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Cat. No. | Product Name | Target | Signaling Pathways |
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T0068 |
Fluphenazine dihydrochloride
氟奋乃静盐酸盐,Prolixin,盐酸氟奋乃静,Fluphenazine hydrochloride |
Dopamine Receptor | GPCR/G Protein; Neuroscience |
Fluphenazine dihydrochloride (Prolixin) 是一种多巴胺受体D1/D2抑制剂。 | |||
T36820 |
Fluphenazine-N-2-chloroethane (hydrochloride)
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Others | Others |
Fluphenazine is a traditional antipsychotic compound that tightly binds the dopamine D2 receptor (Ki = 0.55 nM) and also reversibly inhibits calmodulin at micromolar concentrations. Fluphenazine-N-2-chloroethane is a derivative of fluphenazine that contains an alkylating chlorethylamine chain, which produces irreversible protein binding. It is a relatively selective, irreversible antagonist of D2 receptors both in vitro (IC50 = 100 nM) and in vivo, inactivating approximately 90% of D2 receptors ... |
Cat. No. | Product Name | Target | Signaling Pathways |
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TMIH-0241 |
Fluphenazine-d8 Dihydrochloride
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Fluphenazine-d8 Dihydrochloride 是 Fluphenazine Dihydrochloride 的氘代化合物。Fluphenazine Dihydrochloride 的 CAS 号为 146-56-5。Fluphenazine hydrochloride 是一种多巴胺受体D1/D2抑制剂。 |