAPA 合酶) 显示出抗结核活性,IC50为 30 nM。
T5315 TCA1

TCA-1,TCA 1

Antibacterial; Antibiotic Microbiology/Virology
TCA1 (TCA 1) 是一种小分子,具有抗耐药性和持续性结核病的活性。
T9734 InhA-IN-2

CDK Cell Cycle/Checkpoint
InhA-IN-2直接抑制 InhA,不需要过氧化氢酶过氧化物酶 KatG 的激活。
T0827 Cefsulodin sodium

Cefsulodine sodium,Sulcephalosporin,头孢磺啶钠

Antibacterial; Antibiotic Microbiology/Virology
Cefsulodin sodium (Sulcephalosporin) 是β内酰胺抗生素,对缘脓杆菌和肠杆菌有活性。
T12231 NITD-349

Others; Antibacterial Microbiology/Virology; Others
NITD-349 是MmpL3的抑制剂,它对毒性结核分枝杆菌 H37Rv 显示出高效的抗分枝杆菌活性,MIC50 为 23 nM。
T77730 QST4

Antifungal Microbiology/Virology
QST4 具有抗结核、抗真菌活性,在结核分枝杆菌 Mycobacterium tuberculosis H37Rv 中的 MIC 值为 6.25 μM。
T17176 Salicyl-AMS

Antibacterial Microbiology/Virology
Salicyl-AMS 是一种分支杆菌生长素生物合成抑制剂,能在体外缺铁的情况下抑制分枝杆菌的生长。
T60866 InhA-IN-3

Antibacterial Microbiology/Virology
InhA-IN-3 (TU13) 是一种有效的结核分枝杆菌InhA(烯酰 ACP 还原酶) 抑制剂,具有潜在的抗癌和抗增殖活性,可用于研究结核分枝杆菌感染。
T60073 Antimycobacterial agent-4

4-nitro-N-[4-(2-pyridyl)thiazol-2-yl]benzamide

Antibacterial Microbiology/Virology
Antimycobacterial agent-4 (4-nitro-N-[4-(2-pyridyl)thiazol-2-yl]benzamide) 对结核分枝杆菌具有抗菌活性。
T60877 Mtb ATP synthase-IN-1

ATPase Membrane transporter/Ion channel
Mtb ATP synthase-IN-1 是一种可口服的结核分枝杆菌 (Mtb) ATP 合成抑制剂,可用于研究结核分枝杆菌感染。
T61411 InhA-IN-4

Antibacterial Microbiology/Virology
InhA-IN-4 (TU14) 是一种有效的结核分枝杆菌InhA(烯酰 ACP 还原酶) 抑制剂,具有潜在的抗癌和抗增殖活性,可用于研究结核分枝杆菌感染。
T19464 N6,N6-Dimethyladenosine

N6,N6-二甲基腺苷

Nucleoside Antimetabolite/Analog Cell Cycle/Checkpoint; DNA Damage/DNA Repair
N6,N6-Dimethyladenosine 是存在于牛分枝杆菌 tRNA 中的一种修饰核糖核苷
T110951 Compound F0447-0245

Others Others
Antitubercular agent-33 是一种 2-氨基噻唑衍生物,对于结核分枝杆菌 (Mycobacterium tuberculosis,Mtb)显示出有效的抗结核活性。
T3642 TBA-354

TBA 354

Antibacterial; Antibiotic Microbiology/Virology
TBA-354 有抗结核作用,对结核分枝杆菌 H37Rv 菌株具有活性。
T1629 Rifapentine

MDL473,Rifapentina,Rifapentinum,DL 473,利福喷丁,Priftin,Cyclopentylrifampicin

DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Rifapentine (Rifapentinum) 是可用于肺结核的抗生素。
T72576 Transketolase-IN-4

Antibacterial Microbiology/Virology
Transketolase-IN-4 是一种转酮酶抑制剂 ,IC50值为3.9 μM。Transketolase-IN-4 对结核分枝杆菌 DXS 有抑制作用,IC50 为 114.1 μM。 Transketolase-IN-4 抑制 SW620、LS174T 和 MIA PaCa-2 的肿瘤细胞增殖。
T9830 GSK2556286

GSK286

Antibacterial Microbiology/Virology
GSK2556286 (GSK286) 是一种具有口服活性的结核分枝杆菌 (M. tuberculosis) 抑制剂。GSK2556286 对人巨噬细胞 (macrophages) 生长具有抑制作用,IC50值为 0.07 μM。GSK2556286对多重耐药 (MDR) 或广泛耐药 (XDR) 和药物敏感 (DS) 结核分枝杆菌均有效。
T77683 Methyl quinoline-2-carboxylate

Methyl 2-quinolinecarboxylate

Antibacterial Microbiology/Virology
Methyl quinoline-2-carboxylate (Methyl 2-quinolinecarboxylate) 对结合结核杆菌具有抑制作用。
T27453 GSK1733953A

DG70

Antibacterial Microbiology/Virology
GSK1733953A 可作为一种小分子结核分枝杆菌呼吸抑制剂,对 MenG 活性有抑制作用,IC50 值为 2.6 ± 0.6 μM。GSK1733953A 是一种具有选择性的联苯苯甲酰胺,对结核分枝杆菌去甲基萘醌甲基转移酶的催化甲基化有抑制作用,对结核分枝杆菌H4Rv的MIC为8.37 μg/ml,对耐药菌株的MIC为1.2至9.6 μg/ml。GSK1733953A 是治疗结核病的候选化合物。
T3582 BTZ043

Antibacterial; Antibiotic; DprE1 Microbiology/Virology; Others
BTZ043 是一种 DprE1 的抑制剂,它对结核分枝杆菌 H37Rv 和耻垢分枝杆菌具有纳摩尔杀菌活性,MIC 值分别为 2.3 nM 和 9.2 nM。
T67827 Urease Inhibitor 07

Others Others
Urease Inhibitor 07 是一种异取代金属蛋白酶抑制剂 , 对结核分枝杆菌H37Rv 菌株的潜在活性。
T11497 Ganfeborole HCl

GSK3036656 HCl,GSK656 HCl

Antibacterial Microbiology/Virology
Ganfeborole HCl (GSK3036656 HCl) 是一种具有抗结核活性的小分子化合物,是结核分枝杆菌(Mtb)亮氨酰-tRNA 合成酶(LeuRS;IC50:0.2 μM)的抑制剂。
T78745 Mtb-IN-2

Antibiotic Microbiology/Virology
Mtb-IN-2 是一种具有抗菌活性和低毒性的结核分枝杆菌(Mtb)的小分子化合物,干预蛋氨酸代谢过程,可用于研究结核病。
T0377 Clofazimine

NSC-141046,氯法齐明,氯苯吩嗪

DNA; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Clofazimine (NSC-141046) 是一种具有显著的抗炎效果的亚氨基酚嗪类染料,与其它抗分支杆菌药物联用来治疗AIDS 和克罗恩病。
T21023 Bedaquiline fumarate

TMC 207,R403323,TMC-207,TMC207,R-403323,贝达喹啉富马酸盐,R 403323

Antibacterial; Antibiotic Microbiology/Virology
Bedaquiline fumarate (TMC207) 是二芳基喹啉抗生素,作用于 ATP 合成酶,常用于结核杆菌感染的研究。
T0891 Dapsone

DDS,4,4‘-Sulfonyldianiline,氨苯砜,Bis(4-aminophenyl) sulfone,Sulphadione,4,4'-Diaminodiphenylsulfone,4-Aminophenyl sulfone

Reactive Oxygen Species; Antibacterial; Antibiotic; Parasite Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
Dapsone (Sulphadione) 是具有口服活性和血脑渗透通透性的磺酰类抗生素,具有抑菌、抗细菌和抗原虫活性。它有抗麻风活性,抑制麻风杆菌细胞提取物中叶酸的合成。它可研究皮肤病。
T2585 Bedaquiline

R207910,TMC207,贝达喹啉

Antibacterial; Antibiotic Microbiology/Virology
Bedaquiline (R207910) 是一种二芳基喹啉药物,能同时靶向 c-亚基和 ε-亚基,抑制结核分枝杆菌 (Mtb) F1FO-ATP 合酶。它具有解偶联活性和有用于耐多药结核病的潜力。
T1940 BTB06584

RAAS; ATPase Endocrinology/Hormones; Membrane transporter/Ion channel
BTB06584 是选择性依赖 IF1 的线粒体F1Fo-ATPase 抑制剂,可延迟缺血性细胞死亡。
T63056 Dovramilast

