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Search Results for " lipoxygenase "
Targets Recommended: Lipoxygenase Apoptosis Others Lipoxygenase

200

抑制剂 & 化合物

47

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Cat. No. Product Name Target Signaling Pathways
T8794 4-MMPB

15-Lipoxygenase Inhibitor 1

Apoptosis; Others; Lipoxygenase Apoptosis; Metabolism; Others
4-MMPB (15-Lipoxygenase Inhibitor 1) 是一种选择性15-脂氧合酶抑制剂,其 IC50值为 18 μM,具有前列腺癌的研究潜力。它对大豆 15-脂氧合酶和人 15-脂氧合酶-1 的 IC50 分别为 19.5 μM 和 19.1 μM。
T10151 5-Lipoxygenase-In-1

Lipoxygenase Metabolism
5-Lipoxygenase-In-1 (compound example 4.10) is a 5-Lipoxygenase inhibitor.
T76164 Lipoxygenase, general

Lipoxygenase, general (LOX) 是一种在生化研究中常用的双加氧酶,它能催化如亚油酸和花生四烯酸等多不饱和脂肪酸,生成相应的氢过氧化物。
T75122 5-Lipoxygenase-IN-3

Others Others
5-Lipoxygenase-IN-3 (Compound 14) 是一种5-Lipoxygenase 抑制剂 (IC50: <1 μM)。5-Lipoxygenase-IN-3 可用于炎症性疾病、癌症、中风和阿尔茨海默病的研究。
T8950 CAY10698

Lipoxygenase Metabolism
CAY10698 是选择性的12-Lipoxygenase (12-LOX)抑制剂,IC50=5.1 μM。它对 5-LOX、15-LOX-1、15-LOX-2 和 COX-1/2 无活性。
T8356 FPL 62064

Lipoxygenase; COX Immunology/Inflammation; Metabolism; Neuroscience
FPL 62064 是 5-脂氧合酶和COX 双重抑制剂,具有抗炎活性,对 RBL-1 胞质 5-脂氧合酶和前列腺素合成酶 (环氧化酶) 的IC50值分别为 3.5 和 3.1 μM。
T2367 SKF-86002

SKF86002

p38 MAPK; TNF Apoptosis; MAPK
SKF-86002 是一种可口服的 p38 MAPK 抑制剂,具有抗炎和抗关节炎活性,可用于缓解疼痛的研究。它能抑制脂氧合酶和环氧合酶介导的花生四烯酸代谢,还抑制脂多糖 (LPS) 刺激人单核细胞产生 IL-1 和 TNF-α,IC50为 1 μM。
T4347 ML355

Lipoxygenase Metabolism
ML355 是一种高选择性12-LOX 抑制剂,IC50=0.34 μM,对其他脂氧化酶和环氧化酶有很好的选择性,具有较好的药物动力学特征。
T6243 U-73122

U73122

Phospholipase; Ferroptosis; Lipoxygenase Apoptosis; Metabolism
U-73122 (U73122) 是一种磷脂酶 C 和 5-脂氧合酶抑制剂,对磷脂酶 C 的 IC50值约为 1-2.1 µM。它是一种 PLC 抑制剂,可减少激动剂诱导的血小板和 PMN 中的 Ca2+ 增加。
T16503 PF-4191834

PF-04191834

Lipoxygenase Metabolism
PF-4191834 是 5-Lipoxygenase (5-LOX) 的非铁螯合和非氧化还原抑制剂,IC50 为 229 nM。 PF-4191834 对 5-LOX 的特异性比 12-LOX 和 15-LOX 高约 300 倍,并且对环氧合酶没有活性。 PF-4191834 可用于炎症和疼痛的研究。
T7540 2,5-Di-tert-butylhydroquinone

BHQ,2,5-二特丁基对苯二酚

Calcium Channel; Lipoxygenase; COX Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience
2,5-Di-tert-butylhydroquinone (BHQ) 是一种有效和选择性的内质网 Ca2+-ATPase 抑制剂,可调节5-LO 以及COX-2活性,IC50分别为 1.8 和 14.1 μM。
T21902 ML351

Lipoxygenase Metabolism
ML351 是一种高度特异的15-LOX-1抑制剂,其 IC50=200 nM。它对 T1D 非肥胖糖尿病小鼠模型的血糖异常和β细胞氧化应激有抑制作用。它对相关同工酶 (5-LOX、血小板 12-LOX、15-LOX-2、绵羊 COX-1 和人 COX-2) 表现出良好的选择性(>250倍)。
T6568 Licofelone

利克飞龙,ML-3000

Apoptosis; Lipoxygenase; COX Apoptosis; Immunology/Inflammation; Metabolism; Neuroscience
Licofelone (ML-3000) 是一种 COX/LOX 双重抑制剂,IC50分别为 0.21和0.18 μM,有潜力研究骨关节炎,具有抗炎和抗增殖作用。它可诱导细胞凋亡,减少促炎性白三烯和前列腺素的产生。
T21746 Terameprocol

tetramethyl Nordihydroguaiaretic Acid,EM-1421

HIV Protease Microbiology/Virology; Proteases/Proteasome
Terameprocol (EM-1421) 是 Nordihydroguaiaretic acid 的合成衍生物,是非选择性脂氧合酶抑制剂。
T22398 Phenidone

菲尼酮,1-phenyl-3-pyrazolidinone

Lipoxygenase; COX Immunology/Inflammation; Metabolism; Neuroscience
Phenidone (1-phenyl-3-pyrazolidinone) 是可口服发环氧化酶和脂氧合酶双重抑制剂,可改善实验性自身免疫性脑脊髓炎大鼠的瘫痪,降低自发性高血压大鼠的血压,可用作照片显像剂。
T10098 PGS-IN-1

KME-4

Lipoxygenase; Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism
PGS-IN-1 (KME-4)是一种前列腺素合成酶抑制剂,IC50=0.28 μM。它也可抑制5-脂肪氧合酶的活性,IC50=1.05 μM。
T0477 Zileuton

Abbott 64077,齐留通,A 64077

Ferroptosis; Lipoxygenase; COX Apoptosis; Immunology/Inflammation; Metabolism; Neuroscience
Zileuton (A 64077) 是羟基脲的合成衍生物,是一种选择性的5-脂氧合酶抑制剂,具有平喘特性。
T27026 CJ-13,610

CJ 13610,CJ-13610

Lipoxygenase Metabolism
CJ-13,610 是一种具有口服活性的非氧化还原型 5-脂氧合酶 (5-LOX) 抑制剂。 CJ-13,610 抑制白三烯 B4 的生物合成并调节巨噬细胞中 IL-6 mRNA 的表达。
T6576 Malotilate

