Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T10749 |
Cebranopadol ((1α,4α)stereoisomer)
GRT6005 (1α,4α)stereoisomer |
Others | Others |
Cebranopadol ((1α,4α)stereoisomer) is a stereoisomer of cebranopadol which is a potent ORL-1 agonist. | |||
T5167 |
Cebranopadol
西博帕多,GRT6005 |
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
Cebranopadol (GRT6005) 是镇痛 NOP 和阿片受体激动剂,对人 NOP、μ-阿片 (MOP)、κ-阿片 (KOP) 和 δ-阿片 (DOP) 受体的 Ki 值分别为 0.9、0.7、2.6 和 18 nM。 |