123
21
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T85007 |
10(S)-HOME
HOD |
Others | Others |
10(S)-HOME, an oxylipin, acts as an intermediate in the conversion process of oleic acid into the antibacterial hydroxy fatty acid 7,10-dihydroxy-8(E)-octadecenoic acid within P. aeruginosa. | |||
T16742 |
Rhodamine 110
Rhodamine 110 chloride,RH110,罗丹明110 |
Others | Others |
Rhodamine 110 (RH110) 是灵敏的选择性底物,激发波长为 498 nm,发射波长为 521 nm,可用于测定溶液或活细胞内的蛋白酶。 | |||
T11027 |
DHODH-IN-4
|
Dehydrogenase | Metabolism |
DHODH-IN-4 是人和 Plasmodium falciparum 二氢乳清酸脱氢酶 (DHODH) 的抑制剂,其对 PfDHODH 和 HsDHODH 的IC50 值分别为 4 μM 和 0.18 μM。DHODH-IN-4 (compound 17) 具有抗疟疾活性。 | |||
T11029 |
hDHODH-IN-5
DHODH-IN-7 |
Dehydrogenase | Metabolism |
hDHODH-IN-5 是人源二氢乳清酸脱氢酶的抑制剂 (hDHODH, IC50 = 0.91 μM)。 | |||
T11023 |
DHODH-IN-14
|
Dehydrogenase | Metabolism |
DHODH-IN-14是一种 A771726 的 hydroxyfurazan 类似物。DHODH-IN-14 是一种二氢乳清酸脱氢酶 (DHODH) 抑制剂,对大鼠肝脏 DHODH 的 IC50 为 0.49 μM。DHODH-IN-14 可用于类风湿关节炎。 | |||
T11025 |
hDHODH-IN-3
DHODH-IN-2 |
Dehydrogenase | Metabolism |
hDHODH-IN-3 是人二氢乳清酸脱氢酶的抑制剂,pMIC50 值为 8.6。 hDHODH-IN-3 可以抑制麻疹病毒的复制。 | |||
T11019 |
DHODH-IN-1
|
Dehydrogenase | Metabolism |
DHODH-IN-1 是一种有效的 DHODH 抑制剂 (IC50 = 25 nM) 并抑制嘧啶生物合成途径。 | |||
T11020 |
DHODH-IN-11
|
Dehydrogenase; DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism |
DHODH-IN-11 是一种来氟米特衍生物和弱二氢乳清酸脱氢酶 (DHODH) 抑制剂,pKa 为 5.03 | |||
T19054 |
Rhodamine 800
罗丹明800,罗丹明 800 |
Others | Others |
Rhodamine 800 是近红外荧光染料的一种。 | |||
T11028 |
hDHODH-IN-4
DHODH-IN-5 |
Dehydrogenase | Metabolism |
hDHODH-IN-4 (DHODH-IN-5) 是一种有效的人二氢硼酸脱氢酶 (DHODH) 抑制剂,对人重组 DHODH 的 pIC50 为 7.8。hDHODH-IN-4 抑制麻疹病毒复制,pMIC50 为 8.8。 | |||
T19062 |
Sulforhodamine 101
磺基罗丹明101,磺基罗丹明 101,SR101 |
Others | Others |
Sulforhodamine 101 (SR101) 是一种两性罗丹明红色荧光染料 (excitation/emission: 586/605 nm),常用于神经元形态的研究,并作为星形胶质细胞的细胞类型选择性荧光标记物,在体内和切片制备中都有应用。 | |||
T12438 |
PfDHODH-IN-1
|
Dehydrogenase; Parasite | Metabolism; Microbiology/Virology |
PfDHODH-IN-1 是 Leflunomide 活性代谢物的类似物,具有抗疟疾活性。它是恶性疟原虫二氢乳清酸脱氢酶抑制剂。 | |||
T11022 |
DHODH-IN-13
|
Dehydrogenase | Metabolism |
DHODH-IN-13 是一种 DHODH 抑制剂,对大鼠肝脏的 IC50 为 4.3 μM。 DHODH-IN-13 可用于类风湿性关节炎的研究。 | |||
T11021 |
DHODH-IN-12
|
Dehydrogenase | Metabolism |
DHODH-IN-12 是一种 Leflunomide 衍生物,也是一种二氢乳清酸脱氢酶 (DHODH) 的弱抑制剂,其 pKa 为 5.07。 | |||
T21267 |
HODHBt
|
STAT | JAK/STAT signaling; Stem Cells |
HODHBt 是一种 STAT5-SUMO 蛋白-蛋白相互作用抑制剂。 | |||
TP1865L |
Rhodopsin Epitope Tag acetate
|
Others | Others |
Rhodopsin Epitope Tag acetate 是一种 9 个氨基酸的肽,代表牛视紫红质的 C 末端,广泛用作表位标签。许多抗视紫红质抗体可以识别该表位。 | |||
T19981 |
Rhoduline Acid
Di-J acid,I Acid Imide,NSC 1698 |
||
Rhoduline Acid (Di-J acid)是合成染料的中间体,可用于合成二偶氮染料和四硝唑染料。 | |||
T19063 |
