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Targets Recommended: c-Myc c-Myc

542

抑制剂 & 化合物

173

天然产物

2

化合物库

4

TargetMol 试剂盒

1136

重组蛋白

14

同位素标记化合物

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Cat. No. Product Name
L2130 抗癌细胞代谢库

1268 compounds
1268 种癌细胞代谢相关的生物活性小分子化合物的特有集合,用于肿瘤相关的研究以及抗肿瘤药物的筛选,用于高通量、高内涵筛选;
L2550 谷氨酰胺代谢化合物库

565 compounds
565 种谷氨酰胺代谢相关的分子,可以用于高通量和高内涵筛选;

化合物库

抗癌细胞代谢库
Cat.No: L2130
Compounds: 1268
谷氨酰胺代谢化合物库
Cat.No: L2550
Compounds: 565
Cat. No. Product Name Form Specificity Of Inhibition
C0119B MYC Tag Immunomagnetic Beads

MYC Tag 免疫沉淀磁珠

Suspension in bottle IP, Co-IP
C0119 MYC Tag Immunoprecipitation Kit

MYC Tag 免疫沉淀试剂盒

Suspension in bottle IP, Co-IP
C0051 Penicillin-Streptomycin Solution (100×), Sterile

青霉素-链霉素双抗溶液(100×),灭菌

Solution in bottle
C0052 Penicillin-Streptomycin-Amphotericin B Solution (100×), Sterile

青霉素-链霉素-两性霉素B三抗溶液(100×),灭菌

Solution in bottle

TargetMol 试剂盒

MYC Tag 免疫沉淀磁珠
Cat.No: C0119B
MYC Tag 免疫沉淀试剂盒
Cat.No: C0119
青霉素-链霉素双抗溶液(100×),灭菌
Cat.No: C0051
青霉素-链霉素-两性霉素B三抗溶液(100×),灭菌
Cat.No: C0052
Cat. No. Product Name Target Signaling Pathways
T9061 EN4

EN4 MYC inhibitor

c-Myc Cell Cycle/Checkpoint
EN4 (EN4 MYC inhibitor) 是一种靶向 M​​YC 的半胱氨酸 171 (C171) 的共价配体。它抑制 MYC 转录活性,下调 MYC 靶标,并具有抗肿瘤作用。它对 c-MYC 的选择性高于 N-MYC 和 L-MYC
T3048 10058-F4

c-Myc Inhibitor

c-Myc; Autophagy Autophagy; Cell Cycle/Checkpoint
10058-F4 (c-Myc Inhibitor) 是一种细胞渗透性噻唑烷酮,可特异性抑制 c-Myc-Max 相互作用并防止 c-Myc 靶基因表达的反式激活;诱导细胞周期停滞和凋亡。
TP1315 c-Myc Peptide Trifluoroacetate

Others Others
c-Myc Peptide Trifluoroacetate (145646-22-6 free base) 是一种合成肽,对应于人类 c-myc 蛋白的 C 末端氨基酸 (410-419),参与调控生长相关基因的转录。
TP2311 C-MYC PEPTIDE EPITOPE TFA

Others Others
C-MYC PEPTIDE EPITOPE TFA 是 c-myc 原癌基因的产物,是一种螺旋-环-螺旋亮氨酸拉链磷蛋白,可调节细胞增殖、细胞分化和凋亡中的基因转录。该肽是人类 c-myc 表位。
T39751 MYC-IN-2

Others Others
MYC-IN-2 is a protein-protein inhibitor targeting the MYC protein, designed for use in cancer research.
T3686 10074-G5

c-Myc; Autophagy Autophagy; Cell Cycle/Checkpoint
10074-G5是一种c-Myc-Max 二聚化的抑制剂,IC50值为146 μM。
T15665 KJ Pyr 9

c-Myc; Autophagy Autophagy; Cell Cycle/Checkpoint
KJ Pyr 9 是一种 MYC 的抑制剂,在体外实验中的 Kd 值为 6.5 nM。
T4367 Mycro 3

Mycro-3

c-Myc; Autophagy Autophagy; Cell Cycle/Checkpoint
Mycro 3 在全细胞分析中对 c-Myc 具有强效选择性,可用于胰腺癌的研究。
T72040 c-Myc inhibitor 7

Others Others
c-Myc inhibitor 7是c-Myc 抑制剂和多靶点蛋白降解剂,可有效降解多种肿瘤细胞中的c-Myc、CK1α、GSPT1和IKZF1/2/3蛋白,可用于c-Myc 高表达相关疾病的研究,如癌症、心脑血管疾病和病毒感染。
T4252 ML327

c-Myc; Autophagy Autophagy; Cell Cycle/Checkpoint
ML327 是 MYC 的阻断剂,还可抑制 E-钙粘蛋白转录和逆转上皮间质转化。
T9628 10074-A4

c-Myc Cell Cycle/Checkpoint
10074-A4 是与 c-Myc370-409 结合的 c-Myc 结合化合物,具有抗癌作用,其行为类似于“蛋白质云”周围的“配体云”,具有与非结合配体不同的特征。
TP2179 c-Myc tag Peptide

Others Others
c-Myc Peptide is a useful displacement of c-Myc-tagged fusion proteins bound to anti-c-Myc antibodies in immunoassays. The successful inhibition of antibody binding by c-Myc peptide demonstrates binding is specific. c-Myc peptide participates in the regul
T12134 MYCMI-6

NSC354961

Apoptosis; c-Myc Apoptosis; Cell Cycle/Checkpoint
MYCMI-6 (NSC-354961) 是一种内源性MYC:MAX 蛋白相互作用抑制剂,选择性结合 MYC bHLHZip 域,Kd 值为 1.6 μM。它阻断 MYC 驱动的转录,以 MYC 依赖性的方式抑制肿瘤细胞的生长 ,诱导细胞凋亡。
T12132 MYCi361

NUCC-0196361

c-Myc Cell Cycle/Checkpoint
MYCi361 (NUCC-0196361) 是一种 MYC 抑制剂,抑制肿瘤生长并增强 anti-PD1 免疫疗法,其与 MYC 结合的 Kd 为 3.2 μM。
T60019 VPC-70063

Thiourea, N-[3,5-bis(trifluoromethyl)phenyl]-N'-(phenylmethyl)-

Apoptosis; PARP; c-Myc Apoptosis; Cell Cycle/Checkpoint; Chromatin/Epigenetic; DNA Damage/DNA Repair
VPC-70063 (Thiourea, N-[3,5-bis(trifluoromethyl)phenyl]-N'-(phenylmethyl)-) 是 c-Myc-MAX 的抑制剂。 VPC-70063 的 Myc-Max 转录活性抑制率为 106%,IC50 为 8.9 μM,Myc-Max/UBE2C 下游通路抑制率为 94%。 VPC-70063 可用于抗癌研究。
T9033 BTYNB

MDK6620,BTYNB IMP1 Inhibitor

Others; c-Myc; NF-κB Cell Cycle/Checkpoint; NF-κB; Others
BTYNB (MDK6620) 是IMP1结合 c-Myc mRNA 的有效选择性抑制剂,IC50为 5 μM。它下调 β-TrCP1 mRNA 并减少NF-κB 的激活。它通过损害 IGF2 mRNA 结合蛋白 1 结合来破坏这种增强子功能,可用于癌症研究。
T10352 APTO-253

LOR-253,LT-253

Apoptosis; c-Myc; KLF Apoptosis; Cell Cycle/Checkpoint; MAPK
APTO-253 (LOR-253) 抑制 c-Myc 表达,稳定 G-四链体 DNA,并诱导急性髓细胞白血病细胞的细胞周期停滞和凋亡。 它通过诱导 KLF4 肿瘤抑制因子介导抗癌活性,具有抗关节炎活性。
T9032 MGH-CP1

Others Others
MGH-CP1 是 TEAD2 (IC50:710 nM) 及 TEAD4 (IC50:672 nM) 自棕榈酰化抑制剂,口服有活性,可降低细胞内源性或异位表达的 TEAD 蛋白棕榈酰化水平。MGH-CP1 与 Lats1/2 缺失,是 Myc 的表达受到抑制,阻碍上皮细胞过度增殖,诱导细胞凋亡。
T9370 dCBP-1

Epigenetic Reader Domain; PROTACs Chromatin/Epigenetic; PROTAC
dCBP-1 是基于Cereblon 配体的p300/CBP 的选择性双功能降解剂。dCBP-1可以有效的杀死多发性骨髓瘤细胞,并降低驱动 MYC 表达的致癌增强子活性。
T11284 FIDAS-3

Others; Wnt/beta-catenin; Methionine Adenosyltransferase (MAT) Chromatin/Epigenetic; Cytoskeletal Signaling; Others; Stem Cells
FIDAS-3 是一种强效Wnt 抑制剂,也是一种二苯乙烯衍生物,对甲硫氨酸腺苷转移酶 2A (MAT2A) 的IC50为 4.9 μM。它能够与 S-腺苷甲硫氨酸有效竞争MAT2A 结合,并具有抗癌作用。
T9093 NY2267

Acetic acid, 2-[[6-[2-(cyclohexylamino)-1-[[(4-methoxyphenyl)methyl](2-pyridinylcarbonyl)amino]-2-oxoethyl]-2-naphthalenyl]oxy]-, 1,1-dimethylethyl ester

c-Myc Cell Cycle/Checkpoint
NY2267 (Acetic acid, 2-[[6-[2-(cyclohexylamino)-1-[[(4-methoxyphenyl)methyl](2-pyridinylcarbonyl)amino]-2-oxoethyl]-2-naphthalenyl]oxy]-, 1,1-dimethylethyl ester) 是一种 Myc-Max 相互作用干扰物,抑制 Myc 和 Jun 诱导的转录激活,其 IC50值为 36.5 μM。
T78055 MYC-RIBOTAC

c-Myc Cell Cycle/Checkpoint
MYC-RIBOTAC 是一种针对MYC内部核糖体进入位点(IRES)的核糖核酸酶靶向降解剂(RIBOTAC)。该化合物结合了MYC mRNA的靶向组分以及一种可招募并激活RNA酶L1的小分子。通过降低MYC的mRNA和蛋白质表达水平,MYC-RIBOTAC诱导细胞发生凋亡,应用于抗肿瘤治疗的研究。
T11285 FIDAS-5

Others Others
FIDAS-5 是甲硫氨酸腺苷转移酶 2A 抑制剂(IC50:2.1 μM),具有口服活性。它能够与 S-腺苷甲硫氨酸有效竞争 MAT2A 结合,并具有抗癌作用。
T20533 NNK

Nicotine-derived nitrosamine ketone

Lipoxygenase Metabolism
NNK (Nicotine-derived nitrosamine ketone) 是尼古丁亚硝化衍生物。它可以激活 ERK1/2和 PKCα,并在 Ser70 激活 Bcl2磷酸化,以及在 Thr58和 Ser62激活 c-Myc。它可用于构建肺癌小鼠模型,以及诱导人肺癌细胞的增殖和存活。
T10760 Ceramides Mixture

