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Search Results for " elt "

Targets Recommended: Proton pump Phospholipase Antibacterial

74

抑制剂 & 化合物

23

天然产物

13

重组蛋白

11

同位素标记化合物

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Cat. No.	Product Name	Target	Signaling Pathways
T0674	Lansoprazole 兰索拉唑,A-65006,AG-1749	Proton pump; Phospholipase; Antibacterial	Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
	Lansoprazole (A-65006) 是一种可抑制胃酸生成的质子泵抑制剂。它是中性鞘磷脂酶的外泌体抑制剂。
T10652	Vimseltinib DCC-3014	c-Fms; CSF-1R; c-Kit	Tyrosine Kinase/Adaptors
	Vimseltinib (DCC-3014) 是 c-FMS(CSF-IR) 和 c-Kit 抑制剂，IC50值分别为 <0.01 μM 和 0.1-1 μM。
T3495	Tasimelteon 他司美琼,VEC-162,BMS-214778	Melatonin Receptor; MT Receptor	GPCR/G Protein; Neuroscience
	Tasimelteon (BMS-214778) 是一种褪黑激素受体激动剂，用于治疗盲人的非 24 小时睡眠-觉醒障碍。
T1486	Oseltamivir phosphate GS 4104,磷酸奥司他韦	Influenza Virus	Microbiology/Virology
	Oseltamivir phosphate (GS 4104) 是一种神经氨酸酶抑制剂，可研究流感。
T6825	Eltrombopag Olamine Promacta Olamine,Revolade,艾曲泊帕乙醇胺盐,Eltrombopag diethanolamine salt,SB497115,艾曲波帕乙醇胺盐,SB-497115GR	Thrombin	Proteases/Proteasome
	Eltrombopag Olamine (Eltrombopag diethanolamine salt) 是 Eltrombopag 的口服活性乙醇胺盐，是一种血小板生成素(TPO)受体激动剂，用于血小板减少的某些病症研究。
T11766L	Eltanexor ONO-7706,KPT-8602,ATG-016	Others	Others
	Eltanexor (ONO-7706) 是一种具有口服活性的 exportin-1 (XPO1) 抑制剂。它具有有效的抗白血病活性。 Eltanexor 通过直接靶向 XPO1 抑制 XPO1 依赖性核输出 (EC50=60.9 nM)。 Eltanexor 在一组白血病细胞系中引起半胱天冬酶依赖性细胞凋亡。
T14997	Conteltinib SY-707,CT-707	FAK; PYK2; ALK	Angiogenesis; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
	Conteltinib (CT-707) 是一种靶向FAK、ALK 和 Pyk2 的酶抑制剂，具有抗肿瘤活性。Conteltinib 对 FAK 有明显的抑制作用，通过抑制 YAP 信号传导来克服肝细胞癌中缺氧介导的索拉非尼耐药性，可用于晚期 ALK 阳性非小细胞肺癌和淋巴癌。
T27254	Eltenac B78820,B 78820,B-78820,BY-820,BY820,BY 820	COX	Immunology/Inflammation; Neuroscience
	Eltenac (B78820) 是一种非甾体抗炎剂，是 COX 抑制剂，具有镇痛活性。Eltenac 抑制 COX-1 和 COX-2 ，可用于研究急性呼吸窘迫综合征（ARDS）。
T7637	Deltorphin I Deltorphin 1,Deltorphin I(TFA),Deltorphin C	Opioid Receptor	Endocrinology/Hormones; GPCR/G Protein; Neuroscience
	Deltorphin I 是 δ-阿片受体的激动剂。
T25832	Moveltipril Moveltipril calcium,MC-838,Altiopril calcium	RAAS	Endocrinology/Hormones
	Moveltipril (Moveltipril calcium) 是一种强效血管紧张素转换酶(ACE)抑制剂。
T5186L	Oseltamivir GS 4104	Influenza Virus	Microbiology/Virology
	Oseltamivir (GS 4104) 是一种具有口服活性和高效性的病毒神经氨酸酶（NA），具有抗病毒活性，抑制 A/H3N2，A/H1N2，A/H1N1 和 B 型流感病毒，可用于研究流感和肺炎。
T20166	Deltorphin Deltorphin A,Dermenkephalin	Opioid Receptor	Endocrinology/Hormones; GPCR/G Protein; Neuroscience
	Deltorphin (Dermenkephalin) 是从亚马逊蛙 Phyllomedusa Sauvage 的皮肤中分离出来的。Deltorphin 对阿片受体也有亲和力。
T6462	Deltarasin	PDE; Ras	GPCR/G Protein; MAPK; Metabolism
	Deltarasin 是一种 KRAS-PDEδ 相互作用的小分子抑制剂，与纯化的 PDEδ 结合，Kd 值为 38 nM。
T9950	ElteN378	mTOR	PI3K/Akt/mTOR signaling
	Elte N378 是一种高效的合成 FKBP12 抑制剂，Ki 为 0.5 nM，是一种低原子量配体，其亲和力与大环内酯类雷帕霉素相当。
T7498	Eltoprazine hydrochloride 1-(2,3-二氢苯并[B][1,4]二氧杂芑-5-基)哌嗪,DU 28853 hydrochloride	5-HT Receptor	GPCR/G Protein; Neuroscience
	Eltoprazine hydrochloride (DU 28853 hydrochloride) 是5-HT1A 和5-HT1B 受体激动剂，也是5-HT2C 受体拮抗剂，pEC50分别为9.96、7.19和6.81。
T7746	Eltoprazine dihydrochloride	Others	Others
