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Search Results for " eda "

Targets Recommended: Others PROTAC Linker

62

抑制剂 & 化合物

25

天然产物

15

重组蛋白

6

同位素标记化合物

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Cat. No.	Product Name	Target	Signaling Pathways
T17549	Biotin-EDA	Others; PROTAC Linker	Others; PROTAC
	Biotin-EDA 是一种属于 alkyl chain 类的 PROTAC linker，可用于 PROTAC 分子的合成。
T39373	PNU-EDA-Gly5 PNU-EDA-Gly5	Others; Drug-Linker Conjugates for ADC	Antibody-drug Conjugate/ADC Related; Others
	PNU-EDA-Gly5 is a DNA topoisomerase I inhibitor-based oligo-glycine linker-payload used for the synthesis of antibody-drug conjugates (ADCs). It consists of the DNA topoisomerase I inhibitor PNU-159682 and the linker EDA-Gly5.
T18247	Mal-C2-Gly3-EDA	Others; ADC Linker	Antibody-drug Conjugate/ADC Related; Others
	Mal-C2-Gly3-EDA is a cleavable antibody-drug conjugate (ADC) linker equipped with a Maleimide moiety. It serves the purpose of facilitating the synthesis of ADCs.
T18246	Mal-C2-Gly3-EDA-PNU-159682	Others; Drug-Linker Conjugates for ADC	Antibody-drug Conjugate/ADC Related; Others
	Mal-C2-Gly3-EDA-PNU-159682, a drug-linker conjugate for antibody-drug conjugates (ADC), combines the cleavable ADC linker Mal-C2-Gly3-EDA with the potent ADC cytotoxin PNU-159682.
T75354	RH-EDA	Others	Others
	RH-EDA 是一种基于罗丹明的开启式荧光探针，用于检测生命系统中的羟基自由基。
T74555	EDA-DA	Others	Others
	EDA-DA 是一种 N 末端标记的二肽探针，可用于标记细菌的肽聚糖 (PG)。肽聚糖 (PG) 是绝大多数细菌细胞壁中的一种基本结构，对于分裂和维持细胞形状和静水压力至关重要。
T82842	BODIPY FL EDA free base
	ODIPY FL EDA free base为绿色荧光胺类探针，能通过R-NH2与醛或酮反应形成可逆的席夫碱产物。使用如硼氢化钠或氰硼氢化钠等还原剂，ODIPY FL EDA free base可转化成稳定的胺衍生物，适用于检测修饰或未修饰脱氧核苷酸，以及评估DNA损伤和基因组DNA甲基化情况。
T3979	Emedastine LY188695,依美斯汀,Emadine	Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Emedastine (LY188695) 是一种可口服的，选择性和高亲和力的组胺 H1受体拮抗剂，Ki 值为 1.3 nM。它是苯并咪唑衍生物，可用于过敏性鼻炎、过敏性皮肤疾病和过敏性结膜炎的研究。
T13110	Tedatioxetine hydrobromide Lu AA 24530 hydrobromide	Dopamine Receptor; 5-HT Receptor; Norepinephrine	GPCR/G Protein; Neuroscience
	Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) 是一种血清素-去甲肾上腺素-多巴胺再摄取抑制剂，也是 5-HT2A、5-HT2C、5-HT3 和 α1A-肾上腺素能受体的拮抗剂，可用于治疗抑郁症和焦虑症。
T2410	Nedaplatin 奈达铂,NSC 375101D	DNA/RNA Synthesis	Cell Cycle/Checkpoint; DNA Damage/DNA Repair
	Nedaplatin (NSC-375101D) 是顺铂的衍生物，是肿瘤集落形成单位的 DNA 损伤剂，IC50为94 μM。
T22436	Takeda-6d	VEGFR	Angiogenesis; Tyrosine Kinase/Adaptors
	Takeda-6d 是一种新型、有效的 DFG-out RAF/血管内皮生长因子受体 2 (VEGFR2) 抑制剂，IC50 分别为 7.0 nM 和 2.2 nM。
T36683	Vedaprofen Quadrisol,PM 150,维达洛芬,CERM 10202	COX; Antibacterial; Prostaglandin Receptor	GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience
	Vedaprofen (PM 150) 抑制 COX-1 并通过抗炎活性减少前列腺素 H2 的合成。 Vedaprofen 是一种大肠杆菌滑动钳抑制剂，IC50 为 222 μM，Ki 为 131 μM。
T24850	Takeda103A CMPD103A,Takeda-103A,Takeda-103-A,CMPD-103A,Takeda 103 A	GRK	GPCR/G Protein
	Takeda103A (CMPD103A) 是 GRK2抑制剂。G 蛋白偶联受体是许多生理过程的核心。Takeda103A 对研究心力衰竭具有潜在的研究价值。
T21023	Bedaquiline fumarate TMC 207,R403323,TMC-207,TMC207,R-403323,贝达喹啉富马酸盐,R 403323	Antibacterial; Antibiotic	Microbiology/Virology
	Bedaquiline fumarate (TMC207) 是二芳基喹啉抗生素，作用于 ATP 合成酶，常用于结核杆菌感染的研究。
TD0082	EDANS sodium EDANS sodium salt,EDANS sodium salt [5-((2-Aminoethyl)amino)naphthalene-1-sulfonic acid, sodium salt],5-(2-氨乙基氨)-1-萘磺酸钠盐,5-(2-Aminoethylamino)-1-naphthalenesulfonic acid sodium salt,N-(Aminoethyl)-5-naphthylamine-1-sulfonic Acid Sodium Salt	Others	Others
	EDANS sodium (5-(2-Aminoethylamino)-1-naphthalenesulfonic acid sodium salt) 是开发基于 FRET 的核酸探针的供体，该探针广泛用于实时 PCR 测定。
T23445	Anxiolytic/nonsedative agent-1 TCS 1205	GABA Receptor	Membrane transporter/Ion channel; Neuroscience