Malotilatum,NKK 105,马洛替酯,Kantec

Lipoxygenase Metabolism
Malotilate (Kantec) 是一种抗纤维化物质,是一种口服活性的促肝药,可选择性抑制5-lipoxygenase (5-LOX)(IC50=4.7 μM)。它通过降低肝脏乙醛水平并防止转铁蛋白保留在肝细胞中,从而预防了酒精-吡唑肝炎中肝细胞损伤的发展。
T5200 Indirubin-3'-monoxime

靛玉红-3' -单肟,Indirubin-3'-oxime

GSK-3; Lipoxygenase; CDK Cell Cycle/Checkpoint; Metabolism; PI3K/Akt/mTOR signaling; Stem Cells
Indirubin-3'-monoxime (Indirubin-3'-oxime) 是一种有效的 GSK3β 抑制剂,IC50值为 22 nM。它对 CDK5/p25、CDK1/cyclin B 和CDk2/cyclin E 也有作用,IC50值分别为 100、180 和 250 nM。
T7724 Tepoxalin

RWJ-20485,RWJ20485,ORF20485,替泊沙林,ORF-20485,RWJ 20485,ORF 20485

Lipoxygenase; COX Immunology/Inflammation; Metabolism; Neuroscience
Tepoxalin (RWJ 20485) 是有效的5-脂氧合酶和环氧合酶抑制剂,表现出强大的抗炎活性和较小的胃肠道刺激性。
T19679 Benoxaprofen

氧苯恶唑丙酸,NSC 299582,LY-90459,Benoxaphen. Compound 90459

COX Immunology/Inflammation; Neuroscience
Benoxaprofen (NSC-299582) 是长效的、强效的抗炎和解热化合物,在体外具有较弱的对环氧合酶的抑制作用,也可以抑制脂氧合酶,在一些炎症动物模型中抑制单核细胞迁移。
T24488 MLS000545091

MLS-000545091,MLS 000545091

Others Others
MLS000545091 is a potent and selective human epithelial 15-lipoxygenase-2 mixed-type inhibitor.
T22054 BW 755C

Lipoxygenase Metabolism
BW 755C 是 5-脂氧合酶 (5-LO) 和环氧合酶 (COX) 通路的双重抑制剂。
T12784 RWJ 63556

RWJ-63556

Lipoxygenase; COX Immunology/Inflammation; Metabolism; Neuroscience
RWJ 63556 是一种可口服的 COX-2 selective/5-lipoxygenase 抑制剂,具有抗炎活性。
T24306 L 651896

L651896,L-651896

Leukotriene Receptor; Lipoxygenase GPCR/G Protein; Metabolism
L 651896 是一种新型白三烯生物合成和 5-脂氧合酶抑制剂,可用于研究呼吸系统疾病和心血管疾病。
T16802 Lonapalene

RS4317

Lipoxygenase Metabolism
Lonapalene (RS4317) 是一种 5-脂氧合酶 (5-LO) 抑制剂,具有抗银屑病的功效。Lonapalene 可局部阻断皮肤炎症。
T61211 5-LOX-IN-1

Lipoxygenase Metabolism
5-LOX-IN-1 是一种 5-Lipoxygenase(5-LOX)抑制剂(IC50: 2.3 μM)。5-LOX-IN-1 可用于研究癌症。
T22358 Etalocib

LY293111,VML295

Apoptosis; Leukotriene Receptor; LTR Apoptosis; GPCR/G Protein; Immunology/Inflammation
Etalocib (LY293111) 是一种具有口服活性的白三烯(LTB4)受体的拮抗剂,抑制 [3H]LTB4结合的 Ki 值为 25 nM。它还可诱导凋亡。它抑制 LTB4诱导的钙动员,lC50值为 20 nM。
T16817 S-2474

Lipoxygenase; COX Immunology/Inflammation; Metabolism; Neuroscience
S-2474 是 COX-2 和 5-脂氧合酶的抑制剂 ,具有抗炎活性和神经保护活性,可抑制 Abeta(25 - 35) 和 Abeta(1 - 40) 诱导的细胞死亡。
T60507 Utreloxastat

EPI 857,PTC857

Lipoxygenase Metabolism
Utreloxastat (PTC857) 是一种新型 15-脂氧合酶抑制剂,可用于研究肌萎缩侧索硬化症 。
T27244 Efletirizine

UCB 28754,UCB-28754,UCB28754

Lipoxygenase; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience
Efletirizine (UCB-28754) 是一种组胺受体拮抗剂,对5-脂氧合酶(5-LO)具有抑制作用,对可用于局部治疗过敏疾病。
T9023 Atuliflapon

AZD5718

FLAP Immunology/Inflammation
Atuliflapon (AZD5718) 是可口服的FLAP(5 -脂氧合酶激活蛋白)的抑制剂,IC50值为 2 nM,可用于冠状动脉疾病的研究。
T25737 Linetastine

TMK 688,TMK-688,TMK688

Lipoxygenase; LTR; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience
Linetastine (TMK-688) 是一种 5-脂氧合酶抑制剂(5-LOX),能抑制白三烯的产生,并能拮抗组胺的作用。Linetastine可用于研究哮喘、动脉粥样硬化和消化性溃疡。
T70188 ER-34122

Lipoxygenase Metabolism
ER-34122,一种新型可口服的双重 5-脂氧合酶/环氧合酶抑制剂,在花生四烯酸诱导的耳部炎症模型中具有强大的抗炎活性。
T22502 2-TEDC

Lipoxygenase Metabolism
2-TEDC 是一种有效的脂氧合酶(LOX)抑制剂,对 5-LOX、12-LOX 和 15-LOX 具有抑制作用,IC50 值分别为 0.09 μM、0.013 μM 和 0.5 μM。2-TEDC 可用于研究动脉粥样硬化。
T21821L REV 5901A

REV 5901 HCl,REV 5901A(101910-24-1 Free base)

Leukotriene Receptor; Lipoxygenase; Antibiotic GPCR/G Protein; Metabolism; Microbiology/Virology
REV 5901A (REV 5901 HCl) 是一种具有口服活性的白三烯受体 (leukotriene receptor) 拮抗剂,也是一种 5-脂氧合酶 (5-lipoxygenase) 抑制剂,具有抗菌活性,可减弱小鼠体内结肠癌的生长。REV 5901A 可用于研究哮喘和心肌梗死。
TQ0159 U-73343

U 73343

Phospholipase Metabolism
U-73343 是一种 U-73122 的无活性类似物,能够剂量依赖性的抑制酸分泌,可作为 U-73122 的阴性对照。其中 U 73122 是一种有效的磷脂酶 C (phospholipase C) 和 5-脂氧合酶 (5-LO (5-lipoxygenase)) 抑制剂,对磷脂酶 C 的 IC50值约为 1-2.1 µM。
T77288 KKII5

