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Targets Recommended: ATP Citrate Lyase Isocitrate Dehydrogenase (IDH) Others ADC Linker

386

抑制剂 & 化合物

91

天然产物

2

化合物库

1

TargetMol 试剂盒

12

重组蛋白

22

同位素标记化合物

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Cat. No. Product Name
L3100 造血毒性小分子库

101 compounds
101 种生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
L4900 心血管毒性化合物库

131 compounds
131 种心血管毒性化合物的独特集合,可用于毒理学研究;

化合物库

造血毒性小分子库
Cat.No: L3100
Compounds: 101
心血管毒性化合物库
Cat.No: L4900
Compounds: 131
Cat. No. Product Name Form Specificity Of Inhibition
C0074 Mag Beads COOH High capacity (2.8 μm)

羧基磁珠 (2.8 μm)

Suspension in bottle

TargetMol 试剂盒

羧基磁珠 (2.8 μm)
Cat.No: C0074
Cat. No. Product Name Target Signaling Pathways
T18868 Val-Cit

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Val-Cit 是一种可切割的 ADC 接头,用于合成抗体-药物偶联物。
T18867 Val-Cit-PAB-MMAE

Drug-Linker Conjugates for ADC Antibody-drug Conjugate/ADC Related
Val-Cit-PAB-MMAE 是 ADC 的药物-接头偶联物。它包含 ADC 接头(肽 Val-Cit-PAB)和有效的微管蛋白抑制剂 MMAE。
T17983 Fmoc-Val-Cit-PAB-MMAE

Others; Drug-Linker Conjugates for ADC Antibody-drug Conjugate/ADC Related; Others
Fmoc-Val-Cit-PAB-MMAE 由 ADC 接头 (Fmoc-Val-Cit-PAB) 和强效微管蛋白抑制剂 (MMAE) 组成。 它是一种用于 ADC 的药物-接头偶联物。
T17693 Boc-Val-Cit-PAB

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Boc-Val-Cit-PAB 是一种可切割的 ADC 接头,用于抗体-药物偶联物的合成。
T17213 Val-cit-PAB-OH

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Val-cit-PAB-OH 是可降解ADC 连接剂。
T17691 Boc-Val-Cit-OH

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Boc-Val-Cit-OH 是一种可切割的 ADC 接头,用于合成抗体-药物偶联物。
T4678 Fmoc-Val-Cit-PAB

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Fmoc-Val-Cit-PAB 是一种可降解的抗体-药物偶联的连接剂。
T7767 FMoc-Val-Cit-PAB-PNP

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Fmoc-Val-Cit-PAB-PNP 是一种可降解的 ADC 连接剂,可用于合成抗体偶联药物。
T18321 Mc-Val-Cit-PAB-Cl

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Mc-Val-Cit-PAB-Cl 是一种可切割的 ADC 接头,可用于偶联 MMAE 和抗体以形成抗体-MC-vc-MMAE。
T40303 5-A-RU-PABC-Val-Cit-Fmoc

Others Others
5-A-RU-PABC-Val-Cit-Fmoc 是 5-A-RU 的前体物质之一。5-A-RU 是一种小分子粘膜相关的 MAIT 激活剂,是细菌合成核黄素的前体物质。
T5149 MC-Val-Cit-PAB

N-[6-(2,5-二氢-2,5-二氧代-1H-吡咯-1-基)-1-氧代己基]-L-缬氨酰-N5-(氨基甲酰基)-N-[4-(羟甲基)苯基]-L-鸟氨酰胺

Others; AChR; ADC Linker Antibody-drug Conjugate/ADC Related; Neuroscience; Others
MC-Val-Cit-PAB 是一种组织蛋白酶可裂解的 ADC 接头,用于制备抗体-药物偶联物。
T17692 Boc-Val-Cit-PAB-PNP

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Boc-Val-Cit-PAB-PNP 是一种可切割的 ADC 接头,用于合成抗体-药物偶联物。
T18267 Mal-PEG1-Val-Cit-OH

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Mal-PEG1-Val-Cit-OH是一种在抗体药物偶联体(ADCs)[1]合成中使用的可裂解单元聚乙二醇(PEG)连接器。
T3503 MC-Val-Cit-PABC-PNP

Maleimidocaproyl-L-valine-L-citrulline-p-aminobenzyl alcohol p-nitrophenyl carbonate,马来酰亚胺基己酰-L-缬氨酸-L-瓜氨酸对氨基苄醇 对硝基苯基碳酸脂

Others; AChR; ADC Linker Antibody-drug Conjugate/ADC Related; Neuroscience; Others
MC-Val-Cit-PABC-PNP 是一种组织蛋白酶可裂解的 ADC 肽接头,可用于合成抗体偶联药物。
T39765 Mal-PEG1-Val-Cit-PAB-PNP

Mal-PEG1-Val-Cit-PAB-PNP

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Mal-PEG1-Val-Cit-PAB-PNP is an ADC linker employed in the synthesis of ADCs, enabling cleavage.
T39748 DBCO-PEG4-Val-Cit-PAB-MMAF

DBCO-PEG4-Val-Cit-PAB-MMAF

Others; Drug-Linker Conjugates for ADC Antibody-drug Conjugate/ADC Related; Others
DBCO-PEG4-Val-Cit-PAB-MMAF is a chemical compound that comprises a cleavable 4 unit polyethylene glycol antibody-drug conjugate (ADC) linker known as DBCO-PEG4-Val-Cit-PAB, and a highly effective inhibitor of tubulin polymerization called MMAF. This compound serves as a valuable component in the synthesis of ADCs.
T77847 MC-Val-Cit-PAB-Exatecan

MC-Val-Cit-PAB-DX8951

Others; Drug-Linker Conjugates for ADC Antibody-drug Conjugate/ADC Related; Others
MC-Val-Cit-PAB-Exatecan (MC-Val-Cit-PAB-DX8951) 是一种抗体-活性分子偶联物(ADC)的关键部分,由 DNA 拓扑异构酶 I 抑制剂 DX-8951 和组织蛋白酶敏感的连接子共同构成。
T39307 Azido-PEG4-Val-Cit-PAB-MMAE

Azido-PEG4-Val-Cit-PAB-MMAE

Others; Drug-Linker Conjugates for ADC Antibody-drug Conjugate/ADC Related; Others
Azido-PEG4-Val-Cit-PAB-MMAE is a drug-linker conjugate for antibody-drug conjugates (ADCs), comprising the anti-mitotic agent monomethyl auristatin E (MMAE, a tubulin inhibitor), connected through the cleavable linker Azido-PEG4-Val-Cit-PAB-OH.
T77876 Py-MAA-Val-Cit-PAB-MMAE

AAJ8D6-PY-Val-Cit-MMAE

Others; Drug-Linker Conjugates for ADC Antibody-drug Conjugate/ADC Related; Others
Py-MAA-Val-Cit-PAB-MMAE (AAJ8D6-PY-Val-Cit-MMAE) 是一款ADC Linker,专用于合成抗体药物偶联物Zapadcine-3a (ADC)。Zapadcine-3a 对抗多种肿瘤表现出高效的活性,其作用机理为定位TRAILR2并通过肿瘤细胞内的溶酶体被摄取,进而针对性释放致死的小分子,从而特异性消灭TRAILR2阳性的肿瘤细胞,并能够有效地治愈肿瘤。
T38739 Mal-PEG2-Val-Cit-PABA-PNP