	Anxiolytic/nonsedative agent-1 (TCS 1205) 是一种有效的选择性 GABAA 激动剂。Anxiolytic/nonsedative agent-1 对牛脑膜中的 BzR 显示出明显的亲和力，对 α1β2γ2、α2β2γ2、α5β3γ2 的 Kis 分别为 14、121、239 nM。Anxiolytic/nonsedative agent-1 在体外表现出 α2 选择性功效，在体内表现出抗焦虑选择性作用。
T34795	Tedatioxetine Lu AA 24530,Lu AA-24530,Lu AA24530	Dopamine Receptor; Serotonin Transporter	GPCR/G Protein; Neuroscience
	Tedatioxetine (Lu AA24530) 是一种血清素-去甲肾上腺素-多巴胺再摄取抑制剂（SNDRI），具有抗抑郁作用。Tedatioxetine 可作为 CYP2D6 底物。
T1777	Nintedanib BIBF 1120,Intedanib,尼达尼布	VEGFR; FGFR; FLT; PDGFR; Src	Angiogenesis; Tyrosine Kinase/Adaptors
	Nintedanib (Intedanib) 是一种三重血管激酶抑制剂，抑制 VEGFR1、VEGFR2、VEGFR3 (IC50=34/13/13 nM)，FGFR1、FGFR2、FGFR3 (IC50=69/37/108 nM)，PDGFRα、PDGFRβ (IC50=59/65 nM)。Nintedanib 具有抗肿瘤活性，通过抑制血管生成来抑制肿瘤生长。
T38514	PMEDAP	Others; HIV Protease	Microbiology/Virology; Others; Proteases/Proteasome
	PMEDAP 是有效的人类免疫缺陷病毒 (HIV) 复制抑制剂。它具有抗小鼠巨细胞病毒活性。它有效抑制莫罗尼鼠肉瘤病毒诱导的肿瘤形成和相关死亡率。
T1970	Gedatolisib PF-05212384,PKI-587	PI3K; mTOR	PI3K/Akt/mTOR signaling
	Gedatolisib (PF-05212384) 是一种高效的双重 PI3Kα (IC50:0.4 nM)，PI3Kγ (IC50:5.4 nM) 和 mTOR (IC50:1.6 nM)抑制剂。它在 mTOR 复合物mTORC1和mTORC2中同样有效。
T1073	Dronedarone hydrochloride Dronedarone HCl,SR33589,决奈达隆盐酸盐,盐酸决奈达隆	Potassium Channel; Calcium Channel; Sodium Channel; Adrenergic Receptor; Autophagy	Autophagy; GPCR/G Protein; Membrane transporter/Ion channel; Metabolism; Neuroscience
	Dronedarone hydrochloride (SR33589) 是一种胺碘酮类似物，可抑制 Na+,K+andCa2+的电流，有可能治疗心房颤动。
T26972	Cedazuridine 西达尿苷,(4R)-2'-Deoxy-2',2'-difluoro-3,4,5,6-tetrahydrouridine	DNA Methyltransferase	Chromatin/Epigenetic
	Cedazuridine ((4R)-2'-Deoxy-2',2'-difluoro-3,4,5,6-tetrahydrouridine) 是一种口服的胞苷脱氨酶抑制剂，具有抗肿瘤特性。
T5001	Nintedanib esylate Intedanib,乙磺酸尼达尼布,BIBF 1120 (esylate),尼达尼布乙磺酸盐,Nintedanib Ethanesulfonate Salt,BIBF 1120	VEGFR; FGFR; PDGFR	Angiogenesis; Tyrosine Kinase/Adaptors
	Nintedanib esylate (BIBF 1120 esylate) 是一种有效的三重血管激酶抑制剂，能够抑制 VEGFR1 (IC50:34 nM)、VEGFR2 (IC50:13 nM)、VEGFR3 (IC50:13 nM)，FGFR1 (IC50:69 nM)、FGFR2 (IC50:37 nM)、FGFR3 (IC50:108 nM)，PDGFRα (IC50:59 nM)、PDGFRβ (IC50:65 nM)。
T2585	Bedaquiline R207910,TMC207,贝达喹啉	Antibacterial; Antibiotic	Microbiology/Virology
	Bedaquiline (R207910) 是一种二芳基喹啉药物，能同时靶向 c-亚基和 ε-亚基，抑制结核分枝杆菌 (Mtb) F1FO-ATP 合酶。它具有解偶联活性和有用于耐多药结核病的潜力。
TD0081	EDANS EDANS acid [5-((2-Aminoethyl)amino)naphthalene-1-sulfonic acid],EDANS酸,1,5-EDANS,EDANS acid [5-((2-Aminoethyl)amino)napht	Others	Others
	EDANS (EDANS acid [5-((2-Aminoethyl)amino)naphthalene-1-sulfonic acid]) 是新型的淬灭荧光底物 (fluorogenic substrate)，可利用共振能量转移，分析逆转录病毒蛋白酶。
T0407	Edaravone 依达拉奉右莰醇,依达拉奉,MCI-186	Apoptosis; MMP; Free radical scavengers	Apoptosis; oxidation-reduction; Proteases/Proteasome
	Edaravone (MCI-186) 是一种新型自由基清除剂，能够抑制大鼠与 MMP-9有关的脑出血。
T15198	Edasalonexent CAT-1004	NF-κB	NF-κB
	Edasalonexent (CAT-1004) 是一种可口服的 NF-κB 抑制剂，可用于改善杜氏肌营养不良症。
T76369	CEDAEVFKDSMVPGEK
	CEDAEVFKDSMVPGEK 为大鼠辣椒素受体亚型 1 (VR1) 的多肽序列片段，适用于探测 VR1 的存在、分布及分子形态。
T76067	Dabcyl-KTSAVLQSGFRKME-Edans TFA
	Dabcyl-KTSAVLQSGFRKME-Edans TFA 是一种用于测量蛋白酶酶促活性的荧光肽，具有研究2019-nCoV (COVID-19) 感染潜力的特性。该化合物作为底物，用于相关蛋白酶活性的测定。
T20673	Clofedanol NSC113595,NSC 113595,NSC-113595	Others	Others
	Clofedanol, also known as chlophedianol or antitussin, is used in the treatment of pediatric pertussis.
T39287	Ledaborbactam	Others	Others
	Iedaborbactam, as a beta-lactamase inhibitor (WO2015191907, Example 62), can be used for the research of bacterial infections.
T26818	Binedaline binodaline. Ixprim,SCHA 1059,SCHA1059,Sgd-Sch-1059,SCHA-1059	Others	Others