Lipoxygenase Metabolism
KKII5 是一种有效的脂氧合酶 LOX-1 抑制剂,IC50 为 19 μM。KKII5 抑制脂质过氧化,增强部分化合物活性中心接收电子的能力。
T11487 Fiboflapon

GSK2190915,AM-803

FLAP Immunology/Inflammation
Fiboflapon (GSK2190915) 是一种可口服且具有有效性 5-脂氧合酶激活蛋白 (FLAP) 抑制剂,结合 FLAP 的效价为 2.9 nM,对人血中 LTB4 有抑制作用, IC50 值为 76 nM。
T68155 Tebufelone

Prostaglandin Receptor; LTR GPCR/G Protein; Immunology/Inflammation
Tebufelone 是一种体外高效的CO 抑制剂 ,是一种新型的非甾体抗炎药(NSAID),属于二叔丁基苯酚(DTBP)类,在各种动物模型中显示出强大的抗炎、镇痛和抗网膜炎特性。Tebufelone 能有效地抑制前列腺素(PGE2)的形成,阻止大鼠巨噬细胞(IC50 = 20 microM)和人类全血(IC50 = 22 microM)中脂氧酶途径的产物[白三烯(LTB4)]的体外形成。
T6893 MK-886

MK886,L 663536

Apoptosis; Leukotriene Receptor; COX; PPAR; FLAP Apoptosis; DNA Damage/DNA Repair; GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience
MK-886 (L 663536)是一种细胞可渗透的,具有口服活性的 FLAP (IC50为 30 nM) 和白三烯生物合成 (完整白细胞和人全血中的IC50分别为 3 nM 和 1.1μM) 的抑制剂。它也是一种非竞争性PPARα拮抗剂,可以诱导细胞凋亡。
T10208 A-69412

N-1-(Fur-3-ylethyl)-N-hydroxyurea

Lipoxygenase Metabolism
A-69412 (N-1-(Fur-3-ylethyl)-N-hydroxyurea) 是一种特异性的 5-脂氧合酶 (5-LO) 的可逆抑制剂。 A-69412 能用于哮喘和溃疡性结肠炎,以及其他炎症和过敏症状的研究。
T8844 Diflapolin

Others; FLAP; Epoxide Hydrolase Immunology/Inflammation; Metabolism; Others
Diflapolin 是高活性的双 5-脂氧合酶激活蛋白(FLAP)/可溶性环氧化物水解酶抑制剂,具有显著的抗炎作用和较高的靶向选择性。它抑制分离的 sEH 的活性,IC50为20 nM。它还抑制完整人单核细胞和中性粒细胞中 5-LOX 产物的形成,IC50分别为 30 和 170 nM。
T67908 ThioLox

Lipoxygenase Metabolism
ThioLox 是一种竞争性 15-脂氧合酶-1 (15-LOX-1) 抑制剂(IC50值为12 μM)。ThioLox 显示抗炎和神经保护特性。具有抗炎和神经保护作用,对谷氨酸毒性有很强的保护作用。
T9878 Croconazole

Lipoxygenase; LTR Immunology/Inflammation; Metabolism
Croconazole 对中性粒细胞的 5-脂氧合酶 (5-LOX) 表现出剂量依赖性抑制活性。Croconazole 是一种抗真菌剂。Croconazole 对合成白三烯 B4 (LTB4) 和 5-羟基二十碳四烯酸 (5-HETE) 的 IC50 分别为 7.8 ± 1.7 和 7.6 ± 0.3 μM。
T7530 PD146176

NSC168807

Ferroptosis; Lipoxygenase; Autophagy Apoptosis; Autophagy; Metabolism
PD146176 (NSC-168807) 是一种 15-脂氧合酶(15-LO)抑制剂,抑制兔网织红细胞 15-LO,Ki 为 197 nM,IC50 为 0.54 μM。 它通过刺激老年三重转基因小鼠的自噬来逆转认知障碍、脑淀粉样变性和 tau 病理学。
T68173 ZD-2138

Ici-D2138

Lipoxygenase Metabolism
ZD-2138是一种有效且具有选择性的5-脂氧合酶(5-LOX)的特异性抑制剂,抑制了过敏原诱导的肺支气管收缩,可减少豚鼠孤立气道的神经诱发性快速激肽能收缩。ZD-2138可用来治疗哮喘疾病。
T68037L CBS-1114 HCl

N-Phenylbenzamidrazone hydrochloride,cbs-1114 HCl(46721-85-1 Free base)

Lipoxygenase Metabolism
CBS-1114 HCl (N-Phenylbenzamidrazone hydrochloride) 是一种5-脂氧合酶抑制剂,是一种良好眼睛渗透型号的抗炎化合物。CBS-1114 HCl 可以保持和改善心脏功能,减轻心功能障碍,以及减少患有心血管疾病的受试者的心外膜脂肪组织和/或心包脂肪组织。
T16087 Quiflapon

喹夫拉朋,MK-591

Apoptosis; FLAP Apoptosis; Immunology/Inflammation
Quiflapon (MK-591) 是一种选择性和特异性的FLAP 抑制剂,可诱导细胞凋亡。它也是口服白三烯生物合成抑制剂,在完整的人和诱导的大鼠多形核白细胞 PMNLs 中,其IC50值分别为 3.1 nM 和 6.1 nM。

