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Targets Recommended: 5-HT Receptor HER

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Cat. No. Product Name Target Signaling Pathways
T70044 Sarizotan HCl

EMD 128130 HCl

5-HT Receptor; HER Angiogenesis; GPCR/G Protein; JAK/STAT signaling; Neuroscience; Tyrosine Kinase/Adaptors
Sarizotan HCl (EMD 128130 HCl) 是一种 hERG 通道抑制剂和 5-羟色胺5-HT1A受体激动剂,具有潜在的抗抑郁作用,可用于研究帕金森运动障碍
T40439 Sarizotan

EMD 128130

Others Others
Sarizotan (EMD 128130) is an orally active compound that acts as an agonist for serotonin 5-HT 1A receptors and dopamine receptors. It has shown potent activity with IC 50 values of 6.5 nM for rat 5-HT 1A , 0.1 nM for human 5-HT 1A , 15.1 nM for rat D 2 , 17 nM for human D 2 , 6.8 nM for human D 3 , and 2.4 nM for human D 4.2 .

化合物

Sarizotan HCl
Cat.No: T70044
Synonym: EMD 128130 HCl
Target: 5-HT Receptor, HER
Sarizotan
Cat.No: T40439
Synonym: EMD 128130
Target: Others
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