神经酰胺混合物,神经酰胺

Telomerase DNA Damage/DNA Repair
Ceramides Mixture 是表皮渗透屏障的主要脂质成分,参与生长抑制,细胞周期停滞和端粒酶活性的调节。它是一种内源性神经酰胺,由含羟基和非羟基脂肪酸的神经酰胺组成。
T6010 Idarubicin hydrochloride

盐酸伊达比星,Idamycin,4-demethoxydaunorubicin (NSC256439, 4-DMDR) HCl,4-Demethoxydaunorubicin hydrochloride,Idarubicin HCl,伊达比星盐酸盐,Zavedos

Topoisomerase; Antibacterial; Autophagy; Antifungal Autophagy; DNA Damage/DNA Repair; Microbiology/Virology
Idarubicin hydrochloride (Zavedos) 是一种蒽环类抗白血病药物,能抑制细菌和酵母菌生长,还抑制拓扑异构酶 II,干扰 DNA 复制和 RNA 转录。
T74460 c-Myc inhibitor 5

Others Others
c-Myc inhibitor5 (DA3) 是一种荧光长链桥双嘌呤,可选择性靶向 c-MYCG-四链体(KD16 μM)。c-Myc inhibitor5 显示对 c-MYC 表达的抑制作用,而不是其他 G4 驱动的癌基因。
T75239 c-Myc inhibitor 10

Others Others
c-Myc inhibitor10 (compound 17) 是 c-myc 的抑制剂,表现出一定的的细胞效力,与甲基化的 morpholine 氮的通透性增加一致。
T63359 c-Myc inhibitor 4

Others Others
c-Myc inhibitor 4 是有效的、口服具有活性的 c-Myc-reducing 化合物。C-Myc 是一种重要的原癌基因,与多种肿瘤的发生发展密切相关。
T8658 NEO2734

EP31670

Epigenetic Reader Domain; Histone Acetyltransferase Chromatin/Epigenetic
NEO2734 (EP31670) 是一种具有口服活性的选择性 p300/CBP 和 BET 溴结构域抑制剂,其 IC50值均小于30 nM,可用于前列腺癌的研究。
T72620 c-Myc inhibitor 9

Others Others
c-Myc inhibitor9 是一种c-Myc 抑制剂,logEC50值 ≥6。c-Myc inhibitor9 抑制异种移植裸鼠模型中肿瘤的生长。c-Myc inhibitor9 可用于癌症研究。
T10765 Eragidomide

CC-90009,Cereblon modulator 1

Apoptosis; Ligand for E3 Ligase; Molecular Glues Apoptosis; PROTAC
Cereblon modulator 1 是一种 GSPT1 选择性cereblon (CRBN)E3 连接酶调节剂,以分子胶的方式作用。它通过 CRL4CRBN选择性靶向 GSPT1 进行泛素化和蛋白酶体降解。
T79439 c-Myc inhibitor 12

c-Myc Cell Cycle/Checkpoint
c-Myc inhibitor12 (compound 67h),作为c-Myc抑制剂,具有pEC50值为6.4。
T79438 c-Myc inhibitor 11

c-Myc Cell Cycle/Checkpoint
c-Myc inhibitor11(Compound 67e),一种c-MYC抑制剂(pEC50: 6.4),在大鼠药代动力学评估中表现出高清除率、中等体积分布和短半衰期,适用于癌症研究领域。
T72619 c-Myc inhibitor 8

Others Others
c-Myc inhibitor8 是一种 c-Myc 抑制剂。c-Myc inhibitor8 有效抑制多种癌细胞的细胞活力。c-Myc inhibitor8 在小鼠模型中抑制人前列腺癌和肺癌肿瘤的生长。c-Myc inhibitor8 可用于癌症研究。
T6203 Saxagliptin

BMS-477118,沙克列汀,Onglyza,沙格列汀

Proteasome; DPP-4 Proteases/Proteasome; Ubiquitination
Saxagliptin (BMS-477118) 是一种选择性,可逆性,竞争性和口服活性的二肽基肽酶 4 (DPP-4) (Ki= 0.6-1.3 nM) 抑制剂。Saxagliptin 能够用于 2 型糖尿病的研究。
T0178 Saxagliptin hydrate

沙格列汀单水化合物,Onglyza hydrate,BMS-477118 hydrate

Proteasome; DPP-4 Proteases/Proteasome; Ubiquitination
Saxagliptin hydrate (Onglyza hydrate) 是一种选择性,竞争性,可逆性和口服活性的二肽基肽酶 4 (DPP-4) (Ki= 0.6-1.3 nM) 抑制剂。Saxagliptin hydrate 能够用于 2 型糖尿病的研究。
T12133 MYCi975

NUCC-0200975

c-Myc Cell Cycle/Checkpoint
MYCi975 (NUCC-0200975)是一种具有口服活性的MYC 抑制剂,具有很强的抗肿瘤作用和良好的耐受性,增加肿瘤免疫细胞浸润,增强肿瘤对抗 PD1 免疫研究的敏感性。它破坏 MYC/MAX 相互作用,促进 MYC T58 磷酸化和 MYC 降解,并损害 MYC 驱动的基因表达。
T35626 AMP-Deoxynojirimycin

AMP-DNM

Transferase; Glucosidase Metabolism
AMP-Deoxynojirimycin (AMP-DNM) 是一种有效的神经酰胺葡萄糖基转移酶和 GCase 2 抑制剂。AMP-Deoxynojirimycin 是一种有效的 GlcCer 生物合成抑制剂,可用于研究帕金森和糖尿病。
T67712 Questiomycin A derivatives 13

Others Others
Questiomycin A derivatives 13 是一种 Questiomycin A 衍生物。
T3265 Azathramycin

Desmethyl Azithromycin,阿奇霉素 A,6-Demethylazithromycin,去甲基阿奇霉素,Azaerythromycin A,Azaerythromycin

Antibacterial; Antibiotic Microbiology/Virology
Azathramycin (Desmethyl Azithromycin) 是一种可靶向核糖体的抗生素。
T15735 Leptomycin B

CI 940,LMB,来普霉素B

CRM1; Antibiotic; Antifungal Membrane transporter/Ion channel; Microbiology/Virology
Leptomycin B (LMB) 是一种抗真菌抗生素,可阻断真核细胞周期,抑制蛋白出核转运。Leptomycin 通过半胱氨酸残基处的共价修饰使 CRM1/exportin 1失活。它
T12242 Norvancomycin hydrochloride

Desmethyl-vancomycin hydrochloride,盐酸去甲万古霉素

Antibacterial Microbiology/Virology
Norvancomycin hydrochloride (Desmethyl-vancomycin hydrochloride) 可用于葡萄球菌所致的心内膜炎、骨髓炎、肺炎、败血症或软组织感染。
T67720 Questiomycin A derivatives 21

Others Others
Questiomycin A derivatives 21 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T67720,CAS号为 1807725-36-5。
T21148 Troleandomycin

AI3-50166,Triacetyloleandomycin,Aovine,Micotil,Matromycin T,Cyclamycin

P450; Antibiotic Metabolism; Microbiology/Virology
Troleandomycin (Triacetyloleandomycin) 是一种大环内酯类抗生素,是具有口服活性和特异性的 CYP3A 抑制剂,可诱发记性感言,诱导长期胆汁淤积,可用于研究哮喘疾病。
T11120 Duocarmycin TM

DNA Alkylation; Antibiotic; ADC Cytotoxin Antibody-drug Conjugate/ADC Related; DNA Damage/DNA Repair; Microbiology/Virology
Duocarmycin TM 是一种有抗肿瘤活性的抗生素,也是一种 DNA 烷化剂。
T0788L Spectinomycin dihydrochloride pentahydrate

盐酸大观霉素五水合物,Trobicin,Spectogard,Spectinomycin hydrochloride hydrate

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Spectinomycin dihydrochloride pentahydrate (Spectogard) 是一种广谱氨基环糊精抗生素,可以抑制多种革兰氏阳性和革兰氏阴性生物的生长。
T4267 Tulathromycin A

CP 472295,Draxxin,Tulathromycin,托拉菌素 A

Antibacterial; Antibiotic Microbiology/Virology
Tulathromycin A (CP 472295) 是一种大环内酯类抗生素,靶向细菌核糖体抑制蛋白质合成 (IC50=0.26 µM),具有免疫调节作用。它可研究牛和猪的呼吸道疾病。
T12284 O-Propargyl-Puromycin

OP-puro,O-Propargylpuromycin

Others Others
O-Propargyl-Puromycin (OP-puro) 是一种高效的蛋白质合成抑制剂,是一种嘌呤霉素炔类似物。
T2331 Solithromycin

索利霉素,OP-1068,CEM-101

Antibacterial; Antibiotic Microbiology/Virology
Solithromycin (OP-1068) 是口服可生物利用的抗菌剂,抑制肺炎链球菌、葡萄球菌、金黄色葡萄球菌和流感嗜血杆菌的细胞活力、蛋白质合成和生长速率, IC50 值分别为 7.5 ng/mL、40 ng/mL 和 125 ng/mL。它可与核糖体的大 50S 亚基结合抑制蛋白质生物合成。

