38
3
16
1
Cat. No. | Product Name | ||
---|---|---|---|
L4200 | FDA 上市药物库 | 1729 compounds | |
1729 个FDA 批准药物的独特集合,可用于高通量筛选和高内涵筛选; | |||
L1010 | FDA上市及药典收录分子库 | 3158 compounds | |
3158 个上市及药典分子集合,可用于高通量筛选和高内涵筛选; | |||
L1610 | FDA 上市激酶抑制剂库 | 263 compounds | |
263种靶向激酶的上市药物集合,用于特定靶向激酶,可用于高通量筛选和高内涵筛选; | |||
L4500 | 抗真菌库 | 252 compounds | |
252 个抗真菌活性化合物的独特集合,包含作用于真菌相关靶点的化合物和临床中用于真菌类疾病的药物,是相关疾病药物筛选的有效工具。 | |||
L9900 | 药用辅料化合物库 | 182 compounds | |
182 种 FDA 批准药品中的非活性成分集合 | |||
L5800 | 药物代谢杂质库 | 197 compounds | |
197 种药物异构体/代谢产物的特有集合,可用于高通量、高内涵筛选; | |||
LF9200 | LC 共价筛选化合物库 | 34700 compounds | |
L9410 | 共价抑制剂库 | 1920 compounds | |
1920 种小分子的独特集合,包含已发现的共价抑制剂以及包含某些共价反应基团常见弹头的分子,如氯乙酰基,2-氯丙酰基,丙烯酰基,1-丙-2-炔基,1-丁-2-炔基,酮羰基,二硫键等,可以用于共价抑制剂药物研发; | |||
L3100 | 造血毒性小分子库 | 101 compounds | |
101 种生物活性小分子化合物的特有集合,用于高通量、高内涵筛选; | |||
DF1000 | 片段化合物库 | 11269 compounds | |
ChemDiv’s Fragments Library contains 11,269 compounds. | |||
L6030 | 天然产物衍生物虚筛化合物库 | 163000 compounds | |
16.3万种天然产物衍生物,并且在持续增加中; | |||
L2150 | 抗癌药物库 | 3080 compounds | |
3080 个具有抗癌活性小分子的独特集合,生物活性已经临床前实验证实,可用于高通量、高内涵筛选; | |||
LF8700 | 共价片段化合物库LF | 6500 compounds | |
The resulting Library comprises over 4,000 small-molecule compounds for covalent fragment screening efforts. | |||
L5100 | 含氟化合物库 | 574 compounds | |
574 个含氟化合物的独特集合,可用于高通量筛选和高内涵筛选; | |||
L1500 | GPCR靶点分子库 | 1940 compounds | |
1940 种与 G 蛋白及其耦联受体相关的生物活性小分子化合物,所有小分子都具有良好的生物和药理活性,部分是 FDA 批准的上市药物; | |||
L2110 | 抗癌上市药物库 | 1779 compounds | |
1779 个具有抗癌活性小分子的独特集合,所有化合物都经过了严格的临床前研究和临床试验,由FDA、EMA 或NMPA 批准上市,可用于高通量、高内涵筛选。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T30990 |
CMFDA
5-Chloromethylfluorescein diacetate,Cell Tracker Green,CM-FDA,CM FDA |
||
CMFDA can be used as a fluorescent whole-cell-tracking reagent. | |||
T33276 |
Mefruside
FDA1902,FDA-1902,FDA 1902,FBA-1500,FBA1500,FBA 1500 |
Others | Others |
Mefruside is a diuretic indicated for the treatment of edema and hypertension. | |||
T0459 |
Sulindac
Arthrocine,MK-231,舒林酸,Clinoril,Sulindac sulfoxide |
COX; Autophagy | Autophagy; Immunology/Inflammation; Neuroscience |
Sulindac (Sulindac sulfoxide) 是一种非甾体类抗炎剂,可抑制COX-2的活性,也可抑制 COX-2 的过表达。它是一种亚磺酰基茚衍生物前药,具有潜在的抗肿瘤活性。 | |||
T15458 |
H2DCFDA
2',7'-二氯荧光素二乙酸酯,2',7'-Dichlorodihydrofluorescein diacetate,DCFH-DA |
Reactive Oxygen Species | Immunology/Inflammation; Metabolism; NF-κB |
