Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T40285 |
KRAS G12C inhibitor 18
|
Others | Others |
KRAS G12C inhibitor 18 is a potent, orally active compound that inhibits KRAS G12C and exhibits anti-tumor activities. | |||
T11768 |
KRAS G12C inhibitor 14
|
Ras | GPCR/G Protein; MAPK |
KRAS G12C inhibitor 14 是一种有效的 KRAS G12C 抑制剂(IC50= 18 nM)。 | |||
T62784 |
KRAS inhibitor-18
|
Others | Others |
KRAS inhibitor-18 (compound 3-10) 是一种 KRAS G12C 的有效抑制剂 (IC50: 4.74 μM)。KRAS inhibitor-18 在 MIA PaCA-2,A549 细胞中表现出 p-ERK 抑制作用,IC50s 分别为 66.4,11.1 μM。KRAS inhibitor-18 具有潜力进行胰腺癌、结直肠癌和肺癌的研究。 |