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Targets Recommended: Antibacterial Antibiotic

322

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83

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Cat. No. Product Name Form Specificity Of Inhibition
C0051 Penicillin-Streptomycin Solution (100×), Sterile

青霉素-链霉素双抗溶液(100×),灭菌

Solution in bottle
C0052 Penicillin-Streptomycin-Amphotericin B Solution (100×), Sterile

青霉素-链霉素-两性霉素B三抗溶液(100×),灭菌

Solution in bottle

TargetMol 试剂盒

青霉素-链霉素双抗溶液(100×),灭菌
Cat.No: C0051
青霉素-链霉素-两性霉素B三抗溶液(100×),灭菌
Cat.No: C0052
Cat. No. Product Name Target Signaling Pathways
T14391 Azidamfenicol

Antibacterial; Antibiotic Microbiology/Virology
Azidamfenicol 抑制核糖体肽基转移酶,Ki 为 22 µM。Azidamfenicol 是一种广谱氯霉素类抗生素。
T9680 Irloxacin

Antibacterial Microbiology/Virology
Irloxacin 是一种口服活性的喹诺酮类抗菌剂,在酸性条件下具有更强大的活性。在体外,Irloxacin 对革兰氏阳性菌和革兰氏阴性菌都具有良好的抗菌谱。
T20525 Chloramphenicol palmitate

Antibacterial; Antibiotic Microbiology/Virology
Chloramphenicol palmitate 是一种广谱抗生素,对革兰氏阳性和革兰氏阴性细菌具有活性。 Chloramphenicol palmitate 可用于在含有氯霉素抗性基因的转化细胞中作为细菌选择剂的研究。
T4998L Cefpodoxime (free acid)

Others Others
Cefpodoxime (free acid) 是一种口服的第三代头孢菌素抗生素。除铜绿假单胞菌、肠球菌和脆弱拟杆菌外,它对大多数革兰氏阳性和革兰氏阴性微生物均有效。
T19858 Brodimoprim

DHFR; Antibacterial Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Brodimoprim 是甲氧苄啶的一种类似物,是口服有效的二氢叶酸还原酶抑制剂,对广谱革兰氏阴性和革兰氏阳性细菌具有高度的抑制作用。
T1008 Cephalexin

头孢氨苄,Cefalexin,Cephacillin

Antibacterial; Antibiotic Microbiology/Virology
Cephalexin (Cephacillin) 是一种强口服活性的头孢菌素抗生素。它通过破坏细菌细胞壁的生长来杀死革兰氏阳性和一些革兰氏阴性细菌。它可研究肺炎、链球菌性咽喉炎、细菌性心内膜炎等。
TP1444 Magainin 2

蛙皮素 2

Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Magainin 2是从非洲爪蟾皮肤中分离得到的一种抗菌肽。它对许多革兰氏阴性和革兰氏阳性细菌显示出抗生素活性,对原生动物也有活性。它通过优先与细菌膜中丰富的阴离子磷脂相互作用而发挥细胞毒性作用。
T6582 Mezlocillin Sodium

美洛西林钠,Baycipen

Antibacterial; Antibiotic Microbiology/Virology
Mezlocillin Sodium (Baycipen) 是一种青霉素 β-内酰胺类抗生素,用于治疗由易感染微生物引起的细菌感染。
T3117 Marbofloxacin

马波沙星,Marbofloxacine,Zeniquin,Marbocyl

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Marbofloxacin (Zeniquin) 是一种具有口服活性的氟喹诺酮类广谱抗菌剂。它可研究革兰氏阳性和革兰氏阴性细菌以及支原体引起的感染。
T5006 Flucloxacillin sodium

氟氯西林钠,floxacillin sodium

Antibacterial; Antibiotic Microbiology/Virology
Flucloxacillin sodium (floxacillin sodium) 是一种高活性抗生素,抑制革兰氏阳性和革兰氏阴性菌。
T0116 Balofloxacin

DNA gyrase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Balofloxacin 是一种具有口服活性的氟喹诺酮类抗生素,可通过干扰 DNA 促旋酶来抑制细菌 DNA 的合成,对革兰氏阴性,革兰氏阳性和厌氧菌具有广谱抗菌活性。它可研究呼吸道,肠道和泌尿道感染。
T0396 Pipemidic acid

吡哌酸,Acido pipemidico

Antibacterial; Antibiotic Microbiology/Virology
Pipemidic acid (Acido pipemidico) 是一种新型抗菌剂,对革兰氏阴性菌和某些革兰氏阳性细菌具有活性,可研究肠道、泌尿和胆道感染。
T9066 Merafloxacin

CI 934

SARS-CoV Microbiology/Virology
Merafloxacin (CI 934) 是一种氟喹诺酮类抗菌药物,也被确定为 SARS-CoV-2 的 1 PRF 抑制剂。它对革兰氏阳性菌和革兰氏阴性菌具有体外活性。
T19794 Temafloxacin

替马沙星,Omniflox

Antibiotic Microbiology/Virology
Temafloxacin (Omniflox) 是一种喹诺酮类广谱抗菌剂,对革兰氏阳性菌、革兰氏阴性菌和厌氧菌均有效。
T40475 Ceftobiprole medocaril

BAL5788,头孢比普酯

Antibacterial Microbiology/Virology
Ceftobiprole medocaril (BAL5788) 是 Ceftobiprole 的前药。Ceftobiprole 是一种广谱的头孢菌素,对耐甲氧西林金黄色葡萄球菌具有活性。
T5189 Omadacycline

PTK 0796,Amadacycline

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Omadacycline (Amadacycline) 是一种具有口服活性的氨基甲基环素抗菌剂,是四环素类抗生素。它与 30S 核糖体亚基结合,抑制细菌蛋白质合成。它可用于研究急性细菌性皮肤和皮肤结构感染,感染性肺炎和尿路感染。
TQ0077 Ceftobiprole

Ro 63-9141,BAL 9141,头孢吡普

Antibacterial Microbiology/Virology
Ceftobiprole (Ro 63-9141) 是一种广谱头孢菌素,对甲氧西林耐受的金黄色葡萄球菌的MIC90值为 2 μg/mL。
T0921 Sulfabenzamide

Sultrin,N-Sulfanilylbenzamide,苯甲酰磺胺

Antibacterial; Antibiotic; Autophagy Autophagy; Microbiology/Virology
Sulfabenzamide (N-Sulfanilylbenzamide) 是一种磺胺类抗菌剂,可单独使用或与磺胺噻唑和磺胺乙酰胺一起用作阴道内的局部抗菌制剂。
T0274 Cinoxacin

西诺沙星,Compound 64716

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Cinoxacin (Compound 64716) 是一种喹诺酮类的合成抗生素, 与Oxolinic acid 和 Nalidixic acid 活性相似。
T7865 Danofloxacin

达氟沙星,达诺沙星,Danofloxacino,Danofloxacin free base,Danofloxacine

Others; DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others
Danofloxacin (Danofloxacin free base) free base 是一种具有口服活性第三代氟喹诺酮抗菌剂,对大多数革兰氏阴性和革兰氏阳性细菌,支原体和衣原体物种具有广谱的活性,并通过抑制细菌的 DNA 回转酶发挥抗菌作用。它可用于牛,猪和鸡呼吸道疾病的研究。
T0133 Cefdinir

FK-482,头孢地尼,CI-983,PD 134393

Glutathione Peroxidase; Antibacterial; Antibiotic Metabolism; Microbiology/Virology
Cefdinir (FK-482) 是头孢菌素类中的一种半合成广谱抗生素,对几种革兰氏阴性和革兰氏阳性细菌引起的感染有效。它可研究耳,鼻窦,喉咙和皮肤的常见细菌感染。
T1190 Cefmenoxime hydrochloride

Cefmenoxime hemihydrochloride,SCE-1365 hemihydrochloride,盐酸头孢甲肟

Antibacterial; Antibiotic; Antifection Microbiology/Virology
Cefmenoxime hydrochloride (Cefmenoxime hemihydrochloride) 是一种头孢类抗生素,可通过静脉内或肌肉内给药。 它对大多数常见的革兰氏阳性和革兰氏阴性微生物有活性,是一种肠杆菌科抑制剂,并且对 β-内酰胺酶的水解具有高度抗性。
T0195 Secnidazole

RP-14539,PM-185184,塞克硝唑

Antibiotic; Parasite Microbiology/Virology
Secnidazole (PM-185184) 是一种具有口服活性唑类抗生素,半衰期比甲硝唑更长。它有潜力研究细菌性阴道病。
T12004 Meropenem trihydrate

美罗培南三水合物,SM 7338 trihydrate

Antibacterial; Antibiotic Microbiology/Virology
Meropenem trihydrate (SM 7338 trihydrate) 是一种碳青霉烯抗生素,具有广谱抗菌活性。它对敏感和耐药的杜克氏杆菌 (MIC 值为 0.015-0.12 mg/mL), 淋病奈瑟氏球菌 (MIC 值为 0.02-0.06 mg/mL)和流感嗜血杆菌 (MIC 值为 0.03-0.12 mg/mL) 具有活性。
T6438 Cefoselis Sulfate

FK 037 Sulfate,FK-037,硫酸头孢噻利

Antibacterial; Antibiotic Microbiology/Virology
Cefoselis Sulfate (FK 037 Sulfate) 是一种头孢菌素 β-内酰胺抗生素。它对多种革兰氏阳性和革兰氏阴性生物均表现出良好的活性。它可以透过血脑屏障。
T1000L Chlorhexidine diacetate