	Binedaline is a selective norepinephrine reuptake inhibitor with Ki value of 25 nM.
T131569	Allosedamine	Others	Others
	Allosedamine 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T131569。
T17027	Tedalinab GRC-10693	Cannabinoid Receptor	GPCR/G Protein
	Tedalinab is an effective and selective cannabinoid receptor 2 agonist. Tedalinab has the potential for neuropathic pain and osteoarthritis treatment. Tedalinab has >4700-fold functional selectivity for CB2 over CB1.
T77082	Melredableukin alfa
	Melredableukin alfa (RO-7049665)是一种由人IgG1-κ通过多肽连接子与人突变白细胞介素2(IL2 mutin)融合形成的融合蛋白。它适用于乙型肝炎和溃疡性结肠炎的研究。
T76239	Efrilacedase alfa
	Efrilacedase alfa 是一种活性化合物。Efrilacedase alfa 可用于各种生化研究。
T75369	DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS
	DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS 为一种用于人类疟原虫天冬氨酰蛋白酶的荧光底物，属于荧光染料类。储存条件：需避光。
T82619	Dabsyl-Leu-Gly-Gly-Gly-Ala-Edans
	Dabsyl-Leu-Gly-Gly-Gly-Ala-Edans为标记有Dabsyl荧光基团的肽类化合物。该化合物用于鉴定铜绿假单胞菌LasA蛋白酶的肽酶活性，并呈现酶特异性，适用于相关生物医学研究。
T31092	Credazine BRN 0880257,NIA 20439,SW-670,H-722,Kusakira	Others	Others
	Credazine is a bio-active chemical. Detailed information has not been published.
T60708	Cedazuridine hydrochloride	Others	Others
	Cedazuridine (E7727) (Compound 7a) hydrochloride 是一种可用于研究癌症的，口服有效的胞苷脱氨酶 (CDA) 抑制剂 (IC 50 = 0.4 μM)。
T26549	Acedapsone Atilon,BA 2650,Rodilon,Camilan,Acetamin	Others	Others
	Acedapsone has antimalarial and antimicrobial action, but is mainly used as a depot leprostatic agent.
T21388	Emedastine Difumarate Rapimine,DSSTox_CID_26911,AL-3432A,富马酸依美斯汀,KB-2413,Emedastine fumarate,KB 2413	Others	Others
	Emedastine Difumarate is a selective histamine H1 receptor antagonist with anti-allergic activity, prescribed for allergic conjunctivitis. Upon ocular administration, emedastine causes a dose-dependent inhibition of histamine-stimulated vascular permeabil
T27239	Edaglitazone Edaglitazone sodium,BM-13.1258,RO-2052349-602,依格列宗,R-483,RO-2052349-000	Others	Others
	Edaglitazone is a PPARγ agonist. Edarglitazone restores acute inflammatory responses to cerebral hypoxia-ischemia in the diabetic ob/ob mouse.
T68661	Edatrexate CGP 30694	Others	Others
	Edatrexate (CGP 30694)，即 10-乙基-10-去甲氨基蝶呤，是甲氨蝶呤Methotrexate 的类似物，对耐 MTX 肿瘤具有抗肿瘤活性。Edatrexate 是一种抗叶酸抗代谢物，可用于研究非小细胞肺癌，乳腺癌，非霍奇金淋巴瘤和头颈部癌症的研究。
T69788	Daledalin	Others	Others
	Daledalin is an antidepressant which was synthesized and trialed for depression in the early 1970s, but was never marketed. It is a selective norepinephrine reuptake inhibitor, with no significant effects on the reuptake of serotonin and dopamine, and no antihistamine or anticholinergic properties.
T68229	Nintedanib esylate hemihydrate	Others	Others
	Nintedanib esylate hemihydrate is a potent inhibitor of multiple receptor tyrosine kinases (RTKs) and non-receptor tyrosine kinases (nRTKs).
T39288	Ledaborbactam etzadroxil VNRX-7145	Others	Others
	Ledaborbactam etzadroxil (VNRX-7145) is an orally active inhibitor of Ambler class A, C, and D β-lactamase enzymes.
T35615	Dabcyl-YVADAPV-EDANS
	Dabcyl YVADAPV EDANS 是一种荧光 IL-1β 转化酶 (interleukin-1β converting enzyme, ICE) 底物，可用于检测 ICE 样蛋白酶活性。Dabcyl YVADAPV EDANS 检测荧光的 λex=360 nm，λem=480 nm。
T65192	Fmoc-Glu(Edans)-OH
	Fmoc-Glu(Edans)-OH 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T65192，CAS号为 193475-66-0。
T80587	Alunacedase alfa HrsACE2,GSK 2586881	SARS-CoV	Microbiology/Virology
	Alunacedase alfa (HrsACE2; GSK 2586881) 是一种人源重组的可溶性血管紧张素转化酶 2（hrsACE2）。作为转基因可溶性形态的 ACE2，Alunacedase alfa 能够减少 SARS-CoV-2 与细胞膜结合 ACE2 的竞争性进入，因此具有研究 SARS-CoV-2 的可能性。

