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Search Results for " lipophilic "
Targets Recommended: Parasite

109

抑制剂 & 化合物

7

天然产物

2

重组蛋白

3

同位素标记化合物

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Cat. No. Product Name Target Signaling Pathways
T5639 lufenuron

Fluphenacur,虱螨脲

Parasite Microbiology/Virology
Lufenuron (Fluphenacur) 和几丁质合成抑制剂,可抑制节肢动物的蜕皮,控制蚤和鱼虱。
T15102 Dexamethasone palmitate

地塞米松棕榈酸酯,DXP

Glucocorticoid Receptor Endocrinology/Hormones
Dexamethasone palmitate (DXP) (DXP) 是 Dexamethasone 的前药。Dexamethasone 是糖皮质激素受体激动剂。与Dexamethasone 相比, DXP 对糖皮质激素受体的亲和力低 47 倍。DXP 显示出抗炎活性。
T1065 Baclofen

巴氯芬,Lioresal

GABA Receptor Membrane transporter/Ion channel; Neuroscience
Baclofen (Lioresal) 是 γ-氨基丁酸 (GABA) 的亲脂性衍生物,是可口服的选择性代谢型 GABA-B 受体激动剂,具有高血脑屏障渗透率,用于治疗因脊髓损伤和多发性硬化引起的痉挛。
T19438 Myristyl nicotinate

Tetradecyl nicotinate,肉豆蔻醇烟酸酯

GPR Endocrinology/Hormones; GPCR/G Protein
Myristyl nicotinate (Tetradecyl nicotinate) 是 Nicotinic acid 的亲脂衍生物,是一种酯前药。它能够刺激光损伤的皮肤中的表皮分化,增加皮肤 NAD 含量并增强人皮肤屏障。它被开发用于将烟酸输送到皮肤中,以防止光化性角化病及其发展为皮肤癌。
T21404 Fluticasone furoate

Veramyst,Allermist,Avamys,糠酸氟替卡松,Fluticasone furoate

Glucocorticoid Receptor Endocrinology/Hormones
Fluticasone furoate (Avamys) 是一种合成的三氟化皮质类固醇,衍生自氟替卡松,Kd 为 0.3 nM。Fluticasone furoate 具有有效的抗炎、抗哮喘活性和低全身暴露。Fluticasone furoate 可用作过敏性鼻炎治疗研究的鼻喷雾剂。
T8630 Baclofen hydrochloride

4-amino-3-(4-chlorophenyl)butanoic acid hydron chloride

GABA Receptor Membrane transporter/Ion channel; Neuroscience
Baclofen hydrochloride (4-amino-3-(4-chlorophenyl)butanoic acid hydron chloride) 是一种 GAMMA-AMINOBUTYRIC ACID 衍生物,是一种特异性 GABA-B 受体激动剂。它用于治疗肌肉痉挛,尤其是由于脊髓损伤引起的肌肉痉挛。其治疗效果来自于脊髓和脊髓上部位的作用,通常是减少兴奋性传递。
T1418 Bucladesine sodium

dbcAMP,Dibutyryl-cAMP sodium salt,布拉地新钠盐,Dibutyryl-cAMP,DC2797,Sodium dibutyryl cAMP,Bucladesine,Bucladesine sodium salt

PKA; PDE Metabolism; Tyrosine Kinase/Adaptors
Bucladesine sodium (DC2797) 是一种 cAMP 类似物,具有细胞渗透性。Bucladesine sodium 也是一种 cAMP 依赖性的蛋白激酶 (PKA) 激活剂,一种磷酸二酯 (PDE) 抑制剂。Bucladesine sodium 具有抗炎活性。
T73506 TH-Z93

THZ93

Antibacterial Microbiology/Virology
TH-Z93 是一种有效的 FPPS 抑制剂 (IC50: 90 nM),也是一种亲脂性双膦酸盐。
T15118 DiD perchlorate

Others Others
DiD perchlorate 是一种远红色荧光亲脂性花青染料。它能快速稳定地与磷脂细胞膜结合,能用于细胞追踪。
T67812 Tenifatecan

