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Targets Recommended: Lipoxygenase

635

抑制剂 & 化合物

112

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19

重组蛋白

34

同位素标记化合物

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Cat. No. Product Name Target Signaling Pathways
T39986 LOX-IN-3 dihydrochloride

Lipoxygenase Metabolism
LOX-IN-3 dihydrochloride 是口服有效的赖氨酰氧化酶抑制剂,在纤维化,癌症和/或血管生成方面有研究价值。
T77528 5-LOX-IN-2

Apoptosis; Lipoxygenase Apoptosis; Metabolism
5-LOX-IN-2 是 一种 5-脂氧合酶抑制剂 (5-LOX )抑制剂,从体外实验测得的IC50 值为 0.33 μM。5-LOX-IN-2 以剂量依赖的方式抑制 5-LOX发挥作用。5-LOX-IN-2 可降低肾癌细胞的细胞活性并诱导凋亡 (apoptosis),可用于研究癌症。
T65427 5-LOX inhibitor

1-(sec-Butyl)-4-(4-(4-(4-hydroxyphenyl)piperazin-1-yl)phenyl)-1H-1,2,4-triazol-5(4H)-one

Lipoxygenase Metabolism
5-LOX inhibitor (1-(sec-Butyl)-4-(4-(4-(4-hydroxyphenyl)piperazin-1-yl)phenyl)-1H-1,2,4-triazol-5(4H)-one) 是伊曲康唑杂质之一,是一种选择性 LOX-5 抑制剂。
T77677 12R-LOX-IN-2

Lipoxygenase Metabolism
12R-LOX-IN-2 是一种 12R-脂氧合酶 (12R-LOX) 的抑制剂。12R-LOX-IN-2 抑制咪喹莫特 (IMQ) 诱导银屑病角质形成细胞过度增殖,并抑制细胞集落形成。12R-LOX-IN-2 还降低 IMQ 诱导细胞中 Ki67 的蛋白水平和 IL-17A 的 mRNA 表达。12R-LOX-IN-2 可用于牛皮癣和其他皮肤相关炎症性疾病的研究。
T38006 LOX-IN-3

Others Others
LOX-IN-3, an orally active inhibitor of lysyl oxidase (LOX), holds potential application in the fields of fibrosis, cancer, and angiogenesis research[1].
T61211 5-LOX-IN-1

Lipoxygenase Metabolism
5-LOX-IN-1 是一种 5-Lipoxygenase(5-LOX)抑制剂(IC50: 2.3 μM)。5-LOX-IN-1 可用于研究癌症。
T36169 15-LOX-1 inhibitor 1

Others Others
9c(i472) is an inhibitor of 15-lipoxygenase-1 (15-LO-1; IC50 = 0.19 μM).1 It decreases LPS- and IFN-γ-induced NF- B activity in RAW-Blue cells when used at concentrations of 0.2, 1, and 5 μM. 9c(i472) reduces LPS- and IFN-γ-induced increases in Nos2 expression and lipid peroxidation in RAW 264.7 cells when used at a concentration of 5 μM.
T83457 12R-LOX-IN-1

Others Others
12R-LOX-IN-1(Compound 4a)是一种效能为IC50: 28.25 μM的12R-LOX抑制剂。该化合物能够有效抑制Imiquimod诱导的银屑病角质形成细胞的异常增殖和集落形成能力,同时减少活性氧、Ki67、IL-17A、TNF-α和IL-6的生成,适用于抗银屑病研究。
T78820 5-LOX-IN-5

Lipoxygenase Metabolism
5-LOX-IN-5(Compound 29)作为一种5-LOX抑制剂,拥有56 nM的半抑制浓度(IC50)。它主要被应用于神经退行性疾病的研究领域。
T8356 FPL 62064

Lipoxygenase; COX Immunology/Inflammation; Metabolism; Neuroscience
FPL 62064 是 5-脂氧合酶和COX 双重抑制剂,具有抗炎活性,对 RBL-1 胞质 5-脂氧合酶和前列腺素合成酶 (环氧化酶) 的IC50值分别为 3.5 和 3.1 μM。
T62350 XO/COX/LOX-IN-1

Others Others
XO/COX/LOX-IN-1 是一种黄嘌呤氧化酶/环氧酶/脂氧合酶 XO/COX/LOX 的有效抑制剂。XO/COX/LOX-IN-1 能够用于研究炎症、癌症以及代谢性疾病。
T79158 h15-LOX-2 inhibitor 1

Lipoxygenase Metabolism
h15-LOX-2 inhibitor 1(Comp 105)是一种针对人上皮细胞15-lipoxygenase-2 (h15-LOX-2)的抑制剂,表现出0.34 μM的IC50值。
T62998 COX-2/15-LOX-IN-1

Others Others
COX-2/15-LOX-IN-1 (Compound 14) 是一种 COX-2 和 15-脂氧合酶 (15-LOX)抑制剂,可作用于 COX-1 (IC50: 10.65 μM)、COX-2 (IC50: 0.075 μM) 和 15-LOX (IC50: 2.98 μM)。COX-2-IN-25 具有抗炎作用。
T4347 ML355

Lipoxygenase Metabolism
ML355 是一种高选择性12-LOX 抑制剂,IC50=0.34 μM,对其他脂氧化酶和环氧化酶有很好的选择性,具有较好的药物动力学特征。
T79360 COX-2/15-LOX-IN-2

Lipoxygenase Metabolism
COX-2/15-LOX-IN-2 作为一种效能高的双重抑制剂,对COX-2和15-LOX的IC50值分别为0.065 μM和1.86 μM,显示出显著的抗氧化活性。
T61674 COX-2/5-LOX-IN-1

Others Others
COX-2/5-LOX-IN-1 (compound 3a), a benzothiophen-2-yl pyrazole carboxylic acid derivative, is a potent and dual inhibitor of COX-2 / 5-LOX. It exhibits superior analgesic and anti-inflammatory properties compared to Celecoxib and Indomethacin. COX-2/5-LOX-IN-1 displays strong inhibitory activity against COX-1, COX-2, and 5-LOX, with IC50 values of 12.13 μM, 0.4 μM, and 4.96 μM, respectively [1].
T60630 COX/5-LOX-IN-1

Others Others
COX/5-LOX-IN-1 (compound 6b) 是有效的COX/5-LOX 双重抑制剂,具有用于炎症性疾病研究的潜力。COX/5-LOX-IN-1 对于 COX-1、COX-2 和 5-LOX 酶的IC50值分别为 1.07、0.55 和 0.28 μM。
T61479 LOX-IN-3 dihydrochloride monohydrate

Others Others
LOX-IN-3 dihydrochloride monohydrate (Compound 33) is a lysyl oxidase (LOX) inhibitor with oral activity. It is specifically designed for research purposes in the areas of fibrosis, cancer, and angiogenesis [1].
T61352 COX-2/5-LOX-IN-3

Others Others
COX-2/5-LOX-IN-3 (compound 5b) is a powerful and dual inhibitor of COX-2 and 5-LOX, with IC50 values of 45.73 μM, 5.45 μM, and 4.33 μM for COX-1, COX-2, and 5-LOX, respectively. This compound, COX-2/5-LOX-IN-3, shows promise for the investigation of inflammatory diseases [1].
T79362 COX-2/15-LOX-IN-4

Lipoxygenase Metabolism
COX-2/15-LOX-IN-4(compound 5i)是一种针对COX-2和15-LOX的双重抑制剂,其IC50值分别为0.075 μM和1.97 μM。该化合物能有效地阻止LPS诱发的细胞内促炎细胞因子(IL-6, ROS)的产生,表现出明确的抗炎活性。
T8950 CAY10698

Lipoxygenase Metabolism
CAY10698 是选择性的12-Lipoxygenase (12-LOX)抑制剂,IC50=5.1 μM。它对 5-LOX、15-LOX-1、15-LOX-2 和 COX-1/2 无活性。
T6243 U-73122

U73122

Phospholipase; Ferroptosis; Lipoxygenase Apoptosis; Metabolism
U-73122 (U73122) 是一种磷脂酶 C 和 5-脂氧合酶抑制剂,对磷脂酶 C 的 IC50值约为 1-2.1 µM。它是一种 PLC 抑制剂,可减少激动剂诱导的血小板和 PMN 中的 Ca2+ 增加。
T61910 COX-2/5-LOX-IN-2

Others Others
COX-2/5-LOX-IN-2 是苯并噻吩-2-基吡唑羧酸衍生物。COX-2/5-LOX-IN-2 (5b) 对COX-2和5-LOX 均有抑制作用。COX-2/5-LOX-IN-2 抑制 COX-1、COX-2 和 5-LOX 的IC50s 分别为 5.40、0.01 和 1.78 μM。COX-2/5-LOX-IN-2 显示出超过塞来昔布和吲哚美辛的镇痛和抗炎活性。
T79361 COX-2/15-LOX-IN-3

Lipoxygenase Metabolism
COX-2/15-LOX-IN-3 (compound 5k) 为COX-2/15-LOX的一种双重抑制剂,具有分别为0.075 μM和1.97 μM的IC50值。该化合物能显著抑制LPS诱导的细胞产生促炎细胞因子(IL-6, ROS和NO),表明其具备显著的抗炎活性。
T9108 BI-0115

Lipoxygenase Metabolism
BI-0115 是LOX-1的选择性抑制剂,其IC50值为 5.4 µM,可以阻止细胞摄取氧化低密度脂蛋白。它通过形成同源二聚体配体结合域的二聚体来触发受体抑制。
T16503 PF-4191834

PF-04191834

Lipoxygenase Metabolism
PF-4191834 是 5-Lipoxygenase (5-LOX) 的非铁螯合和非氧化还原抑制剂,IC50 为 229 nM。 PF-4191834 对 5-LOX 的特异性比 12-LOX 和 15-LOX 高约 300 倍,并且对环氧合酶没有活性。 PF-4191834 可用于炎症和疼痛的研究。
T6568 Licofelone