化合物

Cat.No: T17549

Target: Others, PROTAC Linker

Cat.No: T39373

Synonym: PNU-EDA-Gly5

Target: Others, Drug-Linker Conjugates for ADC

Mal-C2-Gly3-EDA

Cat.No: T18247

Target: Others, ADC Linker

Mal-C2-Gly3-EDA-PNU-159682

Cat.No: T18246

Target: Others, Drug-Linker Conjugates for ADC

Cat.No: T75354

Target: Others

Cat.No: T74555

Target: Others

BODIPY FL EDA free base

Cat.No: T82842

Cat.No: T3979

Synonym: LY188695,依美斯汀,Emadine

Target: Histamine Receptor

Tedatioxetine hydrobromide

Cat.No: T13110

Synonym: Lu AA 24530 hydrobromide

Target: Dopamine Receptor, 5-HT Receptor, Norepinephrine

Cat.No: T2410

Synonym: 奈达铂,NSC 375101D

Target: DNA/RNA Synthesis

Cat.No: T22436

Target: VEGFR

Cat.No: T36683

Synonym: Quadrisol,PM 150,维达洛芬,CERM 10202

Target: COX, Antibacterial, Prostaglandin Receptor

Cat.No: T24850

Synonym: CMPD103A,Takeda-103A,Takeda-103-A,CMPD-103A,Takeda 103 A

Target: GRK

Bedaquiline fumarate

Cat.No: T21023

Synonym: TMC 207,R403323,TMC-207,TMC207,R-403323,贝达喹啉富马酸盐,R 403323

Target: Antibacterial, Antibiotic

Cat.No: TD0082

Synonym: EDANS sodium salt,EDANS sodium salt [5-((2-Aminoethyl)amino)naphthalene-1-sulfonic acid, sodium salt],5-(2-氨乙基氨)-1-萘磺酸钠盐,5-(2-Aminoethylamino)-1-naphthalenesulfonic acid sodium salt,N-(Aminoethyl)-5-naphthylamine-1-sulfonic Acid Sodium Salt

Target: Others

Anxiolytic/nonsedative agent-1

Cat.No: T23445

Synonym: TCS 1205

Target: GABA Receptor

Cat.No: T34795

Synonym: Lu AA 24530,Lu AA-24530,Lu AA24530

Target: Dopamine Receptor, Serotonin Transporter

Cat.No: T1777

Synonym: BIBF 1120,Intedanib,尼达尼布

Target: VEGFR, FGFR, FLT, PDGFR, Src

Cat.No: T38514

Target: Others, HIV Protease

Cat.No: T1970

Synonym: PF-05212384,PKI-587

Target: PI3K, mTOR

Dronedarone hydrochloride

Cat.No: T1073

Synonym: Dronedarone HCl,SR33589,决奈达隆盐酸盐,盐酸决奈达隆

Target: Potassium Channel, Calcium Channel, Sodium Channel, Adrenergic Receptor, Autophagy

Cat.No: T26972

Synonym: 西达尿苷,(4R)-2'-Deoxy-2',2'-difluoro-3,4,5,6-tetrahydrouridine

Target: DNA Methyltransferase

Nintedanib esylate

Cat.No: T5001

Synonym: Intedanib,乙磺酸尼达尼布,BIBF 1120 (esylate),尼达尼布乙磺酸盐,Nintedanib Ethanesulfonate Salt,BIBF 1120

Target: VEGFR, FGFR, PDGFR

Cat.No: T2585

Synonym: R207910,TMC207,贝达喹啉

Target: Antibacterial, Antibiotic

Cat.No: TD0081

Synonym: EDANS acid [5-((2-Aminoethyl)amino)naphthalene-1-sulfonic acid],EDANS酸,1,5-EDANS,EDANS acid [5-((2-Aminoethyl)amino)napht

