Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T32770 |
Linsidomine
CV 664 |
Others | Others |
Lincydomine is a smooth muscle relaxant, beneficial to the treatment of unstable angina pectoris, but also can open the respiratory tract of humans and guinea pigs. | |||
T23356 |
Linsidomine hydrochloride
SIN-1 chloride |
Others | Others |
Linsidomine hydrochloride (SIN-1 chloride) 是莫西多明的代谢产物,具有舒张血管、抑制血小板聚集和抗心绞痛的活性。在心肌缺血-再灌注模型中,Linsidomine hydrochloride 减少心肌坏死和再灌注诱导的内皮功能障碍,与海绵体的作用机制涉及一氧化氮的释放有关。 | |||
T0109 |
Molsidomine
Morsydomine,SIN-10,吗多明,Corvaton |
NOD | Immunology/Inflammation; NF-κB |
Molsidomine (Corvaton) 是一种长效的、口服活性的血管扩张药,在肝脏中代谢可被为活性代谢物Linsidomine。 其中Linsidomine 是一种不稳定的化合物,能够产生NO,可用作血管舒张剂。 |