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Targets Recommended: Calcium Channel

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Cat. No. Product Name Target Signaling Pathways
T24239 K201

K-201,JTV 519,JTV-519,K 201

Calcium Channel Membrane transporter/Ion channel; Metabolism
K201 (JTV-519) 是一种 Ca2+ 依赖性阻滞剂,通过稳定兰尼碱受体来防止缺血性心脏和骨骼肌 (SkM) 中的肌质网异常 Ca(2+) 泄漏。
T11732 JTV-519 hemifumarate

K201 hemifumarate

MELK PI3K/Akt/mTOR signaling
JTV-519 hemifumarate,Antiarrhythmic and cardioprotective properties. is a Ca2+-dependent blocker of sarcoplasmic reticulum Ca2+-stimulated ATPase (SERCA) and a partial agonist of ryanodine receptors in striated muscle.
T11731 JTV-519 free base

K201 free base

FLT Angiogenesis; Tyrosine Kinase/Adaptors
JTV-519 free base (K201 free base), recognized for its antiarrhythmic and cardioprotective properties, functions as a Ca2+-dependent blocker of sarcoplasmic reticulum Ca2+-stimulated ATPase (SERCA) and serves as a partial agonist of ryanodine receptors in striated muscle.
T7360 GSK2018682

S1P Receptor; LPL Receptor GPCR/G Protein
GSK2018682 是 1-磷酸鞘氨醇受体S1P1和S1P5激动剂,pEC50值分别为 7.7 和 7.2,可用于多发性硬化的研究。
T71564 GSK2018682 HCl

Others Others
GSK2018682 is a novel sphingosine-1-phosphate receptor 1 (s1p1) and 5 (s1p5) agonist.
T37807 JTV-519 fumarate

Calcium Channel Membrane transporter/Ion channel; Metabolism
JTV-519 fumarate (K201 fumarate) 是 一种 SERCA 阻断剂和兰尼碱受体的部分激动剂,具有抗心律失常和心脏保护作用,可改善肌浆网钙渗漏,可用于研究焦虑症。

化合物

K201
Cat.No: T24239
Synonym: K-201,JTV 519,JTV-519,K 201
Target: Calcium Channel
JTV-519 hemifumarate
Cat.No: T11732
Synonym: K201 hemifumarate
Target: MELK
JTV-519 free base
Cat.No: T11731
Synonym: K201 free base
Target: FLT
GSK2018682
Cat.No: T7360
Synonym:
Target: S1P Receptor, LPL Receptor
GSK2018682 HCl
Cat.No: T71564
Synonym:
Target: Others
JTV-519 fumarate
Cat.No: T37807
Synonym:
Target: Calcium Channel
TargetMol Loading
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