醋酸氯己定,Hibitane diacetate,Chlorhexidine Acetate,Bactigras

CAT; Antibacterial; Antibiotic; Antifection Microbiology/Virology; oxidation-reduction
Chlorhexidine diacetate (Bactigras) 是一种双胍类杀菌剂,能快速消灭革兰氏阳性菌和革兰氏阴性菌。它也用作漱口水以防止口腔菌斑。
T0788L Spectinomycin dihydrochloride pentahydrate

盐酸大观霉素五水合物,Trobicin,Spectogard,Spectinomycin hydrochloride hydrate

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Spectinomycin dihydrochloride pentahydrate (Spectogard) 是一种广谱氨基环糊精抗生素,可以抑制多种革兰氏阳性和革兰氏阴性生物的生长。
T0717L Enoxacin

依诺沙星,NSC 629661,AT 2266,Pd107779,CI 919

DNA/RNA Synthesis; Topoisomerase; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Enoxacin (NSC-629661) 是一种可干扰DNA 复制的氟喹诺酮,抑制细菌 DNA 促旋酶 (IC50=126 µg/ml) 和拓扑异构酶 IV (IC50=26.5 µg/ml)。它是特异性癌症生长抑制剂,可有效抑制革兰氏阳性和阴性细菌。
T1616 Cefotiam hydrochloride

盐酸头孢替安,Pansporin,SCE-963 hydrochloride,Pansporine,头孢替安盐酸盐,Cefotiam dihydrochloride,Halospor

Antibacterial; Antibiotic Microbiology/Virology
Cefotiam hydrochloride (SCE-963 hydrochloride) 是一种肠外头孢菌素类广谱抗生素,对革兰氏阳性菌和革兰氏阴性菌有活性。
T5394 Prulifloxacin

AF 3012,Pruvel,NM441,普卢利沙星

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Prulifloxacin (NM441) 是一种口服有效的氟喹诺酮抗生素 ,对革兰氏阳性和阴性细菌具有广泛活性。它是噻唑喹啉羧酸衍生物 Ulifloxacin 的前药。它有潜力用于下尿路感染和慢性支气管炎。
T0199 Cephradine

Anspor,Cephradin,Velosef,SQ-11436,Sefril,头孢拉定

TOPK; Antibacterial; Antibiotic MAPK; Microbiology/Virology
Cephradine (Anspor) 是广谱口服活性头孢菌素。它对革兰氏阳性和革兰氏阴性病原体都有活性。它已用于泌尿生殖系统、胃肠道和呼吸道感染以及皮肤和软组织感染的研究。它通过直接抑制TOPK 抑制太阳紫外线诱导的皮肤炎症。
T3125 Amikacin sulfate

Amikacin Sulfate Salt,阿米卡霉素硫酸,硫酸阿米卡星

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Amikacin sulfate 是一种氨基糖苷类抗生素,也是卡那霉素的半合成类似物。它具有杀菌作用,直接作用于 30S 和 50S 细菌核糖体亚基,可抑制蛋白质合成。它抑制大多数革兰氏阴性细菌,还抑制易感诺卡氏菌和非结核分枝杆菌引起的感染。
T83705 BING TFA

Blocker of Inter-membrane Stress Responses of Gram-negative Bacteria

BING是一种来源于日本稻田鱼(O. laptipes)的抗菌肽,由液泡蛋白质分选相关蛋白13D样(Vps13D)衍生而来。对包括耐甲氧西林的金黄色葡萄球菌(MRSA; MICs = 4-64 µg/ml)在内的各种革兰氏阴性和革兰氏阳性细菌都有活性。与氨苄西林、阿莫西林和新霉素共同使用时,对抗铜绿假单胞菌(P. aeruginosa)表现出协同效应,并能抑制大肠杆菌(E. coli)对卡那霉素和氨苄西林的抗药性发展。在体内,BING提高了被鳗弧菌(E. tarda)感染的O. laptipes的生存率。
T6706 Ticarcillin sodium

Ticarpen hydrate,Aerugipen hydrate,替卡西林单钠盐单水合物,BRL 2288,AB 2288,Monapen

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Ticarcillin sodium (Aerugipen hydrate) 主要用于抗革兰氏阴性菌, 也能用于研究嗜麦芽感染。
T16028 IMB-XH1

Mcl1-IN-2,7-[(2-吡啶基氨基)-2-噻吩基甲基]-8-喹啉醇

BCL; Antibacterial Apoptosis; Microbiology/Virology
IMB-XH1 (Mcl1-IN-2) 是一种骨髓细胞因子 1 抑制剂。它也是非竞争性的 Delhi metallo-β-lactamase(NDM-1) 抑制剂。它对金属 β-内酰胺酶 NDM-1,IMP-4,ImiS 和 L1 的 IC50值分别为 0.4637 μM,3.980 μM,0.2287 μM 和 1.158 μM。
T1223 Ceftriaxone sodium hydrate

Ceftriaxone Sodium Trihydrate,头孢曲松钠,Ceftriaxone disodium hemiheptahydrate,头孢曲松钠水合物,Ceftriaxone sodium

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Ceftriaxone sodium hydrate 是一种头孢菌素类抗生素,对革兰氏阳性和革兰氏阴性菌均有活性。它具有抗炎和抗氧化作用。
T0717 Enoxacin hydrate

CI-919 hydrate,Enoxacin Sesquihydrate,依诺沙星半水合物,AT-2266 hydrate,依诺沙星倍半水合物

DNA gyrase; DNA/RNA Synthesis; Topoisomerase; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Enoxacin hydrate (AT-2266 hydrate) 是氟喹诺酮,可干扰DNA 复制,抑制细菌 DNA 促旋酶 (IC50=126 µg/ml) 和拓扑异构酶 IV (IC50=26.5 µg/ml)。它是特异性癌症生长抑制剂,抑制革兰氏阳性和阴性细菌。
T6382 Amikacin disulfate

硫酸阿米卡星,Pierami,阿米卡星硫酸盐,BAY-416651 sulfate,BB-K8,Amikacin sulfate

Antibacterial; Antibiotic Microbiology/Virology
Amikacin disulfate (BAY-416651 sulfate) 是氨基糖苷类抗生素,也是卡那霉素的半合成类似物。它具有杀菌作用,直接作用于 30S 和 50S 细菌核糖体亚基,可抑制蛋白质合成。它对大多数革兰氏阴性细菌都有效。它还抑制易感诺卡氏菌和非结核分枝杆菌引起的感染。
T73997 Anti gram-positive/negative bacteria agent 1

Others Others
Anti gram-positive/negative bacteria agent 1 是一种含有基于MECAM的人工铁载体的抗生素化合物。
T6383 Amikacin hydrate

阿米卡星水合物,BAY416651 hydrate

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Amikacin hydrate (BAY416651 hydrate) 是氨基糖苷类抗生素,也是卡那霉素的半合成类似物。它具有杀菌作用,直接作用于 30S 和 50S 细菌核糖体亚基,可抑制蛋白质合成。它还抑制易感诺卡氏菌和非结核分枝杆菌引起的感染。
T20774 Sarafloxacin

A-56620,A 56620,A56620,沙拉沙星

Antibacterial; Antibiotic Microbiology/Virology
Sarafloxacin (A56620) 对革兰氏阳性菌和革兰氏阴性菌具有抗菌活性。
T8352 Phanquinone

Antibacterial Microbiology/Virology
Phanquinone 对广泛的革兰氏阳性和革兰氏阴性生物具有活性。
T11315 Fosmidomycin sodium salt

FR-31564 sodium salt

Antibiotic; Parasite Microbiology/Virology
Fosmidomycin sodium salt (FR-31564 sodium salt) 是一种抗感染类抗生素,具有抗疟疾活性,抑制革兰氏阴性菌和革兰氏阳性菌。
T22314 Doripenem

Antibacterial; Antibiotic Microbiology/Virology
Doripenem 是对革兰氏阳性菌、阴性菌和厌氧菌有效的β-内酰胺广谱抗生素。
T0425 Pefloxacin Mesylate

Pefloxacinium mesylate,甲磺酸培氟沙星

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Pefloxacin Mesylate (Pefloxacinium mesylate) 是一种抗菌化合物,可抑制DNA 旋转酶阻断DNA 复制。
T20711 Hemipyocyanine

1-羟基吩嗪,528-71-2

Amylase Metabolism
Hemipyocyanine (528-71-2) 是一种 α-淀粉酶抑制剂。
T12992 SPR741 acetate

SPR741 acetate,NAB741 acetate,SPR741 acetate (1179330-52-9 free base)

Antibacterial Microbiology/Virology
SPR741 acetate 是衍生自多粘菌素 B 的阳离子肽,通过增加革兰氏阴性细菌外膜的通透性来抑制严重的革兰氏阴性细菌感从而展现出对革兰氏阴性菌的抗菌活性。SPR741 acetate 常与抗生素联合使用来治疗一些疾病。
T6492 Davercin

环酯红霉素,Erythromycin Cyclocarbonate

Antibacterial; Antibiotic Microbiology/Virology
Davercin (Erythromycin Cyclocarbonate) 是 Erythromycin 的衍生物,对革兰氏阳性菌和一些革兰氏阴性菌有活性。
T1640 Ciprofloxacin

Ciproxan,环丙沙星,Ciprobay,Bay o 9867,Bay-09867

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Ciprofloxacin (Bay-09867) 是一种有高抗菌活性的氟喹诺酮类抗生素。
T1037 Doripenem monohydrate