Sulforhodamine B sodium salt
Acid Red 52,Kiton Red 620,磺酰罗丹明B |
Others | Others |
Sulforhodamine B sodium salt (Acid Red 52) 是一种能够定量测定培养细胞的细胞蛋白量的荧光染料,。 | |||
T72083 |
Octadecyl Rhodamine B chloride
|
||
Octadecyl Rhodamine B chloride 也被叫做RBOE, 是一种极性敏感染料,常作为一种发色基团与其他化合物一起使用,可用于给细胞膜染色,在有机分子组装、膜结构及蛋白质结构域中的电子能量转移中都有应用。 | |||
T11546 |
hDHODH-IN-1
|
Dehydrogenase | Metabolism |
hDHODH-IN-1 是有效的人二氢乳清酸脱氢酶抑制剂, 显示出抗炎作用。 | |||
T16743 |
Rhodamine 123
R-22420,罗丹明 123,RH-123,罗丹明123 |
Others | Others |
Rhodamine 123 是一种荧光染料(λex=503 nm, λem=527 nm)。 | |||
T11024 |
DHODH-IN-15
|
Dehydrogenase | Metabolism |
DHODH-IN-15是一种 A771726 的 hydroxyfurazan 类似物。DHODH-IN-15 是一种二氢乳清酸脱氢酶 (DHODH) 抑制剂,对大鼠肝脏 DHODH 的 IC50 为 11 μM。DHODH-IN-15 可用于类风湿关节炎。 | |||
T40168 |
DHODH-IN-16
|
Dehydrogenase | Metabolism |
DHODH-IN-16 是一种有效的二氢乳清酸脱氢酶抑制剂(DHODH,IC50 = 0.396 nM)。 | |||
T67875 |
DHODH-IN-23
|
Dehydrogenase | Metabolism |
DHODH-IN-23是一种 DHODH 抑制剂,具有口服活性。DHODH-IN-23常用于对癌症的研究。 | |||
T8767 |
PfDHODH-IN-2
|
Dehydrogenase; Parasite | Metabolism; Microbiology/Virology |
PfDHODH-IN-2 是一种二氢噻吩酮衍生物,是一种有效的恶性疟原虫二氢乳清酸脱氢酶抑制剂,其IC50值为 1.11 µM。它具有抗疟作用,可研究疟疾。 | |||
T16744 |
Rhodamine 6G
Basic Red 1,罗丹明6G,罗丹明 6G |
Others | Others |
Rhodamine 6G (Basic Red 1) 是一种罗丹明类似物,可用于表征 MRP1 介导的流出的动力学,测定 Pgp 的流出,可用作激光染料和潜在的线粒体探针。 | |||
T11031 |
hDHODH-IN-7
DHODH-IN-9 |
Dehydrogenase | Metabolism |
hDHODH-IN-7 (DHODH-IN-9) 是一种含嗪的类似物,是一种人二氢乳清酸酯脱氢酶抑制剂。hDHODH-IN-7 具有抗病毒作用,pMIC50 为 7.4。 | |||
T26078 |
Rhodblock 6
Rhodblock6,Rhodblock-6 |
ROCK | Cell Cycle/Checkpoint; Cytoskeletal Signaling; Stem Cells |
Rhodblock 6 是一种 Rho 激酶 (ROCK) 抑制剂,可抑制磷酸化 MRLC(肌球蛋白调节轻链)定位,通过特异性抑制 Rho 激酶的活性发挥作用。 | |||
T11030 |
DHODH-IN-8
|
Dehydrogenase | Metabolism |
DHODH-IN-8 是一种人和恶性疟原虫二氢乳清酸脱氢酶的抑制剂,IC50 分别为 0.13 μM 和 47.4 μM,Ki 分别为 0.016 μM 和 5.6 μM。DHODH-IN-8 具有抗疟疾能力。 | |||
T18977 |
Dihydrorhodamine 123
二氢若丹明123,DHR 123 |
Others | Others |
Dihydrorhodamine 123 (DHR 123) 是一种荧光探针 (λex=488 nm,λem=525 nm)。 | |||
T60364 |
DHODH-IN-17
|
Dehydrogenase | Metabolism |
DHODH-IN-17是一种人DHODH抑制剂,IC50为0.40 μM。DHODH-IN-17 是一种 2- 苯胺酰烟酸,可用于研究急性髓系白血病 (AML) 。 | |||
T37320 |
Rhod-FF AM
|
||
Rhod-FF AM is a cell-permeant acetoxymethyl ester of the fluorescent calcium indicator rhod-FF . As rhod-FF AM enters cells, it is hydrolyzed by intracellular esterases to produce rhod-FF. Rhod-FF is a difluorinated analog of the cell-impermeant calcium indicator rhod-2. It has a very low affinity for calcium (Kd = 320 μM). Low affinity calcium indicators are particularly useful for studying compartments with high concentrations of calcium, such as endoplasmic reticulum, where high affinity dyes... | |||
TD0065 |
6-CR110, SE [6-Carboxyrhodamine 110, succinimidyl ester]*Single isomer*
