Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T10419 |
AV-412
MP412 |
EGFR | Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors |
AV-412 (MP412) 是一种EGFR 抑制剂,抑制EGFR、EGFRL858R、EGFRT790M、EGFRL858R/T790M 和 ErbB2 的IC50值分别为0.75、0.5、0.79、2.3 和 19 nM。 | |||
TQ0293 |
AV-412 free base
无盐AV-412,MP-412 free base |
EGFR | Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors |
AV-412 free base is an EGFR inhibitor (IC50s: 0.75, 0.79, 0.5, 2.3, 19 nM for EGFR, EGFR(T790M), EGFR(L858R), EGFR(L858R/T790M) and ErbB2). |