利克飞龙,ML-3000

Apoptosis; Lipoxygenase; COX Apoptosis; Immunology/Inflammation; Metabolism; Neuroscience
Licofelone (ML-3000) 是一种 COX/LOX 双重抑制剂,IC50分别为 0.21和0.18 μM,有潜力研究骨关节炎,具有抗炎和抗增殖作用。它可诱导细胞凋亡,减少促炎性白三烯和前列腺素的产生。
T21746 Terameprocol

tetramethyl Nordihydroguaiaretic Acid,EM-1421

HIV Protease Microbiology/Virology; Proteases/Proteasome
Terameprocol (EM-1421) 是 Nordihydroguaiaretic acid 的合成衍生物,是非选择性脂氧合酶抑制剂。
T7540 2,5-Di-tert-butylhydroquinone

BHQ,2,5-二特丁基对苯二酚

Calcium Channel; Lipoxygenase; COX Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience
2,5-Di-tert-butylhydroquinone (BHQ) 是一种有效和选择性的内质网 Ca2+-ATPase 抑制剂,可调节5-LO 以及COX-2活性,IC50分别为 1.8 和 14.1 μM。
T10098 PGS-IN-1

KME-4

Lipoxygenase; Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism
PGS-IN-1 (KME-4)是一种前列腺素合成酶抑制剂,IC50=0.28 μM。它也可抑制5-脂肪氧合酶的活性,IC50=1.05 μM。
T27026 CJ-13,610

CJ 13610,CJ-13610

Lipoxygenase Metabolism
CJ-13,610 是一种具有口服活性的非氧化还原型 5-脂氧合酶 (5-LOX) 抑制剂。 CJ-13,610 抑制白三烯 B4 的生物合成并调节巨噬细胞中 IL-6 mRNA 的表达。
T21902 ML351

Lipoxygenase Metabolism
ML351 是一种高度特异的15-LOX-1抑制剂,其 IC50=200 nM。它对 T1D 非肥胖糖尿病小鼠模型的血糖异常和β细胞氧化应激有抑制作用。它对相关同工酶 (5-LOX、血小板 12-LOX、15-LOX-2、绵羊 COX-1 和人 COX-2) 表现出良好的选择性(>250倍)。
T22398 Phenidone

菲尼酮,1-phenyl-3-pyrazolidinone

Lipoxygenase; COX Immunology/Inflammation; Metabolism; Neuroscience
Phenidone (1-phenyl-3-pyrazolidinone) 是可口服发环氧化酶和脂氧合酶双重抑制剂,可改善实验性自身免疫性脑脊髓炎大鼠的瘫痪,降低自发性高血压大鼠的血压,可用作照片显像剂。
T8794 4-MMPB

15-Lipoxygenase Inhibitor 1

Apoptosis; Others; Lipoxygenase Apoptosis; Metabolism; Others
4-MMPB (15-Lipoxygenase Inhibitor 1) 是一种选择性15-脂氧合酶抑制剂,其 IC50值为 18 μM,具有前列腺癌的研究潜力。它对大豆 15-脂氧合酶和人 15-脂氧合酶-1 的 IC50 分别为 19.5 μM 和 19.1 μM。
T0477 Zileuton

Abbott 64077,齐留通,A 64077

Ferroptosis; Lipoxygenase; COX Apoptosis; Immunology/Inflammation; Metabolism; Neuroscience
Zileuton (A 64077) 是羟基脲的合成衍生物,是一种选择性的5-脂氧合酶抑制剂,具有平喘特性。
T6576 Malotilate

Malotilatum,NKK 105,马洛替酯,Kantec

Lipoxygenase Metabolism
Malotilate (Kantec) 是一种抗纤维化物质,是一种口服活性的促肝药,可选择性抑制5-lipoxygenase (5-LOX)(IC50=4.7 μM)。它通过降低肝脏乙醛水平并防止转铁蛋白保留在肝细胞中,从而预防了酒精-吡唑肝炎中肝细胞损伤的发展。
T5200 Indirubin-3'-monoxime

靛玉红-3' -单肟,Indirubin-3'-oxime

GSK-3; Lipoxygenase; CDK Cell Cycle/Checkpoint; Metabolism; PI3K/Akt/mTOR signaling; Stem Cells
Indirubin-3'-monoxime (Indirubin-3'-oxime) 是一种有效的 GSK3β 抑制剂,IC50值为 22 nM。它对 CDK5/p25、CDK1/cyclin B 和CDk2/cyclin E 也有作用,IC50值分别为 100、180 和 250 nM。
T7724 Tepoxalin

RWJ-20485,RWJ20485,ORF20485,替泊沙林,ORF-20485,RWJ 20485,ORF 20485

Lipoxygenase; COX Immunology/Inflammation; Metabolism; Neuroscience
Tepoxalin (RWJ 20485) 是有效的5-脂氧合酶和环氧合酶抑制剂,表现出强大的抗炎活性和较小的胃肠道刺激性。
T6893 MK-886

MK886,L 663536

Apoptosis; Leukotriene Receptor; COX; PPAR; FLAP Apoptosis; DNA Damage/DNA Repair; GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience
MK-886 (L 663536)是一种细胞可渗透的,具有口服活性的 FLAP (IC50为 30 nM) 和白三烯生物合成 (完整白细胞和人全血中的IC50分别为 3 nM 和 1.1μM) 的抑制剂。它也是一种非竞争性PPARα拮抗剂,可以诱导细胞凋亡。
T67908 ThioLox

Lipoxygenase Metabolism
ThioLox 是一种竞争性 15-脂氧合酶-1 (15-LOX-1) 抑制剂(IC50值为12 μM)。ThioLox 显示抗炎和神经保护特性。具有抗炎和神经保护作用,对谷氨酸毒性有很强的保护作用。
T1412 Loxapine succinate

Daxolin,Loxapac,Cloxazepin,Loxapine succinate salt,丁二酸洛沙平,琥珀酸洛沙平

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
Loxapine succinate (Loxapac) 是D2/D4多巴胺受体,5-羟色胺受体抑制剂,用于精神分裂症。
T2312 Loxiglumide

CR-1505,氯谷胺

cholecystokinin GPCR/G Protein
Loxiglumide (CR-1505) 是一种缩胆囊素受体拮抗剂。
T1031 Cloxacillin sodium monohydrate

Cloxacillin Sodium,Bactopen,氯唑西林钠一水合物

Antibacterial; Antibiotic Microbiology/Virology
Cloxacillin sodium monohydrate (Cloxacillin Sodium) 有抗菌作用,对Staphylococcus aureus25923 的最小抑菌浓度为256 mg/L。
T9319 Tosufloxacin

tosufloxacin tosilate,托氟沙星,Ozex,7-(3-Aminopyrrolidin-1-yl)-1-(2,4-difluorophenyl)-6-fluoro-4-oxo-1,8-naphthyridine-3-carboxylic acid

Others Others
Tosufloxacin (Ozex) 是一种喹诺酮类抗菌剂,是茶碱代谢的有效抑制剂。
T15777 Loxoribine

RWJ 21757,7-Allyl-8-oxoguanosine,洛索立宾

Influenza Virus; TLR Immunology/Inflammation; Microbiology/Virology
Loxoribine (RWJ 21757) 是一种鸟苷类似物,是一种口服生物可利用的选择性 Toll 样受体 (TLR) 7 激动剂。 具有抗病毒和抗肿瘤活性。它是一种新型的强效免疫刺激剂,具有较广谱的免疫生物学活性。
T22456 Voreloxin hydrochloride

SNS-595 hydrochloride,Vosaroxin,(3S-反式)-1,4-二氢-7-[3-甲氧基-4-(甲基氨基)-1-吡咯烷基]-4-氧代-1-(2-噻唑基)-1,8-萘啶-3-羧酸单盐酸盐

Apoptosis; Topoisomerase Apoptosis; DNA Damage/DNA Repair
Voreloxin hydrochloride (SNS-595 hydrochloride) 是一种新型拓扑异构酶 II 抑制剂,能够诱导 DNA 双链断裂,阻滞 G2 期,引起细胞凋亡。
T1293 Gatifloxacin

BMS 206584-01,PD 135432,CG5501,BMS-206584,AM-1155,加替沙星

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Gatifloxacin (CG5501) 是一种具有广谱抗菌活性的氟喹诺酮类抗生素。它可抑制大肠杆菌 DNA 解旋酶 (IC50=0.109 μg/ml) 和细菌 II 型拓扑异构酶(IC50=13.8 μg/ml)。在动物模型中,它有抗细菌性结膜炎作用。
T0826 Meloxicam

美洛昔康,Movalis,Mobic,Metacam

Apoptosis; COX; Autophagy Apoptosis; Autophagy; Immunology/Inflammation; Neuroscience
Meloxicam (Metacam) 是一种非甾体类抗炎剂,抑制COX 的活性,对 COX-2 和 COX-1 的IC50值分别为 0.49 µM 和 36.6 µM。
T5323 Toloxatone

托洛沙酮,MD 69276

MAO; Monoamine Oxidase Metabolism; Neuroscience
Toloxatone (MD 69276) 是可逆的单胺氧化酶 A (MAOA) 抑制剂,是一种抗抑郁剂。
T6919 Omaveloxolone

RTA-408

Apoptosis; Others; Nrf2; STING Apoptosis; Immunology/Inflammation; Others
Omaveloxolone (RTA-408) 是一种抗氧化炎症调节剂,可激活Nrf2并抑制一氧化氮。它通过抑制 STING 依赖的 NF-κb 信号通路,来抑制破骨细胞的生成。

