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Cat. No. Product Name Target Signaling Pathways
T62852 GSK2945 hydrochloride

Others Others
GSK2945 hydrochloride 是一种叔胺,是一种高特异性的 Rev-erbα/REV-ERBα(小鼠/人反向成红细胞病病毒α) 拮抗剂,他们的 EC50 值分别为 21.5 μM 和 20.8 μM。GSK2945 hydrochloride 能够提高胆固醇 7α-羟化酶 (CYP7A1) 水平和胆固醇代谢。
T11490L GSK2945 hydrochloride (1438071-12-5 free base)

GSK2945 hydrochloride

Others Others
GSK2945 hydrochloride is a highly specific Rev-erbα/REV-ERBα (mouse/human reverse erythroblastosis virus α) antagonist (EC50s: 21.5 μM and 20.8 μM). It enhances cholesterol 7α-hydroxylase (CYP7A1) level and cholesterol metabolism.

化合物

GSK2945 hydrochloride
Cat.No: T62852
Synonym:
Target: Others
GSK2945 hydrochloride (1438071-12-5 free base)
Cat.No: T11490L
Synonym: GSK2945 hydrochloride
Target: Others
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