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Search Results for " ctx "

Targets Recommended: Others

25

抑制剂 & 化合物

1

天然产物

5

重组蛋白

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Cat. No.	Product Name	Target	Signaling Pathways
T2042	CTX-0294885	Others	Others
	CTx0294885 是新型的二苯胺嘧啶化合物，在体外对广泛激酶有抑制作用，可用作琼脂糖凝胶激酶检测试剂。
T71832	CTX-0124143	Histone Acetyltransferase	Chromatin/Epigenetic
	CTX-0124143 是一种组蛋白乙酰转移酶抑制剂，对 KAT6A 的 IC50 值为 1.0μM。CTX-0124143 可用于研究细胞衰老。
TP1289	Cardiotoxin Analog (CTX) IV (6-12) TFA Cardiotoxin Analog (CTX) IV (6-12) (TFA)(115722-23-1,FREE)	Others	Others
	Cardiotoxin Analog (CTX) IV (6-12) TFA(115722-23-1 free base) 是 Cardiotoxin Analog (CTX) IV 的部分肽。从台湾眼镜蛇毒液中分离出的心脏毒素类似物 IV。 CTX IV 是一种独特的蛇毒心脏毒素。
T3715	Acebilustat 阿西鲁司特,CTX-4430	Aminopeptidase; LTR	Immunology/Inflammation; Metabolism
	Acebilustat (CTX-4430) 是一种具有口服活性的白三烯 A4 水解酶抑制剂，可用于炎症研究。
T9167	PF-9363 CTX-3648	Histone Acetyltransferase	Chromatin/Epigenetic
	PF-9363 (CTX-3648) 是一种有效且高选择性的 KAT6A/KAT6B 抑制剂，可用于癌症研究。
TP1455	Cardiotoxin Analog (CTX) IV (6-12) Cardiotoxin Analog (CTX) IV 6-12
	Cardiotoxin Analog (CTX) IV (6-12) is a part peptide of Cardiotoxin Analog (CTX) IV. Cardiotoxin analogues IV isolated from the venom of Taiwan Cobra.
T19251	CTX-0294885 hydrochloride (1439934-41-4 free base) CTX-0294885 hydrochloride	Others	Others
	CTX-0294885 hydrochloride is an agarose-supported kinase capture reagent.
T62049	CTX-712	Others	Others
	CTX-712 是有效的cdc2 样激酶 (CLK) 抑制剂。CTX-712 可以抑制癌症存活和癌细胞生长。
T76734	CTX-471
	CTX-471 是 CD137 的全人源单克隆抗体。CTX-471 对重组人、食蟹猴 CD137 和小鼠 CD137 具有结合亲和力，Kd 值分别为 50 nM、61 nM 和 748 nM。CTX-471 可用于免疫调节和癌症的研究。
T82664	CTX-2026
	CTX-2026是一种与CD277结合的纯人源抗体，在卵巢肿瘤模型中表现出抗肿瘤活性，适用于癌症研究。
T23707	alpha-Conotoxin imi alpha-Ctx-imi
	alpha-Conotoxin imi is a nicotinic acetylcholine receptor ligand.
T72214	CTX-0294885 hydrochloride	Others	Others
	CTX-0294885 hydrochloride 是一种广谱激酶抑制剂，可以从 MDA-MB-231 细胞中捕获 235 种激酶，且可捕获AKT 家族中的所有成员。CTX-0294885 hydrochloride 是一种强大的激酶组信号网络分析试剂，可用于炎症、糖尿病和癌症等疾病的研究。
T15016	CTX1	p53	Apoptosis
	CTX1 is a small molecule activator of p53.
T4584	BMS-813160 BMS 813160	CCR	Immunology/Inflammation; Microbiology/Virology
	BMS-813160 是CCR2/CCR5双重拮抗剂。有用于心血管的研究潜力。
T60050	ANT3310	Antibacterial	Microbiology/Virology
	ANT3310 是一种广谱共价丝氨酸 β-内酰胺酶抑制剂，对 AmpC、CTX-M-15、TEM-1、OXA-48、OXA-23 和 KPC-2 的 IC50 范围为 1 nM 至 175 nM。 ANT3310 可用于细菌感染研究。
T38941	FPI-1523 sodium	Endogenous Metabolite; Antibacterial	Metabolism; Microbiology/Virology
