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Search Results for " kca1.1 "

Targets Recommended: Others

抑制剂 & 化合物

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同位素标记化合物

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Cat. No.	Product Name	Target	Signaling Pathways
T72195	KCa1.1 channel activator-2	Others	Others
	KCa1.1 channel activator-2 (化合物 3F) 是一种槲皮素衍生物，是选择性的血管 KCa1.1 channel 刺激剂。KCa1.1 channel activator-2 具有强效的肌肉松弛活性。
T72194	KCa1.1 channel activator-1	Others	Others
	KCa1.1 channel activator-1 (化合物 1E) 是一种槲皮素衍生物，是选择性的血管 KCa1.1 channel 刺激剂。KCa1.1 channel activator-1 也显示 CaV1.2 channel 通道阻断活性。KCa1.1 channel activator-1 表现出较弱的肌肉松弛活性。
T4294	NS 11021 NS11021	Potassium Channel	Membrane transporter/Ion channel
	NS 11021 (NS11021) 是特异性 Ca2+激活的大电导 K+(KCa1.1)通道激活剂。当浓度高于0.3 μM 时，它通过平行移动通道激活曲线产生更多负电位，以浓度依赖的方式激活 KCa1.1。
T3557	GAL-021 GAL 021	Potassium Channel	Membrane transporter/Ion channel
	GAL-021新型静脉内BKCa-channel 阻滞剂。
T4612	NS309	EGFR; Potassium Channel; HER	Angiogenesis; JAK/STAT signaling; Membrane transporter/Ion channel; Tyrosine Kinase/Adaptors
	NS309 是选择性钙依赖性钾离子通道 SK/IK 的激活剂，在 BK 通道上没有激活作用。
T83868	(±)13,14-EDT (±)13,14-Epoxydocosatrienoic Acid,(±)13,14-EpDoTrE,(±)-Dihomo-13,14-EET	Others	Others
	(±)13,14-EDT是一种氧脂和腎上腺酸的代谢产物，通过细胞色素P450（CYP）途径形成。在50 nM的浓度下，它能激活分离的大鼠冠状小动脉平滑肌细胞中的大导电钙激活钾通道（KCa1.1/BK），并导致分离的猪小动脉扩张（EC50 = 12 pM）。(±)13,14-EDT还能使用TP受体激动剂U-46619预收缩的分离牛冠状动脉放松。
T84609	(±)5(6)-DiHET (±)5,6-DiHETrE	Others	Others
	5(6)-DiHET is a racemic compound synthesized through the action of epoxide hydrolases on 5(6)-EET, encompassing both enantiomeric forms. It serves as a quantitative marker for 5(6)-EET, facilitating its measurement by utilizing the compound's conversion to 5(6)-δ-lactone in solution. Additionally, 5(6)-DiHET activates large-conductance calcium-activated potassium (KCa1.1/BK) channels in rat small coronary artery smooth muscle cells, supporting its biological significance in vascular regulation. ...

化合物

KCa1.1 channel activator-2

Cat.No: T72195

Synonym:

Target: Others

KCa1.1 channel activator-1

Target: Potassium Channel

GAL-021

Cat.No: T3557

Synonym: GAL 021

Target: Potassium Channel

NS309

Cat.No: T4612

Synonym:

Target: EGFR, Potassium Channel, HER

(±)13,14-EDT

Cat.No: T83868

Synonym: (±)13,14-Epoxydocosatrienoic Acid,(±)13,14-EpDoTrE,(±)-Dihomo-13,14-EET

Target: Others

(±)5(6)-DiHET

Cat.No: T84609

Synonym: (±)5,6-DiHETrE

Target: Others

Species：

Expression System：

Tag：

Cat. No.	Product Name	Species	Expression System
TMPH-01028	KCNMA1 Protein, Human, Recombinant K(VCA)alpha,Calcium-activated potassium channel subunit alph...	Human	E. coli
	KCNMA1 Protein, Human, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 17.2 kDa and the accession number is Q12791.

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KCNMA1 Protein, Human, Recombinant

Cat.No: TMPH-01028

Species: Human

Expression System: E. coli

Cat. No.	Product Name	Target	Signaling Pathways
T71303	Flufenamic Acid-d4
	Flufenamic acid-d4 is intended for use as an internal standard for the quantification of flufenamic acid by GC- or LC-MS. Flufenamic acid is a non-steroidal anti-inflammatory drug (NSAID) and COX inhibitor (IC50s = 3 and 9.3 µM for human COX-1 and COX-2, respectively). Flufenamic acid inhibits TNF-α-induced increases in COX-2 levels and NF-κB activation in HT-29 colon cancer cells in a concentration-dependent manner. It inhibits calcium influx induced by fMLP or A23187 in human polymorphonuclear...

同位素标记化合物

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化合物

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同位素标记化合物