化合物

EN4
Cat.No: T9061
Synonym: EN4 MYC inhibitor
Target: c-Myc
10058-F4
Cat.No: T3048
Synonym: c-Myc Inhibitor
Target: c-Myc, Autophagy
c-Myc Peptide Trifluoroacetate
Cat.No: TP1315
Synonym:
Target: Others
C-MYC PEPTIDE EPITOPE TFA
Cat.No: TP2311
Synonym:
Target: Others
MYC-IN-2
Cat.No: T39751
Synonym:
Target: Others
10074-G5
Cat.No: T3686
Synonym:
Target: c-Myc, Autophagy
KJ Pyr 9
Cat.No: T15665
Synonym:
Target: c-Myc, Autophagy
Mycro 3
Cat.No: T4367
Synonym: Mycro-3
Target: c-Myc, Autophagy
c-Myc inhibitor 7
Cat.No: T72040
Synonym:
Target: Others
ML327
Cat.No: T4252
Synonym:
Target: c-Myc, Autophagy
10074-A4
Cat.No: T9628
Synonym:
Target: c-Myc
c-Myc tag Peptide
Cat.No: TP2179
Synonym:
Target: Others
MYCMI-6
Cat.No: T12134
Synonym: NSC354961
Target: Apoptosis, c-Myc
MYCi361
Cat.No: T12132
Synonym: NUCC-0196361
Target: c-Myc
VPC-70063
Cat.No: T60019
Synonym: Thiourea, N-[3,5-bis(trifluoromethyl)phenyl]-N'-(phenylmethyl)-
Target: Apoptosis, PARP, c-Myc
BTYNB
Cat.No: T9033
Synonym: MDK6620,BTYNB IMP1 Inhibitor
Target: Others, c-Myc, NF-κB
APTO-253
Cat.No: T10352
Synonym: LOR-253,LT-253
Target: Apoptosis, c-Myc, KLF
MGH-CP1
Cat.No: T9032
Synonym:
Target: Others
dCBP-1
Cat.No: T9370
Synonym:
Target: Epigenetic Reader Domain, PROTACs
FIDAS-3
Cat.No: T11284
Synonym:
Target: Others, Wnt/beta-catenin, Methionine Adenosyltransferase (MAT)
NY2267
Cat.No: T9093
Synonym: Acetic acid, 2-[[6-[2-(cyclohexylamino)-1-[[(4-methoxyphenyl)methyl](2-pyridinylcarbonyl)amino]-2-oxoethyl]-2-naphthalenyl]oxy]-, 1,1-dimethylethyl ester
Target: c-Myc
MYC-RIBOTAC
Cat.No: T78055
Synonym:
Target: c-Myc
FIDAS-5
Cat.No: T11285
Synonym:
Target: Others
NNK
Cat.No: T20533
Synonym: Nicotine-derived nitrosamine ketone
Target: Lipoxygenase
Ceramides Mixture
Cat.No: T10760
Synonym: 神经酰胺混合物,神经酰胺
Target: Telomerase
Idarubicin hydrochloride
Cat.No: T6010
Synonym: 盐酸伊达比星,Idamycin,4-demethoxydaunorubicin (NSC256439, 4-DMDR) HCl,4-Demethoxydaunorubicin hydrochloride,Idarubicin HCl,伊达比星盐酸盐,Zavedos
Target: Topoisomerase, Antibacterial, Autophagy, Antifungal
c-Myc inhibitor 5
Cat.No: T74460
Synonym:
Target: Others
c-Myc inhibitor 10
Cat.No: T75239
Synonym:
Target: Others
c-Myc inhibitor 4
Cat.No: T63359
Synonym:
Target: Others
NEO2734
Cat.No: T8658
Synonym: EP31670
Target: Epigenetic Reader Domain, Histone Acetyltransferase
c-Myc inhibitor 9
Cat.No: T72620
Synonym:
Target: Others
Eragidomide
Cat.No: T10765
Synonym: CC-90009,Cereblon modulator 1
Target: Apoptosis, Ligand for E3 Ligase, Molecular Glues
c-Myc inhibitor 12
Cat.No: T79439
Synonym:
Target: c-Myc
c-Myc inhibitor 11
Cat.No: T79438
Synonym:
Target: c-Myc
c-Myc inhibitor 8
Cat.No: T72619
Synonym:
Target: Others
Saxagliptin
Cat.No: T6203
Synonym: BMS-477118,沙克列汀,Onglyza,沙格列汀
Target: Proteasome, DPP-4
Saxagliptin hydrate
Cat.No: T0178
Synonym: 沙格列汀单水化合物,Onglyza hydrate,BMS-477118 hydrate
Target: Proteasome, DPP-4
MYCi975
Cat.No: T12133
Synonym: NUCC-0200975
Target: c-Myc
AMP-Deoxynojirimycin
Cat.No: T35626
Synonym: AMP-DNM
Target: Transferase, Glucosidase
Questiomycin A derivatives 13
Cat.No: T67712
Synonym:
Target: Others
Azathramycin
Cat.No: T3265
Synonym: Desmethyl Azithromycin,阿奇霉素 A,6-Demethylazithromycin,去甲基阿奇霉素,Azaerythromycin A,Azaerythromycin
Target: Antibacterial, Antibiotic
Leptomycin B
Cat.No: T15735
Synonym: CI 940,LMB,来普霉素B
Target: CRM1, Antibiotic, Antifungal
Norvancomycin hydrochloride
Cat.No: T12242
Synonym: Desmethyl-vancomycin hydrochloride,盐酸去甲万古霉素
Target: Antibacterial
Questiomycin A derivatives 21
Cat.No: T67720
Synonym:
Target: Others
Troleandomycin
Cat.No: T21148
Synonym: AI3-50166,Triacetyloleandomycin,Aovine,Micotil,Matromycin T,Cyclamycin
Target: P450, Antibiotic
Duocarmycin TM
Cat.No: T11120
Synonym:
Target: DNA Alkylation, Antibiotic, ADC Cytotoxin
Spectinomycin dihydrochloride pentahydrate
Cat.No: T0788L
Synonym: 盐酸大观霉素五水合物,Trobicin,Spectogard,Spectinomycin hydrochloride hydrate
Target: ribosome, Antibacterial, Antibiotic
Tulathromycin A
Cat.No: T4267
Synonym: CP 472295,Draxxin,Tulathromycin,托拉菌素 A
Target: Antibacterial, Antibiotic
O-Propargyl-Puromycin
Cat.No: T12284
Synonym: OP-puro,O-Propargylpuromycin
Target: Others
Solithromycin
Cat.No: T2331
Synonym: 索利霉素,OP-1068,CEM-101
Target: Antibacterial, Antibiotic
Cat. No. Product Name Target Signaling Pathways
TN1892 Lusianthridin

Others; c-Myc Cell Cycle/Checkpoint; Others
Lusianthridin 是来自石斛 Dendrobium venustum 的天然产物。 Lusianthridin 在无毒浓度下表现出抗迁移特性。 Lusianthridin 通过抑制 Src-STAT3 信号传导增强 c-Myc 降解。
T21065 Artemisitene

Others Others
Artemisitene 是青蒿素的氧化形式,是一种抗疟药。青蒿素前体是青蒿素生物合成的重要基础物质,包括青蒿素 B、青蒿素、青蒿酸等。
T3673 Mollugin

大叶茜草素,Rubimaillin

HER; JAK Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells; Tyrosine Kinase/Adaptors
Mollugin (Rubimaillin) 是Rubia cordifolia L.中主要的生物活性成分。它能通过 p38-Smad 信号通路增强 BMP-2 的成骨作用。它通过抑制 TNF-α 诱导的 NF-κB 激活起抗癌疗效。
T4S1173 Agrimol B

仙鹤草酚B,仙鹤草酚 B

Sirtuin; PPAR Chromatin/Epigenetic; DNA Damage/DNA Repair; Metabolism
Agrimol B 是从仙鹤草中分离得到的一种多酚衍生物,可抑制脂肪形成,降低PPARγ的表达,诱导SIRT1易位和表达。
T2764 (S)-10-Hydroxycamptothecin

10-羟喜树碱,10-羟基喜树碱,10-Hydroxycamptothecin,10-HCPT

Apoptosis; Topoisomerase Apoptosis; DNA Damage/DNA Repair
(S)-10-Hydroxycamptothecin (10-HCPT) 是一种从喜树中分离的 DNA 拓扑异构酶 I 抑制剂。它显著诱导细胞凋亡,可研究肝癌、胃癌、结肠癌和白血病。
T6401 Azithromycin

阿奇霉素,Zithromax,CP 62993,XZ-450

Others; Antibacterial; Antibiotic; Autophagy Autophagy; Microbiology/Virology; Others
Azithromycin (CP 62993) 是一种常用于细菌感染研究的大环内酯抗生素。
T2762 Kasugamycin hydrochloride

Kasumin,盐酸春雷霉素

Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Kasugamycin hydrochloride (Kasumin) 是一种能结合 30s 和 70s 核糖体,但不能结合 50s 亚基的抗生素。它模拟 mRNA 核苷酸以破坏 tRNA 结合并抑制经典翻译起始。
T1665 Daptomycin

达托霉素,LY146032

DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Daptomycin (LY146032) 是脂肽类抗生素,在体外快速灭活革兰氏阳性细菌。
T21498 Phleomycin

DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Phleomycin 是在链霉菌中发现的,引起 DNA 切割的抗癌糖肽抗生素之一。 它类似于博来霉素,它结合并插入 DNA 以破坏双螺旋的完整性。
T1335 Mycophenolic acid

霉酚酸,Mycophenolate,RS-61443

Apoptosis; Dehydrogenase; Endogenous Metabolite; Antibacterial; Antibiotic; UGT; Antifungal Apoptosis; Metabolism; Microbiology/Virology
Mycophenolic acid (Mycophenolate) 是一种有效的非竞争性肌苷单磷酸脱氢酶 (IMPDH) 抑制剂,EC50为 0.24 µM。它对多种 RNA 病毒具有抗病毒作用。它也是一种免疫抑制剂,具有抗血管生成和抗肿瘤作用。
T11665 Ionomycin calcium

SQ23377 calcium,罗红霉素钙盐(链霉菌属载体)

Apoptosis; Calcium Channel; Antibacterial; Antibiotic; PKC Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
Ionomycin calcium (SQ23377 calcium) 是选择性钙离子载体,也是一种由 Streptomyces conglobatus 产生的抗生素。它对二价阳离子具有高度特异性,还诱导蛋白激酶 C 激活。Ionomycin 促进细胞凋亡。
T1214 Ribostamycin sulfate

Vistamycin sulfate,硫酸核糖霉素

Antibacterial; Antibiotic Microbiology/Virology
Ribostamycin sulfate (Vistamycin sulfate) 是一种广谱抗菌剂, 在30S 和50S 核糖体亚基结合抑制细菌蛋白质合成, 还抑制蛋白二硫键异构酶分子伴侣活性, 用于药代动力学和肾毒性研究。
T1277 Lincomycin hydrochloride

Lincomycin HCl,NSC 70731,盐酸林可霉素,U10149A

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Lincomycin hydrochloride (U10149A) 是由林可链霉菌产生的抗生素,对革兰氏阳性球菌和厌氧菌具有活性。
T5037 Midecamycin

Antibiotic SF-837,Turimycin P3,Medecamycin A1,Rubimycin,麦迪霉素,Platenomycin B1,Espinomycin A

Antibacterial; Antibiotic Microbiology/Virology
Midecamycin (Medecamycin A1) 是乙酰氧基取代的大环内酯类抗生素,对革兰氏阳性和阴性菌有效。
T6343 Geldanamycin

格尔德霉素,NSC 122750

HSP; Influenza Virus; Tyrosine Kinases; Antibacterial; Antibiotic Cytoskeletal Signaling; Metabolism; Microbiology/Virology; Tyrosine Kinase/Adaptors
Geldanamycin 是一种 HSP90 抑制剂(Kd:1.2 μM),可特异性破坏糖皮质激素受体 (GR)/HSP 的结合。
T1381 Milbemycin oxime

Others; Antibiotic; Parasite Microbiology/Virology; Others
Milbemycin oxime 是一种大环内酯,具有广谱抗寄生虫活性。它由 Milbemycin A4 和 A3 组成。它可结合谷氨酸门控的氯离子通道,可作用于肠道线虫,肺和心脏蠕虫。
T1084 Apramycin sulfate

Nebramycin II,Ai3-29795,硫酸安普霉素,硫酸阿布拉霉素

Antibacterial; Antibiotic Microbiology/Virology
Apramycin sulfate (Nebramycin II) 是一种由黑暗链霉菌产生的兽用氨基糖苷类抗生素。
T21502 Aclacinomycin A

Aclarubicin

Topoisomerase DNA Damage/DNA Repair
Aclacinomycin A (Aclarubicin) 是一种从加利莱链霉菌中分离出的新型蒽环类抗生素,具有抗肿瘤活性。Aclacinomycin A 是拓扑异构酶 I 和 II 的抑制剂,抑制 RNA 活性 。Aclacinomycin A 可用于研究复发性白血病和晚期恶性淋巴瘤。
T6402 Azomycin