CC-11050

PDE Metabolism
Dovramilast (CC-11050) 是一种具有口服活性的磷酸二酯酶4(PDE4)抑制剂,,可以减少促炎介质和细胞因子的产生。Dovramilast 可用于研究结核分枝杆菌感染和红斑狼疮。
T67765 MenA-IN-2

Others Others
MenA-IN-2是一种有效的 1,4-二羟基-2-萘甲酸酯异戊二烯转移酶 (MenA) 抑制剂,对 MenA 的 IC50 值为 22 µM,对结核分枝杆菌 (Mtb) 的 GIC50 值为 10 µM。MenA-IN-2 Mtb 的持续传播具有抑制作用。
T68163 Timcodar

Antibacterial Microbiology/Virology
timcodar 是一种非 FKBP12 结合大环内酯衍生物,是外排泵抑制剂,具有抗菌活性,抑制脂质积累,抑制结核杆菌,可用于研究肥胖。
T0020 Sodium 4-aminosalicylate dihydrate

对氨基水杨酸钠二水合物,Sodium 4-Aminosalicylate,4-Amino-salicylic acid sodium salt

Free radical scavengers; NF-κB; Antibacterial; Antibiotic Microbiology/Virology; NF-κB; oxidation-reduction
Sodium 4-aminosalicylate dihydrate (4-Amino-salicylic acid sodium salt) 是一种抗耐药性结核化合物。
T125120 Cyclo(L-Pro-L-Val)

IκB/IKK; NOS; NF-κB; COX; Antibacterial Immunology/Inflammation; Microbiology/Virology; Neuroscience; NF-κB
Cyclo(L-Pro-L-Val) 是从辣椒溶杆菌AZ2和白斑分枝杆菌果实中提取出的 2,5-二酮哌嗪,具有抗炎活性,对植物病原微生物 (如 R. fascians LMG 3605) 具有毒性活性,能抑制革兰氏阳性植物病原菌。Cyclo(L-Pro-L-Val) 以浓度依赖性方式显著抑制了IKKα、IKKβ、IκBα和NF-κB 的磷酸化以及iNOS 和COX-2的活化,是治疗炎症相关疾病的潜在治疗剂。
T60774 NITD-916

NITD916,NITD 916

Antibiotic Microbiology/Virology
NITD-916 是一种具有口服活性和高度亲脂性的分枝杆菌烯酰还原酶 InhA 抑制剂,IC50 为 570 nM。NITD-916是一种有有效的 4-羟基-2-吡啶酮衍生物, 与 InhA 和 NADH 形成三元复合物,阻止进入脂肪酰基底物结合袋。NITD-916 具有抗结核活性。
T7877 Thiacetazone

氨硫脲,Diazam,Thioacetazone,Neustab,Neotibil

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Thiacetazone (Diazam) 是一种氨基硫脲抗结核剂,也是一种具有口服活性抗生素。它具有抗菌作用,可抑制结核分枝杆菌 H37Rv 的生长,MIC 值为 0.1 μg/mL。
T5400 Q203

IAP6,Telacebec

Antibacterial; Antibiotic Microbiology/Virology
Q203 (Telacebec)是一种中氮杂吡啶酰胺。 在培养基中抑制结核分枝杆菌H37Rv 活性的MIC50值为2.7 nM。
T68025 Zoliprofen

Others Others
Zoliprofen 是一种一种高效的且可口服的非甾体抗炎剂,具有抗炎、解热和镇痛活性,对角叉菜素、制霉菌素、刀豆球蛋白A 诱导的大鼠爪水肿,以及抗大鼠兔血清诱导的骨折或背皮水肿具有抑制作用。Zoliprofen 在大鼠和兔子中对胶原蛋白或花生四烯酸引起的血小板聚集方面比布洛芬和非诺洛芬有效20倍。Zoliprofen 对小鼠内毒素诱导的腹泻和花生四烯酸诱导的兔急性死亡抑制作用显著。
T40520 Thiophene-2

Thiophene-2,TP2

Others Others
Thiophene-2 (TP2) is a targeted inhibitor of polyketide synthase 13 (Pks13), specifically designed to disrupt mycolic acid biosynthesis. By doing so, it effectively induces rapid cell death in mycobacteria. Thiophene-2 demonstrates notable anti-tuberculosis activity and exhibits a minimum inhibitory concentration (MIC) value of 1 μM against Mycobacterium tuberculosis.
T24765 SB-790594-A

SB790594A,SB 790594 A

Others Others
SB-790594-A is a non-cytotoxic Mycobacterium tuberculosis H37Rv inhibitor.
T31688 Ethambutol, (R,R)-

L-Ethambutol

Others Others
Ethambutol, (R, R)- can be used to treat tuberculosis. It is usually used in combination with other tuberculosis medications. It may also be used to treat Mycobacterium avium complex, and Mycobacterium kansasii.
T27477 GSK366A

Others Others
GSK366A is an anti-TB agent against Mycobacterium bovis BCG and Mycobacterium tuberculosis, targeting MmpL3 and inhibiting EchA6.
T25468 GSK1829820A

GSK-1829820-A,GSK 1829820A,GSK 1829820 A,GSK-1829820A

Others Others
GSK1829820A is a Mycobacterium tuberculosis H37Rv non-cytotoxic inhibitor.
T29701 AG 85

AG85,AG-85

Others Others
AG 85 is a major secretion protein of Mycobacterium tuberculosis.
T34177 Pseudopterosin E

Others Others
Pseudopterosin E can act towards Mycobacterium tuberculosis and other pathogens.
T11983 MDRTB-IN-1

Others Others
MDRTB-IN-1 (5aα) is an antibiotic which is against Mycobacterium tuberculosis H37Rv(MIC90 :10.5 μM).
T11594 I2906

Others Others
I2906 showed antimycobacterial and cytotoxic activity against mycobacterium tuberculosis.
T24397 ZTB23(R)

ZTB 23(R),ZTB-23(R)

Others Others
ZTB23(R) is the first potent and selective inhibitor of Mycobacterium tuberculosis Zmp1.

