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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T63014 |
Ivabradine
|
Others | Others |
Ivabradine 是一种有效的、口服具有活力的 HCN (超极化激活的环核苷酸门控) 通道阻滞剂,能够抑制心脏起搏器电流 (If)。Ivabradine 以剂量依赖性的方式降低心率,且不改变血压。Ivabradine 具有抗惊厥、抗缺血和抗心绞痛作用。 | |||
T2535 |
Ivabradine hydrochloride
盐酸伊伐布雷定,S 16257-2,Ivabradine HCl |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Ivabradine hydrochloride (S 16257-2) 是一种可口服的,超极化激活的环核苷酸门控离子通道通道阻滞剂。 | |||
T11695 |
N-Demethyl ivabradine hydrochloride
Ivabradine metabolite N-Demethyl Ivabradine hydrochloride |
Others | Others |
N-Demethyl Ivabradine Hcl is a specific inhibitor of the funny channel.N-Demethyl Ivabradine Hcl is a metabolite of Ivabradine. | |||
T37160 |
8-Demethyl Ivabradine
|
Others | Others |
8-Demethyl Ivabradine is a metabolite derived from Ivabradine, an orally bioavailable cyclic nucleotide-gated (HCN) channel blocker with hyperpolarization-activated properties[1]. | |||
T73976 |
Ivabradine impurity 2
|
Others | Others |
Ivabradine impurity 2 是 Ivabradine 的一个杂质。 Ivabradine 是具有口服活性的,超极化激活的环核苷酸门控离子通道 (HCN) 通道阻滞剂。 | |||
T73975 |
Ivabradine impurity 1
|
Others | Others |
Ivabradine impurity 1 是Ivabradine 的一个杂质。 Ivabradine 是具有口服活性的,超极化激活的环核苷酸门控离子通道 (HCN) 通道阻滞剂。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T11692 |
Ivabradine-d3 hydrochloride
盐酸伊伐布雷定 D3,Ivabradine D3 Hydrochloride |
Others | Others |
Ivabradine hydrochloride is a new If inhibitor with IC50 of 2.9 μM, and used as a pure heart rate lowering agent. Ivabradine D3 Hydrochloride is the deuterium labeled Ivabradine hydrochloride. | |||
T11694 |
Ivabradine-d6 hydrochloride
盐酸伊伐布雷定 D6,Ivabradine D6 hydrochloride |
Others | Others |
Ivabradine hydrochloride is a new If inhibitor with IC50 of 2.9 μM, and used as a pure heart rate lowering agent. Ivabradine D6 hydrochloride is the deuterium labeled Ivabradine hydrochloride. | |||
T19447 |
N-Demethyl Ivabradine D6 Hydrochloride
|
Others | Others |
N-Demethyl Ivabradine D6 Hydrochloride salt is the deuterium labeled N-Demethyl Ivabradine, which is a Ivabradine metabolite. | |||
TMIH-0380 |
N-Desmethyl Ivabradine-d6 HCl
|
||
N-Desmethyl Ivabradine-d6 HCl 是 N-Desmethyl Ivabradine HCl 的氘代化合物。N-Desmethyl Ivabradine HCl 的 CAS 号为 1246638-08-3。 |