Mal-PEG2-Val-Cit-PABA-PNP

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Mal-PEG2-Val-Cit-PABA-PNP is a cleavable linker compound employed in the synthesis of antibody-drug conjugates (ADCs).
T39447 Azide-PEG1-Val-Cit-PABC-OH

Azide-PEG1-Val-Cit-PABC-OH

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Azide-PEG1-Val-Cit-PABC-OH is a one-unit PEG cleavable linker employed for the synthesis of antibody-drug conjugates (ADCs).
T33243 MC-Val-Cit-PAB-VX765

Belnacasan-conjugate,VX765-conjugate,MC-Val-Cit-PABC-VX765

Others Others
MC-VAL-CIT-PAB-VX765 or MC-VAL-CIT-PABC-VX765 is a VX765 derivative that can be conjugated to antibodies, proteins, or polymers for targeted drug delivery. MC-Val- CIT -PAB is a cathepsin cleavable ADC connector, which has been widely used in the preparat
T39579 Mal-(CH2)5-Val-Cit-PAB-Eribulin

Mal-(CH2)5-Val-Cit-PAB-Eribulin

Others; Drug-Linker Conjugates for ADC Antibody-drug Conjugate/ADC Related; Others
Mal-(CH2)5-Val-Cit-PAB-Eribulin is a potent antitumor ADC drug-linker conjugate that utilizes Eribulin, an anti-microtubule agent, connected through the Mal-(CH2)5-Val-Cit-PAB linker.
T18320 MC-Val-Cit-PAB-carfilzomib iodide

MC-Val-Cit-PAB-carfilzomib

Others; Drug-Linker Conjugates for ADC Antibody-drug Conjugate/ADC Related; Others
MC-Val-Cit-PAB-carfilzomib is a potent antitumor drug-linker conjugate for antibody-drug conjugates (ADC), comprising the irreversible proteasome inhibitor carfilzomib, connected through the ADC linker MC-Val-Cit-PAB.
T18324 MC-Val-Cit-PAB-duocarmycin chloride

MC-Val-Cit-PAB-duocarmycin

Others; Drug-Linker Conjugates for ADC Antibody-drug Conjugate/ADC Related; Others
MC-Val-Cit-PAB-duocarmycin is an antibody-drug conjugate (ADC) linker that combines duocarmycin, a potent DNA minor groove-binding alkylating agent, with an antitumor drug through the MC-Val-Cit-PAB linker, exhibiting significant antitumor activity.
T38747 Fmoc-Val-D-Cit-PAB

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Fmoc-Val-D-Cit-PAB is a cleavable linker for antibody-drug-conjugation (ADC).
T38746 Fmoc-D-Val-Cit-PAB

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Fmoc-D-Val-Cit-PAB is a cleavable linker for antibody-drug-conjugation (ADC).
T38748 Fmoc-D-Val-D-Cit-PAB

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Fmoc-D-Val-D-Cit-PAB is a cleavable linker for antibody-drug-conjugation (ADC).
T18323 MC-Val-Cit-PAB-dimethylDNA31

Others; Drug-Linker Conjugates for ADC Antibody-drug Conjugate/ADC Related; Others
MC-Val-Cit-PAB-dimethylDNA31 is a drug-linker conjugate employed in antibody-drug conjugates (ADCs) that exhibits robust antitumor efficacy. This conjugate utilizes the ADC linker, MC-Val-Cit-PAB, to link to the potent antitumor agent dimethylDNA31. Notably, dimethylDNA31 also demonstrates significant bactericidal activity against both persister and stationary-phase Staphylococcus aureus.
T17814 DBCO-Val-Cit-OH

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
DBCO-Val-Cit-OH, a cleavable linker compound, finds utility in the synthesis of antibody-drug conjugates (ADCs)[1].
T39328 SuO-Glu-Val-Cit-PAB-MMAE

Others; Drug-Linker Conjugates for ADC Antibody-drug Conjugate/ADC Related; Others
SuO-Glu-Val-Cit-PAB-MMAE is a chemical compound comprising a cleavable ADC linker, SuO-Glu-Val-Cit-PAB, and a potent tubulin inhibitor known as MMAE. It is utilized in the synthesis of antibody-drug conjugates (ADCs).
T18736 SuO-Val-Cit-PAB-MMAE

Others; Drug-Linker Conjugates for ADC Antibody-drug Conjugate/ADC Related; Others
SuO-Val-Cit-PAB-MMAE is an ADC (antibody-drug conjugate) linker comprising the anti-mitotic monomethyl auristatin E (MMAE, a tubulin inhibitor) connected through the SuO-Val-Cit-PAB peptide.
T17816 DBCO-Val-Cit-PABC-PNP

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
DBCO-Val-Cit-PABC-PNP is a cleavable linker for antibody-drug conjugate (ADC) synthesis[1].
T18511 OPSS-Val-Cit-PAB-OH

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
OPSS-Val-Cit-PAB-OH is an ADC linker utilized for the synthesis of antibody-drug conjugates (ADCs) [1].
T17531 BCN-PEG3-Val-Cit

Others Others
BCN-PEG3-Val-Cit is a PEG-based linker commonly employed in PROTAC synthesis[1]. Additionally, it serves as a cleavable 3 unit PEG linker in the production of antibody-drug conjugates (ADCs)[2].
T18677 SC-Val-Cit-PAB

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
SC-Val-Cit-PAB is a cleavable ADC linker for antibody-drug conjugates (ADCs).
T18307 MC(C5)-Val-Cit

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
MC(C5)-Val-Cit is a cleavable ADC linker employed in ADCs synthesis [1].
T18315 MC-Sq-Cit-PAB-Dolastatin10

Others; Drug-Linker Conjugates for ADC Antibody-drug Conjugate/ADC Related; Others
MC-Sq-Cit-PAB-Dolastatin10 is a potent antitumor drug-linker conjugate for Antibody-Drug Conjugates (ADC), utilizing Dolastatin10 (a tubulin polymerization inhibitor) connected through the MC-Sq-Cit-PAB ADC linker.
T17478 Azido-PEG1-Val-Cit-OH

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Azido-PEG1-Val-Cit-OH is a one-unit cleavable PEG ADC linker employed in the synthesis of antibody-drug conjugates (ADCs)[1].
T28621 RTI-55

ß CIT,ß-CIT,RTI 55,ßCIT

Others Others
RTI-55 is an inhibitor of non-selective dopamine reuptake.
T18753 TCO-PEG1-Val-Cit-OH

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
TCO-PEG1-Val-Cit-OH is a cleavable 1-unit polyethylene glycol (PEG) linker utilized in the synthesis of antibody-drug conjugates (ADCs)[1].
T18301 Mal-Phe-C4-Val-Cit-PAB