SN2310

Others Others
Tenifatecan (SN2310) 是一种高度亲脂性的7-乙基-10-羟基喜树碱(SN)制剂,具有潜在的抗肿瘤活性。
T60151 CP-447697

Complement System Immunology/Inflammation
CP-447697 是亲脂性的 C5a 受体拮抗剂,IC50 值为 31 nM。CP-447697 可用于炎症的研究。
T40857 Calcium ionophore II

Calcium ionophore II,N,N,N′,N′-Tetracyclohexyl-3-oxapentanediamide

Others Others
Calcium ionophore II (N,N,N′,N′-Tetracyclohexyl-3-oxapentanediamide) 是一种亲脂性离子载体,可用于制备钙离子选择性电极。
T17109 TMRM Perchlorate

四甲基若丹明甲酯酸铵,T668

Others Others
TMRM Perchlorate (T668) 是细胞渗透性的阳离子亲脂性红色荧光染料 (λex=530 nm, λem=592 nm)。
T0876 Clioquinol

Chinoform,Iodochlorhydroxyquin,氯碘羟喹

Mitophagy; Antibiotic; Autophagy; Antifungal Autophagy; Microbiology/Virology
Clioquinol (Iodochlorhydroxyquin) 是一种局部抗真菌药,具有抗肿瘤活性。它作为口服抗菌剂,可研究腹泻和皮肤感染。
T40418 DiO

DiOC18(3),3,3'-Dioctadecyloxacarbocyanine perchlorate

Others Others
DiO (DiOC18(3)) 是一种荧光亲脂性示踪剂,可广泛用于标记细胞、细胞器、脂质体、病毒和脂蛋白。
T2405 Revaprazan hydrochloride

盐酸瑞伐拉赞,YH1885

ATPase; COX; Antibacterial Immunology/Inflammation; Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience
Revaprazan hydrochloride (YH1885) 是一种新型酸泵拮抗剂,可降低COX-2的表达,在幽门螺杆菌感染中,显著抑制炎症。
T78393 C12FDG

5-Dodecanoylaminofluorescein di-β-D-Galactopyranoside

C12FDG (5-Dodecanoylaminofluorescein di-β-D-Galactopyranoside) 作为一种亲脂性用于检测β-半乳糖活性的绿色荧光底物,是一种衰老标志物,常与流式细胞仪连用。
TQ0095 Brincidofovir

CMX001,HDP-CDV

Others; Antiviral; HSV Immunology/Inflammation; Microbiology/Virology; Others
Brincidofovir (HDP-CDV) 是 Cidofovir 的一种具有口服活性的亲脂性形式的前体药物,是一种口服长效的抗病毒药物,有广泛的抗 DNA 病毒活性。
T1439 Lacidipine

SN-305,拉西地平,GX-1048,GR-43659X

Apoptosis; Calcium Channel; Reactive Oxygen Species Apoptosis; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; NF-κB
Lacidipine (SN-305) 是一种L 型钙离子通道阻断剂。
T78526 4A3-SC8

4A3 SC8,4A3SC8

Liposome Metabolism
4A3-SC8 为一种具有阳离子基团和亲脂基团的模块化树枝状大分子,可在侵袭性肝癌模型中使小RNA延长生存期,可用于合成脂质纳米颗粒。
T78392 Zinquin ethyl ester

Zinquin ethyl ester为具有特异性的锌离子荧光探针,为Zinquin的亲脂性荧光衍生物,能敏感检测锌离子且可穿透细胞膜。
T36958 BODIPY 505/515

BODIPY 505/515 是一种亲脂性荧光探针,可定位到细胞内的脂质体,已被用于标记脂滴。BODIPY 505/515 已被用于电子显微镜、外荧光显微镜、共聚焦显微镜以及各种藻类物种的流式细胞仪应用中。
T2569 Chlorotrianisene

tris(p-methoxyphenyl)chloroethylene,氯丁烯二烯,CTA,tri-p-anisylchloroethylene,氯烯雌醚,TACE

