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Cat. No. | Product Name | ||
---|---|---|---|
L2700 | 肾上腺素能受体化合物库 | 193 compounds | |
193 种特异靶向肾上腺素受体的生物活性小分子化合物的集合,是相关疾病药物筛选的有效工具; |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T27413 |
Trimebutine CTB salt
GIC1001 |
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
Trimebutine CTB salt (GIC-1001) 是一种阿片受体激动剂,可用于研究疼痛。 | |||
T80478 |
α-Conotoxin GIC
|
||
α-Conotoxin GIC为选择性α3β2烟碱型乙酰胆碱受体拮抗剂,具有IC50值为1.1 nM。 | |||
T8961 |
GW280264X
Carbamic acid |
MMP | Proteases/Proteasome |
GW280264X (Carbamic acid) 是一种 ADAM10/TACE (ADAM17)金属蛋白酶抑制剂。它有效阻断 TACE (ADAM17)和 ADAM10的 IC50分别为 8.0 nM 和 11.5 nM。其中ADAM10/17 能够调节胶质母细胞瘤起始细胞的免疫原性。 | |||
T6516 |
Golgicide A
|
Others; Virus Protease | Microbiology/Virology; Others |
Golgicide A 可抑制柯萨奇病毒 B3 和其他人类肠道病毒的复制。它是一种高度特异性可逆的顺式高尔基体 ADP-核糖基化因子鸟嘌呤核苷酸交换因子抑制剂。 | |||
T9424 |
Temgicoluril
Tetramethylglycoluril,mebikar |
GABA Receptor | Membrane transporter/Ion channel; Neuroscience |
Temgicoluril (mebikar) 具有抗焦虑活性,作用于GABA 受体。 | |||
T38399 |
(Rac)-Golgicide A
(Rac)-GCA |
Virus Protease | Microbiology/Virology |
(Rac)-Golgicide A ((Rac)-GCA) 是 Golgicide A 的一种消旋体。 | |||
T82424 |
Experimental allergic encephalitogenic peptide (human)
|
||
Experimental allergic encephalitogenic peptide (human) 为EAE多肽类化合物,能够诱导豚鼠发生脑脊髓炎。 | |||
T125016 |
4,4'-Di-O-methylellagic acid
|
Others | Others |
4,4'-Di-O-methylellagic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125016,CAS号为 3374-77-4。 | |||
T63825 |
Antiallergic agent-1
|
Others | Others |
Antiallergic agent-1 是 Src 家族激酶抑制剂,是一种新的有价值的先导化合物,具有作为抗过敏剂的潜力。 | |||
T125319 |
Cimicifugic acid F
|
Others | Others |
Cimicifugic acid F 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125319。 | |||
T124973 |
3-O-Methylellagic acid 3'-O-alpha-rhamnopyranoside
|
Others | Others |
3-O-Methylellagic acid 3'-O-alpha-rhamnopyranoside 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124973。 | |||
T126303 |
10alpha-Hydroxyepigambogic acid
|
Others | Others |
10alpha-Hydroxyepigambogic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126303。 | |||
T124627 |
3,4'-Di-O-methylellagic acid
|
Others | Others |
3,4'-Di-O-methylellagic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124627。 | |||
T126415 |
9R-10alpha-Hydroxyepigambogic acid
|
Others | Others |
9R-10alpha-Hydroxyepigambogic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126415。 | |||
T124009 |
30-Hydroxygambogic acid
|
Others | Others |
30-Hydroxygambogic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124009。 | |||
T130680 |
Longicaulenone
|
Others | Others |
Longicaulenone 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T130680。 | |||
T124735 |
3-Methyl ellagic acid
|
Others | Others |
3-Methyl ellagic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T124735。 | |||
T38817 |
Golgicide A-1
GCA-1,Golgicide A-1 |
Others | Others |
