Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T10758L |
Centanafadine hydrochloride
EB-1020 hydrochloride |
Dopamine Receptor; Serotonin Transporter; Adrenergic Receptor; Norepinephrine | GPCR/G Protein; Neuroscience |
Centanafadine hydrochloride (EB-1020 hydrochloride) 是一种去甲肾上腺素(NE)/多巴胺(DA)转运的双抑制剂,还能抑制5-羟色胺(serotonin)转运体。它对人 NE,DA 和5-羟色胺转运体的 IC50值分别为6 nM,38 nM 和 83 nM。 | |||
T10758 |
Centanafadine
EB-1020 |
Others | Others |
Centanafadine is a dual inhibitor of norepinephrine (NE)/dopamine (DA) transporter, also inhibits serotonin transporter (IC50s: 6 nM, 38 nM, and 83 nM for human NE, DA, and serotonin transporter). |