多尼培南(一水合物),S 4661 monohydrate,Doripenem Hydrate,S-4661

Antibacterial; Antibiotic Microbiology/Virology
Doripenem monohydrate (S 4661 monohydrate) 是广谱β-内酰胺抗生素,它对革兰氏阳性,阴性和厌氧菌有抗菌作用。

化合物

Azidamfenicol
Cat.No: T14391
Synonym:
Target: Antibacterial, Antibiotic
Irloxacin
Cat.No: T9680
Synonym:
Target: Antibacterial
Chloramphenicol palmitate
Cat.No: T20525
Synonym:
Target: Antibacterial, Antibiotic
Cefpodoxime (free acid)
Cat.No: T4998L
Synonym:
Target: Others
Brodimoprim
Cat.No: T19858
Synonym:
Target: DHFR, Antibacterial
Cephalexin
Cat.No: T1008
Synonym: 头孢氨苄,Cefalexin,Cephacillin
Target: Antibacterial, Antibiotic
Magainin 2
Cat.No: TP1444
Synonym: 蛙皮素 2
Target: Antibacterial, Antibiotic, Antifungal
Mezlocillin Sodium
Cat.No: T6582
Synonym: 美洛西林钠,Baycipen
Target: Antibacterial, Antibiotic
Marbofloxacin
Cat.No: T3117
Synonym: 马波沙星,Marbofloxacine,Zeniquin,Marbocyl
Target: Topoisomerase, Antibacterial, Antibiotic
Flucloxacillin sodium
Cat.No: T5006
Synonym: 氟氯西林钠,floxacillin sodium
Target: Antibacterial, Antibiotic
Balofloxacin
Cat.No: T0116
Synonym:
Target: DNA gyrase, Antibacterial, Antibiotic
Pipemidic acid
Cat.No: T0396
Synonym: 吡哌酸,Acido pipemidico
Target: Antibacterial, Antibiotic
Merafloxacin
Cat.No: T9066
Synonym: CI 934
Target: SARS-CoV
Temafloxacin
Cat.No: T19794
Synonym: 替马沙星,Omniflox
Target: Antibiotic
Ceftobiprole medocaril
Cat.No: T40475
Synonym: BAL5788,头孢比普酯
Target: Antibacterial
Omadacycline
Cat.No: T5189
Synonym: PTK 0796,Amadacycline
Target: ribosome, Antibacterial, Antibiotic
Ceftobiprole
Cat.No: TQ0077
Synonym: Ro 63-9141,BAL 9141,头孢吡普
Target: Antibacterial
Sulfabenzamide
Cat.No: T0921
Synonym: Sultrin,N-Sulfanilylbenzamide,苯甲酰磺胺
Target: Antibacterial, Antibiotic, Autophagy
Cinoxacin
Cat.No: T0274
Synonym: 西诺沙星,Compound 64716
Target: Topoisomerase, Antibacterial, Antibiotic
Danofloxacin
Cat.No: T7865
Synonym: 达氟沙星,达诺沙星,Danofloxacino,Danofloxacin free base,Danofloxacine
Target: Others, DNA/RNA Synthesis, Antibacterial, Antibiotic
Cefdinir
Cat.No: T0133
Synonym: FK-482,头孢地尼,CI-983,PD 134393
Target: Glutathione Peroxidase, Antibacterial, Antibiotic
Cefmenoxime hydrochloride
Cat.No: T1190
Synonym: Cefmenoxime hemihydrochloride,SCE-1365 hemihydrochloride,盐酸头孢甲肟
Target: Antibacterial, Antibiotic, Antifection
Secnidazole
Cat.No: T0195
Synonym: RP-14539,PM-185184,塞克硝唑
Target: Antibiotic, Parasite
Meropenem trihydrate
Cat.No: T12004
Synonym: 美罗培南三水合物,SM 7338 trihydrate
Target: Antibacterial, Antibiotic
Cefoselis Sulfate
Cat.No: T6438
Synonym: FK 037 Sulfate,FK-037,硫酸头孢噻利
Target: Antibacterial, Antibiotic
Chlorhexidine diacetate
Cat.No: T1000L
Synonym: 醋酸氯己定,Hibitane diacetate,Chlorhexidine Acetate,Bactigras
Target: CAT, Antibacterial, Antibiotic, Antifection
Spectinomycin dihydrochloride pentahydrate
Cat.No: T0788L
Synonym: 盐酸大观霉素五水合物,Trobicin,Spectogard,Spectinomycin hydrochloride hydrate
Target: ribosome, Antibacterial, Antibiotic
Enoxacin
Cat.No: T0717L
Synonym: 依诺沙星,NSC 629661,AT 2266,Pd107779,CI 919
Target: DNA/RNA Synthesis, Topoisomerase, Antibacterial, Antibiotic
Cefotiam hydrochloride
Cat.No: T1616
Synonym: 盐酸头孢替安,Pansporin,SCE-963 hydrochloride,Pansporine,头孢替安盐酸盐,Cefotiam dihydrochloride,Halospor
Target: Antibacterial, Antibiotic
Prulifloxacin
Cat.No: T5394
Synonym: AF 3012,Pruvel,NM441,普卢利沙星
Target: Topoisomerase, Antibacterial, Antibiotic
Cephradine
Cat.No: T0199
Synonym: Anspor,Cephradin,Velosef,SQ-11436,Sefril,头孢拉定
Target: TOPK, Antibacterial, Antibiotic
Amikacin sulfate
Cat.No: T3125
Synonym: Amikacin Sulfate Salt,阿米卡霉素硫酸,硫酸阿米卡星
Target: ribosome, Antibacterial, Antibiotic
BING TFA
Cat.No: T83705
Synonym: Blocker of Inter-membrane Stress Responses of Gram-negative Bacteria
Target:
Ticarcillin sodium
Cat.No: T6706
Synonym: Ticarpen hydrate,Aerugipen hydrate,替卡西林单钠盐单水合物,BRL 2288,AB 2288,Monapen
Target: Others, Antibacterial, Antibiotic
IMB-XH1
Cat.No: T16028
Synonym: Mcl1-IN-2,7-[(2-吡啶基氨基)-2-噻吩基甲基]-8-喹啉醇
Target: BCL, Antibacterial
Ceftriaxone sodium hydrate
Cat.No: T1223
Synonym: Ceftriaxone Sodium Trihydrate,头孢曲松钠,Ceftriaxone disodium hemiheptahydrate,头孢曲松钠水合物,Ceftriaxone sodium
Target: Others, Antibacterial, Antibiotic
Enoxacin hydrate
Cat.No: T0717
Synonym: CI-919 hydrate,Enoxacin Sesquihydrate,依诺沙星半水合物,AT-2266 hydrate,依诺沙星倍半水合物
Target: DNA gyrase, DNA/RNA Synthesis, Topoisomerase, Antibacterial, Antibiotic
Amikacin disulfate
Cat.No: T6382
Synonym: 硫酸阿米卡星,Pierami,阿米卡星硫酸盐,BAY-416651 sulfate,BB-K8,Amikacin sulfate
Target: Antibacterial, Antibiotic
Anti gram-positive/negative bacteria agent 1
Cat.No: T73997
Synonym:
Target: Others
Amikacin hydrate
Cat.No: T6383
Synonym: 阿米卡星水合物,BAY416651 hydrate
Target: Others, Antibacterial, Antibiotic
Sarafloxacin
Cat.No: T20774
Synonym: A-56620,A 56620,A56620,沙拉沙星
Target: Antibacterial, Antibiotic
Phanquinone
Cat.No: T8352
Synonym:
Target: Antibacterial
Fosmidomycin sodium salt
Cat.No: T11315
Synonym: FR-31564 sodium salt
Target: Antibiotic, Parasite
Doripenem
Cat.No: T22314
Synonym:
Target: Antibacterial, Antibiotic
Pefloxacin Mesylate
Cat.No: T0425
Synonym: Pefloxacinium mesylate,甲磺酸培氟沙星
Target: Topoisomerase, Antibacterial, Antibiotic
Hemipyocyanine
Cat.No: T20711
Synonym: 1-羟基吩嗪,528-71-2
Target: Amylase
SPR741 acetate
Cat.No: T12992
Synonym: SPR741 acetate,NAB741 acetate,SPR741 acetate (1179330-52-9 free base)
Target: Antibacterial
Davercin
Cat.No: T6492
Synonym: 环酯红霉素,Erythromycin Cyclocarbonate
Target: Antibacterial, Antibiotic
Ciprofloxacin
Cat.No: T1640
Synonym: Ciproxan,环丙沙星,Ciprobay,Bay o 9867,Bay-09867
Target: Topoisomerase, Antibacterial, Antibiotic
Doripenem monohydrate
Cat.No: T1037
Synonym: 多尼培南(一水合物),S 4661 monohydrate,Doripenem Hydrate,S-4661
Target: Antibacterial, Antibiotic
Cat. No. Product Name Target Signaling Pathways
T2P2937 Nonacosane

Others; Antibacterial Microbiology/Virology; Others
Nonacosane 是从Baphia massaiensis 分离的,是一种由 29 个碳原子组成的直链烷烃,具有植物代谢物和挥发油成分的作用。
T8126 Cefodizime Sodium

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Cefodizime sodium 是一种头孢菌素抗生素,具有抗菌活性。它对肾脏没有毒性,具有良好的耐受性和免疫调节活性,可研究呼吸道和泌尿道的严重感染。
T4S0867 Pogostone

DHELWANGIN,广藿香酮

Apoptosis; Antibacterial; Autophagy Apoptosis; Autophagy; Microbiology/Virology
Pogostone (DHELWANGIN) 是从薄荷中分离出,对革兰氏阴性菌、革兰氏阳性菌、大肠埃希菌等具有强效抗菌、抗真菌活性。它诱导细胞凋亡和自噬。
T8118 Bekanamycin