化合物

LOX-IN-3 dihydrochloride
Cat.No: T39986
Synonym:
Target: Lipoxygenase
5-LOX-IN-2
Cat.No: T77528
Synonym:
Target: Apoptosis, Lipoxygenase
5-LOX inhibitor
Cat.No: T65427
Synonym: 1-(sec-Butyl)-4-(4-(4-(4-hydroxyphenyl)piperazin-1-yl)phenyl)-1H-1,2,4-triazol-5(4H)-one
Target: Lipoxygenase
12R-LOX-IN-2
Cat.No: T77677
Synonym:
Target: Lipoxygenase
LOX-IN-3
Cat.No: T38006
Synonym:
Target: Others
5-LOX-IN-1
Cat.No: T61211
Synonym:
Target: Lipoxygenase
15-LOX-1 inhibitor 1
Cat.No: T36169
Synonym:
Target: Others
12R-LOX-IN-1
Cat.No: T83457
Synonym:
Target: Others
5-LOX-IN-5
Cat.No: T78820
Synonym:
Target: Lipoxygenase
FPL 62064
Cat.No: T8356
Synonym:
Target: Lipoxygenase, COX
XO/COX/LOX-IN-1
Cat.No: T62350
Synonym:
Target: Others
h15-LOX-2 inhibitor 1
Cat.No: T79158
Synonym:
Target: Lipoxygenase
COX-2/15-LOX-IN-1
Cat.No: T62998
Synonym:
Target: Others
ML355
Cat.No: T4347
Synonym:
Target: Lipoxygenase
COX-2/15-LOX-IN-2
Cat.No: T79360
Synonym:
Target: Lipoxygenase
COX-2/5-LOX-IN-1
Cat.No: T61674
Synonym:
Target: Others
COX/5-LOX-IN-1
Cat.No: T60630
Synonym:
Target: Others
LOX-IN-3 dihydrochloride monohydrate
Cat.No: T61479
Synonym:
Target: Others
COX-2/5-LOX-IN-3
Cat.No: T61352
Synonym:
Target: Others
COX-2/15-LOX-IN-4
Cat.No: T79362
Synonym:
Target: Lipoxygenase
CAY10698
Cat.No: T8950
Synonym:
Target: Lipoxygenase
U-73122
Cat.No: T6243
Synonym: U73122
Target: Phospholipase, Ferroptosis, Lipoxygenase
COX-2/5-LOX-IN-2
Cat.No: T61910
Synonym:
Target: Others
COX-2/15-LOX-IN-3
Cat.No: T79361
Synonym:
Target: Lipoxygenase
BI-0115
Cat.No: T9108
Synonym:
Target: Lipoxygenase
PF-4191834
Cat.No: T16503
Synonym: PF-04191834
Target: Lipoxygenase
Licofelone
Cat.No: T6568
Synonym: 利克飞龙,ML-3000
Target: Apoptosis, Lipoxygenase, COX
Terameprocol
Cat.No: T21746
Synonym: tetramethyl Nordihydroguaiaretic Acid,EM-1421
Target: HIV Protease
2,5-Di-tert-butylhydroquinone
Cat.No: T7540
Synonym: BHQ,2,5-二特丁基对苯二酚
Target: Calcium Channel, Lipoxygenase, COX
PGS-IN-1
Cat.No: T10098
Synonym: KME-4
Target: Lipoxygenase, Prostaglandin Receptor
CJ-13,610
Cat.No: T27026
Synonym: CJ 13610,CJ-13610
Target: Lipoxygenase
ML351
Cat.No: T21902
Synonym:
Target: Lipoxygenase
Phenidone
Cat.No: T22398
Synonym: 菲尼酮,1-phenyl-3-pyrazolidinone
Target: Lipoxygenase, COX
4-MMPB
Cat.No: T8794
Synonym: 15-Lipoxygenase Inhibitor 1
Target: Apoptosis, Others, Lipoxygenase
Zileuton
Cat.No: T0477
Synonym: Abbott 64077,齐留通,A 64077
Target: Ferroptosis, Lipoxygenase, COX
Malotilate
Cat.No: T6576
Synonym: Malotilatum,NKK 105,马洛替酯,Kantec
Target: Lipoxygenase
Indirubin-3'-monoxime
Cat.No: T5200
Synonym: 靛玉红-3' -单肟,Indirubin-3'-oxime
Target: GSK-3, Lipoxygenase, CDK
Tepoxalin
Cat.No: T7724
Synonym: RWJ-20485,RWJ20485,ORF20485,替泊沙林,ORF-20485,RWJ 20485,ORF 20485
Target: Lipoxygenase, COX
MK-886
Cat.No: T6893
Synonym: MK886,L 663536
Target: Apoptosis, Leukotriene Receptor, COX, PPAR, FLAP
ThioLox
Cat.No: T67908
Synonym:
Target: Lipoxygenase
Loxapine succinate
Cat.No: T1412
Synonym: Daxolin,Loxapac,Cloxazepin,Loxapine succinate salt,丁二酸洛沙平,琥珀酸洛沙平
Target: Dopamine Receptor, 5-HT Receptor
Loxiglumide
Cat.No: T2312
Synonym: CR-1505,氯谷胺
Target: cholecystokinin
Cloxacillin sodium monohydrate
Cat.No: T1031
Synonym: Cloxacillin Sodium,Bactopen,氯唑西林钠一水合物
Target: Antibacterial, Antibiotic
Tosufloxacin
Cat.No: T9319
Synonym: tosufloxacin tosilate,托氟沙星,Ozex,7-(3-Aminopyrrolidin-1-yl)-1-(2,4-difluorophenyl)-6-fluoro-4-oxo-1,8-naphthyridine-3-carboxylic acid
Target: Others
Loxoribine
Cat.No: T15777
Synonym: RWJ 21757,7-Allyl-8-oxoguanosine,洛索立宾
Target: Influenza Virus, TLR
Voreloxin hydrochloride
Cat.No: T22456
Synonym: SNS-595 hydrochloride,Vosaroxin,(3S-反式)-1,4-二氢-7-[3-甲氧基-4-(甲基氨基)-1-吡咯烷基]-4-氧代-1-(2-噻唑基)-1,8-萘啶-3-羧酸单盐酸盐
Target: Apoptosis, Topoisomerase
Gatifloxacin
Cat.No: T1293
Synonym: BMS 206584-01,PD 135432,CG5501,BMS-206584,AM-1155,加替沙星
Target: Topoisomerase, Antibacterial, Antibiotic
Meloxicam
Cat.No: T0826
Synonym: 美洛昔康,Movalis,Mobic,Metacam
Target: Apoptosis, COX, Autophagy
Toloxatone
Cat.No: T5323
Synonym: 托洛沙酮,MD 69276
Target: MAO, Monoamine Oxidase
Omaveloxolone
Cat.No: T6919
Synonym: RTA-408
Target: Apoptosis, Others, Nrf2, STING
Cat. No. Product Name Target Signaling Pathways
T6S0413 Pectolinarigenin

柳穿鱼黄素,Pectolinaringenin

Others; Lipoxygenase; COX Immunology/Inflammation; Metabolism; Neuroscience; Others
Pectolinarigenin (Pectolinaringenin) 是 COX-2/5-LOX 的双重抑制剂,可抑制炎症病变中类花生酸的形成,具有抗炎活性。
T3399 Psoralidin

Others; Estrogen/progestogen Receptor; Reactive Oxygen Species; Lipoxygenase; Gamma-secretase; Akt; COX; Antibacterial Cytoskeletal Signaling; Endocrinology/Hormones; Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience; NF-κB; Others; PI3K/Akt/mTOR signaling; Proteases/Proteasome; Stem Cells
Psoralidin 是COX-2和5-LOX 的抑制剂,有抗癌,抗菌和抗炎作用。它显著下调NOTCH1信号传导,还极大地诱导活化氧产生。
T8260 4',5-Dihydroxyflavone

Lipoxygenase; Glucosidase Metabolism
4',5-Dihydroxyflavone 是大豆 LOX-1,Ki=102.6 μM。它也是一种酵母 α-葡萄糖苷酶抑制剂,IC50=66 μM。
TQ0180 Chebulagic acid

SARS-CoV; Influenza Virus; Lipoxygenase; COX Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience
Chebulagic acid 是从 Terminalia chebula Retz 中分离出来的一种 COX-LOX 双重抑制剂,有抗炎和抗感染作用。它抑制 SARS-CoV-2病毒的复制,EC50值为 9.76 μM。它还是 M2(S31N)抑制剂和抗流感病毒剂。
T8002 3-Hydroxycoumarin

Lipoxygenase Metabolism
3-hydroxycoumarin 是一种 15-LOX-1的有效氧化还原抑制剂,近期被证明能保护海胆生殖细胞免受紫外线 B 的损伤。
T2807 Caffeic Acid

Lipoxygenase; Endogenous Metabolite; TRP/TRPV Channel Membrane transporter/Ion channel; Metabolism
Caffeic acid 是5-脂氧合酶和 TRPV1离子通道的双重抑制剂。
TN5634 Aureusidin

Auresudidin,金鱼草素,Auresidin

Antioxidant; Reactive Oxygen Species; Lipoxygenase Immunology/Inflammation; Metabolism; NF-κB; oxidation-reduction
Aureusidin (Auresidin) 具有抗氧化和脂氧合酶抑制活性,具有抗炎作用。
TN2330 Phenethyl ferulate

Caffeic Acid 3-Methyl Phenethyl Ester,阿魏酸苯乙酯,阿魏酸苯乙醇酯

Lipoxygenase; COX Immunology/Inflammation; Metabolism; Neuroscience
Phenethyl ferulate (Caffeic Acid 3-Methyl Phenethyl Ester) 对化学诱导的结肠癌具有化学预防特性,可增强偶氮甲烷诱导的结肠肿瘤的细胞凋亡。 它抑制环氧合酶(COX) 和 5-脂氧合酶 (5-LOX) ,IC50 值分别为 4.35 和 5.75 μM。
T5714 5-O-Demethylnobiletin