Estrogen Receptor/ERR; Estrogen/progestogen Receptor; COX Endocrinology/Hormones; Immunology/Inflammation; Neuroscience
Chlorotrianisene (tri-p-anisylchloroethylene) 是长效、可口服、亲脂性高的合成三苯乙烯 (TPE) 衍生物和选择性雌激素受体调节剂,有雌激素活性,也有抗雌激素活性。它还有效抑制COX-1并抑制全血中的血小板聚集。
T36957 BODIPY 493/503

BDP 493/503 lipid stain,Pyrromethene 546

Others Others
BODIPY 493/503 (Pyrromethene 546) 属于亲脂性荧光染料,Ex/Em 为 493/503 nm。 BODIPY 493/503 定位于极性脂质,可用于标记细胞中性脂质含量以及活细胞和固定细胞应用。
T6170 Elesclomol

伊利司莫,STA-4783

Apoptosis; HSP; Reactive Oxygen Species Apoptosis; Cytoskeletal Signaling; Immunology/Inflammation; Metabolism; NF-κB
Elesclomol (STA-4783) 是一种氧化应激诱导剂,也是一种高度亲脂性的铜离子载体。Elesclomol 可以诱导肿瘤细胞凋亡,用于铜死亡相关研究。Elesclomol 还可以抑制 FDX1 介导的 Fe-S 簇生物合成。
T16858 SBE-β-CD

磺丁基-Β-环糊精,Sulfobutylether-β-Cyclodextrin

Others Others
SBE-β-CD (Sulfobutylether-β-Cyclodextrin) 是一种 β-环糊精的衍生物,其磺酸钠盐通过丁基醚间隔基团或磺基丁基醚与亲脂腔隔开。SBE-β-CD 可作为助溶剂,被广泛用于生物学实验中。
T2627 Nolatrexed dihydrochloride

盐酸诺拉曲塞,Thymitaq,AG 337

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Nolatrexed dihydrochloride (Thymitaq) 是一种非竞争性的胸苷酸合酶抑制剂,能够在癌细胞 S 期诱导细胞周期停滞,具有抗癌活性。它与该酶的叶酸辅因子结合位点相互作用,对人胸苷酸合酶的Ki 值为 11 nM。
T11717 JHU395

Apoptosis Apoptosis
JHU395 是一种口服生物利用度高的前药,其活性成分是亲脂性谷氨酸拮抗剂(GA,6-叠氮-5-酮-L-去亚硝基赖氨酸)。JHU395 能有效地将DON输送至恶性周围神经鞘瘤(MPNST)的体外和体内模型中,并在MPNST上显现出显著的抗肿瘤活性。此外,JHU395在血浆中表现出良好的稳定性。
T27624 Iptakalim Hydrochloride

Potassium Channel; AChR Membrane transporter/Ion channel; Neuroscience
Iptakalim hydrochloride 是一种亲脂性的对氨基化合物,是 ATP 敏感的钾通道的开放剂,也是含α4β2的烟碱乙酰胆碱受体拮抗剂。它也是一种 K(ir) 6.1/SUR2B 激活剂,可通过保护内皮功能减轻大鼠缺氧引起的肺动脉高压。
T15378L Gemcitabine elaidate hydrochloride

CO-101 hydrochloride,Gemcitabine elaidate hydrochloride(210829-30-4(free base)),Gemcitabine 5'-elaidate hydrochloride,CP-4126 hydrochloride

Others Others
Gemcitabine elaidate (CP-4126) hydrochloride 是 Gemcitabine 的亲脂性前药。Gemcitabine elaidate hydrochloride 通过酯酶转化为 Gemcitabine 以被磷酸化。Gemcitabine elaidate hydrochloride 可以口服给药,具有抗肿瘤活性。
T15129 DiI

DiIC18(3)

Others Others
DiI (DiIC18(3)) 是一种亲脂性膜染料,通常用作神经元和其它细胞的长期示踪剂。它在进入细胞膜之前荧光非常弱,仅当进入到细胞膜后才可以被激发出很强的橙红色荧光 (λex=549 nm,λem=565 nm)。
T15609 JC-1