化合物

4-MMPB
Cat.No: T8794
Synonym: 15-Lipoxygenase Inhibitor 1
Target: Apoptosis, Others, Lipoxygenase
5-Lipoxygenase-In-1
Cat.No: T10151
Synonym:
Target: Lipoxygenase
Lipoxygenase, general
Cat.No: T76164
Synonym:
Target:
5-Lipoxygenase-IN-3
Cat.No: T75122
Synonym:
Target: Others
CAY10698
Cat.No: T8950
Synonym:
Target: Lipoxygenase
FPL 62064
Cat.No: T8356
Synonym:
Target: Lipoxygenase, COX
SKF-86002
Cat.No: T2367
Synonym: SKF86002
Target: p38 MAPK, TNF
ML355
Cat.No: T4347
Synonym:
Target: Lipoxygenase
U-73122
Cat.No: T6243
Synonym: U73122
Target: Phospholipase, Ferroptosis, Lipoxygenase
PF-4191834
Cat.No: T16503
Synonym: PF-04191834
Target: Lipoxygenase
2,5-Di-tert-butylhydroquinone
Cat.No: T7540
Synonym: BHQ,2,5-二特丁基对苯二酚
Target: Calcium Channel, Lipoxygenase, COX
ML351
Cat.No: T21902
Synonym:
Target: Lipoxygenase
Licofelone
Cat.No: T6568
Synonym: 利克飞龙,ML-3000
Target: Apoptosis, Lipoxygenase, COX
Terameprocol
Cat.No: T21746
Synonym: tetramethyl Nordihydroguaiaretic Acid,EM-1421
Target: HIV Protease
Phenidone
Cat.No: T22398
Synonym: 菲尼酮,1-phenyl-3-pyrazolidinone
Target: Lipoxygenase, COX
PGS-IN-1
Cat.No: T10098
Synonym: KME-4
Target: Lipoxygenase, Prostaglandin Receptor
Zileuton
Cat.No: T0477
Synonym: Abbott 64077,齐留通,A 64077
Target: Ferroptosis, Lipoxygenase, COX
CJ-13,610
Cat.No: T27026
Synonym: CJ 13610,CJ-13610
Target: Lipoxygenase
Malotilate
Cat.No: T6576
Synonym: Malotilatum,NKK 105,马洛替酯,Kantec
Target: Lipoxygenase
Indirubin-3'-monoxime
Cat.No: T5200
Synonym: 靛玉红-3' -单肟,Indirubin-3'-oxime
Target: GSK-3, Lipoxygenase, CDK
Tepoxalin
Cat.No: T7724
Synonym: RWJ-20485,RWJ20485,ORF20485,替泊沙林,ORF-20485,RWJ 20485,ORF 20485
Target: Lipoxygenase, COX
Benoxaprofen
Cat.No: T19679
Synonym: 氧苯恶唑丙酸,NSC 299582,LY-90459,Benoxaphen. Compound 90459
Target: COX
MLS000545091
Cat.No: T24488
Synonym: MLS-000545091,MLS 000545091
Target: Others
BW 755C
Cat.No: T22054
Synonym:
Target: Lipoxygenase
RWJ 63556
Cat.No: T12784
Synonym: RWJ-63556
Target: Lipoxygenase, COX
L 651896
Cat.No: T24306
Synonym: L651896,L-651896
Target: Leukotriene Receptor, Lipoxygenase
Lonapalene
Cat.No: T16802
Synonym: RS4317
Target: Lipoxygenase
5-LOX-IN-1
Cat.No: T61211
Synonym:
Target: Lipoxygenase
Etalocib
Cat.No: T22358
Synonym: LY293111,VML295
Target: Apoptosis, Leukotriene Receptor, LTR
S-2474
Cat.No: T16817
Synonym:
Target: Lipoxygenase, COX
Utreloxastat
Cat.No: T60507
Synonym: EPI 857,PTC857
Target: Lipoxygenase
Efletirizine
Cat.No: T27244
Synonym: UCB 28754,UCB-28754,UCB28754
Target: Lipoxygenase, Histamine Receptor
Atuliflapon
Cat.No: T9023
Synonym: AZD5718
Target: FLAP
Linetastine
Cat.No: T25737
Synonym: TMK 688,TMK-688,TMK688
Target: Lipoxygenase, LTR, Histamine Receptor
ER-34122
Cat.No: T70188
Synonym:
Target: Lipoxygenase
2-TEDC
Cat.No: T22502
Synonym:
Target: Lipoxygenase
REV 5901A
Cat.No: T21821L
Synonym: REV 5901 HCl,REV 5901A(101910-24-1 Free base)
Target: Leukotriene Receptor, Lipoxygenase, Antibiotic
U-73343
Cat.No: TQ0159
Synonym: U 73343
Target: Phospholipase
KKII5
Cat.No: T77288
Synonym:
Target: Lipoxygenase
Fiboflapon
Cat.No: T11487
Synonym: GSK2190915,AM-803
Target: FLAP
Tebufelone
Cat.No: T68155
Synonym:
Target: Prostaglandin Receptor, LTR
MK-886
Cat.No: T6893
Synonym: MK886,L 663536
Target: Apoptosis, Leukotriene Receptor, COX, PPAR, FLAP
A-69412
Cat.No: T10208
Synonym: N-1-(Fur-3-ylethyl)-N-hydroxyurea
Target: Lipoxygenase
Diflapolin
Cat.No: T8844
Synonym:
Target: Others, FLAP, Epoxide Hydrolase
ThioLox
Cat.No: T67908
Synonym:
Target: Lipoxygenase
Croconazole
Cat.No: T9878
Synonym:
Target: Lipoxygenase, LTR
PD146176
Cat.No: T7530
Synonym: NSC168807
Target: Ferroptosis, Lipoxygenase, Autophagy
ZD-2138
Cat.No: T68173
Synonym: Ici-D2138
Target: Lipoxygenase
CBS-1114 HCl
Cat.No: T68037L
Synonym: N-Phenylbenzamidrazone hydrochloride,cbs-1114 HCl(46721-85-1 Free base)
Target: Lipoxygenase
Quiflapon
Cat.No: T16087
Synonym: 喹夫拉朋,MK-591
Target: Apoptosis, FLAP
Cat. No. Product Name Target Signaling Pathways
T3S0153 Xanthatin

苍耳亭,叶黄制菌素

Apoptosis; VEGFR; Lipoxygenase; Wnt/beta-catenin; Antibacterial Angiogenesis; Apoptosis; Cytoskeletal Signaling; Metabolism; Microbiology/Virology; Stem Cells; Tyrosine Kinase/Adaptors
Xanthatin 是一种从Xanthium strumarium 叶子中提取的天然产物,可诱导细胞凋亡。它抑制布鲁氏菌的IC50值为 2.63 μg/ mL,对寄生虫特异性锥虫硫磷还原酶具有不可逆的弱抑制作用。它通过抑制PGE2的合成和 5-脂氧合酶的活性而显示出抗炎活性。
T2807 Caffeic Acid

Lipoxygenase; Endogenous Metabolite; TRP/TRPV Channel Membrane transporter/Ion channel; Metabolism
Caffeic acid 是5-脂氧合酶和 TRPV1离子通道的双重抑制剂。
TQ0180 Chebulagic acid

SARS-CoV; Influenza Virus; Lipoxygenase; COX Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience
Chebulagic acid 是从 Terminalia chebula Retz 中分离出来的一种 COX-LOX 双重抑制剂,有抗炎和抗感染作用。它抑制 SARS-CoV-2病毒的复制,EC50值为 9.76 μM。它还是 M2(S31N)抑制剂和抗流感病毒剂。
T8260 4',5-Dihydroxyflavone

Lipoxygenase; Glucosidase Metabolism
4',5-Dihydroxyflavone 是大豆 LOX-1,Ki=102.6 μM。它也是一种酵母 α-葡萄糖苷酶抑制剂,IC50=66 μM。
T8002 3-Hydroxycoumarin

