Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T69915 |
GX-585
GX585,GX 585 |
Sodium Channel | Membrane transporter/Ion channel |
GX-585 是一种磺胺类化合物,是一种Nav 1.7通道抑制剂,具有镇痛活性,可用于研究神经疼痛和炎症。 | |||
T69914 |
Variegatic acid
|
Others | Others |
Variegatic acid is a natural inhibitor of β-hexosaminidase release and tumor necrosis factor (TNF)-α secretion from rat basophilic leukemia (RBL 2H3) cells, with IC50 values of 10.4 μM and 16.8 μM, respectively, also inhibiting PKC β1 activity with an IC50 value of 36.2 μM. |