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Mal-Phe-C4-Val-Cit-PAB is a cleavable antibody-drug conjugate (ADC) linker featuring a Maleimide functional group. It is employed in the synthesis of ADCs.
T18299 Mal-PEG8-Val-Cit-PAB-MMAE

Others; Drug-Linker Conjugates for ADC Antibody-drug Conjugate/ADC Related; Others
Mal-PEG8-Val-Cit-PAB-MMAE is a cleavable 8 unit PEG ADC linker used in the synthesis of antibody-drug conjugates (ADCs)[1].
T18512 OPSS-Val-Cit-PAB-PNP

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
OPSS-Val-Cit-PAB-PNP is a cleavable linker employed in ADC (antibody-drug conjugates) synthesis [1].
T18328 MC-Val-Cit-PAB-rifabutin

Others; Drug-Linker Conjugates for ADC Antibody-drug Conjugate/ADC Related; Others
MC-Val-Cit-PAB-rifabutin is a drug-linker conjugate designed for antibody-drug conjugates (ADC), featuring the potent antitumor agent rifabutin (a DNA-dependent RNA polymerase inhibitor) connected through the MC-Val-Cit-PAB ADC linker. This configuration endows it with significant antitumor activity.
T17356 Acid-propionylamino-Val-Cit-OH

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
Acid-propionylamino-Val-Cit-OH is a cleavable linker commonly employed in the synthesis of antibody-drug conjugates (ADCs)[1].
T17788 DBCO-(PEG2-Val-Cit-PAB)2

Others; ADC Linker Antibody-drug Conjugate/ADC Related; Others
DBCO-(PEG2-Val-Cit-PAB)2 is a dual cleavable ADC linker for antibody-drug conjugates (ADCs).
T18330 MC-Val-Cit-PAB-vinblastine

Others; Drug-Linker Conjugates for ADC Antibody-drug Conjugate/ADC Related; Others
MC-Val-Cit-PAB-vinblastine is a potent antitumor drug-linker conjugate for Antibody-Drug Conjugates (ADC), featuring vinblastine (a microtubule protein inhibitor) connected through the MC-Val-Cit-PAB ADC linker.
T18327 MC-Val-Cit-PAB-Retapamulin

Others; Drug-Linker Conjugates for ADC Antibody-drug Conjugate/ADC Related; Others
MC-Val-Cit-PAB-Retapamulin is a drug-linker conjugate for antibody-drug conjugates (ADC) that exhibits potent antitumor activity. This compound utilizes Retapamulin, a ribosome inhibitor, connected through the ADC linker MC-Val-Cit-PAB.
T18326 MC-Val-Cit-PAB-MMAF

Others; Drug-Linker Conjugates for ADC Antibody-drug Conjugate/ADC Related; Others
MC-Val-Cit-PAB-MMAF is an antibody-drug conjugate (ADC) component that exhibits antitumor properties through the action of the tubulin inhibitor, monomethyl auristatin F (MMAF), which is connected by a cathepsin-cleavable linker, MC-Val-Cit-PAB.

化合物

Val-Cit
Cat.No: T18868
Synonym:
Target: Others, ADC Linker
Val-Cit-PAB-MMAE
Cat.No: T18867
Synonym:
Target: Drug-Linker Conjugates for ADC
Fmoc-Val-Cit-PAB-MMAE
Cat.No: T17983
Synonym:
Target: Others, Drug-Linker Conjugates for ADC
Boc-Val-Cit-PAB
Cat.No: T17693
Synonym:
Target: Others, ADC Linker
Val-cit-PAB-OH
Cat.No: T17213
Synonym:
Target: Others, ADC Linker
Boc-Val-Cit-OH
Cat.No: T17691
Synonym:
Target: Others, ADC Linker
Fmoc-Val-Cit-PAB
Cat.No: T4678
Synonym:
Target: Others, ADC Linker
FMoc-Val-Cit-PAB-PNP
Cat.No: T7767
Synonym:
Target: Others, ADC Linker
Mc-Val-Cit-PAB-Cl
Cat.No: T18321
Synonym:
Target: Others, ADC Linker
5-A-RU-PABC-Val-Cit-Fmoc
Cat.No: T40303
Synonym:
Target: Others
MC-Val-Cit-PAB
Cat.No: T5149
Synonym: N-[6-(2,5-二氢-2,5-二氧代-1H-吡咯-1-基)-1-氧代己基]-L-缬氨酰-N5-(氨基甲酰基)-N-[4-(羟甲基)苯基]-L-鸟氨酰胺
Target: Others, AChR, ADC Linker
Boc-Val-Cit-PAB-PNP
Cat.No: T17692
Synonym:
Target: Others, ADC Linker
Mal-PEG1-Val-Cit-OH
Cat.No: T18267
Synonym:
Target: Others, ADC Linker
MC-Val-Cit-PABC-PNP
Cat.No: T3503
Synonym: Maleimidocaproyl-L-valine-L-citrulline-p-aminobenzyl alcohol p-nitrophenyl carbonate,马来酰亚胺基己酰-L-缬氨酸-L-瓜氨酸对氨基苄醇 对硝基苯基碳酸脂
Target: Others, AChR, ADC Linker
Mal-PEG1-Val-Cit-PAB-PNP
Cat.No: T39765
Synonym: Mal-PEG1-Val-Cit-PAB-PNP
Target: Others, ADC Linker
DBCO-PEG4-Val-Cit-PAB-MMAF
Cat.No: T39748
Synonym: DBCO-PEG4-Val-Cit-PAB-MMAF
Target: Others, Drug-Linker Conjugates for ADC
MC-Val-Cit-PAB-Exatecan
Cat.No: T77847
Synonym: MC-Val-Cit-PAB-DX8951
Target: Others, Drug-Linker Conjugates for ADC
Azido-PEG4-Val-Cit-PAB-MMAE
Cat.No: T39307
Synonym: Azido-PEG4-Val-Cit-PAB-MMAE
Target: Others, Drug-Linker Conjugates for ADC
Py-MAA-Val-Cit-PAB-MMAE
Cat.No: T77876
Synonym: AAJ8D6-PY-Val-Cit-MMAE
Target: Others, Drug-Linker Conjugates for ADC
Mal-PEG2-Val-Cit-PABA-PNP
Cat.No: T38739
Synonym: Mal-PEG2-Val-Cit-PABA-PNP
Target: Others, ADC Linker
Azide-PEG1-Val-Cit-PABC-OH
Cat.No: T39447
Synonym: Azide-PEG1-Val-Cit-PABC-OH
Target: Others, ADC Linker
MC-Val-Cit-PAB-VX765
Cat.No: T33243
Synonym: Belnacasan-conjugate,VX765-conjugate,MC-Val-Cit-PABC-VX765
Target: Others
Mal-(CH2)5-Val-Cit-PAB-Eribulin
Cat.No: T39579
Synonym: Mal-(CH2)5-Val-Cit-PAB-Eribulin
Target: Others, Drug-Linker Conjugates for ADC
MC-Val-Cit-PAB-carfilzomib iodide
Cat.No: T18320
Synonym: MC-Val-Cit-PAB-carfilzomib
Target: Others, Drug-Linker Conjugates for ADC
MC-Val-Cit-PAB-duocarmycin chloride
Cat.No: T18324
Synonym: MC-Val-Cit-PAB-duocarmycin
Target: Others, Drug-Linker Conjugates for ADC
Fmoc-Val-D-Cit-PAB
Cat.No: T38747
Synonym:
Target: Others, ADC Linker
Fmoc-D-Val-Cit-PAB
Cat.No: T38746
Synonym:
Target: Others, ADC Linker
Fmoc-D-Val-D-Cit-PAB
Cat.No: T38748
Synonym:
Target: Others, ADC Linker
MC-Val-Cit-PAB-dimethylDNA31
Cat.No: T18323
Synonym:
Target: Others, Drug-Linker Conjugates for ADC
DBCO-Val-Cit-OH
Cat.No: T17814
Synonym:
Target: Others, ADC Linker
SuO-Glu-Val-Cit-PAB-MMAE
Cat.No: T39328
Synonym:
Target: Others, Drug-Linker Conjugates for ADC
SuO-Val-Cit-PAB-MMAE
Cat.No: T18736
Synonym:
Target: Others, Drug-Linker Conjugates for ADC
DBCO-Val-Cit-PABC-PNP
Cat.No: T17816
Synonym:
Target: Others, ADC Linker
OPSS-Val-Cit-PAB-OH
Cat.No: T18511
Synonym:
Target: Others, ADC Linker
BCN-PEG3-Val-Cit
Cat.No: T17531
Synonym:
Target: Others
SC-Val-Cit-PAB
Cat.No: T18677
Synonym:
Target: Others, ADC Linker
MC(C5)-Val-Cit
Cat.No: T18307
Synonym:
Target: Others, ADC Linker
MC-Sq-Cit-PAB-Dolastatin10
Cat.No: T18315
Synonym:
Target: Others, Drug-Linker Conjugates for ADC
Azido-PEG1-Val-Cit-OH
Cat.No: T17478
Synonym:
Target: Others, ADC Linker
RTI-55
Cat.No: T28621
Synonym: ß CIT,ß-CIT,RTI 55,ßCIT
Target: Others
TCO-PEG1-Val-Cit-OH
Cat.No: T18753
Synonym:
Target: Others, ADC Linker
Mal-Phe-C4-Val-Cit-PAB
Cat.No: T18301
Synonym:
Target: Others, ADC Linker
Mal-PEG8-Val-Cit-PAB-MMAE
Cat.No: T18299
Synonym:
Target: Others, Drug-Linker Conjugates for ADC
OPSS-Val-Cit-PAB-PNP
Cat.No: T18512
Synonym:
Target: Others, ADC Linker
MC-Val-Cit-PAB-rifabutin
Cat.No: T18328
Synonym:
Target: Others, Drug-Linker Conjugates for ADC
Acid-propionylamino-Val-Cit-OH
Cat.No: T17356
Synonym:
Target: Others, ADC Linker
DBCO-(PEG2-Val-Cit-PAB)2
Cat.No: T17788
Synonym:
Target: Others, ADC Linker
MC-Val-Cit-PAB-vinblastine
Cat.No: T18330
Synonym:
Target: Others, Drug-Linker Conjugates for ADC
MC-Val-Cit-PAB-Retapamulin
Cat.No: T18327
Synonym:
Target: Others, Drug-Linker Conjugates for ADC
MC-Val-Cit-PAB-MMAF
Cat.No: T18326
Synonym:
Target: Others, Drug-Linker Conjugates for ADC
Cat. No. Product Name Target Signaling Pathways
TN7247 Limocitrin 3-O-sophoroside