Golgicide A-1 (GCA-1) is a moderately potent cis-diastereomer variant of Golgicide A (GCA) specifically designed to inhibit mosquito reproduction. | |||
T38818 |
Golgicide A-2
Golgicide A-2,GCA-2 |
Others | Others |
Golgicide A-2 (GCA-2), a derivative of Golgicide A (GCA), is the highly active enantiomer of GCA. It exhibits exceptional selectivity and efficiency in eradicating An. stephensi larvae, thus making it a valuable tool for researching dengue virus-related diseases. | |||
T124889 |
Isocalolongic acid
|
Others | Others |
Isocalolongic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124889,CAS号为 40737-92-6。 | |||
TP2188 |
type I hair keratin fragment [Homo sapiens]/[Ovis aries]/[Rattus norvegicus]
|
Others | Others |
The human type I hair keratin subfamily comprises nine individual members, which can be subdivided into three groups. Group A (hHa1, hHa3-I, hHa3-II, hHa4) and B (hHa7, hHa8) each contains structurally related hair keratins, whereas group C members hHa2, | |||
T60324 |
Fungicide4
|
Others | Others |
Fungicide4 对P. infestans 菌株显示出高活性。 | |||
T32863 |
Longicoricin
|
Others | Others |
Longicoricin is a monotetrahydrofuran Annonaceous acetogenin from Asimina longifolia. | |||
T39882 |
Fungicide5
|
Others | Others |
Fungicide5 is a fungicide candidate targeting succinate dehydrogenase ( K i = 0.095 μM). | |||
T125707 |
Gambogic acid A
|
Others | Others |
Gambogic acid A 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125707。 | |||
T32862 |
Longicin
|
Others | Others |
Longicin is a cytotoxic agent isolated from Asimina longifolia. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T0465 |
Ellagic acid
鞣花酸,Gallogen,Elagostasine |
Hedgehog/Smoothened; Casein Kinase; Reactive Oxygen Species; Topoisomerase; Endogenous Metabolite; PKA; Syk; PKC; Carbonic Anhydrase | Angiogenesis; Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; GPCR/G Protein; Immunology/Inflammation; Metabolism; NF-κB; Stem Cells; Tyrosine Kinase/Adaptors |
Ellagic acid (Gallogen) 是从 Eucalyptus maculata Hook 和 E. Hemipholia F. Muell 的 kino 中分离出来的稠合四环天然产物,是一种有效的,ATP 竞争性的CK2抑制剂,IC50和Ki 值分别为 40 nM 和 20 nM。 | |||
T2883 |
Syringic acid
3,5-dimethyl ether Gallic Acid,SYRA,3,5-dimethoxy-4-hydroxy Benzoic Acid,丁香酸,NSC 2129 |
Others; Endogenous Metabolite; Antibacterial | Metabolism; Microbiology/Virology; Others |
Syringic acid (3,5-dimethoxy-4-hydroxy Benzoic Acid) 能抑制低密度脂蛋白的氧化。 | |||
T5724 |
Neogambogic acid
neo-gambogic acid,新藤黄酸 |
Apoptosis; Others; Antibacterial | Apoptosis; Microbiology/Virology; Others |
Neogambogic acid 是藤黄的有效成分,可诱导细胞凋亡并具有抗癌作用。它有效抑制耐甲氧西林的金黄色葡萄球菌。 | |||
T9328 |
Ellagic Acid Dihydrate
|
P450 | Metabolism |
Ellagic Acid Dihydrate 抑制 CYP1A1 依赖的benzo[a]pyrene 活化。 | |||
T6185 |
Gambogic Acid
藤黄酸,Beta-Guttiferrin,藤黄酸 A,Guttatic Acid,Guttic Acid |
BCL; Autophagy | Apoptosis; Autophagy |