5-DEMETHYLNOBILETIN,去甲基川陈皮素

Leukotriene Receptor; Lipoxygenase GPCR/G Protein; Metabolism
5-O-Demethylnobiletin (5-DEMETHYLNOBILETIN) 是从黄芪中分离出的多甲氧基黄酮,具有抗炎活性,可通过直接抑制 5-LOX 发挥作用,IC50为 0.1 μM。
T5759 S-(+)-Marmesin

(+)-Marmesin,异紫花前胡内酯,(S)-Marmesin,marmesin

Lipoxygenase; COX Immunology/Inflammation; Metabolism; Neuroscience
S-(+)-Marmesin (marmesin) 是一种从木橘成熟树皮中分离得到的香豆素,具有 COX-2/5-LOX 双重抑制活性。
TJS2190 Nordihydroguaiaretic acid

去甲二氢愈创木酸,NDGA,Dihydronorguaiaretic Acid

Antioxidant; Ferroptosis; Lipoxygenase; Autophagy Apoptosis; Autophagy; Metabolism; oxidation-reduction
Nordihydroguaiaretic acid (NDGA) 是从极叉开拉瑞阿提取出的一种天然产物,是脂氧合酶抑制剂,具有抗氧化和清除自由基的特性。
T3S0153 Xanthatin

苍耳亭,叶黄制菌素

Apoptosis; VEGFR; Lipoxygenase; Wnt/beta-catenin; Antibacterial Angiogenesis; Apoptosis; Cytoskeletal Signaling; Metabolism; Microbiology/Virology; Stem Cells; Tyrosine Kinase/Adaptors
Xanthatin 是一种从Xanthium strumarium 叶子中提取的天然产物,可诱导细胞凋亡。它抑制布鲁氏菌的IC50值为 2.63 μg/ mL,对寄生虫特异性锥虫硫磷还原酶具有不可逆的弱抑制作用。它通过抑制PGE2的合成和 5-脂氧合酶的活性而显示出抗炎活性。
TN1097 β-Boswellic acid

Beta-boswellic acid,β-乳香酸

Lipoxygenase; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism
β-Boswellic acid (Beta-boswellic acid) 是从乳香的树胶脂中分离出来的一种天然产物。它是 5-脂氧合酶(5-LO) 产物形成的非还原型抑制剂,其直接与 5-LO 相互作用或阻断其易位。具有抗癌、抗肿瘤和抗高血脂活性。
T3384 Wedelolactone

蟛蜞菊内酯,IKK Inhibitor II

Apoptosis; NF-κB; Lipoxygenase; Caspase Apoptosis; Metabolism; NF-κB; Proteases/Proteasome
Wedelolactone (IKK Inhibitor II) 是来自旱莲草的一种天然产物,通过阻断 IκBα 的磷酸化和降解来抑制细胞中 NF-κB 介导的基因转录,具有抗癌,抗炎和抗氧化活性。
TN1255 3-O-Acetyl-11-hydroxy-beta-boswellic acid

Lipoxygenase Metabolism
3-O-Acetyl-11-hydroxy-beta-boswellic acid 是 5-脂氧合酶抑制剂。
TN1182 11-​Keto-​beta-​boswellic acid

11-Keto-beta-boswellic acid,11-酮基-BETA-乳香酸

Leukotriene Receptor; NF-κB; Lipoxygenase GPCR/G Protein; Metabolism; NF-κB
11-Keto-beta-boswellic acid 是来自乳香的一种五环三萜酸,具有抗炎活性和剂量依赖性心脏保护作用,主要是由于抑制5-脂氧合酶、白三烯、NF-κB 的激活和肿瘤坏死因子 α 的产生。
T6567 Levofloxacin

Levaquin,Cravit,Tavanic,Fluoroquinolone,左氧氟沙星,(-)-Ofloxacin

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Levofloxacin (Fluoroquinolone) 是合成的氟喹诺酮类抗生素,有抑制细菌DNA 旋转酶的超螺旋活性的作用,能阻止DNA 复制。
T1121 Podofilox

鬼臼毒素,Podophyllotoxin,(+)-Shikonin

Microtubule Associated; Topoisomerase Cytoskeletal Signaling; DNA Damage/DNA Repair
Podofilox ((+)-Shikonin) 是从八角莲中分离的一种木脂素,是微管组装和 DNA 拓扑异构酶 II 抑制剂。它对皮肤和粘膜有很强的刺激性,具有角质溶解作用,可用于治疗疣和角化病,具有潜在的抗肿瘤特性。
T1276 Danofloxacin mesylate

甲磺酸达氟沙星,CP 76136-27

DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Danofloxacin mesylate (CP 76136-27) 是一种兽医用氟喹诺酮类抗菌素。
T4S1658 Benzoyloxypaeoniflorin

苯甲酰氧化芍药苷,Benzoyloxypeoniflorin,苯甲酰氧芍药苷

NF-κB; Tyrosinase NF-κB; Proteases/Proteasome
Benzoyloxypaeoniflorin (Benzoyloxypeoniflorin) 是一种酪氨酸酶抑制剂,分离于Paeonia suffruticosa 的根,对mushroom tyrosinase 的 IC50为 0.453 mM。它是一种NF-κB 抑制剂,它通过对血小板聚集和凝血的抑制作用,有助于改善血液循环。
TN1343 8-Geranyloxypsoralen

8-香叶草氧基补骨脂素

Anti-infection; P450; BACE Metabolism; Microbiology/Virology; Neuroscience
8-Geranyloxypsoralen 是一种呋喃香豆素,分离自葡萄柚,是 P450 3A4 的有效抑制剂(IC50:3.93 μM)。
T5744 7-Prenyloxycoumarin

7-(异戊烯基氧基)香豆素,Nsc267697,7-O-Prenylumbelliferone,7-异戊烯氧基香豆素

Antifungal Microbiology/Virology
7-Prenyloxycoumarin (Nsc267697) 是一种 Heracleum dissectum 的天然产物,对乳腺癌具有预防和治疗作用。
T1549 Raloxifene hydrochloride

LY156758 hydrochloride,盐酸雷洛昔芬,Raloxifene HCl,LY139481 hydrochloride,Keoxifene hydrochloride,LY156758 (Keoxifene) HCl

Estrogen Receptor/ERR; Others; MAO; Estrogen/progestogen Receptor; Autophagy Autophagy; Endocrinology/Hormones; Metabolism; Neuroscience; Others
Raloxifene hydrochloride (LY156758 hydrochloride) 是一种选择性且可口服的雌激素受体调节剂,用于预防绝经后妇女的骨质疏松症。它对骨骼和胆固醇代谢具有雌激素激动作用,但对乳腺和子宫组织具有完全的雌激素拮抗作用。
T8384 Gatifloxacin hydrochloride

AM-1155 (hydrochloride),BMS-206584 (hydrochloride),PD135432 (hydrochloride),加替沙星盐酸盐

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Gatifloxacin hydrochloride (AM-1155 hydrochloride) 是一种氟喹诺酮类抗生素,有广谱抗菌活性。它可抑制大肠杆菌 DNA 解旋酶 (IC50=0.109 μg/ml)和细菌 II 型拓扑异构酶(IC50=13.8 μg/ml) 。它在动物模型中,可研究细菌性结膜炎。
T8130 Ciprofloxacin hydrochloride monohydrate

Oftacilox,Ciprofloxacin hydrochloride hydrate,Bay-09867 hydrochloride monohydrate,环丙沙星盐酸盐一水合物,Ceprimax,盐酸环丙沙星(一水物),Ciloxan

Antibacterial; Antibiotic Microbiology/Virology
Ciprofloxacin hydrochloride monohydrate (Bay-09867 hydrochloride monohydrate) 是一种具有高效抗菌活性的氟喹诺酮类抗生素。
TN1025 3,29-O-Dibenzoyloxykarounidiol

Others Others
3,29-O-Dibenzoyloxykarounidiol 是一种苯甲酸三萜烯酯,从 Momordica grosvenori 果实中提取。它能够抑制肿瘤启动子 TPA 诱导的 EB 病毒早期抗原活化。
T8046 Tosufloxacin tosylate hydrate

Tosufloxacin p-Toluenesulfonate Hydrate,A-61827 tosylate hydrate,对甲苯磺酸妥舒沙星水合物,T-3262 Tosylate Hydrate

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Tosufloxacin tosylate hydrate (A-61827 tosylate hydrate) 是一个氟喹诺酮类抗菌剂。
T1306 Norfloxacin

氟哌酸,MK-0366,诺氟沙星

DNA gyrase; Topoisomerase; Endogenous Metabolite; Antibacterial; Antibiotic DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Norfloxacin (MK-0366) 是广谱抗生素,能通过结合DNA 旋转酶抑制革兰氏阳性和阴性菌。
TN5613 3α-Cinnamoyloxy-9β,17-dihydroxy-ent-kaur-15-en-19-oic acid

ent-3β-Cinnamoyloxy-9α,17-dihydroxykaur-15-en-19-oic acid

3α-Cinnamoyloxy-9β,17-dihydroxy-ent-kaur-15-en-19-oic acid 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5613,CAS号为 2186648-60-0。
TN5303 14β,16β-Dihydroxy-3β-(β-D-glucopyranosyloxy)-5α-bufa-20,22-dienolide

14β,16β-Dihydroxy-3β-(β-D-glucopyranosyloxy)-5α-bufa-20,22-dienolide 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5303,CAS号为 1323952-04-0。
TN5555 7α-Galloyloxysweroside

7α-Galloyloxysweroside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5555,CAS号为 2222365-76-4。
TN5683 Ethyl 4-(rhamnosyloxy)benzylcarbamate

Ethyl 4-(rhamnosyloxy)benzylcarbamate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5683,CAS号为 208346-80-9。
T83233 8-Hydroxy-9-isobutyryloxy-10-(2-methylbutanoyl)thymol

8-Hydroxy9,10-diisobutyryloxy-thymol 是从Inula sericophylla中提取的有效萜类化合物。
T83516 (Z)-2-Angeloyloxymethyl-2-butenoic