Limocitrinyle-3-O-β-D-sophoroside

Limocitrin 3-O-sophoroside 是一种可用于生物研究的化合物。
TQ0216 Ercalcitriol

1α,25-Dihydroxy Vitamin D2

Others Others
Ercalcitriol (1α,25-Dihydroxy Vitamin D2) 是维生素 D2 的活性代谢物。 Ercalcitriol 作为维生素 D 的生理活化形式,通过调节正常细胞和转化细胞中的导管素抗菌肽 (CAMP) 和防御素 β-4 (DEFB4) 基因来增强免疫力,从而对抗病原体感染。
T8061 Citronellal

(±)-Citronellal,香茅醛

Others Others
Citronellal ((±)-Citronellal) 是多种芳香植物精油的单萜烯,具有促进睡眠、安定和抗伤害的作用。它可以降低机械伤害感受,且部分通过 NO-cGMP-ATP 敏感型 K⁺渠道通道介导的。
T8069 Triethyl citrate

Others Others
Triethyl citrate 是一种柠檬酸酯,可在纤维素塑料基纳米复合材料中,作为增塑剂使用。
T1591 Ancitabine hydrochloride

NSC 145668 HCl,盐酸环胞苷,Cyclocytidine hydrochloride,Cyclo-CMP hydrochloride,Cyclocytidine HCl,Cyclo-C

Others; DNA/RNA Synthesis; Autophagy Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Others
Ancitabine hydrochloride (NSC 145668 HCl) 是一种天然的抗白血病药物。
T4525 Citraconic acid

2-Methylmaleic Acid,柠康酸,Cis-Methylbutenedioic Acid

Endogenous Metabolite Metabolism
Citraconic acid (2-Methylmaleic Acid) 是由马来酸在2-位具有甲基取代基的二羧酸。
T4S0758 Isoquercitrin-7-O-gentiobioside

槲皮素-3-O-Β-D-葡萄糖-7-O-Β-D-龙胆双糖苷,Quercetin-3-O-beta-D-glucose-7-O-beta-D-gentiobioside,Quercetin-3-O-β-D-glucose-7-O-β-D-gentiobiosiden

Others Others
Quercetin-3-O-β-D-glucose-7-O-β-D-gentiobiosiden (Quercetin-3-O-beta-D-glucose-7-O-beta-D-gentiobioside) 是一种黄酮,来源于 Quercetin 中。
T2852 Citropten

Limettin,Citroptene,Limetin,5, 7-Dimethoxycoumarin,柠美内脂,5,7-二甲氧基香豆素,5,7-Dimethoxycoumarin

Others Others
Citropten 是一种香豆素,分离自佛手柑油中,对 A2058 人黑色素瘤细胞株具有抗增殖作用。
T1508 Decitabine

Dacogen,NSC 127716,地西他滨,Deoxycytidine,5-Aza-2'-deoxycytidine

Apoptosis; Nucleoside Antimetabolite/Analog; DNA Methyltransferase Apoptosis; Cell Cycle/Checkpoint; Chromatin/Epigenetic; DNA Damage/DNA Repair
Decitabine (Deoxycytidine) 是脱氧胞苷类似物,一种 DNA 甲基转移酶抑制剂,具有口服活性。Decitabine 具有抗肿瘤活性和抗代谢活性。Decitabine 诱导细胞周期阻滞和凋亡。
T5257 L-Homocitrulline