H2DCFDA (DCFH-DA) 属于绿色荧光染料,是一种检测细胞内活性氧 (ROS) 的探针 (Ex/Em=488/525 nm),具有细胞膜渗透性。 | |||
T14057 |
6-CFDA
6-羧基荧光素二醋酸,6-Carboxyfluorescein diacetate |
Others | Others |
6-CFDA (6-Carboxyfluorescein diacetate) 是可用于流式细胞术和荧光显微镜的荧光探针,也可以用于活体多光子显微镜研究动物肝胆代谢。 | |||
T18894 |
5(6)-CFDA
CFDA,5-(6)-Carboxyfluorescein diacetate,5(6)-羧基荧光素二乙酸酯 |
Others | Others |
5(6)-CFDA (5-(6)-Carboxyfluorescein diacetate) 是具有细胞渗透性的胺反应型绿色荧光探针(λex: 492 nm; λem: 517 nm),可用于细胞染色分析。 | |||
T14048 |
5-CFDA
5-羧基荧光素二乙酸酯,5-Carboxyfluorescein diacetate |
Others | Others |
5-CFDA (5-Carboxyfluorescein diacetate) 是可透过细胞屏障并被水解为5-carboxyfluorescein,可标记人椎间盘细胞,以便体外荧光显微镜观察。 | |||
T4433 |
6-CFDA N-succinimidyl ester
Carboxyfluorescein diacetate succinimidyl |
Others | Others |
6-CFDA N-succinimidyl ester (Carboxyfluorescein diacetate succinimidyl) 能够自发且不可逆地与游离胺结合。在流式细胞术实验中用于追踪哺乳动物细胞和细菌的细胞分裂。与多种细胞透化剂结合使用,作为一种有效的、非破坏性的荧光染料,可快速检测细菌细胞。 | |||
T83293 |
5-CFDA-AM
|
||
5-CFDA-AM作为一种细胞渗透性的酯酶底物,用于测定酶活性和细胞膜完整性,该化合物为电子中性,其渗透细胞的能力超过CFDA且所需浓度更低。在细胞内部,5-CFDA-AM经酯酶水解生成羧基荧光素,后者带有额外负电荷,因此能更有效地在细胞内保留。 | |||
T72461 |
EFdA-TP tetrasodium
|
Reverse Transcriptase | Microbiology/Virology |
EFdA-TP tetrasodium作为一种核苷逆转录酶(RT)的高效抑制剂,能够作为立即或延迟链终止剂(ICT或DCT)来抑制RT催化的DNA合成,并且能通过多种机制抑制HIV-1 RT。 | |||
T35649 |
EFdA-TP tetraammonium
|
Others | Others |
EFdA-TP tetraammonium is an influential nucleoside reverse transcriptase (RT) inhibitor that effectively prevents RT-mediated DNA synthesis by acting as an immediate or delayed chain terminator (ICT or DCT). Additionally, EFdA-TP tetraammonium exhibits multiple mechanisms of inhibiting HIV-1 RT[1]. | |||
T41110 |
EFdA-TP
|
Others | Others |
EFdA-TP, a highly potent nucleoside reverse transcriptase (RT) inhibitor, exerts its inhibitory effect on RT-catalyzed DNA synthesis through both immediate and delayed chain termination mechanisms, commonly referred to as ICT and DCT, respectively. Additionally, EFdA-TP demonstrates its efficacy in inhibiting HIV-1 RT through multiple pathways. | |||
T30991 |
CM-H2DCFDA
CMH2DCFDA,CM H2DCFDA |
||
CM-H2DCFDA is a fluorescent indicator for reactive oxygen species (ROS) in cells. | |||
T67694 |
ZY-19489
|
Parasite | Microbiology/Virology |
ZY-19489是一种具有抗疟作用的化合物, 是一种潜在的单剂量根治性恶性疟原虫和间日疟原虫疟疾的药物,已获得美国 FDA 的孤儿药认定。 | |||
T22323 |
Enoxaparin sodium
|
Thrombin | Proteases/Proteasome |