Kanamycin B,卡那霉素,卡那霉素 B

Antibacterial; Antibiotic Microbiology/Virology
Bekanamycin (Kanamycin B) 是一种提取自 Streptomyces kanamyceticus 的氨基糖苷类抗生素,抑制一系列革兰氏阳性和阴性细菌。
T0895 Oxytetracycline

土霉素,Terramycin

ribosome; Endogenous Metabolite; Antibacterial; Antibiotic; HSV Metabolism; Microbiology/Virology
Oxytetracycline (Terramycin) 是一种四环素类抗生素。它强力抑制革兰氏阴性和革兰氏阳性细菌。它是一种蛋白质合成抑制剂,可阻止 aminoacil-tRNA 与复杂的核糖体 RNA 结合,具有抗 HSV-1的活性。
T0224 Meropenem

美罗培南,SM 7338

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Meropenem (SM 7338) 是一种具有广谱抗菌活性的碳青霉烯抗生素,对敏感和耐药的淋病奈瑟氏球菌,流感嗜血杆菌和杜克氏杆菌的 MIC 值分别为 0.02-0.06 mg/mL,0.03-0.12 mg/mL 和 0.015-0.12 mg/mL。
T19808 5-Bromo-5-nitro-1,3-dioxane

Bronidox,5-溴-5-硝基-1,3-二噁烷,5-溴-5-硝基-1,3-二恶烷

Others; Antibacterial; Antifungal Microbiology/Virology; Others
5-Bromo-5-nitro-1,3-dioxane (Bronidox) 是一种抗菌化合物,可通过必需蛋白硫醇的氧化抑制酶活性并随后抑制微生物的生长。它有抗革兰氏阳性和革兰氏阴性细菌,以及抗真菌活性。
T8160 EGCG Octaacetate

乙酰化表没食子儿茶素没食子酸酯,乙酰化EGCG

Others; Antibacterial Microbiology/Virology; Others
EGCG Octaacetate 是表没食子儿茶素没食子酸酯的前药,对革兰氏阳性菌和革兰氏阴性菌有潜在抗菌可能。它可下调 PI3K/Akt/NFκB 磷酸化和 p65 乙酰化来降低促炎介质水平,减少小鼠结肠炎引起的结肠癌。
T6624 Oxytetracycline Dihydrate

土霉素二水合物,地霉素,Terramycin Dihydrate

Others; Endogenous Metabolite; Antibacterial; Antibiotic; HSV Metabolism; Microbiology/Virology; Others
Oxytetracycline Dihydrate (Terramycin Dihydrate) 是一种四环素类抗生素,可抑制革兰氏阴性和革兰氏阳性细菌。它是一种蛋白质合成抑制剂,可阻止 aminoacil-tRNA 与复杂的核糖体 RNA 结合,还具有抗 HSV-1的活性。
T0788 Spectinomycin dihydrochloride

淋必治,Spectinomycin 2HCl,盐酸奇霉素,Actinospectacin

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Spectinomycin dihydrochloride (Actinospectacin) 是一种能与细菌核糖体的30S 亚基结合,干扰蛋白质合成的抗生素。
TCS1554 trans-Benzylideneacetone

反式苯亚甲基丙酮,Acetocinnamone,亚苄基丙酮

Phospholipase Metabolism
trans-Benzylideneacetone (Acetocinnamone) 是一种革兰氏阴性致病性线虫细菌嗜线虫(Xenorhabdus nematophila) 的代谢产物,是一种针对磷脂酶 A2 (PLA2) 的酶抑制剂,也是一种免疫抑制剂。
T21430 Oxytetracycline Hydrochloride

Biosolvomycin,盐酸土霉素,Oxytetracycline HCl,Oxytetracycline.HCl,Dalimycin,Oxytetracycline, Sodium Salt,Dalinmycin

Antiviral; Endogenous Metabolite; Antibacterial; HSV Immunology/Inflammation; Metabolism; Microbiology/Virology
Oxytetracycline Hydrochloride (Dalimycin) 是由 Streptomyces rimosus 生产的,一种具有抗菌活性的四环素衍生物。它干扰氨酰-tRNA 与 mRNA-核糖体复合物的结合,从而阻止肽延伸并抑制蛋白质合成。
TN2011 Ombuoside

商陆素-3BETA-芸香糖苷,Ombuin-3beta-rutinoside

Antibacterial Microbiology/Virology
Ombuoside (Ombuin-3beta-rutinoside) 是一种从绞股蓝分离得到的糖苷复合物。它具有抗真菌和抗氧化作用。
TQ0251 (Z)-2-decenoic acid

(Z)-dec-2-enoic acid,(Z)-2-癸烯酸,cis-2-Decenoic acid,cis-dec-2-enoic acid

Others Others
(Z)-2-decenoic acid (cis-dec-2-enoic acid) 是一种由铜绿假单胞菌产生的不饱和脂肪酸。它能够诱导一系列革兰氏阴性细菌(包括铜绿假单胞菌)和革兰氏阳性细菌形成的生物膜发生分散反应。它能够抑制生物膜发育。
T4984 Cefozopran hydrochloride

SCE-2787 hydrochloride

Antifungal Microbiology/Virology
Cefozopran hydrochloride (SCE-2787 hydrochloride) 是一种半合成的非肠道头孢菌素。它是一种广谱抗菌抗生素,能抑制大多数革兰氏阴性和革兰氏阳性菌。
T8261 Ceftazidime Pentahydrate

头孢他啶五水合物,头孢他啶

Antibacterial; Antibiotic Microbiology/Virology
Ceftazidime pentahydrate 是一种β-内酰胺类抗菌剂,对革兰氏阳性和革兰氏阴性需氧细菌有广谱活性,可静脉内或肌肉给药。它对肠杆菌科特别有效,对大多数 β-内酰胺酶具有抗水解作用。
T28764 SF2312

SF-2312,SF 2312

Glucokinase; Antibacterial Metabolism; Microbiology/Virology
SF2312 是一种由放线菌微孢子菌产生的天然膦酸盐抗生素,是高效的糖酵解酶烯醇化酶抑制剂。SF2312 具有抗菌活性,可抑制细菌生长,对革兰氏阴性和革兰氏阴性菌均具有抑制作用。SF2312 抑制人重组 ENO1 和 ENO2。
T8062 Cefazedone

Refosporen,头孢西酮

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Cefazedone (Refosporen) 是一种具有抗革兰氏阳性和革兰氏阴性菌活性的时间依赖性头孢菌素抗生素。
T5757 Loganetin

Antibacterial Microbiology/Virology
Loganetin 是无毒的天然产物,来源于Cornus officinalis Sieb. et Zucc.,可用于耐多药革兰氏阴性菌感染的研究。
T8247 (+)-Aromadendrene

Anti-infection Microbiology/Virology
(+)-Aromadendrene 是一种天然产物,对革兰氏阳性菌和革兰氏阴性菌具有显着的抗菌活性。
T5037 Midecamycin

Antibiotic SF-837,Turimycin P3,Medecamycin A1,Rubimycin,麦迪霉素,Platenomycin B1,Espinomycin A

Antibacterial; Antibiotic Microbiology/Virology
Midecamycin (Medecamycin A1) 是乙酰氧基取代的大环内酯类抗生素,对革兰氏阳性和阴性菌有效。
T1306 Norfloxacin

氟哌酸,MK-0366,诺氟沙星

DNA gyrase; Topoisomerase; Endogenous Metabolite; Antibacterial; Antibiotic DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Norfloxacin (MK-0366) 是广谱抗生素,能通过结合DNA 旋转酶抑制革兰氏阳性和阴性菌。
T1679 Thiostrepton

Thiactin,Bryamycin,Alaninamide,硫链丝菌素

DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Thiostrepton (Alaninamide) 是一种选择性抑制FOXM1的抗生素。FOXM1会与 YAP/TEAD 复合物结合,形成YAP/TEAD/FOXM1 复合物。
T5S0814 Berberine hydrogen sulphate

Berberine Bisulfate,硫酸氢黄连素,Umbellatine Sulfate

Antibacterial Microbiology/Virology
Berberine hydrogen sulphate (Umbellatine Sulfate) 是一种从几种植物中提取的生物碱,对多种微生物具有抗菌活性,包括革兰氏阳性和革兰氏阴性细菌、真菌和原生动物。
T5274 D-​(+)​-​Phenyllactic acid

D-3-苯乳酸,D-3-Phenyllactic acid

Endogenous Metabolite; Antibacterial Metabolism; Microbiology/Virology
D-​(+)​-​Phenyllactic acid (D-3-Phenyllactic acid) 是一种由白地霉分泌得到的抗菌剂,可抑制部分来自人类和食品的革兰氏阳性菌以及来自人类的革兰氏阴性菌。
T0814L Ampicillin

Amcill,D-(-)-α-Aminobenzylpenicillin,Aminobenzylpenicillin,氨苄青霉素,Ampicillin acid

Antibacterial; Antibiotic Microbiology/Virology
Ampicillin (Aminobenzylpenicillin) 属于 β-内酰胺类抗生素,是一种半合成的青霉素。Ampicillin 具有杀菌活性,对各种革兰氏阳性细菌和革兰氏阴性细菌均有抑制活性。
T4889 2,6-Diaminoheptanedioic acid

Others; Endogenous Metabolite Metabolism; Others
2,6-Diaminoheptanedioic acid 是内源性代谢产物的一种。
T8302 Ceftiofur

