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Search Results for " fluphenazine hydrochloride "
Targets Recommended: Dopamine Receptor

2

抑制剂 & 化合物

1

同位素标记化合物

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Cat. No. Product Name Target Signaling Pathways
T0068 Fluphenazine dihydrochloride

氟奋乃静盐酸盐,Prolixin,盐酸氟奋乃静,Fluphenazine hydrochloride

Dopamine Receptor GPCR/G Protein; Neuroscience
Fluphenazine dihydrochloride (Prolixin) 是一种多巴胺受体D1/D2抑制剂。
T36820 Fluphenazine-N-2-chloroethane (hydrochloride)

Others Others
Fluphenazine is a traditional antipsychotic compound that tightly binds the dopamine D2 receptor (Ki = 0.55 nM) and also reversibly inhibits calmodulin at micromolar concentrations. Fluphenazine-N-2-chloroethane is a derivative of fluphenazine that contains an alkylating chlorethylamine chain, which produces irreversible protein binding. It is a relatively selective, irreversible antagonist of D2 receptors both in vitro (IC50 = 100 nM) and in vivo, inactivating approximately 90% of D2 receptors ...

化合物

Fluphenazine dihydrochloride
Cat.No: T0068
Synonym: 氟奋乃静盐酸盐,Prolixin,盐酸氟奋乃静,Fluphenazine hydrochloride
Target: Dopamine Receptor
Fluphenazine-N-2-chloroethane (hydrochloride)
Cat.No: T36820
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
TMIH-0241 Fluphenazine-d8 Dihydrochloride

Fluphenazine-d8 DihydrochlorideFluphenazine Dihydrochloride 的氘代化合物。Fluphenazine Dihydrochloride 的 CAS 号为 146-56-5。Fluphenazine hydrochloride 是一种多巴胺受体D1/D2抑制剂。

同位素标记化合物

Fluphenazine-d8 Dihydrochloride
Cat.No: TMIH-0241
Synonym:
Target:
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