Enoxaparin sodium 是一种低分子量肝素 (LMWH),已获得美国 FDA 批准,可用于医疗管理的 ST 段心肌梗死 (STEMI) 或 STEMI 及随后的经皮冠状动脉介入治疗 (PCI) 患者。它与抗凝血酶结合并增强其作用,并抑制凝血因子 XIa、IXa、Xa 和 IIa(凝血酶),从而防止血栓形成。 | |||
T4027 |
KIN1148
|
Influenza Virus | Microbiology/Virology |
KIN1148 是一种新型小分子佐剂,是IRF3激动剂,用于增强流感疫苗效率。 | |||
T5149 |
MC-Val-Cit-PAB
N-[6-(2,5-二氢-2,5-二氧代-1H-吡咯-1-基)-1-氧代己基]-L-缬氨酰-N5-(氨基甲酰基)-N-[4-(羟甲基)苯基]-L-鸟氨酰胺 |
Others; AChR; ADC Linker | Antibody-drug Conjugate/ADC Related; Neuroscience; Others |
MC-Val-Cit-PAB 是一种组织蛋白酶可裂解的 ADC 接头,用于制备抗体-药物偶联物。 | |||
T0179 |
Ticagrelor
替格瑞洛,替卡格雷,AR-C 126532XX,AZD6140 |
P450; P2Y Receptor | GPCR/G Protein; Metabolism; Neuroscience |
Ticagrelor (AR-C 126532XX) (AZD6140) 是可逆的,可口服的 P2Y12受体拮抗剂,可抑制血小板聚集。 | |||
T3503 |
MC-Val-Cit-PABC-PNP
Maleimidocaproyl-L-valine-L-citrulline-p-aminobenzyl alcohol p-nitrophenyl carbonate,马来酰亚胺基己酰-L-缬氨酸-L-瓜氨酸对氨基苄醇 对硝基苯基碳酸脂 |
Others; AChR; ADC Linker | Antibody-drug Conjugate/ADC Related; Neuroscience; Others |
MC-Val-Cit-PABC-PNP 是一种组织蛋白酶可裂解的 ADC 肽接头,可用于合成抗体偶联药物。 | |||
T7527 |
Frentizole
|
Beta Amyloid | Neuroscience |
Frentizole 是一种 FDA 批准的免疫抑制剂,是一种新型 Aβ-ABAD 相互作用抑制剂。 | |||
T0755 |
Carglumic Acid
Carbaglu,N-Carbamylglutamate,N-Carbamyl-L-glutamic acid,氨甲酰谷氨酸,Carbamylglutamic acid,Carbamino-L-glutamic acid,Ureidoglutaric acid |
Others | Others |
Carglumic Acid (Ureidoglutaric acid) 是一种 N-乙酰谷氨酸 (NAG) 的功能类似物和氨甲酰磷酸合成酶 1(CPS1)的活化剂,可用于与 N-乙酰谷氨酸合成酶 (NAGS) 缺陷相关的急性和慢性高氨血症的研究。 | |||
T6739 |
Zoledronic Acid
CGP-4244,CGP42446A,唑来膦酸,Zoledronate,CGP 42446,ZOL 446,Zometa |
Apoptosis; Rho; Autophagy | Apoptosis; Autophagy; Cell Cycle/Checkpoint |
Zoledronic Acid (ZOL 446) 是一种含氮二磷酸盐,能抑制破骨细胞的分化和凋亡,具有高效的抗骨质再吸收活性,也有抗癌作用。 | |||
T1551 |
Tegaserod maleate
HTF-919,马来酸替加色罗,SDZ-HTF-919 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Tegaserod maleate (SDZ-HTF-919) 是选择性5-HT4受体的部分激动剂和5-HT2B 受体的拮抗剂,用于治疗肠易激综合征和便秘。 | |||
T0918 |
Trimebutine
曲美布汀,Mebutin |
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
Trimebutine (Mebutin) 是阿片受体激动剂,有抗毒蕈碱活性。它是解痉剂,可调节肠道和结肠运动,并通过抗毒蕈碱和弱μ-阿片受体激动剂作用缓解腹痛。 | |||
T0910 |
Terpin hydrate
Terpin Monohydrate,cis-Terpin hydrate,萜品(水合结晶) |
Others | Others |
Terpin hydrate 是一种祛痰药,可除去急慢性支气管炎病人的黏液。 | |||
T20046 |
D & C Red no. 27
D &,Solvent Red 48,C Red no. 27,D and C Red No. 27,Japan Red 218,Phloxine BBN Supra |
||
D&C Red No. 27 Aluminum Lake is a drug and cosmetic synthetic dye. The FDA lists it as a safe additive for drugs and cosmetics as per FDA standards. | |||