Antibacterial; Antibiotic Microbiology/Virology
Ceftiofur 是一种半合成抗生素,对家畜的各种革兰氏阳性和革兰氏阴性菌、好氧菌和厌氧菌均有抗菌活性。
T3501 Colistimethate Sodium

Colistin-1,3,5,9-tetramethanesulfonic A acid,多粘菌素E甲磺酸钠

Others Others
Colistin-1,3,5,9-tetramethanesulfonic A acid 用于治疗选择有限的患者因选定的需氧革兰氏阴性病原体引起的严重感染。
T12830 Sapienic acid sodium

Antibacterial Microbiology/Virology
Sapienic acid sodium,主要存在于皮肤和粘膜中的脂肪酸,对皮肤和口腔内的革兰氏阳性及阴性细菌展现出不同程度的抗菌效果。其对血链球菌、微生物链球菌与核纤梭菌的抗菌活性表现,MBC值分别为31.3 μg/mL、375.0 μg/mL与93.8 μg/mL。
T0958 Penicillin G sodium salt

青霉素钠,Penicillin G Sodium,Benzylpenicillin sodium salt,Benzylpenicillin Sodium

GABA Receptor; Antibacterial; Antibiotic Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience
Penicillin G sodium(Benzylpenicillin sodium) salt 是一种 β-内酰胺类抗生素。
T1313 Nitrofurantoin

Furadantine,呋喃妥因,Macrodantin,Furadonine

Antibacterial; Antibiotic Microbiology/Virology
Nitrofurantoin (Furadantine) 是一种具有口服活性的广谱内酰胺酶抗菌剂。它是一种抗生素,可研究尿路感染。
T8148 Mupirocin calcium hydrate

莫匹罗星钙,Mupirocin calcium

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Mupirocin calcium hydrate 是从Pseudomonas fluorescens 中分离得到的,一种有口服活性的抗生素。它可逆地抑制异亮氨酸转移RNA,并抑制细菌蛋白和RNA 的合成起到抗菌作用。
T2989 4-Hydroxybenzoic acid

p-hydroxybenzoic acid,para-Hydroxybenzoic acid,PHBA,对羟基苯甲酸,4-hydroxybenzoate

Endogenous Metabolite; Antibacterial Metabolism; Microbiology/Virology
4-Hydroxybenzoic acid (4-hydroxybenzoate) 是苯甲酸的酚衍生物,可抑制革兰氏阳性和革兰氏阴性菌,IC50值为160 μg/mL。
T1304 Chlortetracycline hydrochloride

Isphamycin,Chlortetracycline HCl,7-Chlorotetracycline hydrochloride,盐酸金霉素

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Chlortetracycline hydrochloride (Isphamycin) 是一种特异性钙离子载体抗生素, 抑制氨酰 tRNA 结合到核糖体。
T40583 3-Oxo-C14-AHL

N-(3-Oxotetradecanoyl)-DL-homoserine lactone

Others Others
3-Oxo-C14-AHL (N-(3-Oxotetradecanoyl)-DL-homoserine lactone) 是由革兰氏阴性菌产生的群体感应 (QS) 信号分子,可用来提高能农作物的产量。
T20643 Cefoxitin

Rephoxitin,Cefoxitinum

Cell wall; Antibacterial; Antibiotic Immunology/Inflammation; Microbiology/Virology
Cefoxitin (Rephoxitin) 是一种广谱的、可口服的第二代头孢霉素类抗生素。Cefoxitin 干扰细菌细胞壁的合成。其活性谱包括革兰氏阴性和革兰氏阳性菌,通常用于腹腔感染、盆腔感染和某些类型的妇科感染等腹部,对厌氧菌具有高效性。
T8262 Fosfomycin sodium

Fosfomycin Disodium,磷霉素钠

Antibacterial; Antibiotic Microbiology/Virology
Fosfomycin sodium 是一种能透过血脑屏障的广谱抗生素,不可逆地抑制细胞壁合成的早期阶段。它对多种细菌具有杀菌活性,包括耐多药、广泛耐药和耐全药的细菌。
T1100 Polymyxin B Sulfate

Aerosporin,硫酸多粘菌素 B,PMB,Polymyxin B sulphate,硫酸多粘菌素B,Polymyxin B sulfate (1404-26-8 free base),Poly-RX

Antibacterial; Antibiotic Microbiology/Virology
Polymyxin B Sulfate (Poly-RX) 是一个阳离子型表面活性剂抗生素剂,能够提高细胞膜的渗透性。
T1104 Paromomycin Sulfate

Aminosidine sulfate,Paromomycin sulfate salt,硫酸巴龙霉素,巴龙霉素硫酸盐

Antibacterial; Antibiotic; Parasite Microbiology/Virology
Paromomycin Sulfate (Aminosidine sulfate) 是一种广谱氨基糖苷类抗生素 ,是具有杀螨杀菌作用的新霉素衍生物。它通过与细菌 30S 核糖体 A 位点的 RNA 寡核苷酸特异性结合,使 mRNA 的翻译提前终止,并抑制蛋白质合成。它可研究细菌和寄生虫感染。
T11855 Lipopolysaccharides

脂多糖,LPS

Others Others
Lipopolysaccharides (LPS) 是革兰氏阴性细菌细胞壁的一种特有成分,由脂质A、寡糖核心和 O -特异性多糖 (O-antigen) 3个区域组成。Lipopolysaccharides 有利于维持细胞外膜的完整性,保护细菌免受胆汁盐和脂类抗生素的破坏。Lipopolysaccharides 是一种高免疫原性抗原,可以增强免疫反应,可以用于炎症模型构建。
T41078 Lipopolysaccharides, Escherichiacoli

Lipopolysaccharide, E. coli O111:B4

Others Others
Lipopolysaccharides, Escherichiacoli (E. coli O111:B4) 是革兰氏阴性细菌细胞壁的一种特有成分,由脂质A、寡糖核心和 O -特异性多糖 (O-antigen) 3个区域组成。Lipopolysaccharides, Escherichiacoli 有利于维持细胞外膜的完整性,保护细菌免受胆汁盐和脂类抗生素的破坏。Lipopolysaccharides, Escherichiacoli 是一种高免疫原性抗原,可以增强免疫反应,可以用于炎症模型构建。
TN4518 Meridinol

Antifection Microbiology/Virology
Meridinol has wide antimicrobial activity, includes against gram-positive and gram-negative bacteria and fungi.
T26805 Bicyclomycin

Bicozamycin

Others Others
Bicyclomycin is a broad spectrum antibiotic active against Gram-negative bacteria and the Gram-positive bacterium, Micrococcus luteusn.
TN6002 Crenatine

1-Ethyl-4-methoxy-β-carboline

Crenatine possesses antibacterial activity, it is more effective against Gram-positive than Gram-negative bacteria.
T1255L Tobramycin Sulfate

Dartobcin,Nebcine,Tobraneg,Tobrasix

Others Others
Tobramycin Sulfate is a broad-spectrum antibiotic. It is effective against gram-negative bacteria. It especially potent against the Pseudomonas species.
T25971 Polymyxin B2

Polymyxin-B2,PolymyxinB2

Others Others
Polymyxin B2 is an antibiotic primarily utilized for resistant Gram-negative infections. It is derived from the bacterium Bacillus polymyxa.
T16673 Pseudouridimycin

PUM

Others Others
Pseudouridimycin is a C-nucleoside analogue. Pseudouridimycin is an antibiotic and is a selective bacterial RNA polymerase (RNAP) inhibitor. It is effective against both Gram-negative and Gram-positive bacteria.
T4131 Arjunic acid

COX; Antifection Immunology/Inflammation; Microbiology/Virology; Neuroscience
Arjunic acid is a strong antioxidant and a free radical scavenger. Arjunic acid shows activity against Gram-positive and Gram-negative bacteria with MIC values ranging between 1.9 and 15.6 microg/mL.
TN1301 6,8-Diprenylgenistein

6,8-二异戊烯基金雀异黄素,鲁冰花

Antifection Microbiology/Virology
6,8-Diprenylgenistein has antimicrobial activity, it has anti-bacteria activity against Gram-negative and Gram-positive bacteria.
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天然产物