高瓜氨酸,Homo-L-citrulline,Homocitrulline

Others; Endogenous Metabolite Metabolism; Others
L-Homocitrulline (Homocitrulline) 是一种代谢物,可在尿素循环障碍患者的尿液中大量检测到。在某些情况下,由于尿素循环的鸟氨酸供应耗尽而导致的氨甲酰磷酸酯的积累可能是 L-Homocitrulline 和高精氨酸合成增强的原因。
T5087 DL-Isocitric acid trisodium salt

异柠檬酸三钠盐,Isocitric acid trisodium salt

Others; Endogenous Metabolite Metabolism; Others
DL-Isocitric acid trisodium salt 是内源性代谢产物的一种。
T0256 Citric acid trilithium salt tetrahydrate

Lithium citrate tribasic tetrahydrate,柠檬酸三锂盐四水合物,Trilithium citrate tetrahydrate

Dehydrogenase; GSK-3; HIF/HIF Prolyl-Hydroxylase; Antibacterial; GluR Chromatin/Epigenetic; Metabolism; Microbiology/Virology; Neuroscience; PI3K/Akt/mTOR signaling; Stem Cells
Citric acid trilithium salt tetrahydrate (Lithium citrate tribasic tetrahydrate) 是一种用于治疗精神疾病的药物。它也是一种医药和建筑材料, 可用于氨基酸定量分析时的梯度洗脱。
T11589 Hydroxycitric acid tripotassium hydrate

柠檬酸钾一水合物,三水合钾柠檬酸,Potassium citrate monohydrate

ATP Citrate Lyase; HIF/HIF Prolyl-Hydroxylase; HIF Angiogenesis; Chromatin/Epigenetic; Metabolism
Hydroxycitric acid tripotassium hydrate (Potassium citrate monohydrate) 是一种藤黄果的主要活性成分,也是一种柠檬酸的衍生物。它可竞争性抑制柠檬酸裂解酶 (ATP citrate lyase) ,并具有减肥作用。它有效抑制结石形成,并抑制HIF,具有抗氧化,抗炎和抗肿瘤活性。
T1226 Bacitracin

Albac,Ziba-RX,杆菌肽

Antibacterial; Antibiotic Microbiology/Virology
Bacitracin (Ziba-RX) 是一种用于葡萄球菌感染的多肽抗生素。它通过与焦磷酸十一癸烯基结合,起抑制细胞壁生物合成作用。
T8057 Citronellyl acetate

Apoptosis; Others Apoptosis; Others
Citronellyl acetate 是一种植物次生代谢产物,具有杀菌、杀幼虫、杀菌和驱虫杀虫作用,以及抗伤害活性。它在人肝癌细胞中具有促凋亡活性。
T11590 (-)-Hydroxycitric acid

Garcinia acid,(-)-羟基柠檬酸

ATP Citrate Lyase Metabolism
(-)-Hydroxycitric acid (Garcinia acid) 是Garcinia cambogia 果皮中的主要酸。它是 ATP 柠檬酸裂解酶的竞争性抑制剂,能够抑制脂肪酸的合成,减少脂肪生成,控制食物摄入,从而减轻体重。
T3154 Citral

Geranialdehyde,alpha-Citral,柠檬醛,geranial

Others Others
Citral 是一种单萜,从柠檬草精油中获得,具有抗疼痛、抗炎作用。
T4813 L-Citrulline

Endogenous Metabolite Metabolism
L-Citrulline 是一种氨基酸,源自于精氨酸-瓜氨酸途径获得的 l-精氨酸,或脯氨酸、谷氨酰胺和谷氨酸盐的分解代谢过程中产生的鸟氨酸。
TN2151 Rhamnocitrin

Others Others
Rhamnocitrin 是一种分离自黄芪(沙源子)中的类黄酮,具有抗氧化,抗炎和抗动脉粥样硬化活性。它是 DPPH 的清除剂(IC50:28.38 mM)。
TN1124 Neoeriocitrin

AChE Neuroscience
Neoeriocitrin 是一种有效的乙酰胆碱酯酶抑制剂,分离于自百日草,在 MC3T3-E1 中显示出对增殖和成骨分化的活性。
T6S0325 Glycitein

黄豆黄素,Glycetein

Apoptosis; Others Apoptosis; Others
Glycitein (Glycetein) 是一种大豆异黄酮,可研究抗氧化和细胞凋亡。
T12045 (-)-Hydroxycitric acid lactone

藤黄内酯,Garcinia lactone

ATP Citrate Lyase Metabolism
(-)-Hydroxycitric acid lactone (Garcinia lactone) 是一种有效的 ATP-柠檬酸裂解酶抑制剂,能够催化柠檬酸盐线粒体外裂解为草酰乙酸和乙酰辅酶 A,限制了脂肪酸合成所需乙酰辅酶 A 单位的可用性。它是一种减肥药,是一种广受欢迎的减肥食品补充剂。
T0185 Escitalopram

Seroplex,依他普仑,S-(+)-Citalopram,艾司西酞普兰,(S)-Citalopram

Dopamine Receptor; 5-HT Receptor; Serotonin Transporter; Adrenergic Receptor; AChR; Norepinephrine; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Escitalopram (Seroplex) 是一种外消旋 Citalopram 的 S-对映体,是一种选择性 5-羟色胺再摄取抑制剂,Ki=0.89 nM,比 R(-)-enantiomer 结合亲和力高 30 倍。它对多巴胺转运体和去甲肾上腺素转运体均有选择性,是一种研究抑郁症的抗抑郁药。
T0136 Citicoline

CDP-Choline,Citicholine,尼古林,cytidine 5'-diphosphocholine,cytidine diphosphate-choline

Apoptosis; Dopamine Receptor; Endogenous Metabolite Apoptosis; GPCR/G Protein; Metabolism; Neuroscience
Citicoline (CDP-Choline) 是一种合成细胞膜组分磷脂酰胆碱的中间体,有神经保护作用。
T12952 Sodium citrate dihydrate

Citric acid trisodium salt dihydrate,Trisodium citrate dihydrate,二水合柠檬酸钠

Antibacterial Microbiology/Virology
Sodium citrate dihydrate (Trisodium citrate dihydrate) 是一种抗凝血剂,也用为缓冲剂和食品防腐剂。
TN4931 L-Citronellol

(S)-(-)-beta-Citronellol,(S)-(-)-β-Citronellol

Antifungal Microbiology/Virology
L-Citronellol ((S)-(-)-beta-Citronellol) 是一种从天竺葵中分离到的小分子化合物,具有抗真菌活性, 会对真菌膜产生影响。L-Citronellol 在对念珠菌酵母菌作用时与两性霉素B具有协同作用。
T1330 Acitretin

阿曲汀,Ro 10-1670,Etretin

Apoptosis; Retinoid Receptor; Autophagy Apoptosis; Autophagy; Metabolism
Acitretin (Ro 10-1670) 是一种维甲酸,可用于银屑病和阿尔兹海默症的研究。
T0529 Dulcite