Lipoxygenase Metabolism
3-hydroxycoumarin 是一种 15-LOX-1的有效氧化还原抑制剂,近期被证明能保护海胆生殖细胞免受紫外线 B 的损伤。
TN2330 Phenethyl ferulate

Caffeic Acid 3-Methyl Phenethyl Ester,阿魏酸苯乙酯,阿魏酸苯乙醇酯

Lipoxygenase; COX Immunology/Inflammation; Metabolism; Neuroscience
Phenethyl ferulate (Caffeic Acid 3-Methyl Phenethyl Ester) 对化学诱导的结肠癌具有化学预防特性,可增强偶氮甲烷诱导的结肠肿瘤的细胞凋亡。 它抑制环氧合酶(COX) 和 5-脂氧合酶 (5-LOX) ,IC50 值分别为 4.35 和 5.75 μM。
T6S0413 Pectolinarigenin

柳穿鱼黄素,Pectolinaringenin

Others; Lipoxygenase; COX Immunology/Inflammation; Metabolism; Neuroscience; Others
Pectolinarigenin (Pectolinaringenin) 是 COX-2/5-LOX 的双重抑制剂,可抑制炎症病变中类花生酸的形成,具有抗炎活性。
TN5634 Aureusidin

Auresudidin,金鱼草素,Auresidin

Antioxidant; Reactive Oxygen Species; Lipoxygenase Immunology/Inflammation; Metabolism; NF-κB; oxidation-reduction
Aureusidin (Auresidin) 具有抗氧化和脂氧合酶抑制活性,具有抗炎作用。
T9512 Linoleyl alcohol

CIS,CIS-9,12-OCTADECADIENOL,亚麻醇

Others Others
Linoleyl alcohol (CIS,CIS-9,12-OCTADECADIENOL) 是一种脂肪醇,是一种没有α-羧基的 Linoleic acid 的结构类似物。
T3399 Psoralidin

Others; Estrogen/progestogen Receptor; Reactive Oxygen Species; Lipoxygenase; Gamma-secretase; Akt; COX; Antibacterial Cytoskeletal Signaling; Endocrinology/Hormones; Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience; NF-κB; Others; PI3K/Akt/mTOR signaling; Proteases/Proteasome; Stem Cells
Psoralidin 是COX-2和5-LOX 的抑制剂,有抗癌,抗菌和抗炎作用。它显著下调NOTCH1信号传导,还极大地诱导活化氧产生。
T5714 5-O-Demethylnobiletin

5-DEMETHYLNOBILETIN,去甲基川陈皮素

Leukotriene Receptor; Lipoxygenase GPCR/G Protein; Metabolism
5-O-Demethylnobiletin (5-DEMETHYLNOBILETIN) 是从黄芪中分离出的多甲氧基黄酮,具有抗炎活性,可通过直接抑制 5-LOX 发挥作用,IC50为 0.1 μM。
T5759 S-(+)-Marmesin

(+)-Marmesin,异紫花前胡内酯,(S)-Marmesin,marmesin

Lipoxygenase; COX Immunology/Inflammation; Metabolism; Neuroscience
S-(+)-Marmesin (marmesin) 是一种从木橘成熟树皮中分离得到的香豆素,具有 COX-2/5-LOX 双重抑制活性。
TJS2190 Nordihydroguaiaretic acid

去甲二氢愈创木酸,NDGA,Dihydronorguaiaretic Acid

Antioxidant; Ferroptosis; Lipoxygenase; Autophagy Apoptosis; Autophagy; Metabolism; oxidation-reduction
Nordihydroguaiaretic acid (NDGA) 是从极叉开拉瑞阿提取出的一种天然产物,是脂氧合酶抑制剂,具有抗氧化和清除自由基的特性。
T3384 Wedelolactone

蟛蜞菊内酯,IKK Inhibitor II

Apoptosis; NF-κB; Lipoxygenase; Caspase Apoptosis; Metabolism; NF-κB; Proteases/Proteasome
Wedelolactone (IKK Inhibitor II) 是来自旱莲草的一种天然产物,通过阻断 IκBα 的磷酸化和降解来抑制细胞中 NF-κB 介导的基因转录,具有抗癌,抗炎和抗氧化活性。
TN1097 β-Boswellic acid

Beta-boswellic acid,β-乳香酸

Lipoxygenase; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism
β-Boswellic acid (Beta-boswellic acid) 是从乳香的树胶脂中分离出来的一种天然产物。它是 5-脂氧合酶(5-LO) 产物形成的非还原型抑制剂,其直接与 5-LO 相互作用或阻断其易位。具有抗癌、抗肿瘤和抗高血脂活性。
TN1255 3-O-Acetyl-11-hydroxy-beta-boswellic acid

Lipoxygenase Metabolism
3-O-Acetyl-11-hydroxy-beta-boswellic acid 是 5-脂氧合酶抑制剂。
TN1182 11-​Keto-​beta-​boswellic acid

11-Keto-beta-boswellic acid,11-酮基-BETA-乳香酸

Leukotriene Receptor; NF-κB; Lipoxygenase GPCR/G Protein; Metabolism; NF-κB
11-Keto-beta-boswellic acid 是来自乳香的一种五环三萜酸,具有抗炎活性和剂量依赖性心脏保护作用,主要是由于抑制5-脂氧合酶、白三烯、NF-κB 的激活和肿瘤坏死因子 α 的产生。
TN2068 Picrinine

Lipoxygenase Metabolism
Picrinine 是一种从 Alstonia scholaris 的叶子中提取出来的 Akuammiline 生物碱。 Picrinine 具有抗炎活性,通过抑制5-脂氧合酶来发挥作用。
T3879 Silychristin

水飞蓟亭,水飞蓟汀,Silicristin

Lipoxygenase Metabolism
Silychristin (Silicristin) 是甲状腺激素转运体MCT8的有效抑制剂,能强烈抑制 T3 的摄取(IC50:110 nM)。它是一种水飞蓟果实中富含的黄酮类化合物,具有抗氧化作用。
T10821 Cirsiliol

Apoptosis; Lipoxygenase Apoptosis; Metabolism
Cirsiliol是一种特异性5-脂氧合酶 (5-LOX) 抑制剂,是低亲和力的苯二氮卓受体配体。Cirsiliol 抑制 OS 细胞细胞增殖,促进 OS 细胞凋亡,在原位异种肿瘤模型中对 OS 细胞显示出抗肿瘤活性,可用于研究结肠癌。
T6389 Anacardic Acid