	FPI-1523 sodium 是阿维巴坦的衍生物，是一种强效的 β-内酰胺酶抑制剂，对 CTX-M-15 和 OXA-48 的 K d s 分别为 4 nM 和 34 nM。FPI-1523 sodium 对 PBP2 有抑制作用，其 IC 50 为 3.2 μM。FPI-1523 sodium具有相当高的抗菌活性。
T10422	Avibactam free acid NXL-104 free acid	Antibacterial	Microbiology/Virology
	Avibactam (NXL-104) free acid is a covalent and reversible inhibitor of non-β-lactam β-lactamase (IC50s: 8 nM and 5 nM for β-lactamase TEM-1 and CTX-M-15).
T10713	CCR4 antagonist 2	Calcium Channel	Membrane transporter/Ion channel; Metabolism
	CCR4 antagonist 2 (Compound 31) is a novel potent, orally bioavailable small molecule antagonists of CC chemokine receptor 4 (CCR4) that inhibits Treg trafficking into the Tumor Microenvironment without suppressing the number of Treg in healthy tissues. CCR4 antagonist 2 (Compound 31) exhibits IC50 values of Ca2+flux and (chemotaxis) CTX are 40 nM and 70 nM, respectively.
T60874	Avibactam sodium dihydrate	Others	Others
	Avibactam sodium (NXL-104) dihydrate 抑制 CTX-M-15和 β-内酰胺酶 TEM-1，IC50值分别为 5 nM 和 8 nM。Avibactam sodium (NXL-104) dihydrate 是非 β-内酰胺 β-内酰胺酶的可逆共价抑制剂。
T39661	CCR4 antagonist 3 CCR4 antagonist 3	Others	Others
	CCR4 antagonist 3 is an orally active, potent and selective CCR4 antagonist. CCR4 antagonist 3, featuring a novel piperidinyl-azetidine motif, has IC 50 s of 22 nM and 50 nM in the calcium flux and CTX assay. CCR4 antagonist 3 has antitumor activity.
T39662	CCR4 antagonist 3 hydrochloride	Others	Others
	CCR4 antagonist 3 hydrochloride is an orally active, potent and selective CCR4 antagonist. CCR4 antagonist 3, featuring a novel piperidinyl-azetidine motif, has IC 50 s of 22 nM and 50 nM in the calcium flux and CTX assay. CCR4 antagonist 3 has antitumor activity.
T38940	FPI-1523	Others	Others
	FPI-1523, a derivative of Avibactam, is a potent inhibitor of β-lactamase enzymes. It has Kd values of 4 nM and 34 nM for CTX-M-15 and OXA-48, respectively. Additionally, FPI-1523 inhibits PBP2 with an IC50 of 3.2 μM and demonstrates significant antimicrobial activity.
T60711	Avibactam sodium hydrate	Others	Others
	Avibactam sodium hydrate (NXL-104 hydrate) 是 β-内酰胺酶的共价可逆抑制剂，不含β-内酰胺核心。Avibactam sodium hydrate 抑制 β-内酰胺酶CTX-M-15和TEM-1，IC50分别为5 nM 和 8 nM。
T73902	Desacetylcefotaxime	Others	Others
	Desacetylcefotaxime, Cefotaxime的一种体内代谢物，具有类似其母体化合物对多种需氧和厌氧细菌的体外抗菌活性。
T61204	FPI-1465	Others	Others
	FPI-1465 是丝氨酸-β-内酰胺酶和青霉素结合蛋白 (PBP) 的双重抑制剂。FPI-1465 抑制PBP2，IC50为 1.0 μg/mL。FPI-1465 作用于 β-内酰胺酶 CTX-M-15 和 OXA-48，Kd 分别为 0.011 和 5.3 μM。