(Z)-2-Angeloyloxymethyl-2-butenoic acid 是 An anthriscus sylvestris Hoffm. 根部的一种天然产物。
T83558 (3S,4aS,10aS)-3-(Acetyloxy)-2,3,4,4a,10,10a-hexahydro-6-hydroxy-1,1,4a-trimethyl-7-(1-methylethyl)-9(1H)-phenanthrenone

(3S,4aS,10aS)-3-(Acetyloxy)-2,3,4,4a,10,10a-hexahydro-6-hydroxy-1,1,4a-trimethyl-7-(1-methylethyl)-9(1H)-phenanthrenone(化合物3)是从丹参(Salvia miltiorrhiza)根提取的棕榈酸盐。该化合物展现出抗癌活性,对于不同的人类癌症细胞系具有显著的抑制效果,其DC50值分别为:HeLa细胞系25.5 μg/mL、HepG2细胞系37.5 μg/mL以及OVCAR-3细胞系30.2 μg/mL。
TN2938 3-Hydroxy-3-acetonyloxindole

Others Others
3-Hydroxy-3-acetonyloxindole是一种天然产物,属于萝藦科牛奶菜属,其产品编号为 TN2938,CAS号为 33417-17-3。3-Hydroxy-3-acetonyloxindole可用作对照参考。
TN3294 8alpha-(2-Methylacryloyloxy)hirsutinolide 13-O-acetate

NADPH-oxidase; P450; MAO Immunology/Inflammation; Metabolism; Neuroscience
8alpha-(2-Methylacryloyloxy)hirsutinolide 13-O-acetate shows inhibitory activity toward CYP2A6 and MAO-A and MAO-B enzymes.
TN5862 8-Hydroxy-9,10-diisobutyryloxythymol

8-Hydroxy-9,10-diisobutyryloxythymol 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5862,CAS号为 22518-08-7。
TN3302 8 beta-(4-Acetoxy-5-hydroxytigloyloxy)costunolide

Others Others
8 beta-(4-Acetoxy-5-hydroxytigloyloxy)costunolide 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3302,CAS号为 109770-86-7。
TN3301 8beta-(2-Hydroxy-2-methyl-3-oxobutyryloxy)glucozaluzanin C

Others Others
8beta-(2-Hydroxy-2-methyl-3-oxobutyryloxy)glucozaluzanin C 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3301,CAS号为 93395-31-4。
TN2627 14beta-Benzoyloxy-2-deacetylbaccatin VI

Others Others
14beta-Benzoyloxy-2-deacetylbaccatin VI是一种天然产物,属于红豆杉科红豆杉属,其产品编号为 TN2627,CAS号为 705973-69-9。14beta-Benzoyloxy-2-deacetylbaccatin VI可用作对照参考。
T38658 3-(β-D-Glucopyranosyloxy)-1,6-dihydroxy-2-methyl-9,10-anthracenedione

Others Others
3-(β-D-Glucopyranosyloxy)-1,6-dihydroxy-2-methyl-9,10-anthracenedione, also known as an anthraquinone, has been specifically extracted from Rubia cordifolia.
T38657 2-Naphthalenecarboxylic acid, 4-(D-glucopyranosyloxy)-1-hydroxy-3-(3-hydroxy-3-methylbutyl)-, methyl ester

Others Others
2-Naphthalenecarboxylic acid, 4-(D-glucopyranosyloxy)-1-hydroxy-3-(3-hydroxy-3-methylbutyl)-, methyl ester (compound 3) is a naturally occurring substance found in the dried roots of Rubia cordifolia.
TN6331 3β-(4-Hydroxybenzoyloxy)-21β,29-dihydroxyserrat-14-en-24-oic acid

3β-(4-Hydroxybenzoyloxy)-21β,29-dihydroxyserrat-14-en-24-oic acid 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6331,CAS号为 1217268-13-7。
TN6207 7-(6'R-hydroxy-3',7'-dimethylocta-2',7'-dienyloxy)coumarin

7-(6'R-hydroxy-3',7'-dimethylocta-2',7'-dienyloxy)coumarin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6207,CAS号为 118584-19-3。
TN5375 1β,10β-Epoxy-6β-isobutyryloxy-9-oxofuranoeremophilane

1beta,10beta-Epoxy-6beta-isobutyryloxy-9-oxofuranoeremophilane is a natural product from Ligularia fischeri.
TN3277 8-Geranyloxy-5,7-dimethoxycoumarin

Others Others
8-Geranyloxy-5,7-dimethoxycoumarin是一种天然产物,属于芸香科飞龙掌血属,其产品编号为 TN3277,CAS号为 1228175-65-2。8-Geranyloxy-5,7-dimethoxycoumarin可用作对照参考。
TN2987 3Alaph-Tigloyloxypterokaurene L3

Others Others
3Alaph-Tigloyloxypterokaurene L3 is a natural product from Wedelia trilobata.
TN3295 8alpha-(2-Methylacryloyloxy)hirsutinolide

Others Others
8alpha-(2-Methylacryloyloxy)hirsutinolide 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3295,CAS号为 188293-70-1。
TN2849 3-(2-Glucosyloxy-4-methoxyphenyl)propanoic acid

Antifection Microbiology/Virology
2-O-beta-d-Glucosyloxy-4-methoxybenzenepropanoic acid[3-(2-Glucosyloxy-4-methoxyphenyl)propanoic acid] exhibits glutathione S-transferase (GST) inhibitory and antifungal activities.
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天然产物