漆树酸,6-pentadecylsalicylic Acid,Hydroginkgolic acid

Others; Epigenetic Reader Domain; Histone Acetyltransferase; Antibacterial Chromatin/Epigenetic; Microbiology/Virology; Others
Anacardic Acid (6-pentadecylsalicylic Acid) 是从腰果壳中提取液中分离到的酸类物质,是一种组蛋白乙酰转移酶抑制剂,对 p300 和 PCAF 的 IC50值分别为 ∼8.5 μM 和 ∼5 μM。
TN1787 Isomucronulatol 7-O-glucoside

Isomucronulatol 7-O-beta-glucoside,黄芪紫檀烷苷,3-羟基-9,10-二甲氧基紫檀烷

Others Others
Isomucronulatol 7-O-beta-glucoside 具有潜在的抗炎活性,在体外对 LPS 刺激产生的 IL-12 p40 表现出微弱的抑制作用。
T36051 Lipoxin A4

LXA4

Endogenous Metabolite; Interleukin Immunology/Inflammation; Metabolism
Lipoxin A4 (LXA4) 是一种内源性脂氧合酶衍生的类花生酸介质,具有抗炎作用。Lipoxin A4 通过抑制 Nrf2 来减弱 MSU 晶体诱导的 NLRP3 炎症小体激活,通过 FPR2-IRF 途径调节 M1/M2 巨噬细胞极化。Lipoxin 抑制氧化应激和炎症。
TJS0315 4-Methyldaphnetin

7,8-Dihydroxy-4-methylcoumarin,4-甲基瑞香素,DHMC,7,8-二羟基-4-甲基香豆素

Apoptosis; Lipoxygenase Apoptosis; Metabolism
4-Methyldaphnetin (DHMC) 是一种合成 4-甲基香豆素衍生物的前体。它对几种肿瘤细胞株具有选择性的抗增殖和诱导凋亡的作用。它能够清除自由基,显著抑制膜脂过氧化。
T5214 Cholesteryl linoleate

CE(18:2(9Z,12Z)),Cholesterol Linoleate,Linoleic Acid cholesteryl ester,胆甾烯基亚油酸酯

Others; Endogenous Metabolite Metabolism; Others
Cholesteryl linoleate 是低密度脂蛋白和动脉粥样硬化病变中主要的胆固醇酯。它存在于 LDL 中的胆固醇酯,利用 LDL 受体相关蛋白转移到表达 15-脂氧合酶的巨噬细胞和 CHO 细胞的质膜,被氧化形成胆固醇亚油酸氢过氧化物。
TN1308 6-Hydroxyflavanone

Others; Lipoxygenase; COX; GABA Receptor Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience; Others
6-Hydroxyflavanone 是从菖蒲叶中提取分离,通过靶向环氧合酶-2(COX-2),5-脂氧合酶(5-LOX)以及阿片类药物和 GABA-A 受体从而具有抗炎和抗神经性疼痛活性。6-Hydroxyflavanone 在链脲佐菌素诱导的糖尿病神经病变模型中具有抗伤害感受特性。
T4137 4,7-DIHYDROXYCOUMARIN

Others Others
4,7-DIHYDROXYCOUMARIN 是一种天然存在的香豆素衍生物,存在于多种植物中,包括欧芹和洋甘菊。已经发现它可以抑制几种酶的活性,包括细胞色素P450、环氧合酶和脂氧合酶;也可以与DNA 结合,调节基因表达,并抑制细胞周期进展;还可以诱导肿瘤细胞凋亡并减轻炎症。
T6S1699 Shogaol

[6]-Shogaol,姜烯酚,6-姜烯酚,6-Shogaol

Lipoxygenase; Autophagy Autophagy; Metabolism
6-Shogaol (6-Shogaol) 是从生姜中分离的一种天然产物,具有抗癌、抗炎和抗氧化的多种生物活性。
T37974 (S)-Coriolic acid

13(S)-HODE

Lipoxygenase; Mitochondrial Metabolism; PPAR DNA Damage/DNA Repair; Metabolism
(S)-Coriolic acid (13(S)-HODE) 是一种重要的细胞内信号剂,是亚油酸与植物和哺乳动物脂氧合酶反应生成的,在各种生物系统中参与细胞增殖和分化。(S)-Coriolic acid 在 1 μM 左右时,它能抑制肿瘤细胞与血管内皮的粘附,能下调 IRGpIIb/IIIa 受体的表达。(S)-Coriolic acid 是15-脂氧合酶 (15-LOX) 代谢产物,常作为内源性配体激活 PPARγ。(S)-Coriolic acid 诱导线粒体功能障碍 和气道上皮损伤。
T24869 Texasin

IR2,IR 2,IR-2

Others Others
Texasin is a selective inhibitor of human leukocyte 5-lipoxygenase.
TN5196 Turmeronol A

Others Others
Turmeronol A and turmeronol B are inhibitors of soybean lipoxygenase, they inhibited soybean lipoxygenase at the IC50 values of 16 uM and 9 uM, respectively.
TN1813 Jujuboside D

酸枣仁皂苷D,酸枣仁皂甙D

Others Others
Jujuboside D shows lipoxygenase-inhibiting activity.
TN4032 Eugenol benzoate

Others Others
Eugenol benzoate, a potent lipoxygenase inhibitor, has antioxidant activity.
TN5159 Trachelosiaside

Others Others
Trachelosiaside shows moderate activity against lipoxygenase.
TN4331 Isotachioside

Lipoxygenase Metabolism
Isotachioside has15-lipoxygenase (15-LO) inhibitory activities.
TN2688 2,3,4'-Trihydroxy-3',5'-dimethoxypropiophenone

Antioxidant; Lipoxygenase Metabolism; oxidation-reduction
2,3,4'-Trihydroxy-3',5'-dimethoxypropiophenone 是一种天然产物,可从 Parinari hypochrysea (Chrysobalanaceae) 中提取得到。2,3,4'-Trihydroxy-3',5'-dimethoxypropiophenone 具有抗氧化活性且对脂氧合酶具有抑制作用。
TN5017 Sideritoflavone

Opioid Receptor; Prostaglandin Receptor Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation; Neuroscience
Sideritoflavone has anti-inflammatory effect, it is a selective inhibitor of lipoxygenase activity in vitro.
TN7347 9,11-Dehydro-beta-boswellic acid

Others Others
9,11-Dehydro-β-boswellic acid is a compound with urease inhibitory activity and acts as an inhibitor of 5-lipoxygenase (5-LO), a critical enzyme in leukotriene biosynthesis.
T13764 Lycopodine