Galactitol,Dulcitol,Euonymit,NSC 1944,D-Galactitol,Melampyrit,半乳糖醇

Endogenous Metabolite Metabolism
Dulcite (D-Galactitol) 是一种具有微甜味的糖醇,其是半乳糖的代谢分解产物。
TN3194 6''-O-xylosyl-glycitin

Others Others
6''-O-xylosyl-glycitin 是从 Pueraria thunbergiana Benth 的花中分离出来的。
T6S0221 Eriocitrin

eriodictyol 7-rutinoside,圣草次甙,Eriodictyol-7-O-Rutinoside,Eriodictioside,圣草次甙;圣草次苷,Eriodictyol glycoside

Apoptosis; Carbonic Anhydrase Apoptosis; Metabolism
Eriocitrin (Eriodictyol-7-O-Rutinoside) 是从柠檬中分离出来的一种黄酮类天然产物,是强效的抗氧化剂。它通过激活线粒体涉及的内在信号传导途径来触发细胞凋亡。它通过上调 p53、cyclin A、cyclin D3 和 CDK6 使 S 期细胞周期停滞,从而抑制肝癌细胞的增殖。
T5669 Citric acid monohydrate

Others Others
Citric acid monohydrate 是一种存在于柑橘类水果中的三羧酸。柠檬酸因其抗氧化特性而被用作药物制剂中的赋形剂。它保持活性成分的稳定性并用作防腐剂。
T3240 Citronellol

dihydrogeraniol,香茅醇,β-香茅醇,(±)-β-Citronellol

Reactive Oxygen Species Immunology/Inflammation; Metabolism; NF-κB
Citronellol ((±)-β-Citronellol) 是一种单萜类化合物,从头状天竺葵中分离到。它可通过上调 TNF-α,RIP1/RIP3 的活性,下调 caspase-3/caspase-8 的活性,以及增加活性氧 (ROS) 的聚集来诱导肿瘤细胞的坏死性凋亡。
T3237 Lecithin

Phospholutein,卵磷脂,L-α-磷脂酰胆碱,L-α-Phosphatidylcholine,Phosphatidylcholines

Others; Endogenous Metabolite Metabolism; Others
Lecithin (L-α-Phosphatidylcholine) 被认为是安全的常规磷脂源。磷脂能够改变动物细胞膜的脂肪酸组成和微观结构。
T8266 (R)-Citronellol

D-Citronellol,(R)-(+)-β-Citronellol,(R)-3,7-二甲基-6-辛烯醇

Others; Endogenous Metabolite Metabolism; Others
(R)-Citronellol ((R)-(+)-β-Citronellol) 是一种存在于天竺葵精油中的醇单萜。它抑制肥大细胞的脱颗粒,并且不影响咖啡因的苦味感。它能够用于装饰性化妆品,盥洗用品以及非化妆品中。
T13750 L-Fucitol

L-岩藻糖醇,1-Deoxy-D-galactitol

Others Others
L-Fucitol (1-Deoxy-D-galactitol) 是一种糖醇,从肉豆蔻 (Nutmeg) 中分离得到。
TN1299 Desmethylglycitein

4',6,7-三羟基异黄酮,4',6,7-三羟异黄酮,6-羟基大豆苷元,6,7,4'-Trihydroxyisoflavone

PI3K; CDK; PKC Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling
Desmethylglycitein (6,7,4'-Trihydroxyisoflavone) 是大豆中苷元的代谢产物,具有抗氧化性和抗癌活性。它是蛋白激酶 C(PKC)α 的直接抑制剂,抑制正常人皮肤成纤维细胞中的太阳紫外线诱导的基质金属蛋白酶1。它在体内直接结合CDK1和CDK2,抑制 CDK1 和 CDK2 活性。
T2820 Glycitin

黄豆黄苷,Glycitein-7-β-O-glucoside,Glycitein 7-O-β-glucoside

Others; Influenza Virus; Antibacterial Microbiology/Virology; Others
Glycitin (Glycitein 7-O-β-glucoside) 是一种从豆类中分离出来的天然异黄酮,有抗菌,抗病毒和雌激素作用,还有促进骨髓基质细胞和成骨细胞的增殖和抑制骨转换的生物学功能。
T8013 (S)​-​(-​)​-​Citronellal

(S)-(-)-3,7-Dimethyl-6-Octenal,(-)-香茅醛,(-​)​-​Citronellal

Others; Endogenous Metabolite Metabolism; Others
(S)​-​(-​)​-​Citronellal ((S)-(-)-3,7-Dimethyl-6-Octenal) 是存在于Corymbia citriodora 和Cymbopogon nardus 中的一种单萜类化合物。
T7921 β-Cyclocitral

beta-Cyclocitral,β-环柠檬醛

Others Others
β-Cyclocitral 是 β-胡萝卜素的挥发性氧化衍生物,是微囊藻特有的掠食性动物防御信号。它是一种强大的驱虫剂。它是主要的挥发性萜类化合物之一,可以上调防御基因的表达,从而增强过量光照 (EL) 的适应性。
T2871 Quercitrin

Sophoretin,3-rhamnosyl quercetin,Quercetin 3-rhamnoside,Xanthaurine,槲皮苷,Meletin

Reactive Oxygen Species; S6 Kinase; Autophagy Autophagy; Immunology/Inflammation; MAPK; Metabolism; NF-κB; PI3K/Akt/mTOR signaling
Quercitrin (3-rhamnosyl quercetin) 是苦荞麦中的一种天然产物,具有抗炎作用,有用于心血管疾病的研究潜力。
TN7238L Sanguinarine citrate

Sanguinarium citrate,Sanguinarin citrate,Pseudochelerythrine citrate

Antibiotic Microbiology/Virology
Sanguinarine citrate (Pseudochelerythrine chloride) 是一种来源于 Sanguinaria Canadensis 的生物碱,具有抗菌、抗炎和镇痛活性,可用于治疗口腔炎、牙龈出血和喉炎等口腔炎症疾病 。
T1208 Citicoline sodium

Citicoline sodium salt,CDP-choline,胞磷胆碱钠

Apoptosis; Others; Endogenous Metabolite Apoptosis; Metabolism; Others
Citicoline sodium (CDP-choline) 是一种合成细胞膜组分磷脂酰胆碱的中间体,有神经保护作用。
T5S0636 Citric acid

柠檬酸,Citro,Citretten

Apoptosis; Others; Endogenous Metabolite; Antibacterial; Antibiotic Apoptosis; Metabolism; Microbiology/Virology; Others
Citric acid (Citro) 是柑橘类水果中发现的弱有机三羧酸。柠檬酸是食品添加剂和天然防腐剂。
T3766 (-)-vibo-Quercitol

(-)-Viburnitol,(-)-VIBO-栎醇

Others Others
(-)-vibo-Quercitol ((-)-Viburnitol) 是一种羧基糖胺糖苷酶抑制剂。
T2757 Myricitrin

杨梅苷,Myricetrin,Myricitrine

PKC Chromatin/Epigenetic; Cytoskeletal Signaling
Myricitrin (Myricitrine) 是从杨梅根皮中分离出来的类黄酮化合物,具有镇痛作用。它是主要的抗氧化剂。
T6316 Calcitriol

