Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T25629 |
LAQ 824
LAQ824,LAQ-824 |
Others | Others |
LAQ 824 is an inhibitor of histone deacetylase. | |||
T2454 |
Dacinostat
NVP-LAQ824,达西司特,LAQ824 |
HDAC; Autophagy | Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair |
Dacinostat (NVP-LAQ824) 是一种新型 HDAC 抑制剂,IC50 为 32 nM,是 p21 启动子的激活剂。它也可抑制HDAC1的活性,IC50值为 9 nM,主要用于癌症研究。 |