Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T16272 |
Naproxen etemesil
LT-NS 001,MX 1094 |
PDE | Metabolism |
Naproxen is a COX-1 and COX-2 inhibitor (IC50s: 8.72 and 5.15 μM, respectively in cell assay). Naproxen etemesil is a lipophilic and non-acidic prodrug of naproxen. It is hydrolyzed to pharmacologically active Naproxen once absorbed. |