CBIC2

Others Others
JC-1 (CBIC2) 是一种荧光亲脂性羰花青染料,用于测量线粒体膜电位。线粒体膜电位较高时,它在基质中汇聚形成聚合物,可以产生红色荧光(λex=585 nm,λem=590 nm)。线粒体膜电位较低时,它不能聚集在线粒体基质中,以单体形式存在产生绿色荧光(λex=510 nm,λem=527 nm)。
T60774 NITD-916

NITD916,NITD 916

Antibiotic Microbiology/Virology
NITD-916 是一种具有口服活性和高度亲脂性的分枝杆菌烯酰还原酶 InhA 抑制剂,IC50 为 570 nM。NITD-916是一种有有效的 4-羟基-2-吡啶酮衍生物, 与 InhA 和 NADH 形成三元复合物,阻止进入脂肪酰基底物结合袋。NITD-916 具有抗结核活性。
T25360 Eclazolast

RHC2871,RHC-2871,REV2871,REV 2871,RHC 2871

Others Others
Eclazolast (RHC 2871) 是一种亲脂性抗过敏化合物,在肥大细胞模型中抑制介质释放。Eclazolast 通过在细胞内只影响与Fc(epsilon)RI 相关的直接过程而抑制细胞外分泌。Eclazolast 的效果高度依赖于触发细胞的抗原浓度。
T21297 Miriplatin hydrate

SM-11355 (hydrate),Miripla,Miriplatin,SM 11355,SM11355,SM-11355,Miriplatin hydrate

DNA Alkylation DNA Damage/DNA Repair
Miriplatin hydrate (SM-11355 (hydrate)) (MPT)是一种用于TACE 的新型铂类化合物,在肝细胞癌(HCC)的治疗中显示出良好的前景。米铂是一种亲脂性铂复合物,容易悬浮在碘油中,并在肿瘤组织中逐渐释放活性铂化合物。
T6929 Pantoprazole sodium

Pantecta,泮托拉唑钠盐,SKF96022 sodium,SKF96022 (sodium),BY1023 (sodium),泮托拉唑钠,BY-1023 sodium,Pantoloc

Apoptosis; Others; Proton pump; HIF; Autophagy Angiogenesis; Apoptosis; Autophagy; Chromatin/Epigenetic; Membrane transporter/Ion channel; Others
Pantoprazole sodium (Pantecta) 是一种具有口服活性的质子泵抑制剂,是一种取代的苯并咪唑,是H+/K+-ATPase 抑制剂,IC50为 6.8 μM。它可以改善 pH 值稳定性,具有抗分泌和抗溃疡的作用。它联合阿霉素可显著增加肿瘤生长延迟。
T6334 Ridaforolimus

AP23573,Deforolimus,MK-8669

mTOR; Autophagy Autophagy; PI3K/Akt/mTOR signaling
Ridaforolimus (AP23573) 是亲脂性大环内酯类抗生素雷帕霉素的小分子非前药类似物,具有潜在的抗肿瘤活性。它是一种有效和选择性的 mTOR 抑制剂,在 HT-1080 细胞中抑制 S6 磷酸化的 IC50值为 0.2 nM。
T28326 PD 130883

PD-130883,PD130883

Others Others
PD 130883 is a potent lipophilic quinazoline antifolate.
T32257 Janolusimide

Others Others
Janolusimide is a kind of lipophilic tripeptide marine toxin.
T31381 Deoxylimonol

Deoxy-alpha-limonol

Others Others
Deoxylimonol is a lipophilic compound found in human feces.
T13117 Teludipine hydrochloride

GR53992B,GX1296B

Calcium Channel Membrane transporter/Ion channel; Metabolism
Teludipine hydrochloride is a blocker of lipophilic calcium channel.
T23672 AH-1058 HCl

AH 1058 HCl

Others Others
AH-1058 HCl is a lipophilic antiarrhythmic calcium channel blocker.
TD0083 DiIiodide1,1‘-Dioctadecyl-3,3,3’,3‘-tetramethylindocarbocyanine iodide]

DiI碘化物

DiI iodide1 is one of lipophilic fluorescent stains for labeling membranes and other hydrophobic structures. The fluorescence of these environment-sensitive dyes is greatly enhanced when incorporated into membranes or bound to lipophilic biomolecules such as proteins although they are weakly fluorescent in water.
T24473 Mixanpril