	Eltoprazine dihydrochloride 是一种先前开发用于攻击性的药物，已在帕金森病 (PD) 的动物模型和运动障碍 PD 患者中研究了左旋多巴诱导的运动障碍。
T7639	Deltorphin 2 Deltorphin 2(TFA),[D-Ala2]-Deltorphin II	Opioid Receptor	Endocrinology/Hormones; GPCR/G Protein; Neuroscience
	Deltorphin 2 ([D-Ala2]-Deltorphin II) 是一种选择性的 δ 阿片受体肽激动剂，IC50 为 1 nM。
T23717	Ameltolide	Others	Others
	Ameltolide 是一种抗惊厥剂。在动物模型中，它被证明能有效抑制癫痫发作。
T5186	Oseltamivir acid GS 4071,oseltamivir carboxylate,奥斯他伟酸,Ro 64-0802	Influenza Virus; Drug Metabolite	Metabolism; Microbiology/Virology
	Oseltamivir acid (GS 4071) 是Oseltamivir phosphate 的活性代谢产物，是一种有效的流感病毒神经氨酸酶抑制剂和 GS4071 的前药。
T12877L	Seltorexant JNJ-42847922	OX Receptor	GPCR/G Protein; Neuroscience
	Seltorexant (JNJ-42847922) 是一种可口服，高亲和性以及选择性的 orexin-2 受体(OX2R)拮抗剂，对人和大鼠中的 OX2R 的pKi 值分别为 8.0 和 8.1。它穿过血脑屏障，迅速占据大鼠大脑中的 OX2R 结合位点。
T60663L	Oseltamivir acid methyl ester hydrochloride	Others	Others
	Oseltamivir acid methyl ester hydrochloride 是奥司他韦酸的前体形式。它通过羧酸酯酶1 (CES1) 转化为奥司他韦酸。
T2562	Eltrombopag SB-497115,SB-497115-GR,艾曲波帕	Thrombin	Proteases/Proteasome
	Eltrombopag (SB-497115-GR) 是一种具有巨核细胞生成刺激活性的口服活性血小板生成素受体激动剂，可结合并刺激血小板血小板生成素受体，用于血小板减少的某些病症研究。
T1463	Ramelteon 雷美替胺,TAK-375	Melatonin Receptor; MT Receptor	GPCR/G Protein; Neuroscience
	Ramelteon (TAK-375) 是强效高选择性和可口服的 MT1/MT2激动剂，Ki 值分别为 14 和 112 pM，有用于失眠症的研究潜力。
T26367	Reltecimod NSC-37096,P2TA,AB-103,AB103,P-2TA
	Reltecimod, a CD28 antigen inhibitor, is used potentially for the treatment of necrotizing soft tissue infection.
T20166L	Deltorphin acetate Deltorphin acetate(119975-64-3 Free base)	Opioid Receptor	Endocrinology/Hormones; GPCR/G Protein; Neuroscience
	Deltorphin acetate 是一种从青蛙 Phyllomedusa bicolor 的皮肤分泌物中获得的物质，对 δ-阿片受体具有高选择性和亲和力。
T80613	Linvoseltamab REGN5458
	Linvoseltamab为双特异性抗体，针对BCMA(TNFRSF17)与CD3epsilon。该化合物于复发/难治性多发性骨髓瘤(RRMM)模型中展示了良好的安全性和效力。
T23155	Piefeltarraenin ⅠB	Others	Others
	Piefeltarraenin ⅠB is extracted from the whole herb of Picriafel-terrae Lour.
T124900	Delta-9-Tetrahydrocannabivarinic acid	Others	Others
	Delta-9-Tetrahydrocannabivarinic acid 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T124900。
T23976	Deltasonamide 1 Deltasonamide	Others	Others
	Deltasonamide is a potent and selective inhibitor of PDE6δ‐KRas.
T66182	2,3,4,6-Tetra-O-(trimethylsilyl)-D-glucono-delta-lactone	Others	Others
	2,3,4,6-Tetra-O-(trimethylsilyl)-D-glucono-delta-lactone 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T66182，CAS号为 32384-65-9。
T83958	CELT-327	Others	Others
	CELT-327是一种高效且选择性的荧光hA2B/A3腺苷受体拮抗剂，其Kivalues在A2B和A3受体上分别为35.6 nM和45.7 nM。在表达A2B腺苷受体的HCT116细胞中，CELT-327表现出剂量依赖性的膜荧光标记，荧光信号快速扩散并在细胞单层中均匀分布。在活的HCT116紧凑球体中，CELT-327展现出整个球体直径上的均匀染色，可达到球体深层区域。CELT-327可作为荧光腺苷受体探针用于荧光结合分析、活细胞成像、流式细胞术和荧光偏振分析。它是GPCR放射标记配体的合适替代品。激发和发射最大值（λ）分别为589 nm和616 nm。这些波长与作为TR-FRET分析中接受体染料使用兼容，与CoraFluor1 TR-FRET供体一同使用。
T36722	Deltorphin II (trifluoroacetate salt)	Others	Others
	Deltorphin II is a peptide agonist of δ2-opioid receptors.1,2It is selective for δ-opioid receptors over μ- and κ-opioid receptors in radioligand bindings assays (Kis = 0.0033, >1, and >1 μM, respectively) and induces [35S]GTPγS binding in mouse brain membrane preparations (EC50= 0.034 μM). Deltorphin II (0.12 mg/kg) decreases the infarction zone:risk zone ratio in a rat model of myocardial ischemia-reperfusion injury induced by coronary occlusion, an effect that can be reversed by the δ2-opioid...