Gambogic Acid (Guttic Acid) 是来自藤黄树的一种藤黄树脂,抑制 Bcl-XL、Bcl-2、Bcl-W、Bcl-B、Bfl-1和 Mcl-1,IC50分别为 1.47 μM、1.21 μM、2.02 μM、0.66 μM、1.06 μM 和 0.79 μM。 | |||
TQ0180 |
Chebulagic acid
|
SARS-CoV; Influenza Virus; Lipoxygenase; COX | Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience |
Chebulagic acid 是从 Terminalia chebula Retz 中分离出来的一种 COX-LOX 双重抑制剂,有抗炎和抗感染作用。它抑制 SARS-CoV-2病毒的复制,EC50值为 9.76 μM。它还是 M2(S31N)抑制剂和抗流感病毒剂。 | |||
T41017 |
Epigambogic acid
|
||
Epigambogic acid 是一种来自藤黄的小分子化合物,具有抗肿瘤、止咳、祛痰和抗炎活性。 | |||
TN1697 |
Glucosyringic acid
葡萄糖基丁香酸 |
Immunology/Inflammation related | Immunology/Inflammation |
Glucosyringic acid 具有免疫抑制作用,在体外能抑制鼠 B 淋巴细胞的增殖。 | |||
TN7213 |
Ellagic acid 3-O-α-L-rhamnopyranoside
|
Others | Others |
Ellagic acid 3-O-α-L-rhamnopyranoside 是一种天然产物,存在于植物鹅绒委陵菜Potentilla anserina 的块根中。 | |||
TN6177 |
Koenigicine
Koenimbidine,Koenidine |
||
Koenigicine 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6177,CAS号为 24123-92-0。 | |||
T83465 |
10α-Hydroxyepigambogic acid
|
||
10α-Hydroxyepigambogic acid,一种从Garcinia hanburyi中提取的化合物,适用于肿瘤研究领域。 | |||
T83237 |
8,8a-Dihydro-8-hydroxygambogic acid
|
||
8,8a-Dihydro-8-hydroxygambogic acid,一天然产物,从Garcinia hanburyi树脂中分离,具备抗癌活性。 | |||
T81318 |
R-30-Hydroxygambogic acid
|
||
R-30-Hydroxygambogic acid是从藤黄提取的一种聚戊烯酰黄酮外聚体,对K562/R和K562/S两种人白血病细胞系的IC50分别为2.89 μM和1.27 μM。该化合物适用于癌症研究领域。 | |||
T32861 |
Longicautadine
NSC377102,NSC 377102,NSC-377102 |
||
Longicautadine is an alkaloid isolated from stembark of Strychnos chrysophylla. | |||
T8305 |
Ellagic acid (hydrate)
Ellagic Acid hydrate,鞣花酸水合物 |
Antioxidant; Casein Kinase | Metabolism; oxidation-reduction; Stem Cells |
Ellagic acid (hydrate) 是存在于许多水果和蔬菜中的一种天然抗氧化剂,是 ATP 竞争性的 CK2抑制剂,IC50和 Ki 值分别为 40 nM 和 20 nM。 | |||
T80998 |
Thapsigargicin
Thapsigargicine |
||
Thapsigargicin(Thapsigargicine)作为肥大细胞和白细胞的激活剂,能诱导大鼠腹膜肥大细胞及人嗜碱性粒细胞释放组胺,并提升完整人血小板中的细胞质游离钙水平。 | |||
TN6494 |
3-O-methylellagic acid 4'-O-alpha-L-rhamnopyranoside
|
||
3-O-methylellagic acid 4'-O-alpha-L-rhamnopyranoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6494,CAS号为 51768-39-9。 | |||
TN6559 |
Isogambogic acid
|
||
Isogambogic acid shows cytotoxic activiity against KB and drug-resistant KB-V1 cell lines. | |||
TN3652 | Cimicifugic acid B | Others | Others |
Cimicifugic acid B 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3652,CAS号为 205114-66-5。 | |||
TN1234 |
3,3'-Di-O-methylellagic acid-4'-O-β-D-glucopyranoside
3,3'-Di-O-methylellagic acid 4'-glucoside,3,3'-二-O-甲基柔花酸-4'-O-BETA-D-吡喃葡萄糖苷 |
Others | Others |
3,3'-Di-O-methylellagic acid 4'-glucoside is a natural product | |||
TN6255 |
3,7,8-Tri-O-methylellagic acid 2-O-rutinoside
3,3',4'-Tri-O-methylellagic acid 4-O-rutinoside |
||
3,7,8-Tri-O-methylellagic acid 2-O-rutinoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6255,CAS号为 56470-18-9。 | |||
T82478 |
Ellagic acid 4-O-α-L-arabinopyranoside
|
||
Ellagic acid 4-O-α-L-arabinopyranoside,一种具有抗氧化活性的化合物,从Dimocarpus longan Lour, syn. Euphoria longan Lam.(龙眼)中分离得到。 | |||