Lipoxygenase; Caspase Apoptosis; Metabolism; Proteases/Proteasome
Lycopodine, a bioactive compound derived from Lycopodium clavatum spores, effectively inhibits the proliferation of HeLa cells through the induction of apoptosis. This process is mediated by caspase-3 activation. In refractory prostate cancer cells, Lycopodine triggers apoptosis by modulating 5-lipoxygenase and depolarizing the mitochondrial membrane potential, without altering p53 activity.
T60692 Masoprocol

Others Others
Masoprocol (meso-Nordihydroguaiaretic acid) 是口服有效的脂氧合酶 (lipoxygenase) 抑制剂。Masoprocol 具有出抗高血糖活性,可用于 II 型糖尿病的研究。 Masoprocol 可降低体内肝甘油三酯和葡萄糖浓度。
TN4088 Futoenone

PAFR GPCR/G Protein
Futoenone and a series of its derivatives have shown inhibitory activities against matrix metalloproteinases, the molecular modelings of these compounds indicate the preferred binding of the P2' site of the enzymes. Neolignan derivative compounds of the 2,4-diaryl-1,3-dithiolane and futoenone variety exhibit both platelet activating factor receptor(PAF)and 5-lipoxygenase antagonist activity.
TN7391 Caffeoylcalleryanin

Others Others
Caffeoylcalleryanin demonstrated potent inhibitory activity against 15-lipoxygenase (15-LOX), with an IC50 value of 1.59 μM. Furthermore, ethanol extract from A. pulchra leaves (EEAPL) was found to contain compounds exhibiting antiviral properties, particularly effective against Dengue virus type 2 (DENV-2). Among these compounds, Caffeoylcalleryanin emerged as the most potent anti-DENV-2 agent, achieving a selectivity index (SI) of 20.0.
T73776 13-Hydroxyoctadecadienoic acid

Others Others
13-hydroxyoctadecadienoic acid (13-HODE) 是 Linoleic acid 的一种内源性脂氧合酶代谢产物。13-hydroxyoctadecadienoic acid 通过增强磷脂中花生四烯酸 (AA) 的释放来刺激前列环素的产生。
T36878 Sclerotiorin

Others Others
Sclerotiorin is a natural product isolated primarily from Penicillium species. It inhibits soybean lipoxygenase-1 with an IC50 value of 4.2 μM. Sclerotiorin also exhibits a number of other activities including inhibition of cholesterol ester transfer protein (IC50 = 19.4 μM),, inhibition of Grb2-Shc interaction (IC50 = 22 μM),, and antagonism of endothelin receptors (IC50 = 114 and 152 μM for human ETA and ETB, respectively).
TN6458 Acetylshikonin

Acetylshikonin can effectively inhibit tumor cells, it can be used to treat hepatocellular carcinoma cells expressing hepatitis B virus X protein (HBX) by inducing ER stress , an oncoprotein from hepatitis B virus. Acetylshikonin inhibits the production of eicosanoid, is due to the attenuation of cytosolic phospholipase A(2) membrane recruitment via the decrease in [Ca(2+)](i) and to the blockade of cyclooxygenase and 5-lipoxygenase activity.
T36560 (±)9-HpODE

Others Others
(±)9-HpODE is a racemic mixture of the fatty acid hydroperoxide product (9(S)-HpODE) formed from lipoxygenase action on linoleic acid. It shows antimicrobial activity against various fungal and bacterial pathogens and thus may play a role in plant defense. In mammalian species, monocyte-induced oxidization of LDL generates significant amounts of esterified 9-HpODE, which is rapidly reduced to 9-HODE.
T37272 9(S),12(S),13(S)-TriHOME

Others Others
9(S),12(S),13(S)-TriHOME is a linoleic acid-derived oxylipin that has diverse biological activities.1,2,3,4It has been found in various plants and is produced in human eosinophils in a 15-lipoxygenase-dependent, soluble epoxide hydrolase-independent manner.1,59(S),12(S)13(S)-TriHOME inhibits antigen-induced β-hexosaminidase release from RBL-2H3 mast cells (IC50= 28.7 μg/ml).2It inhibits LPS-induced nitric oxide (NO) production in BV-2 microglia (IC50= 40.95 μM).3In vivo, 9(S),12(S),13(S)-TriHOME...

