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Targets Recommended: Apoptosis

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Cat. No. Product Name Target Signaling Pathways
T15337 Forodesine

Immucillin-H,BCX-1777

Apoptosis Apoptosis
Forodesine (BCX-1777) 是一种具有口服活性和高效性的嘌呤核苷磷酸化酶 (PNP) 抑制剂,是一种新的嘌呤核苷类似物,抑制人类淋巴细胞增殖抑制剂,可通过增加 dGTP 水平而诱导白血病细胞凋亡 (apoptosis),可用于研究皮肤T细胞淋巴瘤。
T11313 Forodesine hydrochloride

BCX-1777 hydrochloride,Immucillin-H hydrochloride

Others Others
Forodesine hydrochloride (BCX-1777 hydrochloride), a potent inhibitor of human lymphocyte proliferation, effectively induces apoptosis in leukemic cells by elevating dGTP levels. This compound is an orally active, highly potent purine nucleoside phosphorylase (PNP) inhibitor, demonstrating IC50 values between 0.48 to 1.57 nM across human, mouse, rat, monkey, and dog PNP.

化合物

Forodesine
Cat.No: T15337
Synonym: Immucillin-H,BCX-1777
Target: Apoptosis
Forodesine hydrochloride
Cat.No: T11313
Synonym: BCX-1777 hydrochloride,Immucillin-H hydrochloride
Target: Others
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