化合物

BM212
Cat.No: T7342
Synonym:
Target: Antibacterial
Dup-721
Cat.No: T38359
Synonym:
Target: Antibacterial
AU1235
Cat.No: T10411
Synonym:
Target: Antibacterial
ML406
Cat.No: T8694
Synonym:
Target: Antibacterial, Antibiotic
TCA1
Cat.No: T5315
Synonym: TCA-1,TCA 1
Target: Antibacterial, Antibiotic
InhA-IN-2
Cat.No: T9734
Synonym:
Target: CDK
Cefsulodin sodium
Cat.No: T0827
Synonym: Cefsulodine sodium,Sulcephalosporin,头孢磺啶钠
Target: Antibacterial, Antibiotic
NITD-349
Cat.No: T12231
Synonym:
Target: Others, Antibacterial
QST4
Cat.No: T77730
Synonym:
Target: Antifungal
Salicyl-AMS
Cat.No: T17176
Synonym:
Target: Antibacterial
InhA-IN-3
Cat.No: T60866
Synonym:
Target: Antibacterial
Antimycobacterial agent-4
Cat.No: T60073
Synonym: 4-nitro-N-[4-(2-pyridyl)thiazol-2-yl]benzamide
Target: Antibacterial
Mtb ATP synthase-IN-1
Cat.No: T60877
Synonym:
Target: ATPase
InhA-IN-4
Cat.No: T61411
Synonym:
Target: Antibacterial
N6,N6-Dimethyladenosine
Cat.No: T19464
Synonym: N6,N6-二甲基腺苷
Target: Nucleoside Antimetabolite/Analog
Compound F0447-0245
Cat.No: T110951
Synonym:
Target: Others
TBA-354
Cat.No: T3642
Synonym: TBA 354
Target: Antibacterial, Antibiotic
Rifapentine
Cat.No: T1629
Synonym: MDL473,Rifapentina,Rifapentinum,DL 473,利福喷丁,Priftin,Cyclopentylrifampicin
Target: DNA/RNA Synthesis, Antibacterial, Antibiotic
Transketolase-IN-4
Cat.No: T72576
Synonym:
Target: Antibacterial
GSK2556286
Cat.No: T9830
Synonym: GSK286
Target: Antibacterial
Methyl quinoline-2-carboxylate
Cat.No: T77683
Synonym: Methyl 2-quinolinecarboxylate
Target: Antibacterial
GSK1733953A
Cat.No: T27453
Synonym: DG70
Target: Antibacterial
BTZ043
Cat.No: T3582
Synonym:
Target: Antibacterial, Antibiotic, DprE1
Urease Inhibitor 07
Cat.No: T67827
Synonym:
Target: Others
Ganfeborole HCl
Cat.No: T11497
Synonym: GSK3036656 HCl,GSK656 HCl
Target: Antibacterial
Mtb-IN-2
Cat.No: T78745
Synonym:
Target: Antibiotic
Clofazimine
Cat.No: T0377
Synonym: NSC-141046,氯法齐明,氯苯吩嗪
Target: DNA, Antibacterial, Antibiotic
Bedaquiline fumarate
Cat.No: T21023
Synonym: TMC 207,R403323,TMC-207,TMC207,R-403323,贝达喹啉富马酸盐,R 403323
Target: Antibacterial, Antibiotic
Dapsone
Cat.No: T0891
Synonym: DDS,4,4‘-Sulfonyldianiline,氨苯砜,Bis(4-aminophenyl) sulfone,Sulphadione,4,4'-Diaminodiphenylsulfone,4-Aminophenyl sulfone
Target: Reactive Oxygen Species, Antibacterial, Antibiotic, Parasite
Bedaquiline
Cat.No: T2585
Synonym: R207910,TMC207,贝达喹啉
Target: Antibacterial, Antibiotic
BTB06584
Cat.No: T1940
Synonym:
Target: RAAS, ATPase
Dovramilast
Cat.No: T63056
Synonym: CC-11050
Target: PDE
MenA-IN-2
Cat.No: T67765
Synonym:
Target: Others
Timcodar
Cat.No: T68163
Synonym:
Target: Antibacterial
Sodium 4-aminosalicylate dihydrate
Cat.No: T0020
Synonym: 对氨基水杨酸钠二水合物,Sodium 4-Aminosalicylate,4-Amino-salicylic acid sodium salt
Target: Free radical scavengers, NF-κB, Antibacterial, Antibiotic
Cyclo(L-Pro-L-Val)
Cat.No: T125120
Synonym:
Target: IκB/IKK, NOS, NF-κB, COX, Antibacterial
NITD-916
Cat.No: T60774
Synonym: NITD916,NITD 916
Target: Antibiotic
Thiacetazone
Cat.No: T7877
Synonym: 氨硫脲,Diazam,Thioacetazone,Neustab,Neotibil
Target: Others, Antibacterial, Antibiotic
Q203
Cat.No: T5400
Synonym: IAP6,Telacebec
Target: Antibacterial, Antibiotic
Zoliprofen
Cat.No: T68025
Synonym:
Target: Others
Thiophene-2
Cat.No: T40520
Synonym: Thiophene-2,TP2
Target: Others
SB-790594-A
Cat.No: T24765
Synonym: SB790594A,SB 790594 A
Target: Others
Ethambutol, (R,R)-
Cat.No: T31688
Synonym: L-Ethambutol
Target: Others
GSK366A
Cat.No: T27477
Synonym:
Target: Others
GSK1829820A
Cat.No: T25468
Synonym: GSK-1829820-A,GSK 1829820A,GSK 1829820 A,GSK-1829820A
Target: Others
AG 85
Cat.No: T29701
Synonym: AG85,AG-85
Target: Others
Pseudopterosin E
Cat.No: T34177
Synonym:
Target: Others
MDRTB-IN-1
Cat.No: T11983
Synonym:
Target: Others
I2906
Cat.No: T11594
Synonym:
Target: Others
ZTB23(R)
Cat.No: T24397
Synonym: ZTB 23(R),ZTB-23(R)
Target: Others
Cat. No. Product Name Target Signaling Pathways
T5780 HYPOCRELLIN B

Apoptosis; Parasite; Antifungal Apoptosis; Microbiology/Virology
Hypocrellin B 是从真菌Hypocrella bambusae 和Shiraia bambusicola 中分离得到的一种感光颜料,可用于癌症光动力研究。它是一个凋亡诱导剂,还拥有抗菌和抗利什曼活性。
T1426 Pyrazinamide

Pyrazinoic acid amide,Pyrazinecarboxamide,吡嗪酰胺

Antibacterial; Antibiotic; Autophagy; Fatty Acid Synthase Autophagy; Metabolism; Microbiology/Virology
Pyrazinamide (Pyrazinecarboxamide) 是一种口服抗结核类抗生素。它是一种前药,通过结核分枝杆菌pncA 基因编码的 PZase/烟酰胺酶转化为活性吡嗪酸形式。
TN2730 2,5-Dihydroxybenzaldehyde

Gentisaldehyde,2,5-二羟基苯甲醛

Anti-infection; Antibacterial Microbiology/Virology
2,5-Dihydroxybenzaldehyde (Gentisaldehyde) 是一种天然抗微生物剂,可抑制Mycobacterium avium subsp. paratuberculosis 的生长。它还抑制金黄色葡萄球菌菌株,MIC50为 500 mg/L。
TN2279 Totarol

(+)-Totarol,桃柁酚

Antibacterial; Antifection Microbiology/Virology
Totarol ((+)-Totarol) 对几种致病性革兰氏阳性细菌、结核分枝杆菌具有抗菌作用。
TN5503 Linaroside

Antibacterial Microbiology/Virology
Linaroside 在 6.25 microg mL(-1) 浓度下对结核分枝杆菌、菌株 H(37)Rv 的抗分枝杆菌活性表现出 30%的抑制作用。
T1419 Azithromycin hydrate

CP-62993 dihydrate,阿奇霉素二水物,Azithromycin dihydrate,阿奇霉素二水合物

ribosome; Antibacterial; Antibiotic; Autophagy Autophagy; Microbiology/Virology
Azithromycin hydrate (CP-62993 dihydrate) 是一种大环内酯抗生素,可研究细菌感染。
TN1466 Canthin-6-one

NSC 103003

Antifungal Microbiology/Virology
Canthin-6-one(NSC 103003) 是一种从 Allium neapolitanum 分离出来的生物碱,具有抗菌活性,对结核分枝杆菌具有抑制作用。
T5041 Faropenem sodium

法罗培南,法罗培南钠

Antibacterial; Antibiotic Microbiology/Virology
Faropenem sodium 是一种口服生物可利用的青霉烯类抗生素,能有效杀灭结核分枝杆菌,治疗结核病和社区获得性肺炎。
T5S1285 (+)-(3R,8S)-Falcarindiol

Falcarindiol,镰叶芹二醇

Others Others
(+)-(3R,8S)-Falcarindiol 是一种从胡萝卜中得到的聚乙炔,有抗炎、抗肿瘤和抗脂质过氧化活性。它具有抗分歧杆菌作用,对Mycobacterium tuberculosisH37Ra 的 MIC 和 IC50值分别为 24 μM 和 6 μM。
TN3207 7,3′,4′-Tri-O-methyleriodictyol

Antibiotic Microbiology/Virology
7,3′,4′-Tri-O-methyleriodictyol (7,3',4'-Tri-O-methyleriodictyol) 是一种从Pogostemon cablin的甲醇提取物中分离得到的,具有抗菌、抗氧化、抗肿瘤和抗原生动物活性,抑制结核分枝杆菌感染 ,抑制 SOS 诱导活性。
T5722 Nevadensin

Pedunculin,石吊兰素,5,7-二羟基-6,8,4'-三甲氧基黄酮

Anti-infection; Antibacterial Microbiology/Virology
Nevadensin 是一种重要的草本成分,可抑制雌二醇的生物活化。 它具有抗结核分枝杆菌、镇咳、抗炎、抗高血压等多种药理作用。
TN2233 Spathulenol

Antioxidant; Antifungal Microbiology/Virology; oxidation-reduction
Spathulenol 是一种来自 Aristolochia yunnanensis 的天然成分,具有抗炎、抗氧化、抗增殖、抗溃疡和抗分枝杆菌活性。 Spathulenol 在 DPPH 系统中显示出显著的抗氧化活性,IC50 为 85.60 μg/mL。
TN6714 Geranylgeraniol

FT-0626663,Tetraprenol,CJ24095,CJ 24095,FT0626663,香叶基香叶醇,CJ-24095

Apoptosis Apoptosis
Geranylgeraniol (FT0626663) 是一种类异戊二烯,存在于水果、蔬菜和谷物中,包括大米。 Geranylgeraniol (FT0626663) 抑制生长并诱导各种肿瘤细胞的凋亡。 Geranylgeraniol (FT0626663) 保护单核细胞免受他汀类药物诱导的细胞毒性并抑制分枝杆菌的生长。
TN1019 Beta-mangostin