2-Nitroimidazole,2-硝基咪唑,Ro 05-9129,Amicin

Antibacterial; Antibiotic Microbiology/Virology
Azomycin (Ro 05-9129) 是一种可抑制有氧革兰氏阳性菌和革兰氏阴性菌的生长的抗生素。
T1255 Tobramycin

NSC 180514,妥布霉素,Nebramycin Factor 6,Deoxykanamycin B

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Tobramycin (NSC-180514) 是一种胃肠外给药的广谱氨基糖苷类抗生素,可研究由于敏感生物引起的中度至重度细菌感染疾病。
T21820 Resistomycin

Geliomycin,Heliomycin

Antibiotic Microbiology/Virology
Resistomycin(Geliomycin),一种五环多酮类抗生素,通过触发凋亡展现出强大的抗癌特性。
T5003 Rifamycin sodium

Rifamycin sodium salt,利福霉素钠

Antibacterial; Antibiotic Microbiology/Virology
Rifamycin sodium (Rifamycin sodium salt) salt 是从地中海曲霉或其突变体的发酵中分离出来的一种安沙霉素抗生素家族。它对革兰氏阳性菌和某些革兰氏阴性菌有抗生素活性。
T0793 Kanamycin sulfate

硫酸卡那霉素,Kanamycin monosulfate,Kanamycin A monosulfate,Ophtalmokalixan

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Kanamycin sulfate (Kanamycin monosulfate) 是氨基糖苷类杀菌抗生素,它通过与细菌30S 核糖体结合起作用。
T3607 Leucomycin

吉他霉素,Kitasamycin,Leucomycin V,Turimycin

Antibacterial; Antibiotic Microbiology/Virology
Leucomycin (Turimycin) 是一种由 Streptomyces kitasatoensis 产生的大环内酯类抗生素。
T2481 Ascomycin

FK520,Immunomycin,子囊霉素,FR-900520

Phosphatase; Others; Antibiotic; Parasite; Antifungal Metabolism; Microbiology/Virology; Others
Ascomycin (Immunomycin) 是 Tacrolimus 的乙基类似物,具有免疫抑制特性。它也是一种大环聚酮类抗生素,具有抗疟疾、抗真菌和抗痉挛等多种生物活性。它可防止移植排斥,并具有用于各种皮肤病研究的潜力。
T8347 Rifamycin S

Reactive Oxygen Species; ROS; Antibacterial; Antibiotic Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
Rifamycin S 是一种 DNA 依赖性 RNA 聚合酶抑制剂,是一种醌和一种针对革兰氏阳性细菌的抗生素试剂。它是涉及两个电子的可逆氧化还原系统的氧化形式。它能产生活性氧并抑制微粒体脂质过氧化,可研究肺结核和麻风病。
T67867 Mycaminosyltylonolide

Antibacterial Microbiology/Virology
Mycaminosyltylonolide 是一种大环内酯类抗生素,它是 tyololide 在位置5上具有β - d -mycaminosyl 残基。Mycaminosyltylonolide 是一种有效的抗生素,具有抗菌活性和抑制荧光素酶的合成。
T5530 Mithramycin A

Plicamycin

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Mithramycin A (Plicamycin) 是一种dna 结合的抗肿瘤抗生素,选择性特异性蛋白1 (Sp1)抑制剂,通过降低Sp1蛋白抑制多种肿瘤的生长。特异性蛋白1 (Sp1)是一种锌指转录因子,调节多种细胞功能,促进肿瘤进展。
T67731 Holomycin

N-Demethylthiolutin

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Holomycin (N-Demethylthiolutin) 是二硫代吡咯酮类的次级代谢产物。 HolomycinHolomycin 是一种抗生素次级代谢物,是天然产光杆菌galatheae S2753形成生物膜所必需的,也是一种广谱抗生素。holomycin 通过其烯-二硫基团促进S2753的生物膜形成。 Holomycin 具有抗肿瘤活性,可参与 RNA 合成。
TQ0215 Salinomycin sodium salt

盐霉素钠,Sodium salinomycin,Salinomycin sodium

Apoptosis; Wnt/beta-catenin; Antibacterial; Antibiotic; Autophagy Apoptosis; Autophagy; Cytoskeletal Signaling; Microbiology/Virology; Stem Cells
Salinomycin sodium salt (Sodium salinomycin) 是钾离子载体抗生素,是作用于 Wnt/Fzd/LRP 复合物的Wnt/β-catenin 信号传导抑制剂,能阻断 Wnt 诱导的 LRP6 磷酸化,导致 LRP6 蛋白降解。它选择性抑制人肿瘤干细胞。
T1235 Lincomycin hydrochloride monohydrate

洁霉素盐酸盐,林可霉素,Lincomycin hydrochloride hydrate

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Lincomycin hydrochloride monohydrate (Lincomycin hydrochloride hydrate) 是一种窄谱抗生素, 具有与红霉素相似的效力, 对革兰氏阳性球菌的作用效果很好, 主要抑制细菌细胞蛋白质的合成。
T3675 1-Deoxynojirimycin

Duvoglustat,Moranoline,1-脱氧野尻霉素,moranolin

PI3K; Glucosidase Metabolism; PI3K/Akt/mTOR signaling
1-Deoxynojirimycin (Moranoline) 是一种口服具有活性的 α-葡萄糖苷酶抑制剂。它具有降血糖、减肥和抗病毒的活性。它抑制餐后血糖,预防糖尿病。
T0709 Natamycin

纳他霉素,Pimaricin

Estrogen/progestogen Receptor; Endogenous Metabolite; Antibiotic; Antifungal Endocrinology/Hormones; Metabolism; Microbiology/Virology
Natamycin (Pimaricin) 是由数个链霉菌菌株生产的大环内酯类抗生素,可通过抑制氨基酸和葡萄糖跨质膜的运输来抑制真菌生长。它是一种食品防腐剂,在农业中作抗真菌剂。它可研究真菌性角膜炎。
T13229 Tunicamycin

Influenza Virus; Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Tunicamycin 是一种抗生素的混合物,通过阻断 GlcNAc 磷酸转移酶 (GPT),抑制 N-连接糖基化。Tunicamycin 具有抗肿瘤活性,还具有抗细菌、抗真菌和抗病毒活性。
T8641 Vancomycin

Antibacterial; Antibiotic; Autophagy Autophagy; Microbiology/Virology
Vancomycin 是一种糖肽类抗生素,可以通过改变细胞膜的渗透性并选择性地抑制核糖核酸的合成以发挥抗菌活性。Vancomycin 可以用于治疗所有抗生素均无效的严重感染。
T3629 Gamithromycin

ML-1709460,加米霉素

Antibacterial; Antibiotic Microbiology/Virology
Gamithromycin (ML-1709460) 是一种可抑制 MmmSC 菌株 B237 和 Tan8 生长的大环内酯类抗菌剂,MIC 值分别为 0.00012 和 0.00006 μg/mL。
T14329 Ascamycin

Nucleoside Antimetabolite/Analog; Others; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others
Ascamycin 是一种由链霉菌属产生的 5'-O-磺酰胺核糖核苷抗生素,对黄单胞菌类显示出选择性的抗菌活性,对柠檬黄单胞菌、口蹄疫黄单胞菌和噬菌体具有抑制作用,MIC 值分别为0.4μg/mL、12.5μg/mL 和12.5μg/mL。
T6293 Mycophenolate Mofetil

TM-MMF,吗替麦考酚酯,RS 61443

Apoptosis; Dehydrogenase; Drug Metabolite Apoptosis; Metabolism
Mycophenolate Mofetil (TM-MMF) 是 Mycophenolic acid 的吗啉乙酯前药。它通过抑制肌苷一磷酸脱氢酶抑制从头嘌呤合成,显示出选择性淋巴细胞抗增殖作用。
T8262 Fosfomycin sodium

Fosfomycin Disodium,磷霉素钠

Antibacterial; Antibiotic Microbiology/Virology
Fosfomycin sodium 是一种能透过血脑屏障的广谱抗生素,不可逆地抑制细胞壁合成的早期阶段。它对多种细菌具有杀菌活性,包括耐多药、广泛耐药和耐全药的细菌。
T20699 Daunomycinone

Daunomycinon,Leukaemomycinone C,NSC 109351,NSC-109351,NSC109351

Antibiotic Microbiology/Virology
Daunomycinone (NSC-109351) 是daunomycin 的聚糖,属于抗生素类,是抑制肿瘤的蒽环类化合物的代表性聚糖,可用来治疗癌症和白血病。
T0474 Erythromycin ethylsuccinate

EES,琥乙红霉素

ribosome; HIV Protease; Antibacterial; Antibiotic; Autophagy Autophagy; Microbiology/Virology; Proteases/Proteasome
Erythromycin ethylsuccinate (EES) 是一种由红链霉菌产生的大环内酯类抗生素,有潜力用于多种细菌感染。它具有抗 HIV-1病毒活性。
T17143 Toyocamycin

丰加霉素,Vengicide

Apoptosis; Others; IRE1; Antibiotic; Antifungal Apoptosis; Cell Cycle/Checkpoint; Microbiology/Virology; Others
Toyocamycin (Vengicide) 是放线菌类产生的腺苷类似物,为 X 盒结合蛋白 1 (XBP1) 抑制剂,抑制 IRE1α 诱导的 ATP 依赖性 XBP1 mRNA 的断裂,IC50值为 80 nM。它还诱导凋亡。
T0788 Spectinomycin dihydrochloride

淋必治,Spectinomycin 2HCl,盐酸奇霉素,Actinospectacin

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Spectinomycin dihydrochloride (Actinospectacin) 是一种能与细菌核糖体的30S 亚基结合,干扰蛋白质合成的抗生素。
T15245 Erythromycin estolate

Phtalic anhydride,ilosone

Antibacterial Microbiology/Virology
Erythromycin estolate 是红霉素的衍生物,属于大环内酯类抗生素,常用于研究多种细菌感染。酯酸红霉素对胆汁酸转运有抑制作用,可引起肝损伤,主要是胆汁淤积性肝炎。
T1419 Azithromycin hydrate

CP-62993 dihydrate,阿奇霉素二水物,Azithromycin dihydrate,阿奇霉素二水合物

ribosome; Antibacterial; Antibiotic; Autophagy Autophagy; Microbiology/Virology
Azithromycin hydrate (CP-62993 dihydrate) 是一种大环内酯抗生素,可研究细菌感染。
T6290 Tanespimycin

坦螺旋霉素,17-AAG,CP 127374,NSC 330507,KOS 953

Apoptosis; Mitophagy; HSP; Antibacterial; Antibiotic; Autophagy Apoptosis; Autophagy; Cytoskeletal Signaling; Metabolism; Microbiology/Virology
Tanespimycin (KOS 953) 是一种 Hsp90 抑制剂,可选择性抑制 BT474 肿瘤细胞 Hsp90,IC50为 5 nM。它消耗细胞内 STK38/NDR1,并降低 STK38 激酶活性,还能下调stk38基因表达。
T8504 Dianemycin