T82021	Izeltabart IMGC-936	ADC Antibody	Antibody-drug Conjugate/ADC Related
	Izeltabart（IMGC-936）是一款针对ADAM9的基于Maytansinoid的ADC，由与DM21-C位点特异性偶联的高亲和力人源化抗体构成，使Maytansinoid微管破坏载体通过稳定的三肽连接子进行传递，达到药物-抗体比约为2.0。Izeltabart在ADAM9阳性人类肿瘤细胞系上显示出明显的细胞毒性，并在动物异种移植肿瘤模型中展现出显著的抗肿瘤效果。
T11766	Eltanexor Z-isomer KPT-8602 (Z-isomer)	Others	Others
	Eltanexor Z-isomer exhibits different inhibitory effects on Z138, MM15, 3T3 cell lines, with IC50s of 100 nM-50 μM, < 100 nM, > 30 μM, respectively.Eltanexor Z-isomer is the less active isomer of KPT-8602. KPT-8602 is a potent CRM1 inhibitor.
T83957	CELT-211
	CELT-211是一种强效且选择性的h5HT2B血清素受体荧光配体。它对h5HT2B显示出完全选择性，与h5HT2A、h5HT2C相比，其在放射配体结合测定中针对h5HT2B受体的Ki值为56.3 nM。激发和发射峰值（λ）分别为589和616 nm。这些波长与CoraFlor 1 TR-FRET供体一起使用作为TR-FRET测定中的受体染料是兼容的。
T60663	Oseltamivir acid methyl ester	Others	Others
	Oseltamivir acid methyl ester 是Oseltamivir acid 的前体形式，可通过羧酸酯酶1 (CES1) 转化为Oseltamivir acid。Oseltamivir acid 是神经氨酸酶抑制剂和抗病毒剂。
T12461	PI3Kdelta inhibitor 1	PI3K	PI3K/Akt/mTOR signaling
	PI3Kdelta inhibitor 1 is a potent, selective and orally available inhibitor of PI3Kδ with an IC50 of 1.3 nM.
T82587	Delta (Phospho) Sleep Inducing Peptide DSIP-P
	Delta (Phospho) Sleep Inducing Peptide (DSIP-P) 是促进睡眠效应持久的多肽，能诱导大鼠昼夜运动行为的改变。
T78271	Anti-Mouse TCR gamma/delta Antibody (UC7-13D5)
	Anti-Mouse TCR gamma/delta Antibody为针对小鼠TCR gamma/delta的IgG类免疫抑制抗体，其宿主为亚美尼亚仓鼠。
T10994L2	Deltasonamide 2 (TFA)	PDE	Metabolism
	Deltasonamide 2 TFA is competitive, high affinity PDEδ inhibitor with a Kd of ~385 pM.
T25303	Deltamycin A1	Others	Others
	Deltamycin A1 is a novel macrolide antibiotic.
T131544	Bergenin (Vakerin; Peltophorin; Cuscutin)	Others	Others
	Bergenin (Vakerin; Peltophorin; Cuscutin) 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T131544。
T32375	Kelthane-S Kelthane S	Others	Others
	Kelthane-S is a bioactive chemical.
T70750	Deltibant	Others	Others
	Deltibantis a bradykinin receptor antagonist.
T75770	Deltorphin 2 TFA
	Deltorphin 2 TFA 是一种选择性的 δ 阿片受体肽激动剂。
T41328	Delta-12-Prostaglandin J2
	Delta-12-Prostaglandin J2 在生命科学相关研究中具有广泛的应用。
T78107	Reltecimod TFA AB-103 TFA	Others	Others
	Reltecimod (AB-103) TFA 是一款针对 T 细胞特异性表面糖蛋白CD28(TP44) 的拮抗剂。该化合物能够有效抵御各类细菌感染、细菌产生的外毒素和内毒素，以及电离辐射。其通过特异性目标定位并调节 CD28/B7-2 共刺激通路以减弱炎症反应，但并不完全抑制该通路。Reltecimod TFA 主要用于坏死性软组织感染(NSTIs)的研究。
T26367L	Reltecimod sodium AB 103 sodium,AB-103 sodium,AB103 sodium	Others	Others
	Reltecimod sodium, a CD28 antigen inhibitor, is used potentially for the treatment of necrotizing soft tissue infection.
T4413	Poseltinib	Others	Others
	Poseltinib 是一种具有口服活性，选择性，不可逆的小分子Bruton 酪氨酸激酶 (BTK) 抑制剂，IC50为 1.95 nM，对BTK 的选择性分别是 BMX，TEC 和 TXK 的 0.3，2.3 和 2.4 倍。Poseltinib 可共价结合 BTK 的活性位点 (半胱氨酸 481 残基)，并显示出对 B 细胞受体 (BCR)，Fc 受体 (FcR)，Toll 样受体 (TLR) 介导的信号传导的有效抑制。
T83956	CELT-133	Others	Others
	CELT-133是一种选择性的hα1A肾上腺素能受体荧光拮抗剂。它对α1A显示出完全的选择性，相对于α2A，在放射配体结合实验中的Ki值为5 nM，1 μM时位移为15%。CELT-133对α1肾上腺素能受体的所有亚型都有相同的结合能力。激发和发射峰值(λ)分别是560 nm和571 nm。这些波长与作为TR-FRET实验中接受体染料的使用兼容，同时可以与CoraFluor 1 TR-FRET供体配合使用。

