2
10
1
Cat. No. | Product Name | ||
---|---|---|---|
L6120 | 黄酮类天然产物库 | 514 compounds | |
514 种黄酮类天然产物的独特集合,可用于高通量筛选和高内涵筛选; |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TP2236L |
Cortistatin-8 acetate
Cortistatin-8 acetate(485803-62-1 Free base) |
GHSR | GPCR/G Protein |
Cortistatin-8 acetate 是一种皮质抑素类似物,是一种GHS-R拮抗剂,对生长激素促分泌素受体有抑制作用。Cortistatin-8 acetate 是一种合成皮质抑素衍生的生长素释放肽受体配体,不会改变人类对酰化生长素释放肽或海沙瑞林的内分泌反应。 | |||
TP2236 |
Cortistatin-8
|
Others | Others |
ghrelin receptor antagonist |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1035 |
Hesperidin
橙皮甙,Hesperetin 7-rutinoside,Cirantin,橙皮苷 |
Apoptosis; Reactive Oxygen Species; Endogenous Metabolite; Autophagy | Apoptosis; Autophagy; Immunology/Inflammation; Metabolism; NF-κB |
Hesperidin (Cirantin) 属于黄烷酮糖苷类天然产物,广泛存在于柑橘类水果中。Hesperidin 具有抗氧化活性、抗肿瘤活性和抗过敏活性。 | |||
T0228 |
Methyl-Hesperidin
甲基橙皮甙 |
Akt; PKC | Chromatin/Epigenetic; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling |
Methyl hesperidin 是一种血管扩张剂。 | |||
T7980 |
Hesperidin methylchalcone
|
NF-κB | NF-κB |
Hesperidin methylchalcone 抑制氧化应激,细胞因子产生和NF-κB 活化。它能够抑制炎症和疼痛,具有血管保护作用。 | |||
TN7354 |
(R)-5,3'-Dimethyl hesperidin
|
Others | Others |
Hesperidin analog serves as a reference standard. | |||
TN1733 |
Hesperetin 7-O-glucoside
|
Anti-infection; Antibacterial; HMG-CoA Reductase | Metabolism; Microbiology/Virology |
Hesperetin 7-O-glucoside 是通过 Hesperidin 的酶促转化产生的一种人 HMG-CoA 还原酶抑制剂,具有降压作用,可抑制幽门螺杆菌的生长。 | |||
T2737 |
Neohesperidin
Hesperetin 7-O-neohesperidoside,NSC 31048,新橙皮苷 |
Antioxidant | oxidation-reduction |
Neohesperidin (NSC-31048) 是一种类黄酮化合物,存在于葫芦科植物中,具有抗氧化和抗炎活性。 | |||
T2767 |
Neohesperidin Dihydrochalcone
NHDC,新橙皮苷二氢查尔酮,新橙皮苷二氢查耳酮,Neohesperidin DC,NCI-c60764 |
Reactive Oxygen Species | Immunology/Inflammation; Metabolism; NF-κB |
Neohesperidin Dihydrochalcone (Neohesperidin DC) 是一种合成的糖苷查耳酮,可用作低热量人造甜味剂,添加到各种食品和饮料中。 | |||
TN7424 |
3''-O-Caffeoylhesperidin
|
Others | Others |
T2565 |
Hesperetin
橙皮素 |
Apoptosis; p38 MAPK; 5-HT Receptor; Autophagy; TGF-beta/Smad | Apoptosis; Autophagy; GPCR/G Protein; MAPK; Neuroscience; Stem Cells |
Hesperetin 是一种天然黄烷酮类物质,是人UGT 的广谱抑制剂,可诱导凋亡。 | |||
T0530 |
Flavanone
2-Phenyl-4-chromanone,4-Flavanone,2,3-Dihydroflavone,黄烷酮,2-Phenylchroman-4-one |
Others; Aromatase | Endocrinology/Hormones; Others |
Flavanone (2-Phenylchroman-4-one) 是天然的黄酮类化合物,对人类雌激素合成酶芳香化酶具有抑制作用。 |