Nanchangmycin (free acid)

Antibacterial; Antibiotic Microbiology/Virology
Dianemycin (Nanchangmycin (free acid)) 由Streptomyces nanchangensis 产生的一种聚醚抗生素,抑制革兰氏阳性菌。它也是一种针对 Zika 病毒的广谱抗病毒药物。
T6758 Anisomycin

茴香霉素,Flagecidin,NSC 76712,Wuningmeisu C

Apoptosis; DNA/RNA Synthesis; Antibacterial; Antibiotic; JNK Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; MAPK; Microbiology/Virology
Anisomycin (Flagecidin) 属于细菌抗生素,是一种蛋白合成抑制剂和一种 JNK 激活剂。Anisomycin 通过抑制肽基转移酶或 80S 核糖体系统来干扰蛋白质和 DNA 的合成。
T6740 Bafilomycin A1

巴佛洛霉素A1,巴佛洛霉素 A1

Apoptosis; Proton pump; Antibacterial; Antibiotic; Autophagy Apoptosis; Autophagy; Membrane transporter/Ion channel; Microbiology/Virology
Bafilomycin A1 属于大环内酯类抗生素,是一种 V-ATPase 抑制剂 (IC50=0.44 nM),具有特异性和可逆性。Bafilomycin A1 是自噬晚期阶段抑制剂,阻断自噬体与溶酶体的融合。Bafilomycin A1 也诱导凋亡。
T36818 Questiomycin A

GPR; Antibacterial Endocrinology/Hormones; GPCR/G Protein; Microbiology/Virology
Questiomycin A 是一种在鲜奶油中生产的抗生素,具有抗菌和抗癌活性。 Questiomycin A 抑制细胞保护性 ER 伴侣蛋白 GRP78 的表达。
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天然产物

Lusianthridin
Cat.No: TN1892
Synonym:
Target: Others, c-Myc
Artemisitene
Cat.No: T21065
Synonym:
Target: Others
Mollugin
Cat.No: T3673
Synonym: 大叶茜草素,Rubimaillin
Target: HER, JAK
Agrimol B
Cat.No: T4S1173
Synonym: 仙鹤草酚B,仙鹤草酚 B
Target: Sirtuin, PPAR
(S)-10-Hydroxycamptothecin
Cat.No: T2764
Synonym: 10-羟喜树碱,10-羟基喜树碱,10-Hydroxycamptothecin,10-HCPT
Target: Apoptosis, Topoisomerase
Azithromycin
Cat.No: T6401
Synonym: 阿奇霉素,Zithromax,CP 62993,XZ-450
Target: Others, Antibacterial, Antibiotic, Autophagy
Kasugamycin hydrochloride
Cat.No: T2762
Synonym: Kasumin,盐酸春雷霉素
Target: Antibacterial, Antibiotic, Antifungal
Daptomycin
Cat.No: T1665
Synonym: 达托霉素,LY146032
Target: DNA/RNA Synthesis, Antibacterial, Antibiotic
Phleomycin
Cat.No: T21498
Synonym:
Target: DNA/RNA Synthesis, Antibacterial, Antibiotic
Mycophenolic acid
Cat.No: T1335
Synonym: 霉酚酸,Mycophenolate,RS-61443
Target: Apoptosis, Dehydrogenase, Endogenous Metabolite, Antibacterial, Antibiotic, UGT, Antifungal
Ionomycin calcium
Cat.No: T11665
Synonym: SQ23377 calcium,罗红霉素钙盐(链霉菌属载体)
Target: Apoptosis, Calcium Channel, Antibacterial, Antibiotic, PKC
Ribostamycin sulfate
Cat.No: T1214
Synonym: Vistamycin sulfate,硫酸核糖霉素
Target: Antibacterial, Antibiotic
Lincomycin hydrochloride
Cat.No: T1277
Synonym: Lincomycin HCl,NSC 70731,盐酸林可霉素,U10149A
Target: ribosome, Antibacterial, Antibiotic
Midecamycin
Cat.No: T5037
Synonym: Antibiotic SF-837,Turimycin P3,Medecamycin A1,Rubimycin,麦迪霉素,Platenomycin B1,Espinomycin A
Target: Antibacterial, Antibiotic
Geldanamycin
Cat.No: T6343
Synonym: 格尔德霉素,NSC 122750
Target: HSP, Influenza Virus, Tyrosine Kinases, Antibacterial, Antibiotic
Milbemycin oxime
Cat.No: T1381
Synonym:
Target: Others, Antibiotic, Parasite
Apramycin sulfate
Cat.No: T1084
Synonym: Nebramycin II,Ai3-29795,硫酸安普霉素,硫酸阿布拉霉素
Target: Antibacterial, Antibiotic
Aclacinomycin A
Cat.No: T21502
Synonym: Aclarubicin
Target: Topoisomerase
Azomycin
Cat.No: T6402
Synonym: 2-Nitroimidazole,2-硝基咪唑,Ro 05-9129,Amicin
Target: Antibacterial, Antibiotic
Tobramycin
Cat.No: T1255
Synonym: NSC 180514,妥布霉素,Nebramycin Factor 6,Deoxykanamycin B
Target: ribosome, Antibacterial, Antibiotic
Resistomycin
Cat.No: T21820
Synonym: Geliomycin,Heliomycin
Target: Antibiotic
Rifamycin sodium
Cat.No: T5003
Synonym: Rifamycin sodium salt,利福霉素钠
Target: Antibacterial, Antibiotic
Kanamycin sulfate
Cat.No: T0793
Synonym: 硫酸卡那霉素,Kanamycin monosulfate,Kanamycin A monosulfate,Ophtalmokalixan
Target: ribosome, Antibacterial, Antibiotic
Leucomycin
Cat.No: T3607
Synonym: 吉他霉素,Kitasamycin,Leucomycin V,Turimycin
Target: Antibacterial, Antibiotic
Ascomycin
Cat.No: T2481
Synonym: FK520,Immunomycin,子囊霉素,FR-900520
Target: Phosphatase, Others, Antibiotic, Parasite, Antifungal
Rifamycin S
Cat.No: T8347
Synonym:
Target: Reactive Oxygen Species, ROS, Antibacterial, Antibiotic
Mycaminosyltylonolide
Cat.No: T67867
Synonym:
Target: Antibacterial
Mithramycin A
Cat.No: T5530
Synonym: Plicamycin
Target: DNA/RNA Synthesis
Holomycin
Cat.No: T67731
Synonym: N-Demethylthiolutin
Target: DNA/RNA Synthesis
Salinomycin sodium salt
Cat.No: TQ0215
Synonym: 盐霉素钠,Sodium salinomycin,Salinomycin sodium
Target: Apoptosis, Wnt/beta-catenin, Antibacterial, Antibiotic, Autophagy
Lincomycin hydrochloride monohydrate
Cat.No: T1235
Synonym: 洁霉素盐酸盐,林可霉素,Lincomycin hydrochloride hydrate
Target: ribosome, Antibacterial, Antibiotic
1-Deoxynojirimycin
Cat.No: T3675
Synonym: Duvoglustat,Moranoline,1-脱氧野尻霉素,moranolin
Target: PI3K, Glucosidase
Natamycin
Cat.No: T0709
Synonym: 纳他霉素,Pimaricin
Target: Estrogen/progestogen Receptor, Endogenous Metabolite, Antibiotic, Antifungal
Tunicamycin
Cat.No: T13229
Synonym:
Target: Influenza Virus, Antibacterial, Antibiotic, Antifungal
Vancomycin
Cat.No: T8641
Synonym:
Target: Antibacterial, Antibiotic, Autophagy
Gamithromycin
Cat.No: T3629
Synonym: ML-1709460,加米霉素
Target: Antibacterial, Antibiotic
Ascamycin
Cat.No: T14329
Synonym:
Target: Nucleoside Antimetabolite/Analog, Others, Antibacterial, Antibiotic
Mycophenolate Mofetil
Cat.No: T6293
Synonym: TM-MMF,吗替麦考酚酯,RS 61443
Target: Apoptosis, Dehydrogenase, Drug Metabolite
Fosfomycin sodium
Cat.No: T8262
Synonym: Fosfomycin Disodium,磷霉素钠
Target: Antibacterial, Antibiotic
Daunomycinone
Cat.No: T20699
Synonym: Daunomycinon,Leukaemomycinone C,NSC 109351,NSC-109351,NSC109351
Target: Antibiotic
Erythromycin ethylsuccinate
Cat.No: T0474
Synonym: EES,琥乙红霉素
Target: ribosome, HIV Protease, Antibacterial, Antibiotic, Autophagy
Toyocamycin
Cat.No: T17143
Synonym: 丰加霉素,Vengicide
Target: Apoptosis, Others, IRE1, Antibiotic, Antifungal
Spectinomycin dihydrochloride
Cat.No: T0788
Synonym: 淋必治,Spectinomycin 2HCl,盐酸奇霉素,Actinospectacin
Target: ribosome, Antibacterial, Antibiotic
Erythromycin estolate
Cat.No: T15245
Synonym: Phtalic anhydride,ilosone
Target: Antibacterial
Azithromycin hydrate
Cat.No: T1419
Synonym: CP-62993 dihydrate,阿奇霉素二水物,Azithromycin dihydrate,阿奇霉素二水合物
Target: ribosome, Antibacterial, Antibiotic, Autophagy
Tanespimycin
Cat.No: T6290
Synonym: 坦螺旋霉素,17-AAG,CP 127374,NSC 330507,KOS 953
Target: Apoptosis, Mitophagy, HSP, Antibacterial, Antibiotic, Autophagy
Dianemycin
Cat.No: T8504
Synonym: Nanchangmycin (free acid)
Target: Antibacterial, Antibiotic
Anisomycin
Cat.No: T6758
Synonym: 茴香霉素,Flagecidin,NSC 76712,Wuningmeisu C
Target: Apoptosis, DNA/RNA Synthesis, Antibacterial, Antibiotic, JNK
Bafilomycin A1
Cat.No: T6740
Synonym: 巴佛洛霉素A1,巴佛洛霉素 A1
Target: Apoptosis, Proton pump, Antibacterial, Antibiotic, Autophagy
Questiomycin A
Cat.No: T36818
Synonym:
Target: GPR, Antibacterial
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Cat. No. Product Name Species Expression System
TMPH-01720 c-Myc Protein, Human, Recombinant (His)

Myc proto-oncogene protein,Transcription factor p64...

Human E. coli
Transcription factor that binds DNA in a non-specific manner, yet also specifically recognizes the core sequence 5'-CAC[GA]TG-3'. Activates the transcription of growth-related genes. Binds to the VEGFA promoter, promoting VEGFA production and subsequent sprouting angiogenesis. Regulator of somatic reprogramming, controls self-renewal of embryonic stem cells. Functions with TAF6L to activate target gene expression through RNA polymerase II pause release. c-Myc Protein, Human, Recombinant (His) is...
TMPH-02791 c-Myc Protein, Mouse, Recombinant (GST)

bHLHe39,MYC,Transcription factor p64,Class E basic ...