化合物

Cat.No: T0674

Synonym: 兰索拉唑,A-65006,AG-1749

Target: Proton pump, Phospholipase, Antibacterial

Cat.No: T10652

Synonym: DCC-3014

Target: c-Fms, CSF-1R, c-Kit

Cat.No: T3495

Synonym: 他司美琼,VEC-162,BMS-214778

Target: Melatonin Receptor, MT Receptor

Oseltamivir phosphate

Cat.No: T1486

Synonym: GS 4104,磷酸奥司他韦

Target: Influenza Virus

Eltrombopag Olamine

Cat.No: T6825

Synonym: Promacta Olamine,Revolade,艾曲泊帕乙醇胺盐,Eltrombopag diethanolamine salt,SB497115,艾曲波帕乙醇胺盐,SB-497115GR

Target: Thrombin

Cat.No: T11766L

Synonym: ONO-7706,KPT-8602,ATG-016

Target: Others

Cat.No: T14997

Synonym: SY-707,CT-707

Target: FAK, PYK2, ALK

Cat.No: T27254

Synonym: B78820,B 78820,B-78820,BY-820,BY820,BY 820

Target: COX

Cat.No: T7637

Synonym: Deltorphin 1,Deltorphin I(TFA),Deltorphin C

Target: Opioid Receptor

Cat.No: T25832

Synonym: Moveltipril calcium,MC-838,Altiopril calcium

Target: RAAS

Cat.No: T5186L

Synonym: GS 4104

Target: Influenza Virus

Cat.No: T20166

Synonym: Deltorphin A,Dermenkephalin

Target: Opioid Receptor

Cat.No: T6462

Target: PDE, Ras

Cat.No: T9950

Target: mTOR

Eltoprazine hydrochloride

Cat.No: T7498

Synonym: 1-(2,3-二氢苯并[B][1,4]二氧杂芑-5-基)哌嗪,DU 28853 hydrochloride

Target: 5-HT Receptor

Eltoprazine dihydrochloride

Cat.No: T7746

Target: Others

Cat.No: T7639

Synonym: Deltorphin 2(TFA),[D-Ala2]-Deltorphin II

Target: Opioid Receptor

Cat.No: T23717

Target: Others

Oseltamivir acid

Cat.No: T5186

Synonym: GS 4071,oseltamivir carboxylate,奥斯他伟酸,Ro 64-0802

Target: Influenza Virus, Drug Metabolite

Cat.No: T12877L

Synonym: JNJ-42847922

Target: OX Receptor

Oseltamivir acid methyl ester hydrochloride

Cat.No: T60663L

Target: Others

Cat.No: T2562

Synonym: SB-497115,SB-497115-GR,艾曲波帕

Target: Thrombin

Cat.No: T1463

Synonym: 雷美替胺,TAK-375

Target: Melatonin Receptor, MT Receptor

Cat.No: T26367

Synonym: NSC-37096,P2TA,AB-103,AB103,P-2TA

Deltorphin acetate

Cat.No: T20166L

Synonym: Deltorphin acetate(119975-64-3 Free base)

Target: Opioid Receptor

Cat.No: T80613

Synonym: REGN5458

Piefeltarraenin ⅠB

Cat.No: T23155

Target: Others

Delta-9-Tetrahydrocannabivarinic acid

Cat.No: T124900

Target: Others

Deltasonamide 1

Cat.No: T23976

Synonym: Deltasonamide

Target: Others

2,3,4,6-Tetra-O-(trimethylsilyl)-D-glucono-delta-lactone

Cat.No: T66182

Target: Others

Cat.No: T83958

Target: Others

Deltorphin II (trifluoroacetate salt)

Cat.No: T36722

Target: Others

Cat.No: T82021

Synonym: IMGC-936

Target: ADC Antibody

Eltanexor Z-isomer

Cat.No: T11766

Synonym: KPT-8602 (Z-isomer)

Target: Others

Cat.No: T83957

Oseltamivir acid methyl ester

Cat.No: T60663

Target: Others

PI3Kdelta inhibitor 1

Cat.No: T12461

Target: PI3K

Delta (Phospho) Sleep Inducing Peptide

Cat.No: T82587

Synonym: DSIP-P

Anti-Mouse TCR gamma/delta Antibody (UC7-13D5)

Cat.No: T78271

Deltasonamide 2 (TFA)

Cat.No: T10994L2

Target: PDE

Cat.No: T25303

Target: Others

Bergenin (Vakerin; Peltophorin; Cuscutin)