Pectolinarigenin
Cat.No: T6S0413
Synonym: 柳穿鱼黄素,Pectolinaringenin
Target: Others, Lipoxygenase, COX
Psoralidin
Cat.No: T3399
Synonym:
Target: Others, Estrogen/progestogen Receptor, Reactive Oxygen Species, Lipoxygenase, Gamma-secretase, Akt, COX, Antibacterial
4',5-Dihydroxyflavone
Cat.No: T8260
Synonym:
Target: Lipoxygenase, Glucosidase
Chebulagic acid
Cat.No: TQ0180
Synonym:
Target: SARS-CoV, Influenza Virus, Lipoxygenase, COX
3-Hydroxycoumarin
Cat.No: T8002
Synonym:
Target: Lipoxygenase
Caffeic Acid
Cat.No: T2807
Synonym:
Target: Lipoxygenase, Endogenous Metabolite, TRP/TRPV Channel
Aureusidin
Cat.No: TN5634
Synonym: Auresudidin,金鱼草素,Auresidin
Target: Antioxidant, Reactive Oxygen Species, Lipoxygenase
Phenethyl ferulate
Cat.No: TN2330
Synonym: Caffeic Acid 3-Methyl Phenethyl Ester,阿魏酸苯乙酯,阿魏酸苯乙醇酯
Target: Lipoxygenase, COX
5-O-Demethylnobiletin
Cat.No: T5714
Synonym: 5-DEMETHYLNOBILETIN,去甲基川陈皮素
Target: Leukotriene Receptor, Lipoxygenase
S-(+)-Marmesin
Cat.No: T5759
Synonym: (+)-Marmesin,异紫花前胡内酯,(S)-Marmesin,marmesin
Target: Lipoxygenase, COX
Nordihydroguaiaretic acid
Cat.No: TJS2190
Synonym: 去甲二氢愈创木酸,NDGA,Dihydronorguaiaretic Acid
Target: Antioxidant, Ferroptosis, Lipoxygenase, Autophagy
Xanthatin
Cat.No: T3S0153
Synonym: 苍耳亭,叶黄制菌素
Target: Apoptosis, VEGFR, Lipoxygenase, Wnt/beta-catenin, Antibacterial
β-Boswellic acid
Cat.No: TN1097
Synonym: Beta-boswellic acid,β-乳香酸
Target: Lipoxygenase, DNA/RNA Synthesis
Wedelolactone
Cat.No: T3384
Synonym: 蟛蜞菊内酯,IKK Inhibitor II
Target: Apoptosis, NF-κB, Lipoxygenase, Caspase
3-O-Acetyl-11-hydroxy-beta-boswellic acid
Cat.No: TN1255
Synonym:
Target: Lipoxygenase
11-​Keto-​beta-​boswellic acid
Cat.No: TN1182
Synonym: 11-Keto-beta-boswellic acid,11-酮基-BETA-乳香酸
Target: Leukotriene Receptor, NF-κB, Lipoxygenase
Levofloxacin
Cat.No: T6567
Synonym: Levaquin,Cravit,Tavanic,Fluoroquinolone,左氧氟沙星,(-)-Ofloxacin
Target: Topoisomerase, Antibacterial, Antibiotic
Podofilox
Cat.No: T1121
Synonym: 鬼臼毒素,Podophyllotoxin,(+)-Shikonin
Target: Microtubule Associated, Topoisomerase
Danofloxacin mesylate
Cat.No: T1276
Synonym: 甲磺酸达氟沙星,CP 76136-27
Target: DNA/RNA Synthesis, Antibacterial, Antibiotic
Benzoyloxypaeoniflorin
Cat.No: T4S1658
Synonym: 苯甲酰氧化芍药苷,Benzoyloxypeoniflorin,苯甲酰氧芍药苷
Target: NF-κB, Tyrosinase
8-Geranyloxypsoralen
Cat.No: TN1343
Synonym: 8-香叶草氧基补骨脂素
Target: Anti-infection, P450, BACE
7-Prenyloxycoumarin
Cat.No: T5744
Synonym: 7-(异戊烯基氧基)香豆素,Nsc267697,7-O-Prenylumbelliferone,7-异戊烯氧基香豆素
Target: Antifungal
Raloxifene hydrochloride
Cat.No: T1549
Synonym: LY156758 hydrochloride,盐酸雷洛昔芬,Raloxifene HCl,LY139481 hydrochloride,Keoxifene hydrochloride,LY156758 (Keoxifene) HCl
Target: Estrogen Receptor/ERR, Others, MAO, Estrogen/progestogen Receptor, Autophagy
Gatifloxacin hydrochloride
Cat.No: T8384
Synonym: AM-1155 (hydrochloride),BMS-206584 (hydrochloride),PD135432 (hydrochloride),加替沙星盐酸盐
Target: Topoisomerase, Antibacterial, Antibiotic
Ciprofloxacin hydrochloride monohydrate
Cat.No: T8130
Synonym: Oftacilox,Ciprofloxacin hydrochloride hydrate,Bay-09867 hydrochloride monohydrate,环丙沙星盐酸盐一水合物,Ceprimax,盐酸环丙沙星(一水物),Ciloxan
Target: Antibacterial, Antibiotic
3,29-O-Dibenzoyloxykarounidiol
Cat.No: TN1025
Synonym:
Target: Others
Tosufloxacin tosylate hydrate
Cat.No: T8046
Synonym: Tosufloxacin p-Toluenesulfonate Hydrate,A-61827 tosylate hydrate,对甲苯磺酸妥舒沙星水合物,T-3262 Tosylate Hydrate
Target: Others, Antibacterial, Antibiotic
Norfloxacin
Cat.No: T1306
Synonym: 氟哌酸,MK-0366,诺氟沙星
Target: DNA gyrase, Topoisomerase, Endogenous Metabolite, Antibacterial, Antibiotic
3α-Cinnamoyloxy-9β,17-dihydroxy-ent-kaur-15-en-19-oic acid
Cat.No: TN5613
Synonym: ent-3β-Cinnamoyloxy-9α,17-dihydroxykaur-15-en-19-oic acid
Target:
14β,16β-Dihydroxy-3β-(β-D-glucopyranosyloxy)-5α-bufa-20,22-dienolide
Cat.No: TN5303
Synonym:
Target:
7α-Galloyloxysweroside
Cat.No: TN5555
Synonym:
Target:
Ethyl 4-(rhamnosyloxy)benzylcarbamate
Cat.No: TN5683
Synonym:
Target:
8-Hydroxy-9-isobutyryloxy-10-(2-methylbutanoyl)thymol
Cat.No: T83233
Synonym:
Target:
(Z)-2-Angeloyloxymethyl-2-butenoic
Cat.No: T83516
Synonym:
Target:
(3S,4aS,10aS)-3-(Acetyloxy)-2,3,4,4a,10,10a-hexahydro-6-hydroxy-1,1,4a-trimethyl-7-(1-methylethyl)-9(1H)-phenanthrenone
Cat.No: T83558
Synonym:
Target:
3-Hydroxy-3-acetonyloxindole
Cat.No: TN2938
Synonym:
Target: Others
8alpha-(2-Methylacryloyloxy)hirsutinolide 13-O-acetate
Cat.No: TN3294
Synonym:
Target: NADPH-oxidase, P450, MAO
8-Hydroxy-9,10-diisobutyryloxythymol
Cat.No: TN5862
Synonym:
Target:
8 beta-(4-Acetoxy-5-hydroxytigloyloxy)costunolide
Cat.No: TN3302
Synonym:
Target: Others
8beta-(2-Hydroxy-2-methyl-3-oxobutyryloxy)glucozaluzanin C
Cat.No: TN3301
Synonym:
Target: Others
14beta-Benzoyloxy-2-deacetylbaccatin VI
Cat.No: TN2627
Synonym:
Target: Others
3-(β-D-Glucopyranosyloxy)-1,6-dihydroxy-2-methyl-9,10-anthracenedione
Cat.No: T38658
Synonym:
Target: Others
2-Naphthalenecarboxylic acid, 4-(D-glucopyranosyloxy)-1-hydroxy-3-(3-hydroxy-3-methylbutyl)-, methyl ester
Cat.No: T38657
Synonym:
Target: Others
3β-(4-Hydroxybenzoyloxy)-21β,29-dihydroxyserrat-14-en-24-oic acid
Cat.No: TN6331
Synonym:
Target:
7-(6'R-hydroxy-3',7'-dimethylocta-2',7'-dienyloxy)coumarin
Cat.No: TN6207
Synonym:
Target:
1β,10β-Epoxy-6β-isobutyryloxy-9-oxofuranoeremophilane
Cat.No: TN5375
Synonym:
Target:
8-Geranyloxy-5,7-dimethoxycoumarin
Cat.No: TN3277
Synonym:
Target: Others
3Alaph-Tigloyloxypterokaurene L3
Cat.No: TN2987
Synonym:
Target: Others
8alpha-(2-Methylacryloyloxy)hirsutinolide
Cat.No: TN3295
Synonym:
Target: Others
3-(2-Glucosyloxy-4-methoxyphenyl)propanoic acid
Cat.No: TN2849
Synonym:
Target: Antifection
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Cat. No. Product Name Species Expression System
TMPH-01968 LOX Protein, Human, Recombinant (His & MBP)

LOX,Protein-lysine 6-oxidase,Lysyl oxidase

Human Baculovirus Insect Cells
LOX Protein, Human, Recombinant (His & MBP) is expressed in Baculovirus.
TMPH-03359 LOX Protein, Rat, Recombinant (His)

Lysyl oxidase,Protein-lysine 6-oxidase,Lox

Rat E. coli
Responsible for the post-translational oxidative deamination of peptidyl lysine residues in precursors to fibrous collagen and elastin. Regulator of Ras expression. May play a role in tumor suppression. Plays a role in the aortic wall architecture. LOX Protein, Rat, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 33.0 kDa and the accession number is P16636.
TMPH-02863 LOX Protein, Mouse, Recombinant (His & Myc)

Ras excision protein,Protein-lysine 6-oxidase,Lysyl oxidase,...

Mouse Baculovirus Insect Cells
Responsible for the post-translational oxidative deamination of peptidyl lysine residues in precursors to fibrous collagen and elastin. Regulator of Ras expression. May play a role in tumor suppression. Plays a role in the aortic wall architecture.
TMPH-01969 LOX Protein, Human, Recombinant (His & Myc & SUMO)

Protein-lysine 6-oxidase,LOX,Lysyl oxidase

Human E. coli
Responsible for the post-translational oxidative deamination of peptidyl lysine residues in precursors to fibrous collagen and elastin. Regulator of Ras expression. May play a role in tumor suppression. Plays a role in the aortic wall architecture. LOX Protein, Human, Recombinant (His & Myc & SUMO) is expressed in E. coli expression system with N-10xHis-SUMO and C-Myc tag. The predicted molecular weight is 49.0 kDa and the accession number is P28300.
TMPK-01168 LOX-1 Protein, Mouse, Recombinant (His)

LOXIN,LOX-1,CLEC8A,Ox-LDL receptor 1,S...

Mouse HEK293 Cells
LOX-1 is a transmembrane glycoprotein that binds to and internalizes ox-LDL.LOX-1 gene deletion in mice and anti-LOX-1 therapy has been shown to decrease inflammation, oxidative stress and atherosclerosis. LOX-1 deletion also results in damage from ischemia, making LOX-1 a promising target of therapy for atherosclerosis and related disorders. In this article we focus on the different mechanisms for regulation, signaling and the various effects of LOX-1 in contributing to atherosclerosis.
TMPY-02490 LOX-1 Protein, Human, Recombinant (His)

LOXIN,SCARE1,SLOX1,LOX1,OLR1,oxid...

Human HEK293 Cells
LOX-1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26.5 kDa and the accession number is P78380.
TMPY-03553 15 Lipoxygenase 2 Protein, Human, Recombinant

arachidonate 15-lipoxygenase, type B,ALOX15B,15-

Human Baculovirus Insect Cells
15 Lipoxygenase 2 Protein, Human, Recombinant is expressed in Baculovirus insect cells. The predicted molecular weight is 76 kDa and the accession number is AAH35217.1.
TMPY-03462 15 Lipoxygenase 2 Protein, Human, Recombinant (His & GST)

ALOX15B,arachidonate 15-lipoxygenase, type B,15-

Human Baculovirus Insect Cells
15 Lipoxygenase 2 Protein, Human, Recombinant (His & GST) is expressed in Baculovirus insect cells with His and GST tag. The predicted molecular weight is 103.7 kDa and the accession number is AAH35217.1.
TMPY-03351 LOX-1 Protein, Cynomolgus, Recombinant (His)

oxidized low density lipoprotein (lectin-like) receptor 1,OL...

Cynomolgus HEK293 Cells
LOX-1 Protein, Cynomolgus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26.9 kDa and the accession number is G7PJT2.
TMPY-04066 LOX-1 Protein, Rat, Recombinant (His)

oxidized low density lipoprotein (lectin-like) receptor 1,Ol...

Rat HEK293 Cells
LOX-1 Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 37.9 kDa and the accession number is O70156.
TMPY-03371 LOX-1 Protein, Rat, Recombinant (hFc)

OLR1,Lox1,Oldlr1,oxidized low density lipoprotein (...

Rat HEK293 Cells
LOX-1 Protein, Rat, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 63.9 kDa and the accession number is O70156.
TMPH-00955 ALOX12 Protein, Human, Recombinant (His)

Polyunsaturated fatty acid lipoxygenase ALOX12,LOG1...

Human E. coli
ALOX12 Protein, Human, Recombinant (His) is expressed in E. coli.
TMPY-00203 LOXL2 Protein, Mouse, Recombinant (His)

1110004B06Rik,4930526G11Rik,9430067E15Rik,lysyl oxidase-like...

Mouse HEK293 Cells
Lysyl oxidase homolog 2, also known as Lysyl oxidase-like protein 2, Lysyl oxidase-related protein 2, Lysyl oxidase-related protein WS9-14 and LOXL2, is a secreted protein that belongs to the lysyl oxidase family. LOXL2 contains four SRCR domains. The lysyl oxidase family is made up of five members: lysyl oxidase (LOX) and lysyl oxidase-like 1-4 ( LOXL1, LOXL2, LOXL3, LOXL4 ). All members share conserved C-terminal catalytic domains that provide for lysyl oxidase or lysyl oxidase-like enzyme act...
TMPH-01630 LOXL3 Protein, Human, Recombinant (GST & His)

LOXL3,Lysyl oxidase homolog 3,Lysyl oxidase-like pr...