Others Others
Mixanpril is an RB 105 lipophilic prodrug.
T68515 AZD-1175

Others Others
AZD-1175 is a cannabinoid receptor CB1 antagonist and highly lipophilic compound for the treatment of type 2 diabetes and obesity.
T24300 L 645151

L645151,L-645151

Others Others
L 645151 is an inhibitor of lipophilic CA.
T30841 Cgp 57813

Cgp-57813,Cgp57813

Others Others
CGP 57813 is a lipophilic compound, which can be used as an inhibitor of HIV-1 protease.
T27153 Dexamethasone cipecilate

NS126,NS-126,NS 126

Others Others
Dexamethasone cipecilate is a long-acting intranasal corticosteroid and a highly lipophilic anti-inflammatory corticosteroid.
TD0084 DiI triflate [1,1‘-Dioctadecyl-3,3,3’,3‘-tetramethylindocarbocyanine triflate]

DiI triflate is one of lipophilic fluorescent stains for labeling membranes and other hydrophobic structures. The fluorescence of these environment-sensitive dyes is greatly enhanced when incorporated into membranes or bound to lipophilic biomolecules such as proteins although they are weakly fluorescent in water.
T37936 16-phenoxy tetranor Prostaglandin F2α isopropyl ester

16-phenoxy tetranor Prostaglandin F2α isopropyl ester

Others Others
Prostaglandin F2α (PGF2α) drives luteolysis and smooth muscle contraction by activating the FP receptor. Stable, lipophilic analogs of PGF2α are used to modulate luteolysis and treat glaucoma. 16-phenoxy tetranor Prostaglandin F2α isopropyl ester (16-phenoxy tetranor PGF2α isopropyl ester) is a lipophilic analog of 16-phenoxy tetranor PGF2α. Isopropyl esters of PGs serve as prodrugs, as they are efficiently hydrolyzed in certain tissues to generate the bioactive free acid.