Nonacosane
Cat.No: T2P2937
Synonym:
Target: Others, Antibacterial
Cefodizime Sodium
Cat.No: T8126
Synonym:
Target: Others, Antibacterial, Antibiotic
Pogostone
Cat.No: T4S0867
Synonym: DHELWANGIN,广藿香酮
Target: Apoptosis, Antibacterial, Autophagy
Bekanamycin
Cat.No: T8118
Synonym: Kanamycin B,卡那霉素,卡那霉素 B
Target: Antibacterial, Antibiotic
Oxytetracycline
Cat.No: T0895
Synonym: 土霉素,Terramycin
Target: ribosome, Endogenous Metabolite, Antibacterial, Antibiotic, HSV
Meropenem
Cat.No: T0224
Synonym: 美罗培南,SM 7338
Target: Others, Antibacterial, Antibiotic
5-Bromo-5-nitro-1,3-dioxane
Cat.No: T19808
Synonym: Bronidox,5-溴-5-硝基-1,3-二噁烷,5-溴-5-硝基-1,3-二恶烷
Target: Others, Antibacterial, Antifungal
EGCG Octaacetate
Cat.No: T8160
Synonym: 乙酰化表没食子儿茶素没食子酸酯,乙酰化EGCG
Target: Others, Antibacterial
Oxytetracycline Dihydrate
Cat.No: T6624
Synonym: 土霉素二水合物,地霉素,Terramycin Dihydrate
Target: Others, Endogenous Metabolite, Antibacterial, Antibiotic, HSV
Spectinomycin dihydrochloride
Cat.No: T0788
Synonym: 淋必治,Spectinomycin 2HCl,盐酸奇霉素,Actinospectacin
Target: ribosome, Antibacterial, Antibiotic
trans-Benzylideneacetone
Cat.No: TCS1554
Synonym: 反式苯亚甲基丙酮,Acetocinnamone,亚苄基丙酮
Target: Phospholipase
Oxytetracycline Hydrochloride
Cat.No: T21430
Synonym: Biosolvomycin,盐酸土霉素,Oxytetracycline HCl,Oxytetracycline.HCl,Dalimycin,Oxytetracycline, Sodium Salt,Dalinmycin
Target: Antiviral, Endogenous Metabolite, Antibacterial, HSV
Ombuoside
Cat.No: TN2011
Synonym: 商陆素-3BETA-芸香糖苷,Ombuin-3beta-rutinoside
Target: Antibacterial
(Z)-2-decenoic acid
Cat.No: TQ0251
Synonym: (Z)-dec-2-enoic acid,(Z)-2-癸烯酸,cis-2-Decenoic acid,cis-dec-2-enoic acid
Target: Others
Cefozopran hydrochloride
Cat.No: T4984
Synonym: SCE-2787 hydrochloride
Target: Antifungal
Ceftazidime Pentahydrate
Cat.No: T8261
Synonym: 头孢他啶五水合物,头孢他啶
Target: Antibacterial, Antibiotic
SF2312
Cat.No: T28764
Synonym: SF-2312,SF 2312
Target: Glucokinase, Antibacterial
Cefazedone
Cat.No: T8062
Synonym: Refosporen,头孢西酮
Target: Others, Antibacterial, Antibiotic
Loganetin
Cat.No: T5757
Synonym:
Target: Antibacterial
(+)-Aromadendrene
Cat.No: T8247
Synonym:
Target: Anti-infection
Midecamycin
Cat.No: T5037
Synonym: Antibiotic SF-837,Turimycin P3,Medecamycin A1,Rubimycin,麦迪霉素,Platenomycin B1,Espinomycin A
Target: Antibacterial, Antibiotic
Norfloxacin
Cat.No: T1306
Synonym: 氟哌酸,MK-0366,诺氟沙星
Target: DNA gyrase, Topoisomerase, Endogenous Metabolite, Antibacterial, Antibiotic
Thiostrepton
Cat.No: T1679
Synonym: Thiactin,Bryamycin,Alaninamide,硫链丝菌素
Target: DNA/RNA Synthesis, Antibacterial, Antibiotic
Berberine hydrogen sulphate
Cat.No: T5S0814
Synonym: Berberine Bisulfate,硫酸氢黄连素,Umbellatine Sulfate
Target: Antibacterial
D-​(+)​-​Phenyllactic acid
Cat.No: T5274
Synonym: D-3-苯乳酸,D-3-Phenyllactic acid
Target: Endogenous Metabolite, Antibacterial
Ampicillin
Cat.No: T0814L
Synonym: Amcill,D-(-)-α-Aminobenzylpenicillin,Aminobenzylpenicillin,氨苄青霉素,Ampicillin acid
Target: Antibacterial, Antibiotic
2,6-Diaminoheptanedioic acid
Cat.No: T4889
Synonym:
Target: Others, Endogenous Metabolite
Ceftiofur
Cat.No: T8302
Synonym:
Target: Antibacterial, Antibiotic
Colistimethate Sodium
Cat.No: T3501
Synonym: Colistin-1,3,5,9-tetramethanesulfonic A acid,多粘菌素E甲磺酸钠
Target: Others
Sapienic acid sodium
Cat.No: T12830
Synonym:
Target: Antibacterial
Penicillin G sodium salt
Cat.No: T0958
Synonym: 青霉素钠,Penicillin G Sodium,Benzylpenicillin sodium salt,Benzylpenicillin Sodium
Target: GABA Receptor, Antibacterial, Antibiotic
Nitrofurantoin
Cat.No: T1313
Synonym: Furadantine,呋喃妥因,Macrodantin,Furadonine
Target: Antibacterial, Antibiotic
Mupirocin calcium hydrate
Cat.No: T8148
Synonym: 莫匹罗星钙,Mupirocin calcium
Target: Others, Antibacterial, Antibiotic
4-Hydroxybenzoic acid
Cat.No: T2989
Synonym: p-hydroxybenzoic acid,para-Hydroxybenzoic acid,PHBA,对羟基苯甲酸,4-hydroxybenzoate
Target: Endogenous Metabolite, Antibacterial
Chlortetracycline hydrochloride
Cat.No: T1304
Synonym: Isphamycin,Chlortetracycline HCl,7-Chlorotetracycline hydrochloride,盐酸金霉素
Target: ribosome, Antibacterial, Antibiotic
3-Oxo-C14-AHL
Cat.No: T40583
Synonym: N-(3-Oxotetradecanoyl)-DL-homoserine lactone
Target: Others
Cefoxitin
Cat.No: T20643
Synonym: Rephoxitin,Cefoxitinum
Target: Cell wall, Antibacterial, Antibiotic
Fosfomycin sodium
Cat.No: T8262
Synonym: Fosfomycin Disodium,磷霉素钠
Target: Antibacterial, Antibiotic
Polymyxin B Sulfate
Cat.No: T1100
Synonym: Aerosporin,硫酸多粘菌素 B,PMB,Polymyxin B sulphate,硫酸多粘菌素B,Polymyxin B sulfate (1404-26-8 free base),Poly-RX
Target: Antibacterial, Antibiotic
Paromomycin Sulfate
Cat.No: T1104
Synonym: Aminosidine sulfate,Paromomycin sulfate salt,硫酸巴龙霉素,巴龙霉素硫酸盐
Target: Antibacterial, Antibiotic, Parasite
Lipopolysaccharides
Cat.No: T11855
Synonym: 脂多糖,LPS
Target: Others
Lipopolysaccharides, Escherichiacoli
Cat.No: T41078
Synonym: Lipopolysaccharide, E. coli O111:B4
Target: Others
Meridinol
Cat.No: TN4518
Synonym:
Target: Antifection
Bicyclomycin
Cat.No: T26805
Synonym: Bicozamycin
Target: Others
Crenatine
Cat.No: TN6002
Synonym: 1-Ethyl-4-methoxy-β-carboline
Target:
Tobramycin Sulfate
Cat.No: T1255L
Synonym: Dartobcin,Nebcine,Tobraneg,Tobrasix
Target: Others
Polymyxin B2
Cat.No: T25971
Synonym: Polymyxin-B2,PolymyxinB2
Target: Others
Pseudouridimycin
Cat.No: T16673
Synonym: PUM
Target: Others
Arjunic acid
Cat.No: T4131
Synonym:
Target: COX, Antifection
6,8-Diprenylgenistein
Cat.No: TN1301
Synonym: 6,8-二异戊烯基金雀异黄素,鲁冰花
Target: Antifection
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Cat. No. Product Name Species Expression System
TMPY-03118 ORM2 Protein, Human, Recombinant (His)

AGP-B',ORM2,orosomucoid 2,AGP-B,AGP2

Human HEK293 Cells
ORM2 belongs to the calycin superfamily, lipocalin family. Lipocalins share limited regions of sequence homology and a common tertiary structure architecture. They transport small hydrophobic molecules such as steroids, bilins, retinoids, and lipids. Lipocalins can be found in gram-negative bacteria, vertebrate cells, and invertebrate cells, and plants. They are associated with many biological processes. ORM2 functions as a transport protein in the bloodstream. It is expressed by the liver and s...
TMPY-02204 LBP Protein, Human, Recombinant (His)

BPIFD2,lipopolysaccharide binding protein

Human HEK293 Cells
Lipopolysaccharide binding protein ( LBP ) is a glycoprotein that is synthesized principally by hepatocytes. LBP is a trace plasma protein that binds to the lipid A moiety of bacterial lipopolysaccharides ( LPSs ). LBP binds directly to the outer membrane of Gram-negative bacteria and purified aggregates of extracted endotoxin and catalyzes the delivery of endotoxin to the membrane ( mCD14, GPI-Linked ) and soluble ( sCD14 ) forms of CD14, thereby markedly increasing host cell sensitivity to end...
TMPY-02904 TLR4 Protein, Human, Recombinant (His)

TLR-4,TOLL,toll-like receptor 4,ARMD10,TLR4,CD284

Human Baculovirus Insect Cells
TLR4, also known as TLR-4, is a member of the Toll-like receptor (TLR) family, which plays a fundamental role in pathogen recognition and activation of innate immunity. TLRs are highly conserved from Drosophila to humans and share structural and functional similarities. They recognize pathogen-associated molecular patterns (PAMPs) that are expressed on infectious agents, and mediate the production of cytokines necessary for the development of effective immunity. TLR4 is most abundantly expressed...
TMPH-02773 Lysozyme C-2 Protein, Mouse, Recombinant (His & Myc)

Lysozyme C-2,1,4-beta-N-acetylmuramidase C,Lysozyme C type M...