Topitriol,Rocaltrol,Calcijex,RO215535,骨化三醇,1,25-Dihydroxyvitamin D3

Endogenous Metabolite Metabolism
Calcitriol (1,25-Dihydroxyvitamin D3) 是一种维他命 D 的代谢物,一种维他命 D 受体 (VDR) 的激动剂 (IC50=0.4 nM)。Calcitriol 增加肠道对钙和磷的吸收,并与甲状旁腺激素一起增加了骨吸收。
T20819 Ammonium iron(III) citrate

柠檬酸铁铵,柠檬酸铁 (III) 铵,Ferric ammonium citrate

Others; Ferroptosis Apoptosis; Others
Ammonium iron(III) citrate (Ferric ammonium citrate) 是一种非运铁蛋白结合的铁的生理形式,会引起的细胞内铁超负荷从而导致细胞铁死亡,能增强蛋白质产生。
TN3670 Citromycin

Antifection Microbiology/Virology
Citromycin, an antibiotic, has weakly cytotoxic.
TN1263 3''-O-Galloylmyricitrin

Others Others
3''-O-Galloylmyricitrin is a natural product
TN2934 3''-Galloylquercitrin

Others Others
1. 3''-Galloylquercitrin possesses the activity for PTK inhibition. <br/>
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天然产物

Limocitrin 3-O-sophoroside
Cat.No: TN7247
Synonym: Limocitrinyle-3-O-β-D-sophoroside
Target:
Ercalcitriol
Cat.No: TQ0216
Synonym: 1α,25-Dihydroxy Vitamin D2
Target: Others
Citronellal
Cat.No: T8061
Synonym: (±)-Citronellal,香茅醛
Target: Others
Triethyl citrate
Cat.No: T8069
Synonym:
Target: Others
Ancitabine hydrochloride
Cat.No: T1591
Synonym: NSC 145668 HCl,盐酸环胞苷,Cyclocytidine hydrochloride,Cyclo-CMP hydrochloride,Cyclocytidine HCl,Cyclo-C
Target: Others, DNA/RNA Synthesis, Autophagy
Citraconic acid
Cat.No: T4525
Synonym: 2-Methylmaleic Acid,柠康酸,Cis-Methylbutenedioic Acid
Target: Endogenous Metabolite
Isoquercitrin-7-O-gentiobioside
Cat.No: T4S0758
Synonym: 槲皮素-3-O-Β-D-葡萄糖-7-O-Β-D-龙胆双糖苷,Quercetin-3-O-beta-D-glucose-7-O-beta-D-gentiobioside,Quercetin-3-O-β-D-glucose-7-O-β-D-gentiobiosiden
Target: Others
Citropten
Cat.No: T2852
Synonym: Limettin,Citroptene,Limetin,5, 7-Dimethoxycoumarin,柠美内脂,5,7-二甲氧基香豆素,5,7-Dimethoxycoumarin
Target: Others
Decitabine
Cat.No: T1508
Synonym: Dacogen,NSC 127716,地西他滨,Deoxycytidine,5-Aza-2'-deoxycytidine
Target: Apoptosis, Nucleoside Antimetabolite/Analog, DNA Methyltransferase
L-Homocitrulline
Cat.No: T5257
Synonym: 高瓜氨酸,Homo-L-citrulline,Homocitrulline
Target: Others, Endogenous Metabolite
DL-Isocitric acid trisodium salt
Cat.No: T5087
Synonym: 异柠檬酸三钠盐,Isocitric acid trisodium salt
Target: Others, Endogenous Metabolite
Citric acid trilithium salt tetrahydrate
Cat.No: T0256
Synonym: Lithium citrate tribasic tetrahydrate,柠檬酸三锂盐四水合物,Trilithium citrate tetrahydrate
Target: Dehydrogenase, GSK-3, HIF/HIF Prolyl-Hydroxylase, Antibacterial, GluR
Hydroxycitric acid tripotassium hydrate
Cat.No: T11589
Synonym: 柠檬酸钾一水合物,三水合钾柠檬酸,Potassium citrate monohydrate
Target: ATP Citrate Lyase, HIF/HIF Prolyl-Hydroxylase, HIF
Bacitracin
Cat.No: T1226
Synonym: Albac,Ziba-RX,杆菌肽
Target: Antibacterial, Antibiotic
Citronellyl acetate
Cat.No: T8057
Synonym:
Target: Apoptosis, Others
(-)-Hydroxycitric acid
Cat.No: T11590
Synonym: Garcinia acid,(-)-羟基柠檬酸
Target: ATP Citrate Lyase
Citral
Cat.No: T3154
Synonym: Geranialdehyde,alpha-Citral,柠檬醛,geranial
Target: Others
L-Citrulline
Cat.No: T4813
Synonym:
Target: Endogenous Metabolite
Rhamnocitrin
Cat.No: TN2151
Synonym:
Target: Others
Neoeriocitrin
Cat.No: TN1124
Synonym:
Target: AChE
Glycitein
Cat.No: T6S0325
Synonym: 黄豆黄素,Glycetein
Target: Apoptosis, Others
(-)-Hydroxycitric acid lactone
Cat.No: T12045
Synonym: 藤黄内酯,Garcinia lactone
Target: ATP Citrate Lyase
Escitalopram
Cat.No: T0185
Synonym: Seroplex,依他普仑,S-(+)-Citalopram,艾司西酞普兰,(S)-Citalopram
Target: Dopamine Receptor, 5-HT Receptor, Serotonin Transporter, Adrenergic Receptor, AChR, Norepinephrine, Histamine Receptor
Citicoline
Cat.No: T0136
Synonym: CDP-Choline,Citicholine,尼古林,cytidine 5'-diphosphocholine,cytidine diphosphate-choline
Target: Apoptosis, Dopamine Receptor, Endogenous Metabolite
Sodium citrate dihydrate
Cat.No: T12952
Synonym: Citric acid trisodium salt dihydrate,Trisodium citrate dihydrate,二水合柠檬酸钠
Target: Antibacterial
L-Citronellol
Cat.No: TN4931
Synonym: (S)-(-)-beta-Citronellol,(S)-(-)-β-Citronellol
Target: Antifungal
Acitretin
Cat.No: T1330
Synonym: 阿曲汀,Ro 10-1670,Etretin
Target: Apoptosis, Retinoid Receptor, Autophagy
Dulcite
Cat.No: T0529
Synonym: Galactitol,Dulcitol,Euonymit,NSC 1944,D-Galactitol,Melampyrit,半乳糖醇
Target: Endogenous Metabolite
6''-O-xylosyl-glycitin
Cat.No: TN3194
Synonym:
Target: Others
Eriocitrin
Cat.No: T6S0221
Synonym: eriodictyol 7-rutinoside,圣草次甙,Eriodictyol-7-O-Rutinoside,Eriodictioside,圣草次甙;圣草次苷,Eriodictyol glycoside
Target: Apoptosis, Carbonic Anhydrase
Citric acid monohydrate
Cat.No: T5669
Synonym:
Target: Others
Citronellol
Cat.No: T3240
Synonym: dihydrogeraniol,香茅醇,β-香茅醇,(±)-β-Citronellol
Target: Reactive Oxygen Species
Lecithin
Cat.No: T3237
Synonym: Phospholutein,卵磷脂,L-α-磷脂酰胆碱,L-α-Phosphatidylcholine,Phosphatidylcholines
Target: Others, Endogenous Metabolite
(R)-Citronellol
Cat.No: T8266
Synonym: D-Citronellol,(R)-(+)-β-Citronellol,(R)-3,7-二甲基-6-辛烯醇
Target: Others, Endogenous Metabolite
L-Fucitol
Cat.No: T13750
Synonym: L-岩藻糖醇,1-Deoxy-D-galactitol
Target: Others
Desmethylglycitein
Cat.No: TN1299
Synonym: 4',6,7-三羟基异黄酮,4',6,7-三羟异黄酮,6-羟基大豆苷元,6,7,4'-Trihydroxyisoflavone
Target: PI3K, CDK, PKC
Glycitin
Cat.No: T2820
Synonym: 黄豆黄苷,Glycitein-7-β-O-glucoside,Glycitein 7-O-β-glucoside
Target: Others, Influenza Virus, Antibacterial
(S)​-​(-​)​-​Citronellal
Cat.No: T8013
Synonym: (S)-(-)-3,7-Dimethyl-6-Octenal,(-)-香茅醛,(-​)​-​Citronellal
Target: Others, Endogenous Metabolite
β-Cyclocitral
Cat.No: T7921
Synonym: beta-Cyclocitral,β-环柠檬醛
Target: Others
Quercitrin
Cat.No: T2871
Synonym: Sophoretin,3-rhamnosyl quercetin,Quercetin 3-rhamnoside,Xanthaurine,槲皮苷,Meletin
Target: Reactive Oxygen Species, S6 Kinase, Autophagy
Sanguinarine citrate
Cat.No: TN7238L
Synonym: Sanguinarium citrate,Sanguinarin citrate,Pseudochelerythrine citrate
Target: Antibiotic
Citicoline sodium
Cat.No: T1208
Synonym: Citicoline sodium salt,CDP-choline,胞磷胆碱钠
Target: Apoptosis, Others, Endogenous Metabolite
Citric acid
Cat.No: T5S0636
Synonym: 柠檬酸,Citro,Citretten
Target: Apoptosis, Others, Endogenous Metabolite, Antibacterial, Antibiotic
(-)-vibo-Quercitol
Cat.No: T3766
Synonym: (-)-Viburnitol,(-)-VIBO-栎醇
Target: Others
Myricitrin
Cat.No: T2757
Synonym: 杨梅苷,Myricetrin,Myricitrine
Target: PKC
Calcitriol
Cat.No: T6316
Synonym: Topitriol,Rocaltrol,Calcijex,RO215535,骨化三醇,1,25-Dihydroxyvitamin D3
Target: Endogenous Metabolite
Ammonium iron(III) citrate
Cat.No: T20819
Synonym: 柠檬酸铁铵,柠檬酸铁 (III) 铵,Ferric ammonium citrate
Target: Others, Ferroptosis
Citromycin
Cat.No: TN3670
Synonym:
Target: Antifection
3''-O-Galloylmyricitrin
Cat.No: TN1263
Synonym:
Target: Others
3''-Galloylquercitrin
Cat.No: TN2934
Synonym:
Target: Others
--------- 更多 ---------
Cat. No. Product Name Species Expression System
TMPY-02483 ATP citrate lyase/ACLY Protein, Human, Recombinant (His)