Cat.No: T131544

Target: Others

Cat.No: T32375

Synonym: Kelthane S

Target: Others

Cat.No: T70750

Target: Others

Deltorphin 2 TFA

Cat.No: T75770

Delta-12-Prostaglandin J2

Cat.No: T41328

Cat.No: T78107

Synonym: AB-103 TFA

Target: Others

Reltecimod sodium

Cat.No: T26367L

Synonym: AB 103 sodium,AB-103 sodium,AB103 sodium

Target: Others

Cat.No: T4413

Target: Others

Cat.No: T83956

Target: Others

Cat. No.	Product Name	Target	Signaling Pathways
T5S1025	Picfeltarraenin IA 苦玄参苷IA,Picfeltarraenin A,苦玄参苷 IA	AChE	Neuroscience
	Picfeltarraenin IA (Picfeltarraenin A) 是一种Picriafel-terraeLour (P.fel-terrae) 中提取的三萜类化合物，是一种乙酰胆碱酯酶抑制剂。它可用于感染，癌症和炎症的研究。
T6000	Delta-Tocopherol (+)-DELTA-生育酚,D-DELTA-TOCOPHEROL	Endogenous Metabolite	Metabolism
	Delta-Tocopherol 是维生素 E 的异构体，具有抗氧化活性。
T20754	Deltamethrin Butoss,RU-22974,Esbecythrin,溴氰菊酯,K-Othrin,Decamethrin,RU 22974	Others	Others
	Deltamethrin (RU 22974) 是一种具有神经毒性的拟除虫菊酯杀虫剂，在大鼠中能够产生一系列可逆的运动症状(如包括后肢僵硬、舞蹈性关节炎)。
T4S1024	Picfeltarraenin IB 苦玄参苷IB,苦玄参苷 IB	Others; AChE	Neuroscience; Others
	Picfeltarraenin IB 是一种Picriafel-terraeLour (P.fel-terrae) 中提取的三萜类化合物，是一种乙酰胆碱酯酶抑制剂。它可用于感染，癌症和炎症的研究。
T3844	Deltonin 三角叶薯蓣皂苷	ERK; Others; Akt; Endogenous Metabolite	Cytoskeletal Signaling; MAPK; Metabolism; Others; PI3K/Akt/mTOR signaling
	Deltonin 是从盾叶薯蓣中得到的一种甾体皂苷，抑制ERK1/2和AKT 的活化，具有抗肿瘤活性。
T3S1888	Deltaline 德尔塔林,Deltamine 6-acetate,Eldelin	Others	Others
	Deltaline (Eldelin) 是一种从滇川翠雀花属植物中分离出来的二萜类生物碱。它可用于缓解疼痛的研究，滇川翠雀花属植物也被用于风湿痛、中风引起的麻痹、类风湿性关节炎的研究。
TN3814	Delta 5-avenasterol	Others	Others
	Delta 5-avenasterol has antioxidant activity.
TN3390	alpha-Peltatin	Others	Others
	alpha-Peltatin 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN3390，CAS号为 568-53-6。
TN6697	Delta-Nonalactone
	Delta-Nonalactone 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN6697，CAS号为 3301-94-8。
TN4747	(-)-beta-Peltatin	Others	Others
	(-)-beta-Peltatin has antimitotic, and antineoplastic activities.
TN7422	Peltatoside 7-O-beta-glucopyranoside	Others	Others

TN3817	Delta-Caesalpin	Others	Others
	Delta-Caesalpin 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN3817，CAS号为 7716-14-5。
TN6070	Deltatsine
	Deltatsine是一种天然产物，属于毛茛科翠雀属，其产品编号为 TN6070，CAS号为 92631-66-8。Deltatsine可用作对照参考。
TN3815	Delta 7-avenasterol
	Delta 7-avenasterol has antioxidant activity.
TN2067	Picfeltarraegenin X 苦玄参苷X,Picfeltarraenin X	AChR	Neuroscience
	Picfeltarraenin X shows stronger AChE inhibition than the known AChE inhibitor Tacrine.
TN7332	Delta-9-Tetrahydrocannabinolic acid Δ9-Tetrahydrocannabinolic Acid A	Others	Others
	Delta-9-Tetrahydrocannabinolic acid has been shown to safeguard dopaminergic neurons from cell death induced by MPP(+).
T19274	delta-Valerobetaine Δ-Valerobetaine	Endogenous Metabolite	Metabolism
	delta-Valerobetaine 是一种饮食依赖性肥胖原，是微生物组衍生的代谢物，是三甲胺 N-氧化物 (TMAO) 的前体。delta-Valerobetaine对小鼠的学习和记忆过程有害，可调节抑制性突触传递和神经元网络活动。
TN3505	Beta-Peltoboykinolic acid	Phosphatase	Metabolism
	Beta-Peltoboykinolic acid has in vitro protein tyrosine phosphatase 1B (PTP1B) inhibitory, it inhibits PTP1B with IC50 values of 5.2+/-0.5 microM. It also has cytotoxic activity.
TN3816	delta-Amyrin acetate	Others	Others
	β-Amyrin acetate and β-Amyrin acetate have antidyslipidemic activity.
T83606	(-)-β-Peltatin-5-O-beta-D-glucopyranoside
	(-)-β-Peltatin-5-O-beta-D-glucopyranoside为自P. peltatum L中分离出的活性化合物。
TN2046	Peltatoside 3-阿拉伯糖葡糖基槲皮素	Others	Others
	Peltatoside is a natural product
TN2066	Picfeltarraenin IV	Others	Others
	Picfeltarraenin IV is a natural product from Picria felterrae Lour.
TN2106	Protodeltonin 原三角叶皂苷	BCL; PARP; Caspase	Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Proteases/Proteasome
	Protodeltonin may have anti-thrombotic activity by both improving the anticoagulation activity and inhibiting platelet aggregation action. Protodeltonin can inhibit the proliferation of a panel of established human and murine cancer cell lines in vitro.