Target: Others

Cat.No: T0407

Synonym: 依达拉奉右莰醇,依达拉奉,MCI-186

Target: Apoptosis, MMP, Free radical scavengers

Edasalonexent

Cat.No: T15198

Synonym: CAT-1004

Target: NF-κB

CEDAEVFKDSMVPGEK

Cat.No: T76369

Dabcyl-KTSAVLQSGFRKME-Edans TFA

Cat.No: T76067

Cat.No: T20673

Synonym: NSC113595,NSC 113595,NSC-113595

Target: Others

Cat.No: T39287

Target: Others

Cat.No: T26818

Synonym: binodaline. Ixprim,SCHA 1059,SCHA1059,Sgd-Sch-1059,SCHA-1059

Target: Others

Cat.No: T131569

Target: Others

Cat.No: T17027

Synonym: GRC-10693

Target: Cannabinoid Receptor

Melredableukin alfa

Cat.No: T77082

Efrilacedase alfa

Cat.No: T76239

DABCYL-Glu-Arg-Nle-Phe-Leu-Ser-Phe-Pro-EDANS

Cat.No: T75369

Dabsyl-Leu-Gly-Gly-Gly-Ala-Edans

Cat.No: T82619

Cat.No: T31092

Synonym: BRN 0880257,NIA 20439,SW-670,H-722,Kusakira

Target: Others

Cedazuridine hydrochloride

Cat.No: T60708

Target: Others

Cat.No: T26549

Synonym: Atilon,BA 2650,Rodilon,Camilan,Acetamin

Target: Others

Emedastine Difumarate

Cat.No: T21388

Synonym: Rapimine,DSSTox_CID_26911,AL-3432A,富马酸依美斯汀,KB-2413,Emedastine fumarate,KB 2413