化合物

lufenuron
Cat.No: T5639
Synonym: Fluphenacur,虱螨脲
Target: Parasite
Dexamethasone palmitate
Cat.No: T15102
Synonym: 地塞米松棕榈酸酯,DXP
Target: Glucocorticoid Receptor
Baclofen
Cat.No: T1065
Synonym: 巴氯芬,Lioresal
Target: GABA Receptor
Myristyl nicotinate
Cat.No: T19438
Synonym: Tetradecyl nicotinate,肉豆蔻醇烟酸酯
Target: GPR
Fluticasone furoate
Cat.No: T21404
Synonym: Veramyst,Allermist,Avamys,糠酸氟替卡松,Fluticasone furoate
Target: Glucocorticoid Receptor
Baclofen hydrochloride
Cat.No: T8630
Synonym: 4-amino-3-(4-chlorophenyl)butanoic acid hydron chloride
Target: GABA Receptor
Bucladesine sodium
Cat.No: T1418
Synonym: dbcAMP,Dibutyryl-cAMP sodium salt,布拉地新钠盐,Dibutyryl-cAMP,DC2797,Sodium dibutyryl cAMP,Bucladesine,Bucladesine sodium salt
Target: PKA, PDE
TH-Z93
Cat.No: T73506
Synonym: THZ93
Target: Antibacterial
DiD perchlorate
Cat.No: T15118
Synonym:
Target: Others
Tenifatecan
Cat.No: T67812
Synonym: SN2310
Target: Others
CP-447697
Cat.No: T60151
Synonym:
Target: Complement System
Calcium ionophore II
Cat.No: T40857
Synonym: Calcium ionophore II,N,N,N′,N′-Tetracyclohexyl-3-oxapentanediamide
Target: Others
TMRM Perchlorate
Cat.No: T17109
Synonym: 四甲基若丹明甲酯酸铵,T668
Target: Others
Clioquinol
Cat.No: T0876
Synonym: Chinoform,Iodochlorhydroxyquin,氯碘羟喹
Target: Mitophagy, Antibiotic, Autophagy, Antifungal
DiO
Cat.No: T40418
Synonym: DiOC18(3),3,3'-Dioctadecyloxacarbocyanine perchlorate
Target: Others
Revaprazan hydrochloride
Cat.No: T2405
Synonym: 盐酸瑞伐拉赞,YH1885
Target: ATPase, COX, Antibacterial
C12FDG
Cat.No: T78393
Synonym: 5-Dodecanoylaminofluorescein di-β-D-Galactopyranoside
Target:
Brincidofovir
Cat.No: TQ0095
Synonym: CMX001,HDP-CDV
Target: Others, Antiviral, HSV
Lacidipine
Cat.No: T1439
Synonym: SN-305,拉西地平,GX-1048,GR-43659X
Target: Apoptosis, Calcium Channel, Reactive Oxygen Species
4A3-SC8
Cat.No: T78526
Synonym: 4A3 SC8,4A3SC8
Target: Liposome
Zinquin ethyl ester
Cat.No: T78392
Synonym:
Target:
BODIPY 505/515
Cat.No: T36958
Synonym:
Target:
Chlorotrianisene
Cat.No: T2569
Synonym: tris(p-methoxyphenyl)chloroethylene,氯丁烯二烯,CTA,tri-p-anisylchloroethylene,氯烯雌醚,TACE
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, COX
BODIPY 493/503
Cat.No: T36957
Synonym: BDP 493/503 lipid stain,Pyrromethene 546
Target: Others
Elesclomol
Cat.No: T6170
Synonym: 伊利司莫,STA-4783
Target: Apoptosis, HSP, Reactive Oxygen Species
SBE-β-CD
Cat.No: T16858
Synonym: 磺丁基-Β-环糊精,Sulfobutylether-β-Cyclodextrin
Target: Others
Nolatrexed dihydrochloride
Cat.No: T2627
Synonym: 盐酸诺拉曲塞,Thymitaq,AG 337
Target: DNA/RNA Synthesis
JHU395
Cat.No: T11717
Synonym:
Target: Apoptosis
Iptakalim Hydrochloride
Cat.No: T27624
Synonym:
Target: Potassium Channel, AChR
Gemcitabine elaidate hydrochloride
Cat.No: T15378L
Synonym: CO-101 hydrochloride,Gemcitabine elaidate hydrochloride(210829-30-4(free base)),Gemcitabine 5'-elaidate hydrochloride,CP-4126 hydrochloride
Target: Others
DiI
Cat.No: T15129
Synonym: DiIC18(3)
Target: Others
JC-1
Cat.No: T15609
Synonym: CBIC2
Target: Others
NITD-916
Cat.No: T60774
Synonym: NITD916,NITD 916
Target: Antibiotic
Eclazolast
Cat.No: T25360
Synonym: RHC2871,RHC-2871,REV2871,REV 2871,RHC 2871
Target: Others
Miriplatin hydrate
Cat.No: T21297
Synonym: SM-11355 (hydrate),Miripla,Miriplatin,SM 11355,SM11355,SM-11355,Miriplatin hydrate
Target: DNA Alkylation
Pantoprazole sodium
Cat.No: T6929
Synonym: Pantecta,泮托拉唑钠盐,SKF96022 sodium,SKF96022 (sodium),BY1023 (sodium),泮托拉唑钠,BY-1023 sodium,Pantoloc
Target: Apoptosis, Others, Proton pump, HIF, Autophagy
Ridaforolimus
Cat.No: T6334
Synonym: AP23573,Deforolimus,MK-8669
Target: mTOR, Autophagy
PD 130883
Cat.No: T28326
Synonym: PD-130883,PD130883
Target: Others
Janolusimide
Cat.No: T32257
Synonym:
Target: Others
Deoxylimonol
Cat.No: T31381
Synonym: Deoxy-alpha-limonol
Target: Others
Teludipine hydrochloride
Cat.No: T13117
Synonym: GR53992B,GX1296B
Target: Calcium Channel
AH-1058 HCl
Cat.No: T23672
Synonym: AH 1058 HCl
Target: Others
DiIiodide1,1‘-Dioctadecyl-3,3,3’,3‘-tetramethylindocarbocyanine iodide]
Cat.No: TD0083
Synonym: DiI碘化物
Target:
Mixanpril
Cat.No: T24473
Synonym:
Target: Others
AZD-1175
Cat.No: T68515
Synonym:
Target: Others
L 645151
Cat.No: T24300
Synonym: L645151,L-645151
Target: Others
Cgp 57813
Cat.No: T30841
Synonym: Cgp-57813,Cgp57813
Target: Others
Dexamethasone cipecilate
Cat.No: T27153
Synonym: NS126,NS-126,NS 126
Target: Others
DiI triflate [1,1‘-Dioctadecyl-3,3,3’,3‘-tetramethylindocarbocyanine triflate]
Cat.No: TD0084
Synonym:
Target:
16-phenoxy tetranor Prostaglandin F2α isopropyl ester
Cat.No: T37936
Synonym: 16-phenoxy tetranor Prostaglandin F2α isopropyl ester
Target: Others
Cat. No. Product Name Target Signaling Pathways
TMS2180 Zeaxanthin