Mouse E. coli
Lysozymes have primarily a bacteriolytic function; those in tissues and body fluids are associated with the monocyte-macrophage system and enhance the activity of immunoagents. Lyz2 is active against a range of Gram-positive and Gram-negative bacteria. More effective than Lyz1 in killing Gram-negative bacteria. Lyz1 and Lyz2 are equally effective in killing Gram-positive bacteria. Lysozyme C-2 Protein, Mouse, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-M...
TMPY-02908 BPI Protein, Human, Recombinant (His)

BPIFD1,bactericidal/permeability-increasing protein,rBPI

Human HEK293 Cells
Bactericidal/permeability-increasing protein is a member of the BPI/LBP/Plunc superfamily and BPI/LBP family. It is a cationic protein which can be detected in the azurophilic granule and on the surface of polymorphonuclear leukocytes. Bactericidal/permeability-increasing protein also is a lipopolysaccharide binding protein. It is associated with human neutrophil granules and has bactericidal activity on gram-negative organisms. Bactericidal/permeability-increasing protein contains two domains t...
TMPH-00230 Cathelicidin-6 Protein, Bovine, Recombinant (His & SUMO)

CATHL6,Antibacterial peptide BMAP-27,Myeloid antibacterial p...

Bovine E. coli
Exerts a potent antimicrobial activity against Gram-negative and Gram-positive bacteria, including methicillin-resistant Staphylococcus aureus, and fungi. Cathelicidin-6 Protein, Bovine, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 16.2 kDa and the accession number is P54228.
TMPH-01772 DEFA1 Protein, Human, Recombinant (GST)

MRS,HP1,HP-1,DEFA1,DEF1,Defensin, alpha 1,Neutrophil defensi...

Human E. coli
Defensin 1 and defensin 2 have antibacterial, fungicide and antiviral activities. Has antimicrobial activity against Gram-negative and Gram-positive bacteria. Defensins are thought to kill microbes by permeabilizing their plasma membrane. DEFA1 Protein, Human, Recombinant (GST) is expressed in E. coli expression system with N-GST tag. The predicted molecular weight is 37.2 kDa and the accession number is P59665.
TMPH-03145 Thanatin Protein, Podisus maculiventris, Recombinant (His & KSI)

Thanatin

Podisus maculiventris E. coli
Insect defense peptide with a broad spectrum of activity against Gram-positive and Gram-negative bacteria and fungi. No activity against S.aureus. Stops respiration in bacteria but does not permeabilize their inner membranes. Thanatin Protein, Podisus maculiventris, Recombinant (His & KSI) is expressed in E. coli expression system with N-6xHis-KSI tag. The predicted molecular weight is 17.8 kDa and the accession number is P55788.
TMPH-02544 DEFB4 Protein, Mouse, Recombinant (His & SUMO)

Bdef4,BD-4,Beta-defensin 4,Defensin, beta 4,mBD-4,Defb4

Mouse E. coli
Exhibits antimicrobial activity against Gram-negative bacteria and Gram-positive bacteria. May act as a ligand for C-C chemokine receptor CCR6. Can bind to mouse (but not human) CCR6 and induce chemotactic activity of CCR6-expressing cells. DEFB4 Protein, Mouse, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 20.6 kDa and the accession number is P82019.
TMPH-03100 PMAP-23 Protein, Pig, Recombinant (His & SUMO)

PMAP23,Antibacterial peptide PMAP-23,Myeloid antibacterial p...

Sus scrofa (Pig) E. coli
Exerts antimicrobial activity against both Gram-positive and negative bacteria at concentrations of 2-16 micro molar. Its activity appears to be mediated by its ability to damage bacterial membranes. PMAP-23 Protein, Pig, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 19.0 kDa and the accession number is P49930.
TMPH-01607 LCE3A Protein, Human, Recombinant (His)

Late envelope protein 13,LCE3A,Late cornified envelope prote...

Human E. coli
A structural component of the cornified envelope of the stratum corneum involved in innate cutaneous host defense (Probable). Possesses defensin-like antimicrobial activity against a broad spectrum of Gram-positive and Gram-negative bacteria, both aerobic and anaerobic species. Upon inflammation, may regulate skin barrier repair by shaping cutaneous microbiota composition and immune response to bacterial antigens. LCE3A Protein, Human, Recombinant (His) is expressed in E. coli expression system ...
TMPY-02163 PGLYRP1 Protein, Mouse, Recombinant (His)

Tnfsf3l,peptidoglycan recognition protein 1,PGRP,Tasg7,Tag7,...

Mouse HEK293 Cells
Peptidoglycan recognition protein 1, also known as Peptidoglycan recognition protein short, PGRP-S, PGLYRP1, PGLYRP, PGRP and TNFSF3L, is a secreted protein that belongs to the N-acetylmuramoyl-L-alanine amidase 2 family. PGLYRP1 / PGLYRP is highly expressed in bone marrow. It is weakly expressed in kidney, liver, small intestine, spleen, thymus, peripheral leukocyte, lung, fetal spleen and neutrophils. PGLYRP1 / PGLYRP is a pattern receptor that binds to murein peptidoglycans (PGN) of Gram-posi...
TMPJ-00574 RNASE3 Protein, Human, Recombinant (His)

RNase 3,RNS3,ECP,Eosinophil Cationic Protein,RNASE3,Ribonucl...

Human HEK293 Cells
Ribonuclease 3 (RNASE3) is a basic protein that is localized to the eosinophil primary matrix and belongs to the pancreatic ribonuclease family. RNASE3 is released during degranulation of eosinophils. RNASE3 possesses a wide variety of biological activities. RNASE3 interacts with bacterial lipopolysaccharide (LPS) and lipoteichoic acid (LTA). RNASE3 exhibits antibacterial activity, including cytoplasmic membrane depolarization of preferentially Gram-negative, but also Gram-positive strains. It p...
TMPH-00064 MRJP1 Protein, Apis mellifera, Recombinant (His)

Royalactin,Major royal jelly protein 1,Apalbumin 1,MRJP1,56-...

Apis mellifera P. pastoris (Yeast)
Induces the differentiation of honeybee larvae into queens through an Egfr-mediated signaling pathway. Promotes body size increase by activating p70 S6 kinase, stimulates ovary development by augmenting the titer of vitellogenin (Vg) and juvenile hormone, and reduces developmental time by increasing the activity of mitogen-activated protein kinase and inducing the 20-hydroxyecdysone protein (20E). Most abundant protein found in the royal jelly which is the food of the queen honey bee larva. The ...
TMPK-01242 MD2/LY96 Protein, Human, Recombinant (His)

MD-2,Ly-96,ESOP-1,Lymphocyte antigen 96,LY96,ESOP1

Human E. coli
MD2, a 160-residue accessory glycoprotein, is responsible for the recognition and binding of Gram-negative bacterial membrane component, lipopolysaccharide (LPS).Internalization of pathogen inside the mononuclear phagocytes has also been attributed to MD2 which leads to the clearance of pathogens from the host. MD2/LY96 Protein, Human, Recombinant (His) is expressed in E. coli expression system with C-His tag. The predicted molecular weight is 18.07 kDa and the accession number is Q9Y6Y9-1.
TMPK-00632 MD2/LY96 Protein, Cynomolgus, Recombinant (His)

ESOP-1,LY96,Lymphocyte antigen 96,ESOP1,MD-2

Cynomolgus E. coli
MD2, a 160-residue accessory glycoprotein, is responsible for the recognition and binding of Gram-negative bacterial membrane component, lipopolysaccharide (LPS).Internalization of pathogen inside the mononuclear phagocytes has also been attributed to MD2 which leads to the clearance of pathogens from the host. MD2/LY96 Protein, Cynomolgus, Recombinant (His) is expressed in E. coli expression system with C-His tag. The predicted molecular weight is 17.97 kDa and the accession number is B3Y6B0.
TMPY-03999 MD2/LY96 Protein, Mouse, Recombinant (hFc)

lymphocyte antigen 96,ESOP-1,MD2,MD-2

Mouse HEK293 Cells
LY96 (Lymphocyte Antigen 96, also known as ESOP-1) is a Protein Coding gene. 2 alternatively spliced human isoforms have been reported. This gene encodes a protein that associates with toll-like receptor 4 on the cell surface and confers responsiveness to lipopolysaccharide (LPS), thus providing a link between the receptor and LPS signaling. LY-96 also cooperates with TLR2 in the response to cell wall components from Gram-positive and Gram-negative bacteria. It enhances the TLR4-dependent activa...
TMPH-01540 Intelectin-1/ITLN1 Protein, Human, Recombinant (His & Myc)

Galactofuranose-binding lectin,Endothelial lectin HL-1,Intel...

Human E. coli
Lectin that specifically recognizes microbial carbohydrate chains in a calcium-dependent manner. Binds to microbial glycans that contain a terminal acyclic 1,2-diol moiety, including beta-linked D-galactofuranose (beta-Galf), D-phosphoglycerol-modified glycans, D-glycero-D-talo-oct-2-ulosonic acid (KO) and 3-deoxy-D-manno-oct-2-ulosonic acid (KDO). Binds to glycans from Gram-positive and Gram-negative bacteria, including K.pneumoniae, S.pneumoniae, Y.pestis, P.mirabilis and P.vulgaris. Does not ...
TMPY-02835 DEFB103A Protein, Human, Recombinant (His)

DEFB3,HBP3,defensin, beta 103A,hBD-3,DEFB103,DEFB-3,HBD3,HBP...