T37881 |
Oritavancin(LY-333328)
|
Others | Others |
Oritavancin is a novel semisynthetic glycopeptide antibiotics. On August 6, 2014, the FDA approved oritavancin for treatment of skin infections. Oritavancin possesses potent and rapid bactericidal activity in vitro against a broad spectrum of both resistant and susceptible Gram-positive bacteria, including Staphylococcus aureus, MRSA, enterococci, and streptococci. | |||
T34065 |
Pigment Red 57
Lithol Rubine Na,Japan Red 201,Rubine Red RR 1253,Lithol rubin B |
||
Pigment Red 57, also known as D & C Red No. 6, is a synthetic dye produced from petroleum or coal tar sources; this dye is FDA-approved for use in pharmaceuticals and cosmetics. | |||
T81522 |
Pendetide
GYK-DTPA |
||
Pendetide为一种能与铟(111In)结合的螯合剂,当与Capromab(卡普罗单抗)偶联后,形成Capromab pendetide,此显像剂已获得FDA批准,用于探测前列腺软组织的转移情况。 | |||
T68706 |
Olanzapine HCl
|
Others | Others |
Olanzapine HCl is an atypical antipsychotic. It is approved by the U.S. Food and Drug Administration (FDA) for the treatment of schizophrenia and bipolar disorder. Olanzapine is structurally similar to clozapine and quetiapine. It is a dopamine antagonist and is classified as a thienobenzodiazepine. | |||
T77078 | Maftivimab | ||
Maftivimab (REGN3470-3471-3479) 是线状病毒 (Filovirus) 抑制剂,是食品和活性分子管理局 (FDA) 批准的试剂。 Maftivimab,又名 Atoltivimab、Odesivimab (Inmazeb),可用于扎伊尔埃博拉病毒感染的研究。 | |||
T76848 | Atoltivimab | ||
Atoltivimab (REGN3470) 与 maftivimab/odesivimab (Inmazeb),是美国食品和活性分子管理局 (FDA) 批准的针对扎伊尔埃博拉病毒 (EBOV) 感染的单克隆抗体。 | |||
T25611 |
Lanatoside
Lantoside,ABC lanatoside complex |
Others | Others |
Lanatoside 是一种 FDA 批准的强心苷,已被确定为候选的抗登革热化合物。它也被发现可以促进脉粥样硬化,还具有抗肿瘤活性,可抑制结直肠癌细胞、肝癌细胞的生长。 | |||
T76849 | Bamlanivimab | ||
Bamlanivimab (Anti-Human SARS-CoV-2) 是一种针对COVID-19的单克隆抗体(mAb),于2020年11月获得美国食品药品监督管理局(FDA)的紧急使用授权(EUA)。然而,由于SARS-CoV-2病毒耐药性变体的增多,该授权于2021年4月被撤销。 | |||
T35383 |
Cysteamine bitartrate
Mercaptamine bitartrate |
Others | Others |
Cysteamine bitartrate (Mercaptamine bitartrate)是FDA 批准的胱氨酸消耗氨基硫醇药物(cystine-depleting aminothiol agent),通过参与二硫交换减少溶酶体胱氨酸的积累,用于治疗肾病性胱氨酸病。此外,Cysteamine bitartrate 还具有抗氧化特性。 | |||
T70045 |
HUN47990
|
Others | Others |