β-Mangostin,beta-倒捻子素

Apoptosis; Antibacterial; Parasite Apoptosis; Microbiology/Virology
Beta-mangostin (β-Mangostin) 是存在 Cratoxylum arborescens 中的一种氧杂蒽酮类天然产物,有抗癌和抗菌活性,对结核分枝杆菌的 MIC 值为 6.25 μg/mL。它在体外有抗疟活性,对恶性疟原虫的 IC50值为 3.00 μg/mL。
TN2086 Piperlotine A

Antibacterial Microbiology/Virology
Piperlotine A 是一种可从罗洛胡椒中提取得到的生物碱,具有抗血小板聚集活性。Piperlotine A 在体外试验中显示出对结核分枝杆菌的抑制作用,MIC 值为 50 ug/mL。
T3S1612 kuwanon G

桑黄酮G,Moracenin B,桑黄酮 G,Kuwanone G

Phosphatase; Antibacterial; Bombesin Receptor; AChR; AChE; Glucosidase GPCR/G Protein; Metabolism; Microbiology/Virology; Neuroscience
Kuwanon G (Moracenin B) 是一种从桑树中得到的黄酮类蛙皮素受体拮抗剂,具有杀菌作用。
T14329 Ascamycin

Nucleoside Antimetabolite/Analog; Others; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others
Ascamycin 是一种由链霉菌属产生的 5'-O-磺酰胺核糖核苷抗生素,对黄单胞菌类显示出选择性的抗菌活性,对柠檬黄单胞菌、口蹄疫黄单胞菌和噬菌体具有抑制作用,MIC 值分别为0.4μg/mL、12.5μg/mL 和12.5μg/mL。
TN5684 5,6-Desmethylenedioxy-5-methoxyaglalactone

5,6-Desmethylenedioxy-5-methoxyaglalactone is cytotoxic to small cell lung cancer (NCI-H187) cell line. It has antimycobacterial activity against Mycobacterium tuberculosis H(37)Ra.
T75564 Pomolic acid 3-acetate

Others Others
Pomolic acid 3-acetate 是一种抗结核 (antitubercular) 剂,对 Mycobacterium tuberculosisH37Rv 的 MIC 为 32 μM。
TN1561 Dehydroglaucine

Antifection Microbiology/Virology
Dehydroglaucine is an acetylcholinesterase inhibitor, it shows antimicrobial activity against Staphylococcus aureus, Mycobacterium smegmatis, Candida albicans, and Aspergillus niger.
TN2271 Thalrugosaminine

Antifection Microbiology/Virology
Thalrugosaminine shows promising antibacterial activity with MIC values of 64-128ug/ml and Staphylococcus species is the most sensitive strains. Thalrugosaminine possesses hypotensive activity in rabbits and is active against Mycobacterium smegmatis.
TN5648 Porson

Porson exhibited anti-tubercular activity against Mycobacterium tuberculosis H37Rv in vitro and MICs values of 40.0 μg/mL.
TN4944 Santamarine

Caspase Apoptosis; Proteases/Proteasome
Santamarine has significant anticancer activity, can inhibit L1210 cells because of its cytotoxic,cytostatic and blocking mitosis and reducing uptake of thymidine. Santamarine and reynosin show bactericidal activity against clinical strains of Mycobacterium tuberculosis.
TN4336 Isothymusin

Antifection Microbiology/Virology
Isothymusin( MIC= 200 microg/mL) exhibits inhibition activity against Mycobacterium tuberculosis. It ( IC50=7.7 microg/mL ) exhibits antioxidant activity against the radical scavenging ability of DPPH.
TN3907 Pinosylvin monomethyl ether

(E)-3-Hydroxy-5-methoxystilbene

Antifection Microbiology/Virology
(E)-3-Hydroxy-5-methoxystilbene possesses inhibitory activity against several Gram-positive bacteria, including isolates of methicillin-resistant Staphylococcus aureus (MRSA), Mycobacterium bovis BCG, and avirulent Bacillusanthracis (Sterne strain), among
TN5657 Goniotriol

Goniotriol shows antimycobacterial activity against Mycobacterium tuberculosis (MIC =100 microg/mL). It exhibits antiplasmodial activity against Plasmodium falciparum (IC50=2.6 microg/mL). Goniotriol shows cytotoxicity against cancer cells, KB, BC1, NCI-H
TN4776 Physalin D

TNF; Antifection Apoptosis; Microbiology/Virology
Physalin D shows antimalarial activity; it also exhibits a minimum inhibitory concentration value (MIC) against Mycobacterium tuberculosis H(37)Rv strain of 32 microg/mL. Physalin D displays considerable cytotoxicity against several cancer cell lines. It
TN3924 Eichlerialactone

Others Others
Eichlerialactone and ethyl eichlerianoate show antimycobacterial activity against mycobacterium tuberculosis H37Ra, with minimum inhibitory concentration in the range of 25-50ug/mL; eichlerialactone exhibits good antibacterial activity against both the Gr
TN6069 Thalidezine

Thalidezine, a novel AMPK activator, eliminates apoptosis-resistant cancer cells through energy-mediated autophagic cell death, it can inhibit the growth of mouse L1210 cells in vitro. Thalidezine possesses antimicrobial activity against Mycobacterium sme
TN4953 Sativan

三叶草

Antifection Microbiology/Virology
Sativan possesses a broad spectrum of antimicrobial activity against bacteria and phytopathogenic fungi, it exhibits antituberculosis activity against Mycobacterium tuberculosis H37Rv, with the MIC value of 50 ug/mL.
TN3560 Cabralealactone

Antifection Microbiology/Virology
Cabralealactone displays antimycobacterial activity against Mycobacterium tuberculosis, it is weakly cytotoxic to a breast cancer (BC) cell line, it is moderately active against a small-cell lung cancer (NCI-H187) cell line.
TN3559 Cabraleahydroxylactone

HSV Microbiology/Virology
Cabraleahydroxylactone displays antimycobacterial activity against Mycobacterium tuberculosis, it is weakly cytotoxic to a breast cancer (BC) cell line.It shows antiviral activity against herpes simplex virus type-1 with an IC50 value of 3.20 ug/mL, in comparison with the standard acyclovir (IC50=1.90ug/mL).
T75489 Mildiomycin

Others Others
Mildiomycin是一种针对大麦白粉病具有活性的链轮丝菌抗生素。该化合物能够抑制部分分枝杆菌和红桃菌的生长,然而,对大部分真菌和细菌则显示出无效性。
TN3557 Cabraleadiol

ATPase; Antifection Membrane transporter/Ion channel; Microbiology/Virology
Cabraleadiol displays antimycobacterial activity against Mycobacterium tuberculosis, it also is weakly cytotoxic to a breast cancer (BC) cell line. Cabraleadiol inhibits photosystem II (PS II) and induces the appearance of small G band which is related wi
T75631 Ganorbiformin B

Others Others
Ganorbiformin B是一种具有与灵芝酸相同羊毛甾烷骨架的羊毛甾烷三萜类化合物。其C-3差向异构体灵芝酸T对结核分枝杆菌H37Ra显示出强抗分枝杆菌活性。
T75633 (22S,24E)-3β,22-Diacetoxylanosta-7,9(11),24-trien-26-oic acid

Others Others
(22S,24E)-3β,22-Diacetoxylanosta-7,9(11),24-trien-26-oic acid (compound 15) 为具有抗结核活性的化合物,对结核分枝杆H37Ra的最小抑菌浓度(MIC)为12.5 μg/mL,并展现出对Vero细胞的细胞毒性,其半数抑制浓度(IC50)值为32 μM[1]。
TN5014 Shoreic acid

Antifection; HSV Microbiology/Virology
Shoreic acid exhibits antibacterial activity against E. coli, P. aeruginosa, S. aureus, and B. subtilis with activity indices (AI) of 0.2, 0.3, 0.5 and 0.4, respectively, it also shows antifungal activity against C. albicans and T. mentagrophytes with AI
T72742 (-)-Pinocembrin

(-)-乔松素

Others Others
(-)-Pinocembrin 对 H37Ra 结核分枝杆菌展示了抗菌活性,无论是休眠还是活跃期,其 IC50 值分别为1.11 mg/mL 和 1.21 mg/mL。作为一种抗增殖剂,(-)-Pinocembrin 对于 THP-1、A549、Panc-1、HeLa 和 MCF7 细胞系,IC50 值范围为 1.88 至 11.00 mg/mL。
TN1694 Gliotoxin

