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Targets Recommended: Others

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Cat. No. Product Name Target Signaling Pathways
T37483 Difelikefalin (trifluoroacetate salt)

Others Others
Difelikefalin is a κ-opioid receptor (KOR) agonist.1It activates KOR in HEK293 cells expressing the human receptor (EC50= 0.16 nM in a transactivation assay) and inhibits forskolin-induced cAMP production in R1.G1 mouse thyoma cells (EC50= 0.048 nM). Difelikefalin is selective for KOR over the μ-opioid receptor (MOR; EC50= >1 μM in a transactivation assay). It reduces acetic acid-induced writhing, as well as scratching behavior induced by the KOR antagonist GNTI, in mice (ED50s = 0.07 and 0.05 m...
T69537 Difelikefalin HCl

Others Others
Difelikefalin HCl is a κ-opioid receptor (KOR) agonist. It activates KOR in HEK293 cells expressing the human receptor (EC50 = 0.16 nM in a transactivation assay) and inhibits forskolin-induced cAMP production in R1.G1 mouse thyoma cells (EC50 = 0.048 nM). Difelikefalin HCl is selective for KOR over the μ-opioid receptor (MOR; EC50 = >1 µM in a transactivation assay). It reduces acetic acid-induced writhing, as well as scratching behavior induced by the KOR antagonist GNTI, in mice (ED50s = 0.07...
TP2501 Difelikefalin acetate

Difelikefalin acetate(1024828-77-0 free base),CR 845 acetate,Difelikefalin醋酸盐,FE 202845 acetate

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
Difelikefalin acetate (CR 845 acetate) 是一种外周受限的 kappa 阿片受体激动剂。CR845 表现出低 P450 CYP 抑制和对大脑的低渗透性。
TP2485 difelikefalin acetate(1024828-77-0 Free base)

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
difelikefalin acetate 是酮体和砌块。

化合物

Difelikefalin (trifluoroacetate salt)
Cat.No: T37483
Synonym:
Target: Others
Difelikefalin HCl
Cat.No: T69537
Synonym:
Target: Others
Difelikefalin acetate
Cat.No: TP2501
Synonym: Difelikefalin acetate(1024828-77-0 free base),CR 845 acetate,Difelikefalin醋酸盐,FE 202845 acetate
Target: Opioid Receptor
difelikefalin acetate(1024828-77-0 Free base)
Cat.No: TP2485
Synonym:
Target: Opioid Receptor
TargetMol Loading
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