HUN47990 is a bisphosphonate (BP) prodrug with antitumor activity. HUN47990 potently inhibits the in vitro growth of a variety of tumor cell lines, especially hematopoietic cell lines, at nanomolar concentrations. HUN47990 inhibited the prenylation of the RAP1A small GTPase signaling protein at concentrations as low as 1-10 nM. HUN47990 slowed the growth of human bladder cancer cells in an immunodeficient mouse model. HUN47990 is significantly more active than zoledronic acid, the most active FD... | |||
T70070 |
Cisapride tartrate
|
Others | Others |
Cisapride tartrate is chemically related to metoclopramide, but unlike metoclopramide, it does not cross the blood-brain barrier or have antidopaminergic effects. Cisapride is a serotonin-4 (5-HT4) receptor agonist. Cisapride was indicated for the symptomatic treatment of adult patients with nocturnal heartburn due to gastroesophageal reflux disease. The Food and Drug Administration (FDA) in America stopped the marketing of cisapride as of 14th July 2000. They had received at least 341 reports o... | |||
T14614 |
Biperiden Hydrochloride
KL 373 (Hydrochloride),盐酸比哌立登 |
Others | Others |
Biperiden Hydrochloride (KL 373 Hydrochloride) is an antiparkinsonian agent, which is the selective central M1 cholinoreceptors blocker and it is used for the adjunctive treatment of all forms of Parkinson's disease (postencephalitic, idiopathic, and arte |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2S0850 |
Malic acid
E 296,苹果酸,2-Hydroxysuccinic acid,Hydroxybutanedioic acid,FDA 2018,Deoxytetraric acid,Pomalus acid |
Others; Endogenous Metabolite | Metabolism; Others |
Malic acid (Pomalus acid) 是一种天然存在于水果中的二羧酸,如苹果和梨。Malic acid 在许多酸味或酸味食物中起作用。 | |||
T0845 |
Cyromazine
CGA-72662,Cyromazin,环丙氨嗪 |
Others; Endogenous Metabolite | Metabolism; Others |
Cyromazine (CGA-72662) 是三聚氰胺的环丙基衍生物,是昆虫生长调节剂,用作杀虫剂和杀螨剂,通过影响某些昆虫幼虫阶段的神经系统而起作用。 | |||
T2S1865 |
Octyl gallate
Gallic acid octyl ester,n-Octylgallate,Octyl 3,4,5-trihydroxybenzoate,Progallin O,Stabilizer GA-8,没食子酸辛酯 |
Antioxidant; Influenza Virus; Reactive Oxygen Species; Antibacterial; Antifungal; HSV | Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; oxidation-reduction |
Octyl gallate (Octyl 3,4,5-trihydroxybenzoate) 具有抗菌、抗氧化作用,有选择性和敏感性的荧光特性,广泛用作食品添加剂。它对 HSV-1,水泡性口炎病毒和脊髓灰质炎病毒有显著的抗病毒作用。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TMIJ-0139 |
Ticagrelor-d7
|
||
Ticagrelor-d7 是 Ticagrelor 的氘代化合物。Ticagrelor 的 CAS 号为 274693-27-5。Ticagrelor (AZD6140) 是可逆的,可口服的P2Y12受体拮抗剂,可抑制血小板聚集。 |