Human E. coli
LOXL3 Protein, Human, Recombinant (GST & His) is expressed in E. coli expression system with N-6xHis-GST tag. The predicted molecular weight is 55.7 kDa and the accession number is P58215.
TMPH-01628 LOXL1 Protein, Human, Recombinant

Lysyl oxidase-like protein 1,Lysyl oxidase homolog 1,LOX...

Human E. coli
Active on elastin and collagen substrates. LOXL1 Protein, Human, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 53.0 kDa and the accession number is Q08397.
TMPH-01629 LOXL1 Protein, Human, Recombinant (His)

Lysyl oxidase-like protein 1,LOXL1,Lysyl oxidase ho...

Human E. coli
Active on elastin and collagen substrates.
TMPH-02774 LOXL4 Protein, Mouse, Recombinant (His)

Loxl4,Lysyl oxidase-related protein C,Lysyl oxidase...

Mouse E. coli
May modulate the formation of a collagenous extracellular matrix. LOXL4 Protein, Mouse, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 85.9 kDa and the accession number is Q924C6.
TMPH-00866 ADAMTS14 Protein, Human, Recombinant (His)

A disintegrin and metalloproteinase with thrombospondin moti...

Human E. coli
Has aminoprocollagen type I processing activity in the absence of ADAMTS2. Seems to be synthesized as a latent enzyme that requires activation to display aminoprocollagen peptidase activity. Cleaves lysyl oxidase LOX at a site downstream of its propeptide cleavage site to produce a short LOX form. ADAMTS14 Protein, Human, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 40.2 kDa and the accession number is Q8WXS8.
TMPH-01552 IRF1 Protein, Human, Recombinant (GST & His)

IRF1,Interferon regulatory factor 1

Human Baculovirus Insect Cells
Transcriptional regulator which displays a remarkable functional diversity in the regulation of cellular responses. Regulates transcription of IFN and IFN-inducible genes, host response to viral and bacterial infections, regulation of many genes expressed during hematopoiesis, inflammation, immune responses and cell proliferation and differentiation, regulation of the cell cycle and induction of growth arrest and programmed cell death following DNA damage. Stimulates both innate and acquired imm...

重组蛋白

LOX Protein, Human, Recombinant (His & MBP)
Cat.No: TMPH-01968
Species: Human
Expression System: Baculovirus Insect Cells
LOX Protein, Rat, Recombinant (His)
Cat.No: TMPH-03359
Species: Rat
Expression System: E. coli
LOX Protein, Mouse, Recombinant (His & Myc)
Cat.No: TMPH-02863
Species: Mouse
Expression System: Baculovirus Insect Cells
LOX Protein, Human, Recombinant (His & Myc & SUMO)
Cat.No: TMPH-01969
Species: Human
Expression System: E. coli
LOX-1 Protein, Mouse, Recombinant (His)
Cat.No: TMPK-01168
Species: Mouse
Expression System: HEK293 Cells
LOX-1 Protein, Human, Recombinant (His)
Cat.No: TMPY-02490
Species: Human
Expression System: HEK293 Cells
15 Lipoxygenase 2 Protein, Human, Recombinant
Cat.No: TMPY-03553
Species: Human
Expression System: Baculovirus Insect Cells
15 Lipoxygenase 2 Protein, Human, Recombinant (His & GST)
Cat.No: TMPY-03462
Species: Human
Expression System: Baculovirus Insect Cells
LOX-1 Protein, Cynomolgus, Recombinant (His)
Cat.No: TMPY-03351
Species: Cynomolgus
Expression System: HEK293 Cells
LOX-1 Protein, Rat, Recombinant (His)
Cat.No: TMPY-04066
Species: Rat
Expression System: HEK293 Cells
LOX-1 Protein, Rat, Recombinant (hFc)
Cat.No: TMPY-03371
Species: Rat
Expression System: HEK293 Cells
ALOX12 Protein, Human, Recombinant (His)
Cat.No: TMPH-00955
Species: Human
Expression System: E. coli
LOXL2 Protein, Mouse, Recombinant (His)
Cat.No: TMPY-00203
Species: Mouse
Expression System: HEK293 Cells
LOXL3 Protein, Human, Recombinant (GST & His)
Cat.No: TMPH-01630
Species: Human
Expression System: E. coli
LOXL1 Protein, Human, Recombinant
Cat.No: TMPH-01628
Species: Human
Expression System: E. coli
LOXL1 Protein, Human, Recombinant (His)
Cat.No: TMPH-01629
Species: Human
Expression System: E. coli
LOXL4 Protein, Mouse, Recombinant (His)
Cat.No: TMPH-02774
Species: Mouse
Expression System: E. coli
ADAMTS14 Protein, Human, Recombinant (His)
Cat.No: TMPH-00866
Species: Human
Expression System: E. coli
IRF1 Protein, Human, Recombinant (GST & His)
Cat.No: TMPH-01552
Species: Human
Expression System: Baculovirus Insect Cells
Cat. No. Product Name Target Signaling Pathways
TMIH-0154 Ciprofloxacin-d8

Ciprofloxacin-d8 是 Ciprofloxacin 的氘代化合物。Ciprofloxacin 的 CAS 号为 85721-33-1。Ciprofloxacin是一种有高抗菌活性的氟喹诺酮类抗生素。
TMIH-0306 Lomefloxacin-d5

Lomefloxacin-d5 是 Lomefloxacin 的氘代化合物。
T71984 Enrofloxacin-d5

Enrofloxacin-d5 is intended for use as an internal standard for the quantification of enrofloxacin by GC- or LC-MS. Enrofloxacin is a fluoroquinolone antibiotic. It is active against panels of Campylobacter, E. coli, and Salmonella isolates (mean MIC50s = 0.06, 0.5, and 0.03 µg/ml, respectively). It is also active against equine isolates of L. intracellularis (MICs = 0.125-0.5 µg/ml). Enrofloxacin inhibits bacterial DNA gyrase. In vivo, enrofloxacin (10 mg/kg) increases survival in a mouse model...
TMIJ-0211 Loxoprofen-d4

Loxoprofen-d4 是 Loxoprofen 的氘代化合物。Loxoprofen 的 CAS 号为 68767-14-6。Loxoprofen 是一种非甾体类抗炎药,具有解热作用,可用于缓解疼痛的研究。它是非选择性COX抑制剂,对 COX-1 和 COX-2 的IC50分别为 6.5 和 13.5 μM。
TMIJ-0158 Sitafloxacin-d4

Sitafloxacin-d4 是 Sitafloxacin 的氘代化合物。Sitafloxacin 的 CAS 号为 127254-12-0。Sitafloxacin (Sitafloxacin anhydrous) 是一种具有口服活性的氟喹诺酮类抗生素,具有广谱的抗菌活性。Sitafloxacin 可用于研究呼吸道感染和尿路感染。
TMID-0195 Levofloxacin-d8

Levofloxacin-d8 是 Levofloxacin 的氘代化合物。Levofloxacin 的 CAS 号为 100986-85-4。Levofloxacin是合成的氟喹诺酮类抗生素,有抑制细菌DNA旋转酶的超螺旋活性的作用,能阻止DNA复制。
TMIJ-0293 Difloxacin-d3 hydrochlorid (methyl-d3)

Difloxacin-d3 hydrochlorid (methyl-d3) 是 Difloxacin hydrochlorid 的氘代化合物。Difloxacin hydrochlorid 的 CAS 号为 5522-39-4。
T11113 Duloxetine D3 hydrochloride

(S)-Duloxetine D3 hydrochloride,LY248686 D3 hydrochloride

Others Others
Duloxetine D3 hydrochloride is a serotonin-norepinephrine reuptake inhibitor (SNRI) with a Ki of 4.6 nM, used for treatment of major depressive disorder and generalized anxiety disorder (GAD).Duloxetine D3 hydrochloride ((S)-Duloxetine D3 hydrochloride) i
TMIJ-0079 N-Carbobenzyloxyglycine-d2

N-Carbobenzyloxyglycine-d2 是 N-Carbobenzyloxyglycine 的氘代化合物。N-Carbobenzyloxyglycine 的 CAS 号为 1138-80-3。Z-Glycine (Carbobenzoxyglycine) 是一种药物-脂质结合物,旨在促进脑渗透,基于其亲脂性和与生物膜中脂质的相似性。
TMIJ-0212 trans-Hydroxy Loxoprofen-13C-d3

trans-Hydroxy Loxoprofen-13C-d3 (Mixture of Diastereomers) 是 trans-Hydroxy Loxoprofen 的 13C 和氘代化合物。trans-Hydroxy Loxoprofen 的 CAS 号为 371753-19-4。
TMIJ-0325 Duloxetine-d7 Maleate

Duloxetine-d7 Maleate 是 Duloxetine Maleate 的氘代化合物。Duloxetine Maleate 的 CAS 号为 116817-86-8。
TMID-0079 Norfloxacin-d8

Norfloxacin-d8 是 Norfloxacin 的氘代化合物。Norfloxacin 的 CAS 号为 70458-96-7。Norfloxacin是广谱抗生素,能通过结合DNA旋转酶抑制革兰氏阳性和阴性菌。
TMIH-0398 Norfloxacin-d5

Norfloxacin-d5 是 Norfloxacin 的氘代化合物。
TMIH-0478 rac-Duloxetine-d3

rac-Duloxetine-d3 是 rac-Duloxetine 的氘代化合物。rac-Duloxetine 的 CAS 号为 116817-13-1。
TMIH-0105 Baloxavir-d4