化合物

Cat.No: T2042

Target: Others

Cat.No: T71832

Target: Histone Acetyltransferase

Cardiotoxin Analog (CTX) IV (6-12) TFA

Cat.No: TP1289

Synonym: Cardiotoxin Analog (CTX) IV (6-12) (TFA)(115722-23-1,FREE)

Target: Others

Cat.No: T3715

Synonym: 阿西鲁司特,CTX-4430

Target: Aminopeptidase, LTR

Cat.No: T9167

Synonym: CTX-3648

Target: Histone Acetyltransferase

Cardiotoxin Analog (CTX) IV (6-12)

Cat.No: TP1455

Synonym: Cardiotoxin Analog (CTX) IV 6-12

CTX-0294885 hydrochloride (1439934-41-4 free base)

Cat.No: T19251

Synonym: CTX-0294885 hydrochloride

Target: Others

Cat.No: T62049

Target: Others

Cat.No: T76734

Cat.No: T82664

alpha-Conotoxin imi

Cat.No: T23707

Synonym: alpha-Ctx-imi

CTX-0294885 hydrochloride

Cat.No: T72214

Target: Others

Cat.No: T15016

Target: p53

Cat.No: T4584

Synonym: BMS 813160

Target: CCR

Cat.No: T60050

Target: Antibacterial

FPI-1523 sodium

Cat.No: T38941

Target: Endogenous Metabolite, Antibacterial

Avibactam free acid

Cat.No: T10422

Synonym: NXL-104 free acid

Target: Antibacterial

CCR4 antagonist 2

Cat.No: T10713

Target: Calcium Channel

Avibactam sodium dihydrate

Cat.No: T60874

Target: Others

CCR4 antagonist 3

Cat.No: T39661

Synonym: CCR4 antagonist 3

Target: Others

CCR4 antagonist 3 hydrochloride

Cat.No: T39662

Target: Others

Cat.No: T38940

Target: Others

Avibactam sodium hydrate

Cat.No: T60711

Target: Others

Desacetylcefotaxime

Cat.No: T73902

Target: Others

Cat.No: T61204

Target: Others

Cat. No.	Product Name	Target	Signaling Pathways
T37177	Norcholic Acid	Others	Others
	Norcholic acid is a bile acid and 23-carbon derivative of cholic acid .1Levels of norcholic acid are increased in the urine of patients with liver cirrhosis or cerebrotendinous xanthomatosis (CTX), an inborn error of metabolism characterized by a deficiency in the mitochondrial enzyme sterol 27-hydrolylase (CYP27A1) that leads to progressive neurological symptoms.2,3,4

天然产物

Cat.No: T37177

Target: Others

Species：

Expression System：

Tag：

Cat. No.	Product Name	Species	Expression System
TMPH-03474	Beta-lactamase CTX-M-2 Protein, Salmonella typhimurium, Recombinant bla,Beta-lactamase CTX-M-2,Cefotaximase 2	Salmonella typhimurium	E. coli
	Has cefotaxime-hydrolyzing activity. Beta-lactamase CTX-M-2 Protein, Salmonella typhimurium, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 28.4 kDa and the accession number is P74841.
TMPH-00584	Beta-lactamase CTX-M-1 Protein, E. coli, Recombinant (His) men1,Beta-lactamase MEN-1,Cefotaximase 1,Beta-lactamase ...	E. coli	E. coli
	Broad spectrum beta-lactamase which confers resistance to penicillins, as well as first, second and third-generation cephalosporins.
TMPH-00585	Beta-lactamase CTX-M-1 Protein, E. coli, Recombinant (Yeast, His) Beta-lactamase MEN-1,Cefotaximase 1,bla,men1,Beta-lactamase ...	E. coli	P. pastoris (Yeast)
	Broad spectrum beta-lactamase which confers resistance to penicillins, as well as first, second and third-generation cephalosporins.
TMPH-03036	Cytotoxin 2 Protein, Naja atra, Recombinant (His & Myc) Cardiotoxin 2,CTX A2,Cardiotoxin 1A,Cardiotoxin A2,...	Naja atra	E. coli
	Basic protein that binds to cell membrane and depolarizes cardiomyocytes. It also shows lytic activities, but 2-fold less important than that of CTX-A4. It binds to the integrin alpha-V/beta-3 (ITGAV/ITGB3) with a moderate affinity. It may interact with sulfatides in the cell membrane which induces pore formation and cell internalization and is responsible for cytotoxicity in cardiomyocytes. It also may target the mitochondrial membrane and induce mitochondrial swelling and fragmentation.
TMPH-03037	Alpha-cobratoxin Protein, Naja kaouthia, Recombinant (GST & His & Myc) Alpha-CT,Alpha-Ctx,Alpha-EPTX-Nk2a,Long neurotoxin ...	Naja kaouthia	E. coli
	Monomer: binds with high affinity to muscular (alpha-1-beta-1-gamma-delta/CHRNA1-CHRNB1-CHRNG-CHRND) nAChR (tested on Torpedo californica, Kd=0.2-4.5 nM) and neuronal alpha-7/CHRNA7 nicotinic acetylcholine receptors (Kd=13-105 nM). Also inhibits GABA(A) channels. Heteropentamer targets studied are composed of alpha-1-beta-3-gamma-2 (GABRA1-GABRB3-GABRG2) subunits (IC(50)=236 nM), alpha-1-beta-2-gamma-2 (GABRA1-GABRB2-GABRG2) subunits (IC(50)=469 nM), alpha-2-beta-2-gamma-2 (GABRA2-GABRB2-GABRG2)...

重组蛋白

Beta-lactamase CTX-M-2 Protein, Salmonella typhimurium, Recombinant

Cat.No: TMPH-03474

Species: Salmonella typhimurium

Expression System: E. coli

Beta-lactamase CTX-M-1 Protein, E. coli, Recombinant (His)

Cat.No: TMPH-00584

Species: E. coli

Expression System: E. coli

Beta-lactamase CTX-M-1 Protein, E. coli, Recombinant (Yeast, His)

Cat.No: TMPH-00585

Species: E. coli

Expression System: P. pastoris (Yeast)

Cytotoxin 2 Protein, Naja atra, Recombinant (His & Myc)

Cat.No: TMPH-03036

Species: Naja atra

Expression System: E. coli

Alpha-cobratoxin Protein, Naja kaouthia, Recombinant (GST & His & Myc)

Cat.No: TMPH-03037

Species: Naja kaouthia

Expression System: E. coli

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