天然产物

Picfeltarraenin IA

Cat.No: T5S1025

Synonym: 苦玄参苷IA,Picfeltarraenin A,苦玄参苷 IA

Target: AChE

Delta-Tocopherol

Cat.No: T6000

Synonym: (+)-DELTA-生育酚,D-DELTA-TOCOPHEROL

Target: Endogenous Metabolite

Cat.No: T20754

Synonym: Butoss,RU-22974,Esbecythrin,溴氰菊酯,K-Othrin,Decamethrin,RU 22974

Target: Others

Picfeltarraenin IB

Cat.No: T4S1024

Synonym: 苦玄参苷IB,苦玄参苷 IB

Target: Others, AChE

Cat.No: T3844

Synonym: 三角叶薯蓣皂苷

Target: ERK, Others, Akt, Endogenous Metabolite

Cat.No: T3S1888

Synonym: 德尔塔林,Deltamine 6-acetate,Eldelin

Target: Others

Delta 5-avenasterol

Cat.No: TN3814

Target: Others

Cat.No: TN3390

Target: Others

Delta-Nonalactone

Cat.No: TN6697

(-)-beta-Peltatin

Cat.No: TN4747

Target: Others

Peltatoside 7-O-beta-glucopyranoside

Cat.No: TN7422

Target: Others

Delta-Caesalpin

Cat.No: TN3817

Target: Others

Cat.No: TN6070

Delta 7-avenasterol

Cat.No: TN3815

Picfeltarraegenin X

Cat.No: TN2067

Synonym: 苦玄参苷X,Picfeltarraenin X

Target: AChR

Delta-9-Tetrahydrocannabinolic acid

Cat.No: TN7332

Synonym: Δ9-Tetrahydrocannabinolic Acid A

Target: Others

delta-Valerobetaine

Cat.No: T19274

Synonym: Δ-Valerobetaine

Target: Endogenous Metabolite

Beta-Peltoboykinolic acid

Cat.No: TN3505

Target: Phosphatase

delta-Amyrin acetate

Cat.No: TN3816

Target: Others

(-)-β-Peltatin-5-O-beta-D-glucopyranoside

Cat.No: T83606

Cat.No: TN2046

Synonym: 3-阿拉伯糖葡糖基槲皮素

Target: Others

Picfeltarraenin IV

Cat.No: TN2066

Target: Others

Cat.No: TN2106

Synonym: 原三角叶皂苷

Target: BCL, PARP, Caspase

Species：

Expression System：

Tag：

Cat. No.	Product Name	Species	Expression System
TMPY-01429	RELT/TNFRSF19L Protein, Human, Recombinant (His) TRLT,TNFRSF19L,RELT tumor necrosis factor receptor	Human	HEK293 Cells
	RELT/TNFRSF19L Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 15.7 kDa and the accession number is A0A024R5N3.
TMPY-01029	RELT/TNFRSF19L Protein, Human, Recombinant (His & hFc) TRLT,TNFRSF19L,RELT tumor necrosis factor receptor	Human	HEK293 Cells
	RELT/TNFRSF19L Protein, Human, Recombinant (His & hFc) is expressed in HEK293 mammalian cells with His and hFc tag. The predicted molecular weight is 42 kDa and the accession number is A0A024R5N3.
TMPJ-00272	RELT/TNFRSF19L Protein, Human, Recombinant (hFc) RELT,TNFRSF19L,Receptor expressed in lymphoid tissu...	Human	HEK293 Cells
	Tumor necrosis factor receptor superfamily member 19L (TNFRSF19L), also known as Receptor expressed in lymphoid tissues and RELT, is a member of the TNF-receptor superfamily. TNFRSF19L is a single-pass type membrane protein and contains one TNFR-Cys repeat. TNFRSF19L is highly expressed in spleen, lymph node, thymus, peripheral blood leukocytes, bone marrow and fetal liver. It has been shown TNFRSF19L activates the NF-kappaB pathway and selectively binds TNF receptor-associated factor 1 (TRAF1)....
TMPH-03534	Delta-hemolysin Protein, S. aureus, Recombinant (His & KSI) hld,Delta-hemolysin,Delta-toxin,Delt	Staphylococcus aureus	E. coli
	Lyses erythrocytes and many other mammalian cells. Delta-hemolysin Protein, S. aureus, Recombinant (His & KSI) is expressed in E. coli expression system with N-6xHis-KSI tag. The predicted molecular weight is 18.3 kDa and the accession number is P0A0M1.
TMPH-01434	Hemoglobin subunit delta/HBD Protein, Human, Recombinant (GST & His) HBD,Hemoglobin delta chain,Hemoglobin subunit d...	Human	E. coli
	Involved in oxygen transport from the lung to the various peripheral tissues. Hemoglobin subunit delta/HBD Protein, Human, Recombinant (GST & His) is expressed in E. coli expression system with N-6xHis-GST tag. The predicted molecular weight is 47.5 kDa and the accession number is P02042.
TMPH-00811	Hepatitis delta virus genotype I (HDV) Small delta antigen Protein (His & Myc) Small delta antigen,p24	HDV	P. pastoris (Yeast)
	Promotes both transcription and replication of genomic RNA. Following virus entry into host cell, provides nuclear import of HDV RNPs thanks to its nuclear localization signal. May interact with host RNA polymerase II thereby changing its template requirement from DNA to RNA. RNA pol II complex would then acts as an RNA-directed RNA polymerase, and transcribe and replicate HDV genome. Hepatitis delta virus genotype I (HDV) Small delta antigen Protein (His & Myc) is expressed in yeast with N-6xHi...
TMPY-04531	p38 delta/MAPK13 Protein, Human, Recombinant (GST), Activated in vitro P38 δ/MAPK13,MAPK13,PRKM13,MAPK-13,p38δ,p38delta,mi...	Human	Baculovirus Insect Cells