6-羧基罗丹明110琥珀酰亚胺酯(单一化合物) |
||
6-CR110, SE [6-Carboxyrhodamine 110, succinimidyl ester]*Single isomer* is a Fluorescein for peptide and oligonucleotide labeling. Compared to fluorescein labeling reagents such as FITC and FAM, CR110 reagents give more photostable and pH-independent bioconjugates that have the absorption maximum around the preferred 488 nm excitation wavelength. They are photostable alternative reagents superior to FITC and FAM. | |||
TD0067 |
5(6)-ROX [5-(and 6)-Carboxy-X-rhodamine] *Mixed isomers*
|
||
ROX dyes have a strong red fluorescence.Their excitation and emission wavelengths are longer than those of traditional rhodamine dyes.They are used as labels for peptides, proteins, and other biological ligands.5-ROX, 6-ROx, and their mixture of 5(6) -RoX | |||
T34320 |
Rhodexin A
|
Others | Others |
Rhodexin A is a cardetonic agent of the plant Rhodea japonica. | |||
T70017 |
13(S)HODE Ethanolamide
|
Others | Others |
13(S)HODE Ethanolamide is a biochemical used to inhibit the adhesion of tumor cells | |||
T37862 |
9(R)-HODE
|
Others | Others |
9(R)-HODE is one of several monohydroxylated products of linoleic acid. All known mammalian lipoxygenases appear to catalyze the oxygenation of arachidonic and linoleic acid to give products having strictly the (S) configuration at the site of oxygen insertion. However, both human umbilical vein endothelial cells and bovine aorta endothelial cells have been shown to produce 9(R)-HODE when incubated with linoleic acid. The physiological function of 9(R)-HODE and the enzyme that catalyzes its form... | |||
T76138 |
Phosphodiesterase
|
Others | Others |
Phosphodiesterase(PDE) 是一种可以催化环核苷酸3 '环磷酸键水解的酶,常用于生化研究。Phosphodiesterase 可作为第二信使分子 cAMP 和 cGMP 介导的信号转导的重要调节因子。根据其对环核苷酸的特异性也可以分别不同类型,如 PDE1-PDE11,在多种疾病方面也具有一定的潜力。 | |||
T64146 |
RORγt/DHODH-IN-3
|
Others | Others |
RORγt/DHODH-IN-3 (compound (S)-14d) 是一种有效的、口服具有活力 RORγt (IC50: 0.098 μM) 和 DHODH (IC50: 0.432 μM) 的双重抑制剂。RORγt/DHODH-IN-1 具有明显的体内抗炎作用。 | |||
T34321 |
Rhododendrol, (+/-)-
AI3-31843 |
Others | Others |
Rhododendrol, (+/-)-, is an aromatic compound that may be useful in the treatment of hepatic diseases. However, this product is a known pro-oxidant which can be toxic to melanocytes. | |||
T32584 |
Lathodoratin
|
Others | Others |
Lathodoratin is a bioactive chemical. | |||
T126500 |
Trichodermamide C
|
Others | Others |
Trichodermamide C 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126500,CAS号为 1036712-09-0。 | |||
T125826 |
Apiosylrhododendrin
|
Others | Others |
Apiosylrhododendrin 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125826,CAS号为 146609-83-8。 | |||
T38209 |