Human E. coli
Beta-defensin 3 is a member of the defensin family. Defensin family is comprised by microbicidal and cytotoxic peptides made by neutrophils. Members of the beta-defensin 3 family are highly similar in protein sequence. Beta-defensin 3 shows antimicrobial activity against Gram-positive bacteria S.aureus and S.pyogenes, Gram-negative bacteria P.aeruginosa and E.coli and the yeast C.albicans. Beta-defensin 3 is abundantly expressed in skin and tonsils, and to a lesser extent in trachea, uterus, kid...
TMPY-03728 CCL28 Protein, Human, Recombinant (His)

MEC,SCYA28,chemokine (C-C motif) ligand 28,CCK1

Human E. coli
CCL28 chemokine is expressed by epithelial cells of various mucosal tissues. This chemokine binds to CCR3 and CCR10 receptors and plays an essential role in the IgA antibody secreting cells (IgA-ASC) homing to mucosal surfaces and lactating mammary gland as well. Besides, CCL28 has been shown to exert a potent antimicrobial activity against both Gram-negative and Gram-positive bacteria and fungi. The potent antimicrobial function of CCL28 combined with its wide distribution in mucosal tissues an...
TMPY-02375 acnB Protein, E. coli, Recombinant

yacI,yacJ

E. coli E. coli
Escherichia coli contains two major aconitases (Acns), AcnA and AcnB. They are distantly related monomeric Fe-S proteins that contain different arrangements of four structural domains. acnA is specifically subject to SoxRS-mediated activation, whereas acnB encodes the major aconitase that is synthesized earlier in the growth cycle than AcnA. It is concluded that AcnB is the major citric acid cycle enzyme. Aconitate hydratase 2 (acnB) catalyzes the isomerization of citrate to isocitrate via cis-a...
TMPH-02671 Gasdermin-D Protein, Mouse, Recombinant (His & Myc)

Gasdermin-D,Gasdermin domain-containing protein 1,Gsdmd

Mouse E. coli
Precursor of a pore-forming protein that plays a key role in host defense against pathogen infection and danger signals. This form constitutes the precursor of the pore-forming protein: upon cleavage, the released N-terminal moiety (Gasdermin-D, N-terminal) binds to membranes and forms pores, triggering pyroptosis.; Promotes pyroptosis in response to microbial infection and danger signals. Produced by the cleavage of gasdermin-D by inflammatory caspases CASP1 or CASP4/CASP11 in response to canon...

重组蛋白

ORM2 Protein, Human, Recombinant (His)
Cat.No: TMPY-03118
Species: Human
Expression System: HEK293 Cells
LBP Protein, Human, Recombinant (His)
Cat.No: TMPY-02204
Species: Human
Expression System: HEK293 Cells
TLR4 Protein, Human, Recombinant (His)
Cat.No: TMPY-02904
Species: Human
Expression System: Baculovirus Insect Cells
Lysozyme C-2 Protein, Mouse, Recombinant (His & Myc)
Cat.No: TMPH-02773
Species: Mouse
Expression System: E. coli
BPI Protein, Human, Recombinant (His)
Cat.No: TMPY-02908
Species: Human
Expression System: HEK293 Cells
Cathelicidin-6 Protein, Bovine, Recombinant (His & SUMO)
Cat.No: TMPH-00230
Species: Bovine
Expression System: E. coli
DEFA1 Protein, Human, Recombinant (GST)
Cat.No: TMPH-01772
Species: Human
Expression System: E. coli
Thanatin Protein, Podisus maculiventris, Recombinant (His & KSI)
Cat.No: TMPH-03145
Species: Podisus maculiventris
Expression System: E. coli
DEFB4 Protein, Mouse, Recombinant (His & SUMO)
Cat.No: TMPH-02544
Species: Mouse
Expression System: E. coli
PMAP-23 Protein, Pig, Recombinant (His & SUMO)
Cat.No: TMPH-03100
Species: Sus scrofa (Pig)
Expression System: E. coli
LCE3A Protein, Human, Recombinant (His)
Cat.No: TMPH-01607
Species: Human
Expression System: E. coli
PGLYRP1 Protein, Mouse, Recombinant (His)
Cat.No: TMPY-02163
Species: Mouse
Expression System: HEK293 Cells
RNASE3 Protein, Human, Recombinant (His)
Cat.No: TMPJ-00574
Species: Human
Expression System: HEK293 Cells
MRJP1 Protein, Apis mellifera, Recombinant (His)
Cat.No: TMPH-00064
Species: Apis mellifera
Expression System: P. pastoris (Yeast)
MD2/LY96 Protein, Human, Recombinant (His)
Cat.No: TMPK-01242
Species: Human
Expression System: E. coli
MD2/LY96 Protein, Cynomolgus, Recombinant (His)
Cat.No: TMPK-00632
Species: Cynomolgus
Expression System: E. coli
MD2/LY96 Protein, Mouse, Recombinant (hFc)
Cat.No: TMPY-03999
Species: Mouse
Expression System: HEK293 Cells
Intelectin-1/ITLN1 Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-01540
Species: Human
Expression System: E. coli
DEFB103A Protein, Human, Recombinant (His)
Cat.No: TMPY-02835
Species: Human
Expression System: E. coli
CCL28 Protein, Human, Recombinant (His)
Cat.No: TMPY-03728
Species: Human
Expression System: E. coli
acnB Protein, E. coli, Recombinant
Cat.No: TMPY-02375
Species: E. coli
Expression System: E. coli
Gasdermin-D Protein, Mouse, Recombinant (His & Myc)
Cat.No: TMPH-02671
Species: Mouse
Expression System: E. coli
Cat. No. Product Name Target Signaling Pathways
TMID-0079 Norfloxacin-d8

Norfloxacin-d8 是 Norfloxacin 的氘代化合物。Norfloxacin 的 CAS 号为 70458-96-7。Norfloxacin是广谱抗生素,能通过结合DNA旋转酶抑制革兰氏阳性和阴性菌。
TMID-0271 Miloxacin-d3

Miloxacin-d3 是 Miloxacin 的氘代化合物。Miloxacin 的 CAS 号为 37065-29-5。
TMIH-0154 Ciprofloxacin-d8

Ciprofloxacin-d8 是 Ciprofloxacin 的氘代化合物。Ciprofloxacin 的 CAS 号为 85721-33-1。Ciprofloxacin是一种有高抗菌活性的氟喹诺酮类抗生素。
T37250 Cefazolin-13C2,15N

Cefazolin-13C2,15N

Cefazolin-13C2,15N is intended for use as an internal standard for the quantification of cefazolin by GC- or LC-MS. Cefazolin is a broad-spectrum cephalosporin antibiotic that is active in vitro against various Gram-positive and Gram-negative bacteria (MICs = 0.2-12.5 μg/ml). It also inhibits the growth of clinical isolates of S. aureus, E. coli, P. mirabilis, and K. pneumoniae (MICs = 0.1-25 μg/ml). In vivo, cefazolin protects against S. aureus, E. coli, and P. mirabilis infection in mice (ED50...
TMIJ-0059 Moxifloxacin-d4

Moxifloxacin-d4 是 Moxifloxacin 的氘代化合物。Moxifloxacin 的 CAS 号为 151096-09-2。Moxifloxacin 是一种8-甲氧基喹诺酮类口服有效抗菌药物,用于急性细菌性鼻窦炎,慢性支气管炎的急性细菌性加重和感染性肺炎的研究。
TMID-0281 Moxifloxacin-13C-d3

Moxifloxacin-13C-d3 是 Moxifloxacin 的 13C 和氘代化合物。Moxifloxacin 的 CAS 号为 151096-09-2。Moxifloxacin 是一种8-甲氧基喹诺酮类口服有效抗菌药物,用于急性细菌性鼻窦炎,慢性支气管炎的急性细菌性加重和感染性肺炎的研究。
TMIJ-0327 Cefpodoxime-d3 Acid

Cefpodoxime-d3 Acid 是 Cefpodoxime Acid 的氘代化合物。Cefpodoxime Acid 的 CAS 号为 80210-62-4。Cefpodoxime (free acid) 是一种口服的第三代头孢菌素抗生素。除铜绿假单胞菌、肠球菌和脆弱拟杆菌外,它对大多数革兰氏阳性和革兰氏阴性微生物均有效。
TMID-0290 Cefpodoxime proxetil-d3

Cefpodoxime proxetil-d3 是 Cefpodoxime proxetil 的氘代化合物。Cefpodoxime proxetil 的 CAS 号为 87239-81-4。Cefpodoxime Proxetil 是一种口服的广谱型抗生素。它与青霉素结合蛋白结合,抑制肽聚糖的合成,干扰细菌细胞壁的生物合成。
TMID-0072 Imipenem-d4

Imipenem-d4 是 Imipenem 的氘代化合物。Imipenem 的 CAS 号为 64221-86-9。Imipenem (MK0787) 是一种噻吩霉素衍生物,属于抗生素类,具有抗菌活性,对革兰氏阳性和革兰氏阴性菌具有部分的抑制作用。Imipenem 可用于研究碳青霉烯类非易感性感染和铜绿假单胞菌生物膜感染。

同位素标记化合物

Norfloxacin-d8
Cat.No: TMID-0079
Synonym:
Target:
Miloxacin-d3
Cat.No: TMID-0271
Synonym:
Target:
Ciprofloxacin-d8
Cat.No: TMIH-0154
Synonym:
Target:
Cefazolin-13C2,15N
Cat.No: T37250
Synonym: Cefazolin-13C2,15N
Target:
Moxifloxacin-d4
Cat.No: TMIJ-0059
Synonym:
Target:
Moxifloxacin-13C-d3
Cat.No: TMID-0281
Synonym:
Target:
Cefpodoxime-d3 Acid
Cat.No: TMIJ-0327
Synonym:
Target:
Cefpodoxime proxetil-d3
Cat.No: TMID-0290
Synonym:
Target:
Imipenem-d4
Cat.No: TMID-0072
Synonym:
Target:
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