Apoptosis; NF-κB; Wnt/beta-catenin; COX; PKA; Antibacterial; Antifection Apoptosis; Cytoskeletal Signaling; Immunology/Inflammation; Microbiology/Virology; Neuroscience; NF-κB; Stem Cells; Tyrosine Kinase/Adaptors
Gliotoxin 是一种次生代谢产物,由A. fumigatus 分泌,可以抑制巨噬细胞的吞噬作用和其他免疫细胞的免疫功能。它通过阻止 IκB 降解来抑制诱导型NF-κB 活性,从而诱导宿主细胞凋亡。它可以激活PKA 并增加细胞内 cAMP 浓度,调节肌动蛋白细胞骨架重排以促进A. fumigatus 内化到肺上皮细胞。
TN1378 α-Viniferin

ALPHA-VINIFERIN,Alpha-葡萄素

P450; NO Synthase; Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism
α-Viniferin 也称为2-芳基苯并呋喃类黄酮,是前列腺素H2合成酶抑制剂。具有抗阿尔茨海默病、抗结核、抗肿瘤、抗炎、抗糖尿病等多种药理活性
T38330 Collinin

Others Others
Collinin is a coumarin that has been found in Z. schinifolium and has diverse biological activities.1,2,3,4 It is active against drug-susceptible and -resistant strains of M. tuberculosis (MIC50s = 3.13-6.25 μg/ml).1 Collinin inhibits LPS-induced nitric oxide (NO) production (IC50 = 5.9 μM) and reduces COX-2 protein levels in RAW 264.7 cells.2 It completely inhibits aggregation of isolated rabbit platelets induced by arachidonic acid , collagen, or platelet activating factor (PAF) when used at a...

天然产物

HYPOCRELLIN B
Cat.No: T5780
Synonym:
Target: Apoptosis, Parasite, Antifungal
Pyrazinamide
Cat.No: T1426
Synonym: Pyrazinoic acid amide,Pyrazinecarboxamide,吡嗪酰胺
Target: Antibacterial, Antibiotic, Autophagy, Fatty Acid Synthase
2,5-Dihydroxybenzaldehyde
Cat.No: TN2730
Synonym: Gentisaldehyde,2,5-二羟基苯甲醛
Target: Anti-infection, Antibacterial
Totarol
Cat.No: TN2279
Synonym: (+)-Totarol,桃柁酚
Target: Antibacterial, Antifection
Linaroside
Cat.No: TN5503
Synonym:
Target: Antibacterial
Azithromycin hydrate
Cat.No: T1419
Synonym: CP-62993 dihydrate,阿奇霉素二水物,Azithromycin dihydrate,阿奇霉素二水合物
Target: ribosome, Antibacterial, Antibiotic, Autophagy
Canthin-6-one
Cat.No: TN1466
Synonym: NSC 103003
Target: Antifungal
Faropenem sodium
Cat.No: T5041
Synonym: 法罗培南,法罗培南钠
Target: Antibacterial, Antibiotic
(+)-(3R,8S)-Falcarindiol
Cat.No: T5S1285
Synonym: Falcarindiol,镰叶芹二醇
Target: Others
7,3′,4′-Tri-O-methyleriodictyol
Cat.No: TN3207
Synonym:
Target: Antibiotic
Nevadensin
Cat.No: T5722
Synonym: Pedunculin,石吊兰素,5,7-二羟基-6,8,4'-三甲氧基黄酮
Target: Anti-infection, Antibacterial
Spathulenol
Cat.No: TN2233
Synonym:
Target: Antioxidant, Antifungal
Geranylgeraniol
Cat.No: TN6714
Synonym: FT-0626663,Tetraprenol,CJ24095,CJ 24095,FT0626663,香叶基香叶醇,CJ-24095
Target: Apoptosis
Beta-mangostin
Cat.No: TN1019
Synonym: β-Mangostin,beta-倒捻子素
Target: Apoptosis, Antibacterial, Parasite
Piperlotine A
Cat.No: TN2086
Synonym:
Target: Antibacterial
kuwanon G
Cat.No: T3S1612
Synonym: 桑黄酮G,Moracenin B,桑黄酮 G,Kuwanone G
Target: Phosphatase, Antibacterial, Bombesin Receptor, AChR, AChE, Glucosidase
Ascamycin
Cat.No: T14329
Synonym:
Target: Nucleoside Antimetabolite/Analog, Others, Antibacterial, Antibiotic
5,6-Desmethylenedioxy-5-methoxyaglalactone
Cat.No: TN5684
Synonym:
Target:
Pomolic acid 3-acetate
Cat.No: T75564
Synonym:
Target: Others
Dehydroglaucine
Cat.No: TN1561
Synonym:
Target: Antifection
Thalrugosaminine
Cat.No: TN2271
Synonym:
Target: Antifection
Porson
Cat.No: TN5648
Synonym:
Target:
Santamarine
Cat.No: TN4944
Synonym:
Target: Caspase
Isothymusin
Cat.No: TN4336
Synonym:
Target: Antifection
Pinosylvin monomethyl ether
Cat.No: TN3907
Synonym: (E)-3-Hydroxy-5-methoxystilbene
Target: Antifection
Goniotriol
Cat.No: TN5657
Synonym:
Target:
Physalin D
Cat.No: TN4776
Synonym:
Target: TNF, Antifection
Eichlerialactone
Cat.No: TN3924
Synonym:
Target: Others
Thalidezine
Cat.No: TN6069
Synonym:
Target:
Sativan
Cat.No: TN4953
Synonym: 三叶草
Target: Antifection
Cabralealactone
Cat.No: TN3560
Synonym:
Target: Antifection
Cabraleahydroxylactone
Cat.No: TN3559
Synonym:
Target: HSV
Mildiomycin
Cat.No: T75489
Synonym:
Target: Others
Cabraleadiol
Cat.No: TN3557
Synonym:
Target: ATPase, Antifection
Ganorbiformin B
Cat.No: T75631
Synonym:
Target: Others
(22S,24E)-3β,22-Diacetoxylanosta-7,9(11),24-trien-26-oic acid
Cat.No: T75633
Synonym:
Target: Others
Shoreic acid
Cat.No: TN5014
Synonym:
Target: Antifection, HSV
(-)-Pinocembrin
Cat.No: T72742
Synonym: (-)-乔松素
Target: Others
Gliotoxin
Cat.No: TN1694
Synonym:
Target: Apoptosis, NF-κB, Wnt/beta-catenin, COX, PKA, Antibacterial, Antifection
α-Viniferin
Cat.No: TN1378
Synonym: ALPHA-VINIFERIN,Alpha-葡萄素
Target: P450, NO Synthase, Prostaglandin Receptor
Collinin
Cat.No: T38330
Synonym:
Target: Others
Cat. No. Product Name Species Expression System
TMPH-03022 PstP Protein, Mycobacterium tuberculosis, Recombinant

PP2C-family Ser/Thr phosphatase,pstP,Serine/threonine protei...

Mycobacterium tuberculosis E. coli
Plays an important role in regulating cell division and growth by reversible phosphorylation signaling. May play important roles in regulating cellular metabolism and signaling pathways, which could mediate the growth and development of the cell. Plays a role in establishing and maintaining infection. PstP Protein, Mycobacterium tuberculosis, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 25.3 kDa and the accession number is P9WHW4.
TMPH-03000 ATase Protein, Mycobacterium tuberculosis, Recombinant (His)

ATase,Glutamine phosphoribosylpyrophosphate amidotransferase...

Mycobacterium tuberculosis E. coli
Catalyzes the formation of phosphoribosylamine from phosphoribosylpyrophosphate (PRPP) and glutamine. ATase Protein, Mycobacterium tuberculosis, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 56.5 kDa and the accession number is P9WHQ6.
TMPH-03008 ENR Protein, Mycobacterium tuberculosis, Recombinant (His)

FAS-II enoyl-ACP reductase,Enoyl-ACP reductase,Enoyl-[acyl-c...

Mycobacterium tuberculosis E. coli
ENR Protein, Mycobacterium tuberculosis, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 32.6 kDa and the accession number is P9WGR0.
TMPH-03010 EsxB Protein, Mycobacterium tuberculosis, Recombinant (His)

ESAT-6-like protein EsxB,10 kDa culture filtrate antigen CFP...

Mycobacterium tuberculosis P. pastoris (Yeast)
A secreted protein. Acts as a strong host T-cell antigen. Involved in translocation of bacteria from the host (human) phagolysosome to the host cytoplasm. Might serve as a chaperone to prevent uncontrolled membrane lysis by its partner EsxA.
TMPH-02999 uL2 Protein, Mycobacterium tuberculosis, Recombinant (His)

rplB,50S ribosomal protein L2,Large ribosomal subunit protei...