Hodgkinsine
|
Others | Others |
Hodgkinsine is a pyrrolidinoindoline alkaloid that has been found inP. colorataand has analgesic activity.1It increases latency to paw licking in the hot plate test and latency to tail withdrawal in the tail-flick test in mice when administered at a dose of 5 mg/kg. 1.Amador, T.A., Verotta, L., Nunes, D.S., et al.Antinociceptive profile of hodgkinsinePlanta Med.66(8)770-772(2000) | |||
T64845 |
Rhodamine-6G N-Phenyl-thiosemicarbazide
|
Others | Others |
1-(3',6'-Bis(ethylamino)-2',7'-dimethyl-3-oxospiro[isoindoline-1,9'-xanthen]-2-yl)-3-phenylthiourea 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T64845。 | |||
T123823 |
Isorhodoptilometrin
|
Others | Others |
Isorhodoptilometrin 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T123823,CAS号为 97995-25-0。 | |||
T34933 |
Trichodesmic acid
(+)-Trichodesmic acid |
Others | Others |
Trichodesmic acid is a new bisabolane-type sesquiterpene. | |||
T63148 |
DHODH-IN-20
|
Others | Others |
DHODH-IN-20 (Compound 133) 是一种 DHODH 的有效抑制剂。其中 DHODH 是一种含铁的黄素依赖性酶,存在于人类线粒体的内膜中。DHODH-IN-20 对肿瘤的生长具有抑制作用。DHODH-IN-20 具有潜力进行急性髓细胞白血病的研究。 | |||
T67239 |
Tetrakis[(S)-(+)-(1-adamantyl)-(N-phthalimido)acetato]dirhodium(II)
|
Others | Others |
Tetrakis[(S)-(+)-(1-adamantyl)-(N-phthalimido)acetato]dirhodium(II) 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T67239,CAS号为 909389-99-7。 | |||
TD0066 |
5(6)-TAMRA [5-(and-6)-Carboxytetramethylrhodamine] *Mixed isomers*
|
||
5(6)-TAMRA contains a carboxylic acid that can be used to react with primary amines via carbodiimide activation of the carboxylic acid. This bright, orange-fluorescent dye produces conjugates with absorption/emission maxima of ~555/580 nm. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T19924 |
Rhododendrol
Betuligenol,Frambinol,杜鹃醇 |
Others | Others |
Rhododendrol (Frambinol) 是一种黑色素合成物,防止雄性小鼠高脂饮食引起的体重升高和增加雄性小鼠白色脂肪细胞的脂肪分解。Rhododendrol 可用作美白/美白化妆品抑制剂。 | |||
T3852 |
Rhodiosin
|
Antioxidant; AChE | Neuroscience; oxidation-reduction |
Rhodiosin 是从红景天的根中分离的特异性非竞争性细胞色素 P450 2D6 抑制剂,IC50=0.761 μM,Ki=0.769 μM。它有 DPPH 自由基清除活性,IC50=27.7 μM。它抑制乙酰胆碱酯酶,IC50范围为 57.50 至 2.43 μg/mL。 | |||
T5S0527 |
Rhodojaponin III
闹羊花素 Ⅲ,闹羊花毒素III |
Others | Others |
Rhodojaponin III 是二萜类化合物,提取于Rhododendron molle 叶子,具有抗炎作用。 | |||
T4S0528 |
Rhodojaponin V
闹羊花素 V,闹羊花毒素V |
Others; Antibacterial | Microbiology/Virology; Others |
Rhodojaponin V 是一种从Rhododendron molle 叶子中获得的二萜类化合物,具有抗炎作用。 | |||
T2S2043 |
Dracorhodin perchlorate
Dracorhodin perochlorate,血竭素高氯酸盐,Dracohodin perochlorate |
Apoptosis; Others | Apoptosis; Others |
Dracorhodin perchlorate 是来源于中药血竭的一种天然产物。它抑制细胞生长,并以剂量和时间依赖性方式诱导成纤维细胞凋亡,将细胞周期阻滞在 G1 期,可作为抗乳腺癌的候选药物。 | |||