Mouse E. coli
Transcription factor that binds DNA in a non-specific manner, yet also specifically recognizes the core sequence 5'-CAC[GA]TG-3'. Activates the transcription of growth-related genes. Binds to the VEGFA promoter, promoting VEGFA production and subsequent sprouting angiogenesis. Regulator of somatic reprogramming, controls self-renewal of embryonic stem cells. Functions with TAF6L to activate target gene expression through RNA polymerase II pause release. c-Myc Protein, Mouse, Recombinant (GST) is...
TMPH-01721 c-Myc Protein, Human, Recombinant (Avi & His & MBP), Biotinylated

BHLHE39,Class E basic helix-loop-helix protein 39,Transcript...

Human E. coli
Transcription factor that binds DNA in a non-specific manner, yet also specifically recognizes the core sequence 5'-CAC[GA]TG-3'. Activates the transcription of growth-related genes. Binds to the VEGFA promoter, promoting VEGFA production and subsequent sprouting angiogenesis. Regulator of somatic reprogramming, controls self-renewal of embryonic stem cells. Functions with TAF6L to activate target gene expression through RNA polymerase II pause release. c-Myc Protein, Human, Recombinant (Avi & H...
TMPH-01775 N-myc Protein, Human, Recombinant (His)

MYCN,Class E basic helix-loop-helix protein 37,N-

Human P. pastoris (Yeast)
Positively regulates the transcription of MYCNOS in neuroblastoma cells. N-myc Protein, Human, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 51.6 kDa and the accession number is P04198.
TMPH-01801 NME2 Protein, Human, Recombinant (His & Myc)

NME2,nm23-H2,Histidine protein kinase NDKB,Nucleoside diphos...

Human E. coli
NME2 Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 24.2 kDa and the accession number is P22392.
TMPY-02888 MAX Protein, Human, Recombinant (His & GST)

MYC associated factor X,bHLHd4

Human Baculovirus Insect Cells
MYC associated factor X contains 1 basic helix-loop-helix (bHLH) domain and belongs to the MAX family. It is highly expressed in the brain, heart, and lung while lower levels are seen in the liver, kidney, and skeletal muscle. MYC associated factor X can form homodimers and heterodimers with other family members, which include Mad, Mxi1, and Myc. Myc is an oncoprotein implicated in cell proliferation, differentiation, and apoptosis. The homodimers and heterodimers compete for a common DNA target...
TMPH-00857 ABAT Protein, Human, Recombinant (His & Myc & SUMO)

L-AIBAT,GABA aminotransferase,GABA transaminase,GABA-T,(S)-3...

Human E. coli
Catalyzes the conversion of gamma-aminobutyrate and L-beta-aminoisobutyrate to succinate semialdehyde and methylmalonate semialdehyde, respectively. Can also convert delta-aminovalerate and beta-alanine. ABAT Protein, Human, Recombinant (His & Myc & SUMO) is expressed in E. coli expression system with N-10xHis-SUMO and C-Myc tag. The predicted molecular weight is 73.3 kDa and the accession number is P80404.
TMPJ-01040 MAX Protein, Human, Recombinant (His)

Protein Max,MAX,bHLHd4,Myc-Associated Factor X,Clas...

Human E. coli
Myc-Associated Factor X (MAX) is a member of the basic helix-loop-helix leucine zipper (bHLHZ) family of transcription factors. It contains 1 basic helix-loop-helix (bHLH) domain. It is found in the brain, heart, and lung at high levels while lower levels are seen in the liver, kidney, and skeletal muscle. MAX forms a sequence-specific DNA-binding protein complex with MYC or MAD which recognizes the core sequence 5'-CAC[GA]TG-3'. The MYC-MAX complex is a transcriptional activator, whereas the MA...
TMPY-03443 NDRG1 Protein, Human, Recombinant (His)

TARG1,PROXY1,RIT42,NDR1,DRG1,RTP,TDD5,CMT4D,CAP43,NMSL,N-

Human E. coli
NDRG1 gene is a member of the N-Myc downregulated gene family which belongs to the alpha/beta hydrolase superfamily. NDRG1 is a cytoplasmic protein involved in stress responses, hormone responses, cell growth, and differentiation. NDRG1 is necessary for p53-mediated caspase activation and apoptosis. Mutations in the NDRG1 gene are a cause of Charcot-Marie-Tooth disease type 4D, and expression of this gene may be a prognostic indicator for several types of cancer. NDRG1 is a stress-responsive pro...
TMPJ-01097 ZBTB17 Protein, Human, Recombinant (His)

MIZ1,ZNF60,Myc-Interacting Zinc Finger Protein 1,ZN...

Human E. coli
Zinc Finger and BTB Domain-Containing Protein 17 (ZBTB17) belongs to the Kruppel C2H2-type zinc finger protein family. ZBTB17 may function as a housekeeping DNA-binding protein that regulates the expression of specific genes, it has been shown to bind to the promoters of adenovirus major late protein and cyclin D1 and activate transcription. ZBTB17 may has growth arrest activity, probably through inhibition of cell cycle progression. ZBTB17 required for early embryonic development during gastrul...
TMPH-03372 Sharpin Protein, Rat, Recombinant (His & Myc)

Sharpin,Shank-associated RH domain-interacting protein

Rat E. coli
Sharpin Protein, Rat, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 47.7 kDa and the accession number is Q9EQL9.
TMPH-01949 PML Protein, Human, Recombinant (His & Myc)

PML,Tripartite motif-containing protein 19,RING-type E3 SUMO...

Human Baculovirus Insect Cells
PML Protein, Human, Recombinant (His & Myc) is expressed in Baculovirus insect cells with N-10xHis and C-Myc tag. The predicted molecular weight is 24.5 kDa and the accession number is P29590.
TMPH-01262 PRKN Protein, Human, Recombinant (His & Myc)

Parkinson juvenile disease protein 2,E3 ubiquitin-protein li...

Human Baculovirus Insect Cells
PRKN Protein, Human, Recombinant (His & Myc) is expressed in Baculovirus insect cells with N-10xHis and C-Myc tag. The predicted molecular weight is 55.6 kDa and the accession number is O60260.
TMPH-02949 HADHA Protein, Mouse, Recombinant (His & Myc)

Trifunctional enzyme subunit alpha, mitochondrial,TP-alpha,H...

Mouse E. coli
HADHA Protein, Mouse, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 52.1 kDa and the accession number is Q8BMS1.
TMPH-02795 Myoglobin Protein, Mouse, Recombinant (His & Myc)

Mb,Nitrite reductase MB,Myoglobin,Pseudoperoxidase MB

Mouse HEK293 Cells
Serves as a reserve supply of oxygen and facilitates the movement of oxygen within muscles. Myoglobin Protein, Mouse, Recombinant (His & Myc) is expressed in HEK293 mammalian cells with N-10xHis and C-Myc tag. The predicted molecular weight is 21.9 kDa and the accession number is P04247.
TMPH-01378 GIPR Protein, Human, Recombinant (His & Myc)

GIPR,Glucose-dependent insulinotropic polypeptide receptor,G...

Human HEK293 Cells
This is a receptor for GIP. The activity of this receptor is mediated by G proteins which activate adenylyl cyclase. GIPR Protein, Human, Recombinant (His & Myc) is expressed in HEK293 mammalian cells with N-10xHis and C-Myc tag. The predicted molecular weight is 18.5 kDa and the accession number is P48546.
TMPH-00924 AMELX Protein, Human, Recombinant (His & Myc)

AMGX,AMG,Amelogenin, X isoform

Human Baculovirus Insect Cells
AMELX Protein, Human, Recombinant (His & Myc) is expressed in Baculovirus.
TMPH-00961 Aspartoacylase Protein, Human, Recombinant (His & Myc)

Aminoacylase-2,ACY2,ACY-2,ASP,ASPA,Aspartoacylase

Human HEK293 Cells
Aspartoacylase Protein, Human, Recombinant (His & Myc) is expressed in HEK293.
TMPH-01981 NPEPPS Protein, Human, Recombinant (His & Myc)

Cytosol alanyl aminopeptidase,NPEPPS,Puromycin-sens...

Human Baculovirus Insect Cells
NPEPPS Protein, Human, Recombinant (His & Myc) is expressed in Baculovirus.
TMPH-00920 FTO Protein, Human, Recombinant (His & Myc)

U6 small nuclear RNA (2'-O-methyladenosine-N(6)-)-demethylas...

Human E. coli
FTO Protein, Human, Recombinant (His & Myc) is expressed in E. coli.
TMPH-02517 APOD Protein, Mouse, Recombinant (His & Myc)

Apolipoprotein D,ApoD,Apo-D

Mouse E. coli
APOD occurs in the macromolecular complex with lecithin-transport and binding of bilin. Appears to be able to transport a variety of ligands in a number of different contexts. APOD Protein, Mouse, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 26.9 kDa and the accession number is P51910.
TMPH-00872 CHRNE Protein, Human, Recombinant (His & Myc)

Acetylcholine receptor subunit epsilon,ACHRE,CHRNE

Human E. coli
After binding acetylcholine, the AChR responds by an extensive change in conformation that affects all subunits and leads to opening of an ion-conducting channel across the plasma membrane. CHRNE Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 32.5 kDa and the accession number is Q04844.
TMPH-01080 Ceruloplasmin Protein, Human, Recombinant (His & Myc)

CP,Ceruloplasmin,Ferroxidase ceruloplasmin,Cuproxidase cerul...

Human E. coli
Ceruloplasmin is a blue, copper-binding (6-7 atoms per molecule) glycoprotein. It has ferroxidase activity oxidizing Fe(2+) to Fe(3+) without releasing radical oxygen species. It is involved in iron transport across the cell membrane. Provides Cu(2+) ions for the ascorbate-mediated deaminase degradation of the heparan sulfate chains of GPC1. May also play a role in fetal lung development or pulmonary antioxidant defense. Ceruloplasmin Protein, Human, Recombinant (His & Myc) is expressed in E. co...
TMPH-02431 Legumain Protein, Cynomolgus, Recombinant (His & Myc)

Legumain,Protease, cysteine 1,Asparaginyl endopeptidase,LGMN

Cynomolgus Baculovirus Insect Cells
Has a strict specificity for hydrolysis of asparaginyl bonds. Can also cleave aspartyl bonds slowly, especially under acidic conditions. Required for normal lysosomal protein degradation in renal proximal tubules. Required for normal degradation of internalized EGFR. Plays a role in the regulation of cell proliferation via its role in EGFR degradation. May be involved in the processing of proteins for MHC class II antigen presentation in the lysosomal/endosomal system. Legumain Protein, Cynomolg...
TMPH-02643 Enteropeptidase Protein, Mouse, Recombinant (His & Myc)

Serine protease 7,Prss7,Transmembrane protease serine 15,Ent...