Anchovyxanthin,All-Trans-Zeaxanthin,玉米

Antioxidant; Endogenous Metabolite Metabolism; oxidation-reduction
Zeaxanthin (All-Trans-Zeaxanthin) 是食物获得类胡萝卜素,存在于眼睛的黄斑部,具有抗氧化活性。
T2A2509 Laurocapram

月桂氮酮,Tranzone,Azone,N-Lauryl caprolactam,N-0252,月桂氮卓酮,N-Dodecylcaprolactam

Others Others
Laurocapram (N-Lauryl caprolactam) 是吸收促进剂,对于亲脂性和亲水性物质都是一种最有效的吸收剂。
T16747 Riboflavin Tetrabutyrate

Reactive Oxygen Species Immunology/Inflammation; Metabolism; NF-κB
Riboflavin Tetrabutyrate 是一种亲脂性黄素衍生物,具有抗氧化和脂质过氧化物去除活性。
T8021 Dibenzoyl Thiamine

Bentiamine,二苯甲酰硫胺素

Others Others
Dibenzoyl Thiamine (Bentiamine) 是一种硫胺素的衍生物。它在体内被迅速吸收,并转化成硫胺素。
T29352 2-Hydroxydecanoic acid

(±)-α-hydroxy Decanoic Acid,羟基癸酸,(±)-2-hydroxy Decanoic Acid,alpha-Hydroxydecanoic acid,2-hydroxy Decylic Acid,2-Hydroxydecanoate

Others Others
2-Hydroxydecanoic acid ((±)-α-hydroxy Decanoic Acid) 是一种在好氧菌 P. ovalis 的脂多糖部分的亲脂部分中发现的脂肪酸。
TL0004 FERULIC ACID METHYL ESTER

阿魏酸甲酯,Methyl ferulate,Methyl 4'-hydroxy-3'-methoxycinnamate

p38 MAPK; Autophagy Autophagy; MAPK
FERULIC ACID METHYL ESTER (Methyl ferulate) 是从大百部中分到的阿魏酸衍生物,具有抗氧化和抗炎作用。在原发性骨髓源性巨噬细胞中,它抑制 COX-2 的表达,降低 p-p38和 p-JNK 的水平。它能够透过细胞膜和血脑屏障,清除自由基,可研究神经退行性疾病。
T79989 Funiculosin

Antibiotic Microbiology/Virology
Funiculosin为一种中性亲脂性抗生素,能够抑制DNA及RNA病毒,并具备抗真菌活性。在初级鸡胚成纤维细胞中,Funiculosin可有效抑制致病真菌引发的感染。