Mycobacterium tuberculosis E. coli
One of the primary rRNA binding proteins. Required for association of the 30S and 50S subunits to form the 70S ribosome, for tRNA binding and peptide bond formation. It has been suggested to have peptidyltransferase activity; this is somewhat controversial. Makes several contacts with the 16S rRNA in the 70S ribosome. uL2 Protein, Mycobacterium tuberculosis, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 34.7 kDa and the accession ...
TMPH-03021 PstP Protein, Mycobacterium tuberculosis, Recombinant (His)

Mycobacterial Ser/Thr phosphatase,PP2C-family Ser/Thr phosph...

Mycobacterium tuberculosis E. coli
Plays an important role in regulating cell division and growth by reversible phosphorylation signaling. May play important roles in regulating cellular metabolism and signaling pathways, which could mediate the growth and development of the cell. Plays a role in establishing and maintaining infection.
TMPH-03196 PYCR Protein, Mycobacterium tuberculosis, Recombinant (His & Myc)

PCA reductase,Pyrroline-5-carboxylate reductase,proC

Mycobacterium tuberculosis E. coli
Catalyzes the reduction of 1-pyrroline-5-carboxylate (PCA) to L-proline. PYCR Protein, Mycobacterium tuberculosis, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 37.6 kDa and the accession number is P9WHU7.
TMPH-02996 KsdD Protein, Mycobacterium smegmatis, Recombinant (His & Myc)

3-oxosteroid 1-dehydrogenase,3-keto-Delta(4)-steroid Delta(1...

Mycolicibacterium smegmatis E. coli
Catalyzes the elimination of the C-1 and C-2 hydrogen atoms of the A-ring from the polycyclic ring structure of 3-ketosteroids. Is also involved in the formation of 1,4-androstadiene-3,17-dione (ADD) from 4-androstene-3,17-dione (AD) to. KsdD Protein, Mycobacterium smegmatis, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 68.9 kDa and the accession number is A0R4S9.
TMPH-00758 EspK Protein, Mycobacterium tuberculosis, Recombinant (His & Myc)

espK,ESX-1 secretion-associated protein EspK

Mycobacterium tuberculosis E. coli
May act as a chaperone that facilitates EspB secretion through an interaction with EccCb1.
TMPH-03016 MPT64 Protein, Mycobacterium tuberculosis, Recombinant (His)

Immunogenic protein MPT64,Antigen MPT64,mpt64

Mycobacterium tuberculosis P. pastoris (Yeast)
MPT64 Protein, Mycobacterium tuberculosis, Recombinant (His) is expressed in Yeast.
TMPH-03004 Ag85A Protein, Mycobacterium tuberculosis, Recombinant (His)

Diacylglycerol acyltransferase/mycolyltransferase Ag85A,Fibr...

Mycobacterium tuberculosis E. coli
Ag85A Protein, Mycobacterium tuberculosis, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 34.1 kDa and the accession number is P9WQP2.
TMPH-03001 MT2731 Protein, Mycobacterium tuberculosis, Recombinant (His)

Antitoxin MT2731

Mycobacterium tuberculosis P. pastoris (Yeast)
Antitoxin component of a type II toxin-antitoxin (TA) system. Neutralizes the effect of cognate toxin MT2730. MT2731 Protein, Mycobacterium tuberculosis, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 9.7 kDa and the accession number is P9WJ10.
TMPH-02998 Porin MspA Protein, Mycobacterium smegmatis, Recombinant (His)

mspA,Porin MspA

Mycobacterium smegmatis E. coli
Porin MspA Protein, Mycobacterium smegmatis, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 25.4 kDa and the accession number is A0QR29.
TMPH-03612 SodC Protein, Mycobacterium tuberculosis, Recombinant (His & Myc)

Superoxide dismutase [Cu-Zn],sodC

Mycobacterium tuberculosis E. coli
Destroys radicals which are normally produced within the cells and which are toxic to biological systems. May play a role in favoring mycobacterial survival in phagocytes. SodC Protein, Mycobacterium tuberculosis, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 28.1 kDa and the accession number is P9WGE8.
TMPH-02993 DisA Protein, Mycobacterium paratuberculosis, Recombinant (His & Myc)

disA,c-di-AMP synthase,DNA integrity scanning protein DisA,D...

Mycobacterium paratuberculosis E. coli
Participates in a DNA-damage check-point. DisA forms globular foci that rapidly scan along the chromosomes searching for lesions.; Has also diadenylate cyclase activity, catalyzing the condensation of 2 ATP molecules into cyclic di-AMP (c-di-AMP). c-di-AMP likely acts as a signaling molecule that may couple DNA integrity with a cellular process. DisA Protein, Mycobacterium paratuberculosis, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predict...
TMPH-03019 MPT51 Protein, Mycobacterium tuberculosis, Recombinant (His & SUMO)

MPT51/MPB51 antigen,mpt51

Mycobacterium tuberculosis E. coli
May have a role in host tissue attachment, whereby ligands may include the serum protein fibronectin and small sugars. MPT51 Protein, Mycobacterium tuberculosis, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 44.5 kDa and the accession number is P9WQN6.
TMPH-02995 MAP_1030 Protein, Mycobacterium paratuberculosis, Recombinant (His)

Probable transcriptional regulatory protein MAP_1030

Mycobacterium paratuberculosis P. pastoris (Yeast)
MAP_1030 Protein, Mycobacterium paratuberculosis, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 28.8 kDa and the accession number is P62039.
TMPH-03018 MeTAP1 Protein, Mycobacterium tuberculosis, Recombinant (His)

Peptidase M,map-1,Methionine aminopeptidase 1

Mycobacterium tuberculosis E. coli
Removes the N-terminal methionine from nascent proteins. The N-terminal methionine is often cleaved when the second residue in the primary sequence is small and uncharged (Met-Ala-, Cys, Gly, Pro, Ser, Thr, or Val). Requires deformylation of the N(alpha)-formylated initiator methionine before it can be hydrolyzed. MeTAP1 Protein, Mycobacterium tuberculosis, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 32.9 kDa and the accession ...
TMPH-03012 HBHA Protein, Mycobacterium tuberculosis, Recombinant (His & Myc)

Adhesin,Heparin-binding hemagglutinin,hbhA

Mycobacterium tuberculosis E. coli
Required for extrapulmonary dissemination. Mediates adherence to epithelial cells by binding to sulfated glycoconjugates present at the surface of these cells. HBHA Protein, Mycobacterium tuberculosis, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 28.8 kDa and the accession number is P9WIP8.
TMPH-02997 Dps Protein, Mycobacterium smegmatis, Recombinant (His & SUMO)

Neutrophil-activating protein A,NAP A,HP-NAP,Bacterioferriti...

Mycobacterium smegmatis E. coli
Protects DNA from oxidative damage by sequestering intracellular Fe(2+) ion and storing it in the form of Fe(3+) oxyhydroxide mineral. One hydrogen peroxide oxidizes two Fe(2+) ions, which prevents hydroxyl radical production by the Fenton reaction. It protects DNA from hydroxyl radical-mediated cleavage. Binds DNA with no apparent sequence specificity without self-aggregation nor promotion of DNA condensation. Is unable to protect DNA from DNase-mediated cleavage. Dps Protein, Mycobacterium sme...
TMPH-03014 MPT63 Protein, Mycobacterium tuberculosis, Recombinant (His)

mpt63,Antigen MPT63,16 kDa immunoprotective extracellular pr...

Mycobacterium tuberculosis E. coli
N/A. MPT63 Protein, Mycobacterium tuberculosis, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 17.7 kDa and the accession number is P9WIP0.
TMPH-03007 Ag85C Protein, Mycobacterium tuberculosis, Recombinant (His)

Acyl-CoA:diacylglycerol acyltransferase,Fibronectin-binding ...

Mycobacterium tuberculosis E. coli
Ag85C Protein, Mycobacterium tuberculosis, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 36.1 kDa and the accession number is P9WQN8.
TMPH-02409 LprG Protein, Mycobacterium tuberculosis, Recombinant (His & Myc)

27 kDa lipoprotein,lprG,Triacylglyceride transfer protein Lp...

Mycobacterium tuberculosis E. coli
LprG Protein, Mycobacterium tuberculosis, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 29.2 kDa and the accession number is P9WK44.
TMPH-03002 FtsQ Protein, Mycobacterium tuberculosis, Recombinant (His & Myc)

ftsQ,Cell division protein FtsQ

Mycobacterium tuberculosis E. coli
Essential cell division protein. FtsQ Protein, Mycobacterium tuberculosis, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 28.2 kDa and the accession number is P9WNA0.
TMPH-03011 EsxH Protein, Mycobacterium tuberculosis, Recombinant (His & SUMO)

Low molecular weight protein antigen 7,esxH,10 kDa antigen C...