Target: Others

Cat.No: T27239

Synonym: Edaglitazone sodium,BM-13.1258,RO-2052349-602,依格列宗,R-483,RO-2052349-000

Target: Others

Cat.No: T68661

Synonym: CGP 30694

Target: Others

Cat.No: T69788

Target: Others

Nintedanib esylate hemihydrate

Cat.No: T68229

Target: Others

Ledaborbactam etzadroxil

Cat.No: T39288

Synonym: VNRX-7145

Target: Others

Dabcyl-YVADAPV-EDANS

Cat.No: T35615

Fmoc-Glu(Edans)-OH

Cat.No: T65192

Alunacedase alfa

Cat.No: T80587

Synonym: HrsACE2,GSK 2586881

Target: SARS-CoV

Cat. No.	Product Name	Target	Signaling Pathways
T3862	Irigenin	NF-κB; Integrin	Cytoskeletal Signaling; NF-κB
	Irigenin 可通过特异性和选择性地阻断 Extra Domain A 域的 C-C 环上α9β1和α4β1整合素结合位点，介导其抗转移作用。可通过增强胃癌细胞中促凋亡分子的表达来敏化 TRAIL 诱导的凋亡，具有抗癌作用。
T3S0081	Oxypeucedanin (+-)-Oxypeucedanin,氧化前胡素,Oxypeucadanin	Potassium Channel	Membrane transporter/Ion channel
	Oxypeucedanin ((+-)-Oxypeucedanin) 是呋喃香豆素衍生物，分离自Angelica dahurica。它是选择性开放通道阻滞剂，可抑制hKv1.5通道电流，IC50值为 76 nM。它延长心脏动作电位持续时间，是潜在的抗心律失常试剂。它通过抑制癌细胞迁移来诱导细胞凋亡。
T7056	Dronedarone 决奈达隆,SR 33589	P450; Potassium Channel; Calcium Channel; Sodium Channel; Adrenergic Receptor; AChR; Autophagy	Autophagy; GPCR/G Protein; Membrane transporter/Ion channel; Metabolism; Neuroscience
	Dronedarone (SR 33589) 是一种胺碘酮类似物，对治疗心房颤动可能有效。它是CYP3A4的底物和中度抑制剂。它是多种离子电流的有效阻滞剂，通过非竞争性结合到肾上腺素能受体显示出抗肾上腺素能的效果。
T5763	Sedanolide	Others; Autophagy	Autophagy; Others
	Sedanolide 是从伞形科的种子油中分离出的一种天然苯酞，具有抗炎和抗氧化活性。
T6S0078	Oxypeucedanin hydrate Prangolarin Hydrate,水合氧化前胡素	Antioxidant	oxidation-reduction
	Oxypeucedanin hydrate (Prangolarin Hydrate) 是一种分离自D. anethifolia 中的天然香豆素化合物，存在于几种植物中，具有抗感染和抗真菌活性。
T5808	(-)-Oxypeucedanin hydrate 水合氧化前胡素,OXYPEUCEDANIN HYDRATE	Others	Others
	(-)-Oxypeucedanin hydrate 是一种呋喃香豆素衍生物，分离自Ducrosia anethifolia 中。
T13816	(+)-Peusedanol (+)-白花前胡醇,白花前胡醇	Others	Others
	(+)-Peusedanol 是一种香豆素，从滨海前胡中分离出来。
TN5212	Uvedalin	Others	Others
	Uvedalin shows cytotoxicity against HeLa, HL-60, and Murine B16-F10 melanoma cell lines.
TN4758	Peucedanol 3'-O-glucoside	Others	Others
	Peucedanol 3'-O-glucoside 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN4758，CAS号为 65891-61-4。
T75620	(+)-Oxypeucedanin methanolate	Others	Others
	(+)-Oxypeucedanin methanolate (compound 9) 是一种天然产物，可抑制前列腺素 E2 的产生。
TN4755	Peucedanocoumarin I	Others	Others
	Peucedanocoumarin I是一种天然产物，属于伞形科前胡属，其产品编号为 TN4755，CAS号为 130464-55-0。Peucedanocoumarin I可用作对照参考。
TN3645	Chlorouvedalin	Others	Others
	Chlorouvedalin 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN3645，CAS号为 24694-80-2。
TC0029	Peucedanin	Others	Others
	Peucedanin 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TC0029，CAS号为 133-26-6。
TMA2563	Pedalitin	Tyrosinase	Proteases/Proteasome
	Pedalitin is a mixed-type inhibitor of tyrosinase. In the assay of α-glucosidase inhibition, rosmarinic acid is a competitive inhibitor, whereas both methyl rosmarinate and Pedalitin are mixed-type inhibitors.
TN4757	Peucedanocoumarin III	Others	Others
	Peucedanocoumarin Ⅲ can induce rice resistance to blast disease.
TN4756	Peucedanocoumarin II	Others	Others
	Peucedanocoumarin II shows only partial relaxation.
TN6851	Iso-oxypeucedanin
	Iso-oxypeucedanin is a natural product.
T81532	Pedaliin 6''-acetate
	Pedaliin 6''-acetate (compound 10) 为甘青青兰中分离得到的天然产物，具有抗氧化活性，并能对抗DOX诱导的H9c2心肌细胞毒性，表现出细胞保护效应，其EC50为19.1 μM。
TN4759	Peucedanol 7-O-glucoside	Others	Others
	Peucedanol 7-O-glucoside 是一种天然产物，可用于生命科学领域的相关研究。其产品编号为 TN4759，CAS号为 65853-04-5。
T41136	Azedarachol	Others	Others
	Azedarachol possesses antifeedant activity.
TN5546	Pedaliin Pedalin,Pedalitin 6-O-glucoside,Glucosyl-6-pedalitin	Antioxidant	oxidation-reduction
	Pedaliin 是从芝麻 (Sesamum indicum L)和藏药Dracocephalum tanguticum Maxim 地上部分提取的一种黄酮类化合物。Pedaliin 在体外显示出抗氧化和抗结肠癌作用，可用于研究心脑血管疾病。
T83521	(S)-7-O-Methylpeucedanol 3′-O-β-D-glucopyranoside
	(S)-7-O-Methylpeucedanol 3'-O-β-D-glucopyranoside 为一种香豆素糖苷[sup][1]。
TN6027	Pedatisectine F 2-Methyl-6-(1,2,3,4-tetrahydroxybutyl)pyrazine
	Pedatisectine F是一种天然产物，属于天南星科半夏属，其产品编号为 TN6027，CAS号为 206757-32-6。Pedatisectine F可用作对照参考。
T81505	Peucedanoside A
	Peucedanoside A，一种从Peucedanum praeretorum Dunn根部分离得到的苷类化合物。
TN7289	Cedarwood terpenes	Others	Others
	Cedarwood terpenes是源自雪松木的天然萜烯混合物。

天然产物

Cat.No: T3862

Target: NF-κB, Integrin

Cat.No: T3S0081

Synonym: (+-)-Oxypeucedanin,氧化前胡素,Oxypeucadanin

Target: Potassium Channel

Cat.No: T7056

Synonym: 决奈达隆,SR 33589

Target: P450, Potassium Channel, Calcium Channel, Sodium Channel, Adrenergic Receptor, AChR, Autophagy