TN1011 |
Rhodionin
|
P450; AChE | Metabolism; Neuroscience |
Rhodionin 是从红景天的根中分离的特异性非竞争性细胞色素 P450 2D6 抑制剂,IC50=0.761 μM,Ki=0.769 μM。它有 DPPH 自由基清除活性,IC50为 19.49 μM。它抑制乙酰胆碱酯酶,IC50范围为 57.50 至 2.43 μg/mL。 | |||
T7975 |
Rhodamine B
罗丹明B,Rhodamine B,罗丹明 B,Tetraethylrhodamine,Brilliant Pink B,Basic Violet 1,Rhodamine O |
Others | Others |
Rhodamine B (Brilliant Pink B) 是荧光染料,常用于染色纺织品、肥皂、纸张、皮革和药品。 | |||
T5S0526 |
Rhodojaponin II
闹羊花素 II,闹羊花毒素II |
Others | Others |
Rhodojaponin II 是 Rhododendron molle 叶子中获得的二萜类化合物,具有抗炎作用。 | |||
TN4909 | (+)-Rhododendrol | Others | Others |
(+)-Rhododendrol shows anti-inflammatory effects, it can suppress the NO production by activated macrophages in vivo. | |||
TN6252 | Isostephodeline | ||
Isostephodeline 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6252,CAS号为 56648-85-2。 | |||
T3833 |
Sanshodiol
|
Others | Others |
Sanshodiol是一种天然产物,属于芸香科花椒属,其产品编号为 T3833,CAS号为 54854-91-0。Sanshodiol可用作对照参考。 | |||
TN6261 |
Stephodeline
|
||
Stephodeline 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6261,CAS号为 56596-12-4。 | |||
T40741 |
Dracorhodin
|
Others | Others |
Dracorhodin, the primary constituent found in the sanguis draconis extract, is a flavylium compound classified within the anthocyanin family. Notably, dracorhodin possesses the ability to elicit vasodilation. | |||
T13868 |
Rhodiolin
|
Others | Others |
Rhodiolin is a natural product(flavonoid) isolated from Rhodiola fastigita. | |||
TN6173 |
Rhodomyrtosone I
|
||
Rhodomyrtosone I 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6173,CAS号为 1402725-98-7。 | |||
TN2155 |
Rhodiocyanoside A
|
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Rhodiocyanoside A has antiallergic activity, it exhibits inhibitory activity on the histamine release from rat peritoneal exudate cells sensitized with anti-DNP IgE and inhibits the PCA reaction in rats. | |||
TN7421 |
Beta-Dimorphecolic acid (9(S)-HODE)
|
Others | Others |
Dexamethasone exhibits anti-inflammatory activity. | |||
TN3269 |
8,9-Didehydro-7-hydroxydolichodial
|
Others | Others |
8,9-Didehydro-7-hydroxydolichodial是一种天然产物,属于败酱科败酱属,其产品编号为 TN3269,CAS号为 97856-19-4。8,9-Didehydro-7-hydroxydolichodial可用作对照参考。 | |||
T40627 |
Trichodesmine
|
Others | Others |
Trichodesmine, a dehydropyrrolizidine alkaloid, exhibits hepatotoxic, pneumotoxic, and neurotoxic effects in vivo. | |||
T34931 |
Trichodecenin II
Trichodecenin-II,4-Decenoyl-gly-gly-leu-aib-gly-leu-lol |
Others | Others |
Trichodecenin II is a peptaibol isolated from Trichoderma viride. | |||
TN6133 |
Rhodomyrtone
Rhodomyrtone A |
||
Rhodomyrtone 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6133,CAS号为 468757-69-9。 |