Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T71060 |
IST-622
|
Others | Others |
IST-622 is a unique topoisomerase inhibitor, showing significant growth-inhibitory effects against large-cell lung cancer (Lu-116) and gastric adenocarcinoma (St-4). | |||
T71059 |
Ranitidine bismuth citrate
IST 622,雷尼替丁枸橼酸盐 |
Others | Others |
Ranitidine bismuth citrate 为一种口服活性的组胺H2受体(Histamine H2-receptor)拮抗剂,其IC50值为3.3 μM,对SARS-CoV-2感染细胞显示高选择性。该化合物还是治疗幽门螺杆菌(Helicobacter Pylori)感染的常用试剂,其MIC90为16 ng/L。 |