Cat.No: T5763

Target: Others, Autophagy

Oxypeucedanin hydrate

Cat.No: T6S0078

Synonym: Prangolarin Hydrate,水合氧化前胡素

Target: Antioxidant

(-)-Oxypeucedanin hydrate

Cat.No: T5808

Synonym: 水合氧化前胡素,OXYPEUCEDANIN HYDRATE

Target: Others

Cat.No: T13816

Synonym: (+)-白花前胡醇,白花前胡醇

Target: Others

Cat.No: TN5212

Target: Others

Peucedanol 3'-O-glucoside

Cat.No: TN4758

Target: Others

(+)-Oxypeucedanin methanolate

Cat.No: T75620

Target: Others

Peucedanocoumarin I

Cat.No: TN4755

Target: Others

Cat.No: TN3645

Target: Others

Cat.No: TC0029

Target: Others

Cat.No: TMA2563

Target: Tyrosinase

Peucedanocoumarin III

Cat.No: TN4757

Target: Others

Peucedanocoumarin II

Cat.No: TN4756

Target: Others

Iso-oxypeucedanin

Cat.No: TN6851

Pedaliin 6''-acetate

Cat.No: T81532

Peucedanol 7-O-glucoside

Cat.No: TN4759

Target: Others

Cat.No: T41136

Target: Others

Cat.No: TN5546

Synonym: Pedalin,Pedalitin 6-O-glucoside,Glucosyl-6-pedalitin

Target: Antioxidant

(S)-7-O-Methylpeucedanol 3′-O-β-D-glucopyranoside

Cat.No: T83521

Pedatisectine F

Cat.No: TN6027

Synonym: 2-Methyl-6-(1,2,3,4-tetrahydroxybutyl)pyrazine

Peucedanoside A

Cat.No: T81505

Cedarwood terpenes

Cat.No: TN7289

Target: Others

Species：

Expression System：

Tag：

Cat. No.	Product Name	Species	Expression System
TMPY-01932	EDA2R Protein, Human, Recombinant (His) EDAA2R,ectodysplasin A2 receptor,EDA-A2R,T...	Human	HEK293 Cells
	EDA2R Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 16.7 kDa and the accession number is Q9HAV5-1.
TMPJ-01211	EDA2R Protein, Mouse, Recombinant (His) EDA-A2R,Tumor necrosis factor receptor superfamily ...	Mouse	HEK293 Cells
	Tumor necrosis factor receptor superfamily member 27, also known as XEDAR and EDA2R, is a type III transmembrane protein of the TNFR superfamily. EDA2R consists of extracellular domain (ECD) with 3 cysteine-rich repeats and a single transmembrane domain but lacks an N-terminal signal peptide. EDA2R is widely expressed, notably in embryonic basal epidermal cells and maturing hair follicles. Even though it does not contain a cytoplasmic death domain, EDA2R can associate with Fas and induce EDA‑A2 ...
TMPY-00294	EDA2R Protein, Human, Recombinant (hFc) EDA-A2R,EDAA2R,ectodysplasin A2 receptor,X...	Human	HEK293 Cells
	EDA2R Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 41.3 kDa and the accession number is Q9HAV5-1.
TMPY-01636	EDAR Protein, Human, Recombinant (hFc) DL,EDA1R,ED5,EDA3,ED3,HRM1,ectodysplasin A...	Human	HEK293 Cells
	EDAR Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 44.6 kDa and the accession number is Q9UNE0-1.
TMPY-01637	EDAR Protein, Human, Recombinant (His) ED3,DL,ectodysplasin A receptor,ED1R,EDA1R,HRM1,	Human	HEK293 Cells
	EDAR Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 19 kDa and the accession number is Q9UNE0-1.
TMPY-03029	EDA2R Protein, Rat, Recombinant (His) ectodysplasin A2 receptor	Rat	HEK293 Cells
	EDA2R Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 16.7 kDa and the accession number is D3ZAX4.
TMPY-00301	EDA2R Protein, Cynomolgus, Recombinant (His) ectodysplasin A2 receptor	Cynomolgus	HEK293 Cells
	EDA2R Protein, Cynomolgus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 16.6 kDa and the accession number is A0A2K5TKN6.
TMPY-03682	EDA2R Protein, Cynomolgus, Recombinant (hFc) ectodysplasin A2 receptor	Cynomolgus	HEK293 Cells
	EDA2R Protein, Cynomolgus, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 38.4 kDa and the accession number is A0A5F8A4K0.
TMPY-02935	EDA2R Protein, Rat, Recombinant (hFc) ectodysplasin A2 receptor	Rat	HEK293 Cells
	EDA2R Protein, Rat, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 42.3 kDa and the accession number is D3ZAX4.
TMPY-03124	EDA2R Protein, Mouse, Recombinant (hFc) Xedar,TNFRSF27,9430060M22Rik,ectodysplasin A2 recep...	Mouse	HEK293 Cells
	EDA2R Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 42.4 kDa and the accession number is Q8BX35.
TMPJ-01370	EDAR Protein, Mouse, Recombinant (hFc) Ectodysplasin-A receptor,Anhidrotic ectodysplasin receptor 1...	Mouse	HEK293 Cells
	Ectodysplasin A receptor (EDAR) is a type I transmembrane protein of the TNF-α receptor superfamily which plays a key role in ectodermal differentiation. EDAR was encoded by the mouse downless gene and defective in human dominant and recessive forms of autosomal hypohidrotic ectodermal dysplasia (EDA) syndrome. The extracellular domain of EDAR contains 14 cysteine residues, six of which approximate the TNFRSF cysteine-rich region, the cytoplasmic domain contains a region with homology to the dea...
TMPY-03638	EDAR Protein, Cynomolgus, Recombinant (His) ectodysplasin A receptor	Cynomolgus	HEK293 Cells
	EDAR Protein, Cynomolgus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 21.4 kDa and the accession number is F7GZI3.
TMPY-03253	EDAR Protein, Cynomolgus, Recombinant (hFc) ectodysplasin A receptor	Cynomolgus	HEK293 Cells
	EDAR Protein, Cynomolgus, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 44.6 kDa.
TMPY-02826	EDAR Protein, Rat, Recombinant (hFc) ectodysplasin A receptor	Rat	HEK293 Cells
	EDAR Protein, Rat, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 44.4 kDa and the accession number is NP_001178828.1.
TMPY-00069	Dromedary camel coronavirus (DcCoV)(strain HKU23-368F) Nucleoprotein/DcCoV-NP Protein (His) DcCoV-NP	DcCoV	Baculovirus Insect Cells
	Dromedary camel coronavirus (DcCoV)(strain HKU23-368F) Nucleoprotein/DcCoV-NP Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 50.8 kDa and the accession number is X2JHN2.

