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Search Results for " fenspiride-d5 "
Targets Recommended: Others

3

抑制剂 & 化合物

1

同位素标记化合物

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Cat. No. Product Name Target Signaling Pathways
T71139 EXP3892

Others Others
EXP3892 is an angiotensin II receptor antagonist.
T0383 Fenspiride hydrochloride

Fenspiride HCl,Pneumorel,Fluiden,Decaspiride,盐酸芬司必利

Adrenergic Receptor; PDE; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience
Fenspiride hydrochloride (Decaspiride) 是一种口服活性的非甾体抗炎剂,是 H1-组胺受体的拮抗剂,可用于呼吸系统疾病的研究。
T60417 Fenspiride

Others Others
Fenspiride 是 H1-组胺受体的拮抗剂。 Fenspiride 是一种具有口服活性的非甾体类抗炎药,可用于治疗呼吸道感染和中耳炎。 Fenspiride 抑制磷酸二酯酶 4 和磷酸二酯酶 3 的活性,-logIC50 值分别为 4.16+/-0.09 和 3.44+/-0.12。 磷酸二酯酶 5 活性也受到抑制,-logIC50 值约为 3.8。

化合物

EXP3892
Cat.No: T71139
Synonym:
Target: Others
Fenspiride hydrochloride
Cat.No: T0383
Synonym: Fenspiride HCl,Pneumorel,Fluiden,Decaspiride,盐酸芬司必利
Target: Adrenergic Receptor, PDE, Histamine Receptor
Fenspiride
Cat.No: T60417
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T71141 Fenspiride-d5

Fenspiride-d5 is intended for use as an internal standard for the quantification of fenspiride by GC- or LC-MS. Fenspiride is an antagonist of histamine H1 receptors and a non-steroidal anti-inflammatory drug (NSAID). It inhibits histamine-induced contraction of isolated guinea pig trachea but not histamine-induced inotropy of isolated guinea pig heart. It also inhibits phosphodiesterase 4 (PDE4), PDE5, and PDE3 (IC50s = 69, ~158, and 363 µM, respectively, in isolated human bronchi derived from ...

同位素标记化合物

Fenspiride-d5
Cat.No: T71141
Synonym:
Target:
TargetMol Loading
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