	p38 delta/MAPK13 Protein, Human, Recombinant (GST), Activated in vitro is expressed in Baculovirus insect cells with GST tag. The predicted molecular weight is 68.4 kDa and the accession number is O15264.
TMPH-00056	Delta-AITX-Avd1c Protein, Anemonia sulcata, Recombinant (His) ATX II,Delta-AITX-Avd1c,Toxin II,Delta-act...	Anemonia sulcata	P. pastoris (Yeast)
	Binds specifically to voltage-gated sodium channels (Nav) (site 3), thereby delaying their inactivation. Has a strong effect on crustaceans and insects (DmNav1) and a weaker effect on mammals. This toxin is highly potent at mammalian Nav1.1/SCN1A (EC(50)=6.01 nM) and Nav1.2/SCN2A (EC(50)=7.88 nM). It has also great activity on Nav1.5/SCN5A (EC(50)=49.05 nM), Nav1.4/SCN4A (EC(50)=109.49 nM) and Nav1.6/SCN8A (EC(50)=about 180 nM) and is less potent on Nav1.3/SCN3A (EC(50)=759.22 nM) (when measured...
TMPH-00810	Hepatitis delta virus genotype I (HDV) Large delta antigen Protein (His & Myc) p27,Large delta antigen	HDV	P. pastoris (Yeast)
	Following virus entry into host cell, provides nuclear import of HDV RNPs thanks to its nuclear localization signal. Needs co-infection with hepatitis B virus to provide surface proteins, otherwise there is no packaging or budding. Packages the HDV ribonucleoprotein in hepatitis B virus empty particles. Interacts with both HDV genomic RNA and cytoplasmic tail of HBsAg. May inhibit viral RNA replication. Hepatitis delta virus genotype I (HDV) Large delta antigen Protein (His & Myc) is expressed i...
TMPH-00025	DELTA-actitoxin-Aeq1a Protein, Acinetobacter baumannii, Recombinant (His & SUMO) 1,2-CTD,catA,Catechol 1,2-dioxygenase	Acinetobacter baylyi	E. coli
	DELTA-actitoxin-Aeq1a Protein, Acinetobacter baumannii, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 50.3 kDa and the accession number is P07773.
TMPH-02473	14-3-3 zeta/delta Protein, Mouse, Recombinant (His & SUMO) Ywhaz,14-3-3 protein zeta/delta,SEZ-2,KCIP-1,Protei...	Mouse	E. coli
	Adapter protein implicated in the regulation of a large spectrum of both general and specialized signaling pathways. Binds to a large number of partners, usually by recognition of a phosphoserine or phosphothreonine motif. Binding generally results in the modulation of the activity of the binding partner. Induces ARHGEF7 activity on RAC1 as well as lamellipodia and membrane ruffle formation. In neurons, regulates spine maturation through the modulation of ARHGEF7 activity. 14-3-3 zeta/delta Prot...
TMPY-04551	p38 delta/MAPK13 Protein, Human, Recombinant (GST) MAPK13,p38δ,PRKM13,MAPK-13,mitogen-activated protein kinase ...	Human	Baculovirus Insect Cells
	p38 delta/MAPK13 Protein, Human, Recombinant (GST) is expressed in Baculovirus insect cells with GST tag. The predicted molecular weight is 68.4 kDa and the accession number is O15264.
TMPH-00818	Delta-theraphotoxin-Hm1a Protein, Heteroscodra maculata, Recombinant (His & Myc & SUMO) Kappa-TRTX-Hm1a,Delta-TRTX-Hm1a,Heteroscodratoxin-1...	Heteroscodra maculata	E. coli
	Delta-theraphotoxin-Hm1a Protein, Heteroscodra maculata, Recombinant (His & Myc & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO and C-Myc tag. The predicted molecular weight is 21.5 kDa and the accession number is P60992.

重组蛋白

RELT/TNFRSF19L Protein, Human, Recombinant (His)

Cat.No: TMPY-01429

Species: Human

Expression System: HEK293 Cells

RELT/TNFRSF19L Protein, Human, Recombinant (His & hFc)

Cat.No: TMPY-01029

Species: Human

Expression System: HEK293 Cells

RELT/TNFRSF19L Protein, Human, Recombinant (hFc)

Cat.No: TMPJ-00272

Species: Human

Expression System: HEK293 Cells

Delta-hemolysin Protein, S. aureus, Recombinant (His & KSI)

Cat.No: TMPH-03534

Species: Staphylococcus aureus

Expression System: E. coli

Hemoglobin subunit delta/HBD Protein, Human, Recombinant (GST & His)

Cat.No: TMPH-01434

Species: Human

Expression System: E. coli

Hepatitis delta virus genotype I (HDV) Small delta antigen Protein (His & Myc)

Cat.No: TMPH-00811

Species: HDV

Expression System: P. pastoris (Yeast)

p38 delta/MAPK13 Protein, Human, Recombinant (GST), Activated in vitro

Cat.No: TMPY-04531

Species: Human

Expression System: Baculovirus Insect Cells

Delta-AITX-Avd1c Protein, Anemonia sulcata, Recombinant (His)

Cat.No: TMPH-00056

Species: Anemonia sulcata

Expression System: P. pastoris (Yeast)

Hepatitis delta virus genotype I (HDV) Large delta antigen Protein (His & Myc)

Cat.No: TMPH-00810

Species: HDV

Expression System: P. pastoris (Yeast)