重组蛋白

EDA2R Protein, Human, Recombinant (His)

Cat.No: TMPY-01932

Species: Human

Expression System: HEK293 Cells

EDA2R Protein, Mouse, Recombinant (His)

Cat.No: TMPJ-01211

Species: Mouse

Expression System: HEK293 Cells

EDA2R Protein, Human, Recombinant (hFc)

Cat.No: TMPY-00294

Species: Human

Expression System: HEK293 Cells

EDAR Protein, Human, Recombinant (hFc)

Cat.No: TMPY-01636

Species: Human

Expression System: HEK293 Cells

EDAR Protein, Human, Recombinant (His)

Cat.No: TMPY-01637

Species: Human

Expression System: HEK293 Cells

EDA2R Protein, Rat, Recombinant (His)

Cat.No: TMPY-03029

Species: Rat

Expression System: HEK293 Cells

EDA2R Protein, Cynomolgus, Recombinant (His)

Cat.No: TMPY-00301

Species: Cynomolgus

Expression System: HEK293 Cells

EDA2R Protein, Cynomolgus, Recombinant (hFc)

Cat.No: TMPY-03682

Species: Cynomolgus

Expression System: HEK293 Cells

EDA2R Protein, Rat, Recombinant (hFc)

Cat.No: TMPY-02935

Species: Rat

Expression System: HEK293 Cells

EDA2R Protein, Mouse, Recombinant (hFc)

Cat.No: TMPY-03124

Species: Mouse

Expression System: HEK293 Cells

EDAR Protein, Mouse, Recombinant (hFc)

Cat.No: TMPJ-01370

Species: Mouse

Expression System: HEK293 Cells

EDAR Protein, Cynomolgus, Recombinant (His)

Cat.No: TMPY-03638

Species: Cynomolgus

Expression System: HEK293 Cells

EDAR Protein, Cynomolgus, Recombinant (hFc)

Cat.No: TMPY-03253

Species: Cynomolgus

Expression System: HEK293 Cells

EDAR Protein, Rat, Recombinant (hFc)

Cat.No: TMPY-02826

Species: Rat

Expression System: HEK293 Cells

Dromedary camel coronavirus (DcCoV)(strain HKU23-368F) Nucleoprotein/DcCoV-NP Protein (His)

Cat.No: TMPY-00069

Species: DcCoV

Expression System: Baculovirus Insect Cells

Cat. No.	Product Name	Target	Signaling Pathways
TMIH-0370	N-Desbutyl Dronedarone-d7 HCl
	N-Desbutyl Dronedarone-d7 HCl 是 N-Desbutyl Dronedarone HCl 的氘代化合物。N-Desbutyl Dronedarone HCl 的 CAS 号为 197431-02-0。
T19273	Debutyldronedarone D7 SR-35021 D7	Others	Others
	Debutyldronedarone D7 is deuterium-labeled Debutyldronedarone, which is the main circulating active metabolite of dronedarone in the body.
TMIJ-0138	Dronedarone-d6 HCl
	Dronedarone-d6 HCl 是 Dronedarone HCl 的氘代化合物。Dronedarone HCl 的 CAS 号为 141625-93-6。Dronedarone Hydrochloride 是一种胺碘酮类似物，可抑制Na+,K+andCa2+的电流，有可能治疗心房颤动。
TMIJ-0333	Nintedanib-d8
	Nintedanib-d8 是 Nintedanib 的氘代化合物。Nintedanib 的 CAS 号为 656247-17-5。Nintedanib 是一种有效的三重血管激酶抑制剂，能够抑制VEGFR1 (IC50:34 nM)、VEGFR2 (IC50:13 nM)、VEGFR3 (IC50:13 nM)，FGFR1 (IC50:69 nM)、FGFR2 (IC50:37 nM)、FGFR3 (IC50:108 nM)，PDGFRα (IC50:59 nM)、PDGFRβ (IC50:65 nM)。
TMIH-0393	Nintedanib-13C-d3
	Nintedanib-13C-d3 是 Nintedanib 的 13C 和氘代化合物。Nintedanib 的 CAS 号为 656247-17-5。Nintedanib 是一种有效的三重血管激酶抑制剂，能够抑制VEGFR1 (IC50:34 nM)、VEGFR2 (IC50:13 nM)、VEGFR3 (IC50:13 nM)，FGFR1 (IC50:69 nM)、FGFR2 (IC50:37 nM)、FGFR3 (IC50:108 nM)，PDGFRα (IC50:59 nM)、PDGFRβ (IC50:65 nM)。
T11152	Edaravone-d5 MCI-186 D5	Others	Others
	Edaravone, a novel and potent free radical scavenger, effectively prevents MMP-9-related brain hemorrhage in rats treated with tissue plasminogen activator. Its deuterium-labeled variant, Edaravone D5, retains the original compound's attributes while offering isotopic labeling benefits.

同位素标记化合物

N-Desbutyl Dronedarone-d7 HCl

Cat.No: TMIH-0370

Debutyldronedarone D7

Cat.No: T19273

Synonym: SR-35021 D7

Target: Others

Dronedarone-d6 HCl

Cat.No: TMIJ-0138

Cat.No: TMIJ-0333

Nintedanib-13C-d3

Cat.No: TMIH-0393

Cat.No: T11152

Synonym: MCI-186 D5

Target: Others

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