天然产物

Zeaxanthin
Cat.No: TMS2180
Synonym: Anchovyxanthin,All-Trans-Zeaxanthin,玉米
Target: Antioxidant, Endogenous Metabolite
Laurocapram
Cat.No: T2A2509
Synonym: 月桂氮酮,Tranzone,Azone,N-Lauryl caprolactam,N-0252,月桂氮卓酮,N-Dodecylcaprolactam
Target: Others
Riboflavin Tetrabutyrate
Cat.No: T16747
Synonym:
Target: Reactive Oxygen Species
Dibenzoyl Thiamine
Cat.No: T8021
Synonym: Bentiamine,二苯甲酰硫胺素
Target: Others
2-Hydroxydecanoic acid
Cat.No: T29352
Synonym: (±)-α-hydroxy Decanoic Acid,羟基癸酸,(±)-2-hydroxy Decanoic Acid,alpha-Hydroxydecanoic acid,2-hydroxy Decylic Acid,2-Hydroxydecanoate
Target: Others
FERULIC ACID METHYL ESTER
Cat.No: TL0004
Synonym: 阿魏酸甲酯,Methyl ferulate,Methyl 4'-hydroxy-3'-methoxycinnamate
Target: p38 MAPK, Autophagy
Funiculosin
Cat.No: T79989
Synonym:
Target: Antibiotic
Cat. No. Product Name Species Expression System
TMPJ-01412 LRP-12 Protein, Human, Recombinant (His)

LRP-12,ST7,Suppressor of Tumorigenicity 7 Protein,LRP12,Low-...

Human HEK293 Cells
Low-Density Lipoprotein Receptor-Related Protein 12 (LRP12) belongs to the LDLR family. LRP12 is a type I transmembrane protein annd widely expressed in heart, skeletal muscle, brain, lung, placenta and pancreas. LRP12 contains 2 CUB domain and 5 LDL-receptor class A domain. LRP12 has been shown to interact with GNB2L1, ZFYVE9 and ITGB1BP3. LRP12 is a receptor probably, which may be involved in the internalization of lipophilic molecules and/or signal transduction. In addition, LRP12 may act as ...
TMPY-01679 LCN1 Protein, Human, Recombinant (His)

TLC,MGC71975,TP,VEGP,Lipocalin 1,PMFA

Human HEK293 Cells
Lipocalin-1, also known as Von Ebner gland protein, VEG protein, Tear Prealbumin, VEGP, Tear lipocalin, and LCN1 is a secreted protein that belongs to the calycin superfamily and Lipocalin family. Human Lipocalin-1 / VEGP was originally described as a major protein of human tear fluid, which was thought to be tear specific. Lipocalin-1 / VEGP is identical to lingual von Ebner's gland protein and is also produced in the prostate, nasal mucosa, and tracheal mucosa. Homologous proteins have been fo...

重组蛋白

LRP-12 Protein, Human, Recombinant (His)
Cat.No: TMPJ-01412
Species: Human
Expression System: HEK293 Cells
LCN1 Protein, Human, Recombinant (His)
Cat.No: TMPY-01679
Species: Human
Expression System: HEK293 Cells
Cat. No. Product Name Target Signaling Pathways
TMID-0245 Pindolol-d7

Pindolol-d7 是 Pindolol 的氘代化合物。Pindolol 的 CAS 号为 13523-86-9。Pindolol 是一种非选择性β-阻断剂,局部的β-肾上腺素能受体激动剂活性,也作为5-HT1A受体部分拮抗剂,Ki为33nM。它是非心脏选择性的,具有内在的拟交感神经作用。
TMIJ-0497 Lacidipine-d10

Lacidipine-d10 是 Lacidipine 的氘代化合物。Lacidipine 的 CAS 号为 103890-78-4。Lacidipine 是一种L型钙离子通道阻断剂。
TMID-0096 P-CRESOL-d3 (METHYL-d3)

P-CRESOL-d3 (METHYL-d3) 是 P-CRESOL 的氘代化合物。P-CRESOL 的 CAS 号为 106-44-5。p-Cresol 是一种部分亲脂性部分,在正常条件下与血浆蛋白(接近 100%)强烈结合。对甲酚通过结合代谢,主要是硫酸化和葡萄糖醛酸化,但未结合的对甲酚至少部分通过尿液去除。

同位素标记化合物

Pindolol-d7
Cat.No: TMID-0245
Synonym:
Target:
Lacidipine-d10
Cat.No: TMIJ-0497
Synonym:
Target:
P-CRESOL-d3 (METHYL-d3)
Cat.No: TMID-0096
Synonym:
Target:
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