Mouse HEK293 Cells
Responsible for initiating activation of pancreatic proteolytic proenzymes (trypsin, chymotrypsin and carboxypeptidase A). It catalyzes the conversion of trypsinogen to trypsin which in turn activates other proenzymes including chymotrypsinogen, procarboxypeptidases, and proelastases.
TMPH-02908 AICDA Protein, Mouse, Recombinant (His & Myc)

Single-stranded DNA cytosine deaminase,Cytidine aminohydrola...

Mouse E. coli
Single-stranded DNA-specific cytidine deaminase. Involved in somatic hypermutation (SHM), gene conversion, and class-switch recombination (CSR) in B-lymphocytes by deaminating C to U during transcription of Ig-variable (V) and Ig-switch (S) region DNA. Required for several crucial steps of B-cell terminal differentiation necessary for efficient antibody responses. May also play a role in the epigenetic regulation of gene expression by participating in DNA demethylation.
TMPH-02807 NPTXR Protein, Mouse, Recombinant (His & Myc)

Neuronal pentraxin receptor,Nptxr

Mouse Baculovirus Insect Cells
May be involved in mediating uptake of synaptic material during synapse remodeling or in mediating the synaptic clustering of AMPA glutamate receptors at a subset of excitatory synapses.
TMPH-02863 LOX Protein, Mouse, Recombinant (His & Myc)

Ras excision protein,Protein-lysine 6-oxidase,Lysyl oxidase,...

Mouse Baculovirus Insect Cells
Responsible for the post-translational oxidative deamination of peptidyl lysine residues in precursors to fibrous collagen and elastin. Regulator of Ras expression. May play a role in tumor suppression. Plays a role in the aortic wall architecture.
TMPH-01565 IARS Protein, Human, Recombinant (His & Myc)

Isoleucine--tRNA ligase, cytoplasmic,Isoleucyl-tRNA syntheta...

Human E. coli
Catalyzes the specific attachment of an amino acid to its cognate tRNA in a 2 step reaction: the amino acid (AA) is first activated by ATP to form AA-AMP and then transferred to the acceptor end of the tRNA.
TMPH-00133 AcMNPV Major capsid Protein (His & Myc)

VP39,P39

AcMNPV E. coli
Most abundant structural protein of the nucleocapsid produced during the infection cycle. The monomers are arranged in stacked rings around the nucleoprotein core. AcMNPV Major capsid Protein (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 46.4 kDa and the accession number is P17499.
TMPH-01898 PARL Protein, Human, Recombinant (Myc)

Mitochondrial intramembrane cleaving protease PARL,Presenili...

Human E. coli
Required for the control of apoptosis during postnatal growth. Essential for proteolytic processing of an antiapoptotic form of OPA1 which prevents the release of mitochondrial cytochrome c in response to intrinsic apoptotic signals. Required for the maturation of PINK1 into its 52kDa mature form after its cleavage by mitochondrial-processing peptidase (MPP). Promotes changes in mitochondria morphology regulated by phosphorylation of P-beta domain. PARL Protein, Human, Recombinant (Myc) is expre...
TMPH-01900 DDX5 Protein, Human, Recombinant (His & Myc)

HELR,RNA helicase p68,HLR1,G17P1,DEAD box protein 5,Probable...

Human E. coli
DDX5 Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 74.1 kDa and the accession number is P17844.
TMPH-00973 DHX36 Protein, Human, Recombinant (His & Myc)

DEAH-box protein 36,G4R1,ATP-dependent DNA/RNA helicase DHX3...

Human E. coli
DHX36 Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 18.2 kDa and the accession number is Q9H2U1.
TMPH-01606 BAG6 Protein, Human, Recombinant (His & Myc)

BAG-6,Protein G3,BAG family molecular chaperone regulator 6,...

Human Baculovirus Insect Cells
BAG6 Protein, Human, Recombinant (His & Myc) is expressed in Baculovirus insect cells with N-10xHis and C-Myc tag. The predicted molecular weight is 38.7 kDa and the accession number is P46379.
TMPH-02930 TREX1 Protein, Mouse, Recombinant (His & Myc)

3'-5' exonuclease TREX1,Three-prime repair exonuclease 1,Tre...

Mouse E. coli
TREX1 Protein, Mouse, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 41.1 kDa and the accession number is Q91XB0.
TMPH-02491 SCD1 Protein, Mouse, Recombinant (His & Myc)

Stearoyl-CoA desaturase 1,Scd1,Delta(9)-desaturase 1,Fatty a...

Mouse E. coli
SCD1 Protein, Mouse, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 18.4 kDa and the accession number is P13516.
TMPH-02899 VRK1 Protein, Mouse, Recombinant (His & Myc)

Vaccinia-related kinase 1,Serine/threonine-protein kinase 51...

Mouse E. coli
VRK1 Protein, Mouse, Recombinant (His & Myc) is expressed in E. coli expression system with N-6xHis and C-Myc tag. The predicted molecular weight is 55.2 kDa and the accession number is Q80X41.
TMPH-01327 FBXO48 Protein, Human, Recombinant (His & Myc)

F-box protein 48,F-box only protein 48,FBXO48

Human E. coli
FBXO48 Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 25.7 kDa and the accession number is Q5FWF7.
TMPH-02007 RIPK1 Protein, Human, Recombinant (His & Myc)

Receptor-interacting protein 1,Receptor-interacting serine/t...

Human E. coli
RIPK1 Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 49.4 kDa and the accession number is Q13546.
TMPH-02893 SVS4 Protein, Mouse, Recombinant (His & Myc)

Seminal vesicle protein 2,Seminal vesicle secretory protein ...

Mouse E. coli
N/A. SVS4 Protein, Mouse, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 17.8 kDa and the accession number is P18419.
TMPH-03330 Mcpt4 Protein, Rat, Recombinant (His & Myc)

Mast cell protease IV,Mast cell protease 4,Mcpt4

Rat E. coli
N/A. Mcpt4 Protein, Rat, Recombinant (His & Myc) is expressed in E. coli expression system with N-6xHis and C-Myc tag. The predicted molecular weight is 30.5 kDa and the accession number is P97592.
TMPH-01030 CAPN14 Protein, Human, Recombinant (His & Myc)

Calpain-14,Calcium-activated neutral proteinase 14,CAPN14,CA...

Human Baculovirus Insect Cells
Calcium-regulated non-lysosomal thiol-protease. CAPN14 Protein, Human, Recombinant (His & Myc) is expressed in Baculovirus insect cells with N-10xHis and C-Myc tag. The predicted molecular weight is 78.6 kDa and the accession number is A8MX76.
TMPH-02484 ADAMTS13 Protein, Mouse, Recombinant (His & Myc)

ADAM-TS 1,A disintegrin and metalloproteinase with thrombosp...

Mouse E. coli
Cleaves the vWF multimers in plasma into smaller forms thereby controlling vWF-mediated platelet thrombus formation. ADAMTS13 Protein, Mouse, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 32.7 kDa and the accession number is Q769J6.
TMPH-02682 GSTM3 Protein, Mouse, Recombinant (His & Myc)

GST class-mu 3,Gstm3,Glutathione S-transferase Mu 3,Glutathi...

Mouse E. coli
Conjugation of reduced glutathione to a wide number of exogenous and endogenous hydrophobic electrophiles. GSTM3 Protein, Mouse, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 33.0 kDa and the accession number is P19639.
TMPH-01203 DCAF16 Protein, Human, Recombinant (His & Myc)

C4orf30,DCAF16,DDB1- and CUL4-associated factor 16

Human E. coli
Functions as a substrate recognition component for CUL4-DDB1 E3 ubiquitin-protein ligase complex, which mediates ubiquitination and proteasome-dependent degradation of nuclear proteins. DCAF16 Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 31.2 kDa and the accession number is Q9NXF7.
TMPH-01579 KRT19 Protein, Human, Recombinant (His & Myc)

Cytokeratin-19,KRT19,Keratin, type I cytoskeletal 19,Keratin...

Human Baculovirus Insect Cells
Involved in the organization of myofibers. Together with KRT8, helps to link the contractile apparatus to dystrophin at the costameres of striated muscle. KRT19 Protein, Human, Recombinant (His & Myc) is expressed in Baculovirus insect cells with N-10xHis and C-Myc tag. The predicted molecular weight is 48 kDa and the accession number is P08727.
TMPH-00922 ALPK1 Protein, Human, Recombinant (His & Myc)

KIAA1527,Lymphocyte alpha-protein kinase,Alpha-protein kinas...

Human Baculovirus Insect Cells
ALPK1 Protein, Human, Recombinant (His & Myc) is expressed in Baculovirus.
TMPH-00914 ALKAL2 Protein, Human, Recombinant (His & Myc)

FAM150B,AUG-alpha,Augmentor alpha,ALK and LTK ligand 2

Human Baculovirus Insect Cells
ALKAL2 Protein, Human, Recombinant (His & Myc) is expressed in Baculovirus.
TMPH-02033 RPE65 Protein, Human, Recombinant (His & Myc)

Retinol isomerase,Retinoid isomerohydrolase,All-trans-retiny...

Human Baculovirus Insect Cells
RPE65 Protein, Human, Recombinant (His & Myc) is expressed in Baculovirus.
TMPH-02800 SIRT5 Protein, Mouse, Recombinant (His & Myc)

Regulatory protein SIR2 homolog 5,Sirt5,NAD-dependent protei...

Mouse Baculovirus Insect Cells
SIRT5 Protein, Mouse, Recombinant (His & Myc) is expressed in Baculovirus.
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重组蛋白