DELTA-actitoxin-Aeq1a Protein, Acinetobacter baumannii, Recombinant (His & SUMO)

Cat.No: TMPH-00025

Species: Acinetobacter baylyi

Expression System: E. coli

14-3-3 zeta/delta Protein, Mouse, Recombinant (His & SUMO)

Cat.No: TMPH-02473

Species: Mouse

Expression System: E. coli

p38 delta/MAPK13 Protein, Human, Recombinant (GST)

Cat.No: TMPY-04551

Species: Human

Expression System: Baculovirus Insect Cells

Delta-theraphotoxin-Hm1a Protein, Heteroscodra maculata, Recombinant (His & Myc & SUMO)

Cat.No: TMPH-00818

Species: Heteroscodra maculata

Expression System: E. coli

Cat. No.	Product Name	Target	Signaling Pathways
TMIH-0485	Ramelteon-d3
	Ramelteon-d3 是 Ramelteon 的氘代化合物。Ramelteon 的 CAS 号为 196597-26-9。Ramelteon 是强效高选择性和可口服的MT1/MT2激动剂，Ki值分别为 14 和 112 pM，有用于失眠症的研究潜力。
TMIH-0356	Monohydroxylated ramelteon (II)-d3
	Monohydroxylated ramelteon (II)-d3 是 Monohydroxylated ramelteon (II) 的氘代化合物。Monohydroxylated ramelteon (II) 的 CAS 号为 896736-21-3。
TMIH-0411	Oseltamivir-d3 acid
	Oseltamivir-d3 acid 是 Oseltamivir acid 的氘代化合物。Oseltamivir acid 的 CAS 号为 196618-13-0。
TMIH-0486	Ramelteon-d5
	Ramelteon-d5 是 Ramelteon 的氘代化合物。Ramelteon 的 CAS 号为 196597-26-9。Ramelteon 是强效高选择性和可口服的MT1/MT2激动剂，Ki值分别为 14 和 112 pM，有用于失眠症的研究潜力。
TMIH-0412	Oseltamivir-d3 acid(3R,4S,5S)
	Oseltamivir-d3 acid(3R,4S,5S) 是 Oseltamivir acid(3R,4S,5S) 的氘代化合物。
TMIJ-0061	Oseltamivirphosphate-d5
	Oseltamivirphosphate-d5 是 Oseltamivirphosphate 的氘代化合物。Oseltamivirphosphate 的 CAS 号为 204255-11-8。
T70035	Tasimelteon-d5
	Tasimelteon-d5 is intended for use as an internal standard for the quantification of tasimelteon by GC- or LC-MS. Tasimelteon is a melatonin (MT) receptor agonist. It selectively binds MT1 and MT2 receptors over a panel of 160 additional receptors and enzymes at 10 µM. Tasimelteon inhibits forskolin-induced cAMP accumulation with EC50 values of 0.79 and 1 nM in NIH3T3 cells expressing the MT1 or MT2 receptor, respectively. Formulations containing tasimelteon have been used in the treatment of no...
TMID-0032	Oseltamivir-d3
	Oseltamivir-d3 是 Oseltamivir 的氘代化合物。Oseltamivir 的 CAS 号为 196618-13-0。Oseltamivir (GS 4104) 是一种具有口服活性和高效性的病毒神经氨酸酶（NA），具有抗病毒活性，抑制 A/H3N2，A/H1N2，A/H1N1 和 B 型流感病毒，可用于研究流感和肺炎。
TMIJ-0071	Oseltamivir-13C-d3 Acid
	Oseltamivir-13C-d3 Acid 是 Oseltamivir Acid 的 13C 和氘代化合物。Oseltamivir Acid 的 CAS 号为 187227-45-8。Oseltamivir acid是Oseltamivir phosphate 的活性代谢产物，是一种有效的流感病毒神经氨酸酶抑制剂和 GS4071 的前药。
TMIJ-0230	Oseltamivir EP Impurity C-d3 HCl
	Oseltamivir EP Impurity C-d3 HCl 是 Oseltamivir EP Impurity C HCl 的氘代化合物。Oseltamivir EP Impurity C HCl 的 CAS 号为 1415963-60-8。
T38602	(E/Z)-Eltrombopag 13C4 (E/Z)-Eltrombopag 13C4,(E/Z)-SB-497115 13C4
	(E/Z)-Eltrombopag 13C4 ((E/Z)-SB-497115 13C4) is a mixture complex of E-Eltrombopag and Z-Eltrombopag, with 13C labeled. Z-Eltrombopag is a thrombopoietin (TPO) receptor agonist developed for certain conditions that lead to thrombocytopenia.

同位素标记化合物

Cat.No: TMIH-0485

Monohydroxylated ramelteon (II)-d3

Cat.No: TMIH-0356

Oseltamivir-d3 acid

Cat.No: TMIH-0411

Cat.No: TMIH-0486

Oseltamivir-d3 acid(3R,4S,5S)

Cat.No: TMIH-0412

Oseltamivirphosphate-d5

Cat.No: TMIJ-0061

Cat.No: T70035

Cat.No: TMID-0032

Oseltamivir-13C-d3 Acid

Cat.No: TMIJ-0071

Oseltamivir EP Impurity C-d3 HCl

Cat.No: TMIJ-0230

(E/Z)-Eltrombopag 13C4

Cat.No: T38602

Synonym: (E/Z)-Eltrombopag 13C4,(E/Z)-SB-497115 13C4

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