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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2508 |
Binimetinib
ARRY-438162,ARRY-162,MEK162 |
MEK; Autophagy | Autophagy; MAPK |
Binimetinib (ARRY-162) 是一种可口服的选择性 MEK1/2抑制剂,抑制MEK 的IC50为 12 nM。 | |||
T28862 |
ST-168
ST168,ST 168 |
Others | Others |
ST-168 is a potent inhibitor of PI3K and MEK. ST-168 displays improved PI3K and MEK1 isoform inhibition. ST-168 demonstrated a 2.8-, 2.7-, 23-, and 2.5-fold improved inhibition toward the PI3Kα, PI3Kβ, PI3Kδ, and PI3Kγ isoforms and a 2.2-fold improvement |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TMIH-0117 |
Binimetinib-13C-d3
|
||
Binimetinib-13C-d3 是 Binimetinib 的 13C 和氘代化合物。Binimetinib 的 CAS 号为 606143-89-9。Binimetinib 是一种可口服的选择性MEK1/2抑制剂,抑制MEK的IC50为 12 nM。 |