天然产物

Xanthatin
Cat.No: T3S0153
Synonym: 苍耳亭,叶黄制菌素
Target: Apoptosis, VEGFR, Lipoxygenase, Wnt/beta-catenin, Antibacterial
Caffeic Acid
Cat.No: T2807
Synonym:
Target: Lipoxygenase, Endogenous Metabolite, TRP/TRPV Channel
Chebulagic acid
Cat.No: TQ0180
Synonym:
Target: SARS-CoV, Influenza Virus, Lipoxygenase, COX
4',5-Dihydroxyflavone
Cat.No: T8260
Synonym:
Target: Lipoxygenase, Glucosidase
3-Hydroxycoumarin
Cat.No: T8002
Synonym:
Target: Lipoxygenase
Phenethyl ferulate
Cat.No: TN2330
Synonym: Caffeic Acid 3-Methyl Phenethyl Ester,阿魏酸苯乙酯,阿魏酸苯乙醇酯
Target: Lipoxygenase, COX
Pectolinarigenin
Cat.No: T6S0413
Synonym: 柳穿鱼黄素,Pectolinaringenin
Target: Others, Lipoxygenase, COX
Aureusidin
Cat.No: TN5634
Synonym: Auresudidin,金鱼草素,Auresidin
Target: Antioxidant, Reactive Oxygen Species, Lipoxygenase
Linoleyl alcohol
Cat.No: T9512
Synonym: CIS,CIS-9,12-OCTADECADIENOL,亚麻醇
Target: Others
Psoralidin
Cat.No: T3399
Synonym:
Target: Others, Estrogen/progestogen Receptor, Reactive Oxygen Species, Lipoxygenase, Gamma-secretase, Akt, COX, Antibacterial
5-O-Demethylnobiletin
Cat.No: T5714
Synonym: 5-DEMETHYLNOBILETIN,去甲基川陈皮素
Target: Leukotriene Receptor, Lipoxygenase
S-(+)-Marmesin
Cat.No: T5759
Synonym: (+)-Marmesin,异紫花前胡内酯,(S)-Marmesin,marmesin
Target: Lipoxygenase, COX
Nordihydroguaiaretic acid
Cat.No: TJS2190
Synonym: 去甲二氢愈创木酸,NDGA,Dihydronorguaiaretic Acid
Target: Antioxidant, Ferroptosis, Lipoxygenase, Autophagy
Wedelolactone
Cat.No: T3384
Synonym: 蟛蜞菊内酯,IKK Inhibitor II
Target: Apoptosis, NF-κB, Lipoxygenase, Caspase
β-Boswellic acid
Cat.No: TN1097
Synonym: Beta-boswellic acid,β-乳香酸
Target: Lipoxygenase, DNA/RNA Synthesis
3-O-Acetyl-11-hydroxy-beta-boswellic acid
Cat.No: TN1255
Synonym:
Target: Lipoxygenase
11-​Keto-​beta-​boswellic acid
Cat.No: TN1182
Synonym: 11-Keto-beta-boswellic acid,11-酮基-BETA-乳香酸
Target: Leukotriene Receptor, NF-κB, Lipoxygenase
Picrinine
Cat.No: TN2068
Synonym:
Target: Lipoxygenase
Silychristin
Cat.No: T3879
Synonym: 水飞蓟亭,水飞蓟汀,Silicristin
Target: Lipoxygenase
Cirsiliol
Cat.No: T10821
Synonym:
Target: Apoptosis, Lipoxygenase
Anacardic Acid
Cat.No: T6389
Synonym: 漆树酸,6-pentadecylsalicylic Acid,Hydroginkgolic acid
Target: Others, Epigenetic Reader Domain, Histone Acetyltransferase, Antibacterial
Isomucronulatol 7-O-glucoside
Cat.No: TN1787
Synonym: Isomucronulatol 7-O-beta-glucoside,黄芪紫檀烷苷,3-羟基-9,10-二甲氧基紫檀烷
Target: Others
Lipoxin A4
Cat.No: T36051
Synonym: LXA4
Target: Endogenous Metabolite, Interleukin
4-Methyldaphnetin
Cat.No: TJS0315
Synonym: 7,8-Dihydroxy-4-methylcoumarin,4-甲基瑞香素,DHMC,7,8-二羟基-4-甲基香豆素
Target: Apoptosis, Lipoxygenase
Cholesteryl linoleate
Cat.No: T5214
Synonym: CE(18:2(9Z,12Z)),Cholesterol Linoleate,Linoleic Acid cholesteryl ester,胆甾烯基亚油酸酯
Target: Others, Endogenous Metabolite
6-Hydroxyflavanone
Cat.No: TN1308
Synonym:
Target: Others, Lipoxygenase, COX, GABA Receptor
4,7-DIHYDROXYCOUMARIN
Cat.No: T4137
Synonym:
Target: Others
Shogaol
Cat.No: T6S1699
Synonym: [6]-Shogaol,姜烯酚,6-姜烯酚,6-Shogaol
Target: Lipoxygenase, Autophagy
(S)-Coriolic acid
Cat.No: T37974
Synonym: 13(S)-HODE
Target: Lipoxygenase, Mitochondrial Metabolism, PPAR
Texasin
Cat.No: T24869
Synonym: IR2,IR 2,IR-2
Target: Others
Turmeronol A
Cat.No: TN5196
Synonym:
Target: Others
Jujuboside D
Cat.No: TN1813
Synonym: 酸枣仁皂苷D,酸枣仁皂甙D
Target: Others
Eugenol benzoate
Cat.No: TN4032
Synonym:
Target: Others
Trachelosiaside
Cat.No: TN5159
Synonym:
Target: Others
Isotachioside
Cat.No: TN4331
Synonym:
Target: Lipoxygenase
2,3,4'-Trihydroxy-3',5'-dimethoxypropiophenone
Cat.No: TN2688
Synonym:
Target: Antioxidant, Lipoxygenase
Sideritoflavone
Cat.No: TN5017
Synonym:
Target: Opioid Receptor, Prostaglandin Receptor
9,11-Dehydro-beta-boswellic acid
Cat.No: TN7347
Synonym:
Target: Others
Lycopodine
Cat.No: T13764
Synonym:
Target: Lipoxygenase, Caspase
Masoprocol
Cat.No: T60692
Synonym:
Target: Others
Futoenone
Cat.No: TN4088
Synonym:
Target: PAFR
Caffeoylcalleryanin
Cat.No: TN7391
Synonym:
Target: Others
13-Hydroxyoctadecadienoic acid
Cat.No: T73776
Synonym:
Target: Others
Sclerotiorin
Cat.No: T36878
Synonym:
Target: Others
Acetylshikonin
Cat.No: TN6458
Synonym:
Target:
(±)9-HpODE
Cat.No: T36560
Synonym:
Target: Others
9(S),12(S),13(S)-TriHOME
Cat.No: T37272
Synonym:
Target: Others
Cat. No. Product Name Species Expression System
TMPY-03553 15 Lipoxygenase 2 Protein, Human, Recombinant

arachidonate 15-lipoxygenase, type B,ALOX15B,15-LOX...

Human Baculovirus Insect Cells
15 Lipoxygenase 2 Protein, Human, Recombinant is expressed in Baculovirus insect cells. The predicted molecular weight is 76 kDa and the accession number is AAH35217.1.
TMPY-03462 15 Lipoxygenase 2 Protein, Human, Recombinant (His & GST)

ALOX15B,arachidonate 15-lipoxygenase, type B,15-LOX...

Human Baculovirus Insect Cells
15 Lipoxygenase 2 Protein, Human, Recombinant (His & GST) is expressed in Baculovirus insect cells with His and GST tag. The predicted molecular weight is 103.7 kDa and the accession number is AAH35217.1.
TMPH-00955 ALOX12 Protein, Human, Recombinant (His)

Polyunsaturated fatty acid lipoxygenase ALOX12,LOG1...

Human E. coli
ALOX12 Protein, Human, Recombinant (His) is expressed in E. coli.
TMPY-01481 FLAP Protein, Human, Recombinant (His)

FLAP,arachidonate 5-lipoxygenase-activating protein

Human Baculovirus Insect Cells
Arachidonate 5-Lipoxygenase-Activating Protein (ALOX5AP), also known as FLAP, belongs to the MAPEG family. ALOX5AP/FLAP is an essential partner of 5-LO for this process. The FLAP (ALOX5AP) gene has been linked to risk for myocardial infarction, stroke and restenosis, reigniting pharmaceutical interest in this target. It had been found that ALOX5AP/FLAP is a key enzyme in leukotriene formation, in both human pulmonary microvascular endothelial cells and a transformed human brain endothelial cell ...

重组蛋白

15 Lipoxygenase 2 Protein, Human, Recombinant
Cat.No: TMPY-03553
Species: Human
Expression System: Baculovirus Insect Cells
15 Lipoxygenase 2 Protein, Human, Recombinant (His & GST)
Cat.No: TMPY-03462
Species: Human
Expression System: Baculovirus Insect Cells
ALOX12 Protein, Human, Recombinant (His)
Cat.No: TMPH-00955
Species: Human
Expression System: E. coli
FLAP Protein, Human, Recombinant (His)
Cat.No: TMPY-01481
Species: Human
Expression System: Baculovirus Insect Cells
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