c-Myc Protein, Human, Recombinant (His)
Cat.No: TMPH-01720
Species: Human
Expression System: E. coli
c-Myc Protein, Mouse, Recombinant (GST)
Cat.No: TMPH-02791
Species: Mouse
Expression System: E. coli
c-Myc Protein, Human, Recombinant (Avi & His & MBP), Biotinylated
Cat.No: TMPH-01721
Species: Human
Expression System: E. coli
N-myc Protein, Human, Recombinant (His)
Cat.No: TMPH-01775
Species: Human
Expression System: P. pastoris (Yeast)
NME2 Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-01801
Species: Human
Expression System: E. coli
MAX Protein, Human, Recombinant (His & GST)
Cat.No: TMPY-02888
Species: Human
Expression System: Baculovirus Insect Cells
ABAT Protein, Human, Recombinant (His & Myc & SUMO)
Cat.No: TMPH-00857
Species: Human
Expression System: E. coli
MAX Protein, Human, Recombinant (His)
Cat.No: TMPJ-01040
Species: Human
Expression System: E. coli
NDRG1 Protein, Human, Recombinant (His)
Cat.No: TMPY-03443
Species: Human
Expression System: E. coli
ZBTB17 Protein, Human, Recombinant (His)
Cat.No: TMPJ-01097
Species: Human
Expression System: E. coli
Sharpin Protein, Rat, Recombinant (His & Myc)
Cat.No: TMPH-03372
Species: Rat
Expression System: E. coli
PML Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-01949
Species: Human
Expression System: Baculovirus Insect Cells
PRKN Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-01262
Species: Human
Expression System: Baculovirus Insect Cells
HADHA Protein, Mouse, Recombinant (His & Myc)
Cat.No: TMPH-02949
Species: Mouse
Expression System: E. coli
Myoglobin Protein, Mouse, Recombinant (His & Myc)
Cat.No: TMPH-02795
Species: Mouse
Expression System: HEK293 Cells
GIPR Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-01378
Species: Human
Expression System: HEK293 Cells
AMELX Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-00924
Species: Human
Expression System: Baculovirus Insect Cells
Aspartoacylase Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-00961
Species: Human
Expression System: HEK293 Cells
NPEPPS Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-01981
Species: Human
Expression System: Baculovirus Insect Cells
FTO Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-00920
Species: Human
Expression System: E. coli
APOD Protein, Mouse, Recombinant (His & Myc)
Cat.No: TMPH-02517
Species: Mouse
Expression System: E. coli
CHRNE Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-00872
Species: Human
Expression System: E. coli
Ceruloplasmin Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-01080
Species: Human
Expression System: E. coli
Legumain Protein, Cynomolgus, Recombinant (His & Myc)
Cat.No: TMPH-02431
Species: Cynomolgus
Expression System: Baculovirus Insect Cells
Enteropeptidase Protein, Mouse, Recombinant (His & Myc)
Cat.No: TMPH-02643
Species: Mouse
Expression System: HEK293 Cells
AICDA Protein, Mouse, Recombinant (His & Myc)
Cat.No: TMPH-02908
Species: Mouse
Expression System: E. coli
NPTXR Protein, Mouse, Recombinant (His & Myc)
Cat.No: TMPH-02807
Species: Mouse
Expression System: Baculovirus Insect Cells
LOX Protein, Mouse, Recombinant (His & Myc)
Cat.No: TMPH-02863
Species: Mouse
Expression System: Baculovirus Insect Cells
IARS Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-01565
Species: Human
Expression System: E. coli
AcMNPV Major capsid Protein (His & Myc)
Cat.No: TMPH-00133
Species: AcMNPV
Expression System: E. coli
PARL Protein, Human, Recombinant (Myc)
Cat.No: TMPH-01898
Species: Human
Expression System: E. coli
DDX5 Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-01900
Species: Human
Expression System: E. coli
DHX36 Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-00973
Species: Human
Expression System: E. coli
BAG6 Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-01606
Species: Human
Expression System: Baculovirus Insect Cells
TREX1 Protein, Mouse, Recombinant (His & Myc)
Cat.No: TMPH-02930
Species: Mouse
Expression System: E. coli
SCD1 Protein, Mouse, Recombinant (His & Myc)
Cat.No: TMPH-02491
Species: Mouse
Expression System: E. coli
VRK1 Protein, Mouse, Recombinant (His & Myc)
Cat.No: TMPH-02899
Species: Mouse
Expression System: E. coli
FBXO48 Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-01327
Species: Human
Expression System: E. coli
RIPK1 Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-02007
Species: Human
Expression System: E. coli
SVS4 Protein, Mouse, Recombinant (His & Myc)
Cat.No: TMPH-02893
Species: Mouse
Expression System: E. coli
Mcpt4 Protein, Rat, Recombinant (His & Myc)
Cat.No: TMPH-03330
Species: Rat
Expression System: E. coli
CAPN14 Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-01030
Species: Human
Expression System: Baculovirus Insect Cells
ADAMTS13 Protein, Mouse, Recombinant (His & Myc)
Cat.No: TMPH-02484
Species: Mouse
Expression System: E. coli
GSTM3 Protein, Mouse, Recombinant (His & Myc)
Cat.No: TMPH-02682
Species: Mouse
Expression System: E. coli
DCAF16 Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-01203
Species: Human
Expression System: E. coli
KRT19 Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-01579
Species: Human
Expression System: Baculovirus Insect Cells
ALPK1 Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-00922
Species: Human
Expression System: Baculovirus Insect Cells
ALKAL2 Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-00914
Species: Human
Expression System: Baculovirus Insect Cells
RPE65 Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-02033
Species: Human
Expression System: Baculovirus Insect Cells
SIRT5 Protein, Mouse, Recombinant (His & Myc)
Cat.No: TMPH-02800
Species: Mouse
Expression System: Baculovirus Insect Cells
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Cat. No. Product Name Target Signaling Pathways
TMIH-0359 Mycophenolic Acid-d3 Phenyl Glucuronide

Mycophenolic Acid-d3 Phenyl Glucuronide 是 Mycophenolic Acid Phenyl Glucuronide 的氘代化合物。Mycophenolic Acid Phenyl Glucuronide 的 CAS 号为 31528-44-6。Mycophenolic acid glucuronide是人血浆中mycophenolic acid的葡糖甙代谢产物。
TMID-0284 Vancomycin-d12 TFA

Vancomycin-d12 TFA 是 Vancomycin TFA 的氘代化合物。Vancomycin TFA 的 CAS 号为 1404-90-6。Vancomycin 是一种抗生素,用于通过阻止细菌生长来治疗严重的细菌感染。它还改变细胞膜的渗透性并选择性地抑制核糖核酸的合成。
TMID-0283 Vancomycin-13C-d3

Vancomycin-13C-d3 是 Vancomycin 的 13C 和氘代化合物。Vancomycin 的 CAS 号为 1404-90-6。Vancomycin 是一种抗生素,用于通过阻止细菌生长来治疗严重的细菌感染。它还改变细胞膜的渗透性并选择性地抑制核糖核酸的合成。
TMIJ-0087 Mycophenolic acid-13C-d3

Mycophenolic acid-13C-d3 是 Mycophenolic acid 的 13C 和氘代化合物。Mycophenolic acid 的 CAS 号为 24280-93-1。Mycophenolic acid 是一种有效的非竞争性肌苷单磷酸脱氢酶 (IMPDH) 抑制剂,EC50为 0.24 µM。它对多种 RNA 病毒具有抗病毒作用。它也是一种免疫抑制剂,具有抗血管生成和抗肿瘤作用。
TMID-0086 Mycophenolate Mofetil-d4

Mycophenolate Mofetil-d4 是 Mycophenolate Mofetil 的氘代化合物。Mycophenolate Mofetil 的 CAS 号为 128794-94-5。Mycophenolate mofetil 是 Mycophenolic acid 的吗啉乙酯前药。它通过抑制肌苷一磷酸脱氢酶抑制从头嘌呤合成,显示出选择性淋巴细胞抗增殖作用。
T12691 Rapamycin-d3

AY-22989-d3,Sirolimus-d3

Others Others
Rapamycin-d3 is the deuterium labeled Rapamycin. Rapamycin is a potent and specific inhibitor of mTOR(IC50 of 0.1 nM in HEK293 cells).
TMIJ-0181 Clindamycin-13C-d3

Clindamycin-13C-d3 是 Clindamycin 的 13C 和氘代化合物。Clindamycin 的 CAS 号为 18323-44-9。Clindamycin 从细菌核糖体中解离肽基-tRNA,破坏细菌蛋白质合成。 它是一种半合成广谱抗生素,由母体化合物林可霉素化学修饰而成。
TMIJ-0111 Azithromycin-13C-d3

Azithromycin-13C-d3 是 Azithromycin 的 13C 和氘代化合物。Azithromycin 的 CAS 号为 83905-01-5。Azithromycin是一种常用于细菌感染研究的大环内酯抗生素。
TMIJ-0281 Lincomycin-d3

Lincomycin-d3 是 Lincomycin 的氘代化合物。Lincomycin 的 CAS 号为 7179-49-9。Lincomycin hydrochloride monohydrate 是一种窄谱抗生素, 具有与红霉素相似的效力, 对革兰氏阳性球菌的作用效果很好, 主要抑制细菌细胞蛋白质的合成。
TMIJ-0340 Lincomycin-13C-d3

Lincomycin-13C-d3 是 Lincomycin 的 13C 和氘代化合物。Lincomycin 的 CAS 号为 7179-49-9。Lincomycin hydrochloride monohydrate 是一种窄谱抗生素, 具有与红霉素相似的效力, 对革兰氏阳性球菌的作用效果很好, 主要抑制细菌细胞蛋白质的合成。
TMIH-0221 Erythromycin-13C-d3

Erythromycin-13C-d3 是 Erythromycin 的 13C 和氘代化合物。
T12135 Mycophenolic acid-d3

Mycophenolate-d3,Mycophenolate D3

Others; Antibacterial Microbiology/Virology; Others
Mycophenolic acid-d3 (Mycophenolate-d3) 是 Mycophenolic acid 的衍生物。Mycophenolic acid 是一种降低GTP 水平和损害RNA 聚合酶II (RNAP II)转录延伸的化合物,促进了近端位点的使用,能够逆转虫草素对选择性聚腺苷化的作用。
TMIJ-0109 Erythromycin Ethylsuccinate-13C-d3

Erythromycin Ethylsuccinate-13C-d3 是 Erythromycin Ethylsuccinate 的 13C 和氘代化合物。Erythromycin Ethylsuccinate 的 CAS 号为 1264-62-6。Erythromycin Ethylsuccinate是一种由红链霉菌产生的大环内酯类抗生素,有潜力用于多种细菌感染。它具有抗HIV-1病毒活性。
TMIJ-0110 Clarithromycin-13C-d3

Clarithromycin-13C-d3 是 Clarithromycin 的 13C 和氘代化合物。Clarithromycin 的 CAS 号为 81103-11-9。Clarithromycin 具有广谱的抗菌活性。它抑制CYP3A4催化的三唑仑 α-羟基化,IC50(Ki) 值为 56 (43) μM。它抑制 HERG 钾电流。它可削弱连接 hERG1 和 PI3K 的信号通路影响自噬流 。

同位素标记化合物

Mycophenolic Acid-d3 Phenyl Glucuronide
Cat.No: TMIH-0359
Synonym:
Target:
Vancomycin-d12 TFA
Cat.No: TMID-0284
Synonym:
Target:
Vancomycin-13C-d3
Cat.No: TMID-0283
Synonym:
Target:
Mycophenolic acid-13C-d3
Cat.No: TMIJ-0087
Synonym:
Target:
Mycophenolate Mofetil-d4
Cat.No: TMID-0086
Synonym:
Target:
Rapamycin-d3
Cat.No: T12691
Synonym: AY-22989-d3,Sirolimus-d3
Target: Others
Clindamycin-13C-d3
Cat.No: TMIJ-0181
Synonym:
Target:
Azithromycin-13C-d3
Cat.No: TMIJ-0111
Synonym:
Target:
Lincomycin-d3
Cat.No: TMIJ-0281
Synonym:
Target:
Lincomycin-13C-d3
Cat.No: TMIJ-0340
Synonym:
Target:
Erythromycin-13C-d3
Cat.No: TMIH-0221
Synonym:
Target:
Mycophenolic acid-d3
Cat.No: T12135
Synonym: Mycophenolate-d3,Mycophenolate D3
Target: Others, Antibacterial
Erythromycin Ethylsuccinate-13C-d3
Cat.No: TMIJ-0109
Synonym:
Target:
Clarithromycin-13C-d3
Cat.No: TMIJ-0110
Synonym:
Target:
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