TN1203 |
2,3,8-Tri-O-methylellagic acid
2,3,8-三邻甲基鞣花酸 |
Antifection | Microbiology/Virology |
2,3,8-tri-O-Methyl ellagic acid has antimicrobial activity agaist Vibro cholera, Staphylococcus aureus, Klebsiella pneumoniae, Pseudomonas aeruginosa, Bacillus cereus, Escherichia coli. | |||
TN6226 |
3-O-Methylellagic acid 4-O-rhamnoside
|
||
3-O-Methylellagic acid 4-O-rhamnoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6226,CAS号为 639089-97-7。 | |||
TN6149 |
Digicitrin
|
||
Digicitrin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6149,CAS号为 5065-10-1。 | |||
TN1978 |
Neochebulagic acid
新诃黎勒酸 |
Others | Others |
Neochebulagic acid is a natural product | |||
TN6156 |
3,4,3'-Tri-O-methylflavellagic acid
|
||
3,4,3'-Tri-O-methylflavellagic acid 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6156,CAS号为 13756-49-5。 | |||
TN1242 |
3,3'-Di-O-methylellagic acid
3,8-Di-O-methylellagic acid,3,3'-O-二甲基鞣花酸 |
Others; TNF; Antifection | Apoptosis; Microbiology/Virology; Others |
3,3'-Di-O-methylellagic acid reveals moderate antibacterial activity, it also shows strong DPPH radical scavenging activities with SC50 of 123.3 ug/mL. It has a lower capacity of stimulating murine peritoneal macrophages to release nitric oxide and tumoural-alpha necrose factor | |||
T75665 |
3-O-Methylellagic acid
|
Others | Others |
3-O-Methylellagic acid 是一种天然产物,从Myrciaria cauliflora 中分离得到,具有抗炎活性。3-O-Methylellagic acid 对葡萄糖转运有抑制作用。3-O-Methylellagic acid 具有抗菌活性,对葡萄球菌 ATCC 25923 菌株作用的 MIC 值为 32 μg/mL。 | |||
TN7498 |
Ellagic acid 4-O-alpha-L-arabinofuranoside
|
Others | Others |
TN2482 |
1,2,3-Tri-O-methyl-7,8-methyleneflavellagic acid
|
Others | Others |
1,2,3-Tri-O-methyl-7,8-methyleneflavellagic acid 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2482,CAS号为 69251-99-6。 | |||
T82344 |
Gambogic acid B
|
||
Gambogic acid B,一种从Garcinia hanburyi树脂中分离得到的活性化合物,对A549、HCT116 和 MDA-MB-231 细胞显示细胞毒性,其IC50值分别为1.60 μM、6.88 μM 和 0.87 μM。 | |||
T81232 |
S-30-Hydroxygambogic acid
|
||
S-30-Hydroxygambogic acid,一聚戊烯酰黄酮外聚体,源自藤黄。针对人白血病细胞系K562/R及K562/S,其IC50值别为4.49 μM与3.61 μM。S-30-Hydroxygambogic acid主用于癌症研究领域。 | |||
T75546 |
Ellagic acid 4-O-β-D-xylopyranoside
|
Others | Others |
Ellagic acid 4-O-β-D-xylopyranoside,天然鞣花单宁,展现抗菌活性。同时,作为黄嘌呤氧化酶 (xanthine oxidase) 抑制剂,其50为 2.1 μg/mL。 |
Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPH-00444 |
GSTP1 Protein, Cricetulus longicaudatus, Recombinant (His & Myc)
GST class-pi,GSTP1,Glutathione S-transferase P |
Chinese hamster | E. coli |
GSTP1 Protein, Cricetulus longicaudatus, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPH-00445 |
GSTP1 Protein, Cricetulus longicaudatus, Recombinant (His)
Glutathione S-transferase P,GST class-pi,GSTP1 |
Chinese hamster | P. pastoris (Yeast) |
GSTP1 Protein, Cricetulus longicaudatus, Recombinant (His) is expressed in Yeast. |