Baloxavir-d4 是 Baloxavir 的氘代化合物。Baloxavir 的 CAS 号为 1985605-59-1。Baloxavir 是衍生自前药 Baloxavir marboxil,是流感病毒聚合酶 PA 亚基的一流帽依赖性核酸内切酶抑制剂。它抑制病毒 RNA 的转录和复制,具有强大的抗病毒活性。
TMIJ-0136 Moxifloxacin-d4 HCl

Moxifloxacin-d4 HCl 是 Moxifloxacin HCl 的氘代化合物。Moxifloxacin HCl 的 CAS 号为 186826-86-8。Moxifloxacin Hydrochloride是一种口服有效的 8-甲氧基喹诺酮类抗菌药物,可研究感染性肺炎,急性细菌性鼻窦炎和慢性支气管炎的急性细菌性加重。
TMID-0194 Ofloxacin-d8

Ofloxacin-d8 是 Ofloxacin 的氘代化合物。Ofloxacin 的 CAS 号为 82419-36-1。Ofloxacin是可抑制细菌DNA旋转酶的一种氟喹诺酮类抗生素。
TMIJ-0288 Danofloxacin-d3

Danofloxacin-d3 是 Danofloxacin 的氘代化合物。Danofloxacin 的 CAS 号为 112398-08-0。Danofloxacin free base 是一种具有口服活性第三代氟喹诺酮抗菌剂,对大多数革兰氏阴性和革兰氏阳性细菌,支原体和衣原体物种具有广谱的活性,并通过抑制细菌的 DNA 回转酶发挥抗菌作用。它可用于牛,猪和鸡呼吸道疾病的研究。
TMID-0271 Miloxacin-d3

Miloxacin-d3 是 Miloxacin 的氘代化合物。Miloxacin 的 CAS 号为 37065-29-5。
TMIH-0364 Naloxone-d5

Naloxone-d5 是 Naloxone 的氘代化合物。
TMIJ-0015 Ciprofloxacin-d8 Hydrochloride

Ciprofloxacin-d8 Hydrochloride 是 Ciprofloxacin Hydrochloride 的氘代化合物。Ciprofloxacin Hydrochloride 的 CAS 号为 93107-08-5。Ciprofloxacin hydrochloride是一种高抗菌活性的氟喹诺酮类抗生素。
TMIH-0472 Rac Loxoprofen sodium-d3

Rac Loxoprofen sodium-d3 是 Rac Loxoprofen sodium 的氘代化合物。Rac Loxoprofen sodium 的 CAS 号为 68767-14-6。Loxoprofen 是一种非甾体类抗炎药,具有解热作用,可用于缓解疼痛的研究。它是非选择性COX抑制剂,对 COX-1 和 COX-2 的IC50分别为 6.5 和 13.5 μM。
TMIJ-0059 Moxifloxacin-d4

Moxifloxacin-d4 是 Moxifloxacin 的氘代化合物。Moxifloxacin 的 CAS 号为 151096-09-2。Moxifloxacin 是一种8-甲氧基喹诺酮类口服有效抗菌药物,用于急性细菌性鼻窦炎,慢性支气管炎的急性细菌性加重和感染性肺炎的研究。
TMID-0270 Pefloxacin-d5

Pefloxacin-d5 是 Pefloxacin 的氘代化合物。Pefloxacin 的 CAS 号为 70458-92-3。
T10181 6-beta-Naloxol D5 hydrochloride

6β-Naloxol D5 hydrochloride

Others Others
6-beta-Naloxol D5 hydrochloride is a deuterium-labeled opioid antagonist, closely related to naloxone, that serves as an effective compound in the field of chemical research.
TMIH-0305 Lomefloxacin-d5 hydrochloride

Lomefloxacin-d5 hydrochloride 是 Lomefloxacin hydrochloride 的氘代化合物。Lomefloxacin hydrochloride 的 CAS 号为 98079-51-7。Lomefloxacin是一种广谱喹诺酮类抗生素,具有抗菌活性。它可研究支气管炎、尿路感染、结膜炎、外耳炎和中耳炎。
TMIH-0300 Levofloxacin-d3

Levofloxacin-d3 是 Levofloxacin 的氘代化合物。Levofloxacin 的 CAS 号为 100986-85-4。Levofloxacin是合成的氟喹诺酮类抗生素,有抑制细菌DNA旋转酶的超螺旋活性的作用,能阻止DNA复制。
TMIH-0406 Ofloxacin-d3

Ofloxacin-d3 是 Ofloxacin 的氘代化合物。
TMIH-0205 Duloxetine-d3 HCl

Duloxetine-d3 HCl 是 Duloxetine HCl 的氘代化合物。Duloxetine HCl 的 CAS 号为 136434-34-9。Duloxetine hydrochloride 是一种 5-羟色胺-去甲肾上腺素重吸收 (serotonin-norepinephrine reuptake) 抑制剂 (SNRI),Ki=4.6 nM,可用于广泛性焦虑症的研究。
T11998 Meloxicam-d3

Meloxicam D4

Others Others
Meloxicam D4 is deuterium labeled Meloxicam. Meloxicam is a non-steroidal antiinflammatory agent, inhibits COX activity,(Target:COX-1; IC50: 36.6 μM ;(Target:COX-2; IC50: 0.49 μM).
TMIJ-0037 Sarafloxacin-d8 Hydrochloride

Sarafloxacin-d8 Hydrochloride 是 Sarafloxacin Hydrochloride 的氘代化合物。Sarafloxacin Hydrochloride 的 CAS 号为 91296-87-6。Sarafloxacin hydrochloride是一种抗菌化合物。
TMIJ-0213 Naloxone-d5 HCl

Naloxone-d5 HCl 是 Naloxone HCl 的氘代化合物。Naloxone HCl 的 CAS 号为 357-08-4。Naloxone hydrochloride 是一种特异性、没有激动剂活性的opiate拮抗剂。它是 mu、delta 和 kappa 阿片受体的竞争性拮抗剂。
TMIJ-0300 Duloxetine-d7

Duloxetine-d7 是 Duloxetine 的氘代化合物。Duloxetine 的 CAS 号为 116539-59-4。Duloxetine 是一种 5 羟色胺-去甲肾上腺素重吸收 (serotonin-norepinephrine reuptake) 抑制剂,Ki=4.6 nM,可作用于广泛性焦虑症的研究。
TMID-0281 Moxifloxacin-13C-d3

Moxifloxacin-13C-d3 是 Moxifloxacin 的 13C 和氘代化合物。Moxifloxacin 的 CAS 号为 151096-09-2。Moxifloxacin 是一种8-甲氧基喹诺酮类口服有效抗菌药物,用于急性细菌性鼻窦炎,慢性支气管炎的急性细菌性加重和感染性肺炎的研究。

同位素标记化合物

Ciprofloxacin-d8
Cat.No: TMIH-0154
Synonym:
Target:
Lomefloxacin-d5
Cat.No: TMIH-0306
Synonym:
Target:
Enrofloxacin-d5
Cat.No: T71984
Synonym:
Target:
Loxoprofen-d4
Cat.No: TMIJ-0211
Synonym:
Target:
Sitafloxacin-d4
Cat.No: TMIJ-0158
Synonym:
Target:
Levofloxacin-d8
Cat.No: TMID-0195
Synonym:
Target:
Difloxacin-d3 hydrochlorid (methyl-d3)
Cat.No: TMIJ-0293
Synonym:
Target:
Duloxetine D3 hydrochloride
Cat.No: T11113
Synonym: (S)-Duloxetine D3 hydrochloride,LY248686 D3 hydrochloride
Target: Others
N-Carbobenzyloxyglycine-d2
Cat.No: TMIJ-0079
Synonym:
Target:
trans-Hydroxy Loxoprofen-13C-d3
Cat.No: TMIJ-0212
Synonym:
Target:
Duloxetine-d7 Maleate
Cat.No: TMIJ-0325
Synonym:
Target:
Norfloxacin-d8
Cat.No: TMID-0079
Synonym:
Target:
Norfloxacin-d5
Cat.No: TMIH-0398
Synonym:
Target:
rac-Duloxetine-d3
Cat.No: TMIH-0478
Synonym:
Target:
Baloxavir-d4
Cat.No: TMIH-0105
Synonym:
Target:
Moxifloxacin-d4 HCl
Cat.No: TMIJ-0136
Synonym:
Target:
Ofloxacin-d8
Cat.No: TMID-0194
Synonym:
Target:
Danofloxacin-d3
Cat.No: TMIJ-0288
Synonym:
Target:
Miloxacin-d3
Cat.No: TMID-0271
Synonym:
Target:
Naloxone-d5
Cat.No: TMIH-0364
Synonym:
Target:
Ciprofloxacin-d8 Hydrochloride
Cat.No: TMIJ-0015
Synonym:
Target:
Rac Loxoprofen sodium-d3
Cat.No: TMIH-0472
Synonym:
Target:
Moxifloxacin-d4
Cat.No: TMIJ-0059
Synonym:
Target:
Pefloxacin-d5
Cat.No: TMID-0270
Synonym:
Target:
6-beta-Naloxol D5 hydrochloride
Cat.No: T10181
Synonym: 6β-Naloxol D5 hydrochloride
Target: Others
Lomefloxacin-d5 hydrochloride
Cat.No: TMIH-0305
Synonym:
Target:
Levofloxacin-d3
Cat.No: TMIH-0300
Synonym:
Target:
Ofloxacin-d3
Cat.No: TMIH-0406
Synonym:
Target:
Duloxetine-d3 HCl
Cat.No: TMIH-0205
Synonym:
Target:
Meloxicam-d3
Cat.No: T11998
Synonym: Meloxicam D4
Target: Others
Sarafloxacin-d8 Hydrochloride
Cat.No: TMIJ-0037
Synonym:
Target:
Naloxone-d5 HCl
Cat.No: TMIJ-0213
Synonym:
Target:
Duloxetine-d7
Cat.No: TMIJ-0300
Synonym:
Target:
Moxifloxacin-13C-d3
Cat.No: TMID-0281
Synonym:
Target:
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