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Targets Recommended: Others

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Cat. No. Product Name Target Signaling Pathways
T36109 L Moses dihydrochloride

Others Others
High affinity and selective cell-permeable p300/CBP-associated factor (PCAF) inhibitor (Ki = 47 nM). Exhibits no significant activity against a panel of 48 other bromodomains except GCN5 (Kd = 600 nM). Exhibits >4500-fold selectivity for PCAF over BRD4. Also exhibits metabolic stability in mouse and human liver microsomes and no observable cytotoxicity in peripheral blood mononuclear cells (PBMC). Moustakim et al (2017) Discovery of a PCAF bromodomain chemical probe. Angew.Chem.Int.Ed. 56 827 P...
T62424 L-Moses dihydrochloride

Others Others
L-Moses (L-45) dihydrochloride 是一个有效的、选择性 p300/CBP 相关因子 (PCAF) 溴结构域 (Brd) 抑制剂 (Kd: 126 nM)。

化合物

L Moses dihydrochloride
Cat.No: T36109
Synonym:
Target: Others
L-Moses dihydrochloride
Cat.No: T62424
Synonym:
Target: Others
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