Mycobacterium tuberculosis E. coli
EsxH, in complex with EsxG, disrupts ESCRT function and impairs host phagosome maturation, thereby promoting intracellular bacterial growth. The complex acts by interacting, via EsxH, with the host hepatocyte growth factor-regulated tyrosine kinase substrate (HGS/HRS), a component of the ESCRT machinery.
TMPH-03006 Ag85B Protein, Mycobacterium tuberculosis, Recombinant (His)

30 kDa extracellular protein,Diacylglycerol acyltransferase/...

Mycobacterium tuberculosis P. pastoris (Yeast)
Ag85B Protein, Mycobacterium tuberculosis, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 32.7 kDa and the accession number is P9WQP0.
TMPH-02990 Alpha-crystallin Protein, Mycobacterium bovis, Recombinant (His)

14 kDa antigen,Acr,16 kDa antigen,HSP 16.3

Mycobacterium bovis Baculovirus Insect Cells
Acts as a chaperone. Alpha-crystallin Protein, Mycobacterium bovis, Recombinant (His) is expressed in Baculovirus insect cells with C-9xHis tag. The predicted molecular weight is 18.1 kDa and the accession number is P0A5B8.
TMPH-03017 CYP51 Protein, Mycobacterium tuberculosis, Recombinant (His & Myc)

Cytochrome P450-14DM,Sterol 14alpha-demethylase,Sterol 14-al...

Mycobacterium tuberculosis Baculovirus Insect Cells
Its precise biological substrate is not known. Catalyzes C14-demethylation of lanosterol, 24,25-dihydrolanosterol and obtusifoliol which is critical for ergosterol biosynthesis. It transforms lanosterol into 4,4'-dimethyl cholesta-8,14,24-triene-3-beta-ol.
TMPH-03003 Ag85A Protein, Mycobacterium tuberculosis, Recombinant (His & SUMO)

Diacylglycerol acyltransferase/mycolyltransferase Ag85A,Acyl...

Mycobacterium tuberculosis E. coli
Ag85A Protein, Mycobacterium tuberculosis, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 44.6 kDa and the accession number is P9WQP2.
TMPH-02994 MAP_1030 Protein, Mycobacterium paratuberculosis, Recombinant (E. coli, His)

Probable transcriptional regulatory protein MAP_1030

Mycobacterium paratuberculosis E. coli
MAP_1030 Protein, Mycobacterium paratuberculosis, Recombinant (E. coli, His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 32.8 kDa and the accession number is P62039.
TMPH-03015 MPT64 Protein, Mycobacterium tuberculosis, Recombinant (E. coli, His)

mpt64,Antigen MPT64,Immunogenic protein MPT64

Mycobacterium tuberculosis E. coli
N/A. MPT64 Protein, Mycobacterium tuberculosis, Recombinant (E. coli, His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 26.4 kDa and the accession number is P9WIN9.
TMPH-03020 MTR Protein, Mycobacterium tuberculosis, Recombinant (His & Myc & SUMO)

mtr,Mycothione reductase,Mycothiol-disulfide reductase,NADPH...

Mycobacterium tuberculosis E. coli
Catalyzes the NAD(P)H-dependent reduction of mycothione (the oxidized disulfide form of mycothiol) to mycothiol.
TMPH-02992 FbpB Protein, Mycobacterium kansasii, Recombinant (His & Myc & SUMO)

fbpB,30 kDa extracellular protein,Extracellular alpha-antige...

Mycobacterium kansasii E. coli
FbpB Protein, Mycobacterium kansasii, Recombinant (His & Myc & SUMO) is expressed in E. coli expression system with N-10xHis-SUMO and C-Myc tag. The predicted molecular weight is 50.6 kDa and the accession number is P21160.
TMPH-03023 AmiB2 Protein, Mycobacterium tuberculosis, Recombinant (His & Myc & SUMO)

Putative amidase AmiB2

Mycobacterium tuberculosis E. coli
AmiB2 Protein, Mycobacterium tuberculosis, Recombinant (His & Myc & SUMO) is expressed in E. coli.
TMPH-02989 ESAT-6 Protein, Mycobacterium bovis, Recombinant (His & Myc)

ESAT-6,6 kDa early secretory antigenic target,esxA

Mycobacterium bovis E. coli
A secreted protein. Acts as a strong host T-cell antigen. Plays a number of roles in modulating the host's immune response to infection as well as being responsible for bacterial escape into the host cytoplasm. ESAT-6 Protein, Mycobacterium bovis, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 17.2 kDa and the accession number is P0A565.
TMPH-03009 EsxB Protein, Mycobacterium tuberculosis, Recombinant (E. coli, His)

ESAT-6-like protein EsxB,esxB,10 kDa culture filtrate antige...

Mycobacterium tuberculosis E. coli
A secreted protein. Acts as a strong host T-cell antigen. Involved in translocation of bacteria from the host (human) phagolysosome to the host cytoplasm. Might serve as a chaperone to prevent uncontrolled membrane lysis by its partner EsxA. EsxB Protein, Mycobacterium tuberculosis, Recombinant (E. coli, His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 14.7 kDa and the accession number is P9WNK4.
TMPH-03013 HRP1 Protein, Mycobacterium tuberculosis, Recombinant (His & Myc & SUMO)

hrp1,Hypoxic response protein 1

Mycobacterium tuberculosis E. coli
Unlike some other CBS-domain containing proteins does not seem to bind AMP.
TMPH-03005 Ag85B Protein, Mycobacterium tuberculosis, Recombinant (E. coli, His)

30 kDa extracellular protein,DGAT,Fbps B,Diacylglycerol acyl...

Mycobacterium tuberculosis E. coli
Ag85B Protein, Mycobacterium tuberculosis, Recombinant (E. coli, His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 36.2 kDa and the accession number is P9WQP0.
TMPH-02991 Alpha-crystallin Protein, Mycobacterium bovis, Recombinant (E. coli, His)

14 kDa antigen,Acr,16 kDa antigen,HSP 16.3

Mycobacterium bovis E. coli
Acts as a chaperone. Alpha-crystallin Protein, Mycobacterium bovis, Recombinant (E. coli, His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 20.1 kDa and the accession number is P0A5B8.
TMPH-01258 DAG1 Protein, Human, Recombinant (His & Myc)

Dystrophin-associated glycoprotein 1,Dystroglycan,Dystroglyc...

Human Baculovirus Insect Cells
The dystroglycan complex is involved in a number of processes including laminin and basement membrane assembly, sarcolemmal stability, cell survival, peripheral nerve myelination, nodal structure, cell migration, and epithelial polarization.; Extracellular peripheral glycoprotein that acts as a receptor for extracellular matrix proteins containing laminin-G domains. Receptor for laminin-2 (LAMA2) and agrin in peripheral nerve Schwann cells. Also acts as a receptor for laminin LAMA5.; Transmembra...
TMPY-01033 IL-32 Protein, Human, Recombinant (isoform alpha, His)

IL-32δ,IL-32beta,IL32,TAIFc,IL-32γ,白介素,IL-32 Protein(isoform...

Human HEK293 Cells
IL-32 is a recently discovered cytokine that induces various proinflammatory cytokines (TNF-alpha, IL-1beta, IL-6) and chemokines in both human and mouse cells through the NF-kappaB and p38 MAPK inflammatory signal pathways. It is regulated robustly by other major proinflammatory cytokines and is crucial to inflammation and immune responses. Four of the IL-32 isoforms (alpha, beta, gamma, and delta) are the most representative IL-32 transcripts, and the gamma isoform of IL-32 is the most active,...

重组蛋白

PstP Protein, Mycobacterium tuberculosis, Recombinant
Cat.No: TMPH-03022
Species: Mycobacterium tuberculosis
Expression System: E. coli
ATase Protein, Mycobacterium tuberculosis, Recombinant (His)
Cat.No: TMPH-03000
Species: Mycobacterium tuberculosis
Expression System: E. coli
ENR Protein, Mycobacterium tuberculosis, Recombinant (His)
Cat.No: TMPH-03008
Species: Mycobacterium tuberculosis
Expression System: E. coli
EsxB Protein, Mycobacterium tuberculosis, Recombinant (His)
Cat.No: TMPH-03010
Species: Mycobacterium tuberculosis
Expression System: P. pastoris (Yeast)
uL2 Protein, Mycobacterium tuberculosis, Recombinant (His)
Cat.No: TMPH-02999
Species: Mycobacterium tuberculosis
Expression System: E. coli
PstP Protein, Mycobacterium tuberculosis, Recombinant (His)
Cat.No: TMPH-03021
Species: Mycobacterium tuberculosis
Expression System: E. coli
PYCR Protein, Mycobacterium tuberculosis, Recombinant (His & Myc)
Cat.No: TMPH-03196
Species: Mycobacterium tuberculosis
Expression System: E. coli
KsdD Protein, Mycobacterium smegmatis, Recombinant (His & Myc)
Cat.No: TMPH-02996
Species: Mycolicibacterium smegmatis
Expression System: E. coli
EspK Protein, Mycobacterium tuberculosis, Recombinant (His & Myc)
Cat.No: TMPH-00758
Species: Mycobacterium tuberculosis
Expression System: E. coli
MPT64 Protein, Mycobacterium tuberculosis, Recombinant (His)
Cat.No: TMPH-03016
Species: Mycobacterium tuberculosis
Expression System: P. pastoris (Yeast)
Ag85A Protein, Mycobacterium tuberculosis, Recombinant (His)
Cat.No: TMPH-03004
Species: Mycobacterium tuberculosis
Expression System: E. coli
MT2731 Protein, Mycobacterium tuberculosis, Recombinant (His)
Cat.No: TMPH-03001
Species: Mycobacterium tuberculosis
Expression System: P. pastoris (Yeast)
Porin MspA Protein, Mycobacterium smegmatis, Recombinant (His)
Cat.No: TMPH-02998
Species: Mycobacterium smegmatis
Expression System: E. coli
SodC Protein, Mycobacterium tuberculosis, Recombinant (His & Myc)
Cat.No: TMPH-03612
Species: Mycobacterium tuberculosis
Expression System: E. coli
DisA Protein, Mycobacterium paratuberculosis, Recombinant (His & Myc)
Cat.No: TMPH-02993
Species: Mycobacterium paratuberculosis
Expression System: E. coli
MPT51 Protein, Mycobacterium tuberculosis, Recombinant (His & SUMO)
Cat.No: TMPH-03019
Species: Mycobacterium tuberculosis
Expression System: E. coli
MAP_1030 Protein, Mycobacterium paratuberculosis, Recombinant (His)
Cat.No: TMPH-02995
Species: Mycobacterium paratuberculosis
Expression System: P. pastoris (Yeast)
MeTAP1 Protein, Mycobacterium tuberculosis, Recombinant (His)
Cat.No: TMPH-03018
Species: Mycobacterium tuberculosis
Expression System: E. coli
HBHA Protein, Mycobacterium tuberculosis, Recombinant (His & Myc)
Cat.No: TMPH-03012
Species: Mycobacterium tuberculosis
Expression System: E. coli
Dps Protein, Mycobacterium smegmatis, Recombinant (His & SUMO)
Cat.No: TMPH-02997
Species: Mycobacterium smegmatis
Expression System: E. coli
MPT63 Protein, Mycobacterium tuberculosis, Recombinant (His)
Cat.No: TMPH-03014
Species: Mycobacterium tuberculosis
Expression System: E. coli
Ag85C Protein, Mycobacterium tuberculosis, Recombinant (His)
Cat.No: TMPH-03007
Species: Mycobacterium tuberculosis
Expression System: E. coli
LprG Protein, Mycobacterium tuberculosis, Recombinant (His & Myc)
Cat.No: TMPH-02409
Species: Mycobacterium tuberculosis
Expression System: E. coli
FtsQ Protein, Mycobacterium tuberculosis, Recombinant (His & Myc)
Cat.No: TMPH-03002
Species: Mycobacterium tuberculosis
Expression System: E. coli
EsxH Protein, Mycobacterium tuberculosis, Recombinant (His & SUMO)
Cat.No: TMPH-03011
Species: Mycobacterium tuberculosis
Expression System: E. coli
Ag85B Protein, Mycobacterium tuberculosis, Recombinant (His)
Cat.No: TMPH-03006
Species: Mycobacterium tuberculosis
Expression System: P. pastoris (Yeast)
Alpha-crystallin Protein, Mycobacterium bovis, Recombinant (His)
Cat.No: TMPH-02990
Species: Mycobacterium bovis
Expression System: Baculovirus Insect Cells
CYP51 Protein, Mycobacterium tuberculosis, Recombinant (His & Myc)
Cat.No: TMPH-03017
Species: Mycobacterium tuberculosis
Expression System: Baculovirus Insect Cells
Ag85A Protein, Mycobacterium tuberculosis, Recombinant (His & SUMO)
Cat.No: TMPH-03003
Species: Mycobacterium tuberculosis
Expression System: E. coli
MAP_1030 Protein, Mycobacterium paratuberculosis, Recombinant (E. coli, His)
Cat.No: TMPH-02994
Species: Mycobacterium paratuberculosis
Expression System: E. coli
MPT64 Protein, Mycobacterium tuberculosis, Recombinant (E. coli, His)
Cat.No: TMPH-03015
Species: Mycobacterium tuberculosis
Expression System: E. coli
MTR Protein, Mycobacterium tuberculosis, Recombinant (His & Myc & SUMO)
Cat.No: TMPH-03020
Species: Mycobacterium tuberculosis
Expression System: E. coli
FbpB Protein, Mycobacterium kansasii, Recombinant (His & Myc & SUMO)
Cat.No: TMPH-02992
Species: Mycobacterium kansasii
Expression System: E. coli
AmiB2 Protein, Mycobacterium tuberculosis, Recombinant (His & Myc & SUMO)
Cat.No: TMPH-03023
Species: Mycobacterium tuberculosis
Expression System: E. coli
ESAT-6 Protein, Mycobacterium bovis, Recombinant (His & Myc)
Cat.No: TMPH-02989
Species: Mycobacterium bovis
Expression System: E. coli
EsxB Protein, Mycobacterium tuberculosis, Recombinant (E. coli, His)
Cat.No: TMPH-03009
Species: Mycobacterium tuberculosis
Expression System: E. coli
HRP1 Protein, Mycobacterium tuberculosis, Recombinant (His & Myc & SUMO)
Cat.No: TMPH-03013
Species: Mycobacterium tuberculosis
Expression System: E. coli
Ag85B Protein, Mycobacterium tuberculosis, Recombinant (E. coli, His)
Cat.No: TMPH-03005
Species: Mycobacterium tuberculosis
Expression System: E. coli
Alpha-crystallin Protein, Mycobacterium bovis, Recombinant (E. coli, His)
Cat.No: TMPH-02991
Species: Mycobacterium bovis
Expression System: E. coli
DAG1 Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-01258
Species: Human
Expression System: Baculovirus Insect Cells
IL-32 Protein, Human, Recombinant (isoform alpha, His)
Cat.No: TMPY-01033
Species: Human
Expression System: HEK293 Cells
Cat. No. Product Name Target Signaling Pathways
T11817 Lansoprazole Sulfide D4

Proton pump Membrane transporter/Ion channel
Lansoprazole Sulfide D4 is a deuterium labeled Lansoprazole Sulfide. Lansoprazole Sulfide is an orally active anti-TB (Mycobacterium tuberculosis) agent with IC50 values of 0.59 μM intracellularly and 0.46 μM in broth.Lansoprazole Sulfide is an active metabolite of the proton pump inhibitor Lansoprazole.
T31813 Fludalanine

MK641,D-Alanine-2-d, 3-fluoro-,3-Fluoro-D-(2-2H)alanine

Fludalanine (MK641), an analogue of D-alanine, irreversiably inactivates racemase and also inhibits synthase. When used in combination with cycloserine, it has been found to be more active against a variety of non-mycobacterium organisms than fludalanine
TMID-0123 Rifapentine-d9

Rifapentine-d9 是 Rifapentine 的氘代化合物。Rifapentine 的 CAS 号为 61379-65-5。Rifapentine是可用于肺结核的抗生素。
TMIJ-0179 Faropenem-d7 Sodium Salt

Faropenem-d7 Sodium Salt 是 Faropenem Sodium Salt 的氘代化合物。Faropenem Sodium Salt 的 CAS 号为 122547-49-3。Faropenem sodium 是一种口服生物可利用的青霉烯类抗生素,能有效杀灭结核分枝杆菌,治疗结核病和社区获得性肺炎。

同位素标记化合物

Lansoprazole Sulfide D4
Cat.No: T11817
Synonym:
Target: Proton pump
Fludalanine
Cat.No: T31813
Synonym: MK641,D-Alanine-2-d, 3-fluoro-,3-Fluoro-D-(2-2H)alanine
Target:
Rifapentine-d9
Cat.No: TMID-0123
Synonym:
Target:
Faropenem-d7 Sodium Salt
Cat.No: TMIJ-0179
Synonym:
Target:
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