ATPCL,ACL,ATP citrate lyase,CLATP

Human Baculovirus Insect Cells
ATP citrate lyase, also known as Acly or Acl, is the primary enzyme responsible for the synthesis of cytosolic acetyl-CoA in many tissues. The enzyme is composed of two polymer chains which are polypeptides in human. ATP citrate lyase is responsible for catalyzing the conversion of citrate and CoA into acetyl-CoA and oxaloacetate, along with the hydrolysis of ATP. A definitive role for ATP citrate lyase in tumorigenesis has emerged from ATP citrate lyase RNAi and chemical inhibitor studies, show...
TMPY-00085 Calcitonin receptor Protein, Human, Recombinant (aa 1-153, hFc)

CTR,CTR1,CT-R,calcitonin receptor,CRT

Human HEK293 Cells
Calcitonin receptor Protein, Human, Recombinant (aa 1-153, hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 42.1 kDa and the accession number is P30988-2.
TMPY-00066 Procalcitonin/CALCA Protein, Human, Recombinant (His)

KC,CGRP,CALC1,Procalcitonin,CT,calcitonin-...

Human HEK293 Cells
Procalcitonin/CALCA Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 14.2 kDa and the accession number is P01258-1.
TMPH-00400 DHAK Protein, Citrobacter freundii, Recombinant (His & SUMO)

Dihydroxyacetone kinase,dhaK,Glycerone kinase,DHA kinase

Citrobacter freundii E. coli
Catalyzes the phosphorylation of dihydroxyacetone. DHAK Protein, Citrobacter freundii, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 35.9 kDa and the accession number is P45510.
TMPY-04120 Procalcitonin/CALCA Protein, Human, Recombinant (mFc)

Procalcitonin,CGRP,CGRP-I,calcitonin-relat...

Human HEK293 Cells
Procalcitonin/CALCA Protein, Human, Recombinant (mFc) is expressed in HEK293 mammalian cells with mFc tag. The predicted molecular weight is 39.2 kDa and the accession number is P01258-1.
TMPH-03412 Citrate synthase Protein, Rickettsia australis, Recombinant (His & Myc)

gltA,Citrate synthase

Rickettsia australis E. coli
Citrate synthase Protein, Rickettsia australis, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 53.6 kDa and the accession number is P51039.
TMPY-02413 Isocitrate dehydrogenase/IDH1 Protein, Human, Recombinant (His)

HEL-S-26,HEL-216,IDP,IDCD,PICD,IDH,isocitrate dehyd...

Human E. coli
Isocitrate dehydrogenase/IDH1 Protein, Human, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 48 kDa and the accession number is O75874.
TMPY-04070 Citrate Synthase Protein, Human, Recombinant (His)

citrate synthase

Human Baculovirus Insect Cells
Chondroitin sulphate (CS) glycosaminoglycan chains on cell and extracellular matrix proteoglycans (PGs) can no longer be regarded as merely hydrodynamic space fillers. Overwhelming evidence over recent years indicates that sulphation motif sequences within the CS chain structure are a source of significant biological information to cells and their surrounding environment. CS sulphation motifs have been shown to interact with a wide variety of bioactive molecules, e.g. cytokines, growth factors, ...
TMPY-00317 Calcitonin receptor Protein, Human, Recombinant (aa 25-154, hFc)

CTR,calcitonin receptor,CRT,CTR1,CT-R

Human HEK293 Cells
Calcitonin receptor Protein, Human, Recombinant (aa 25-154, hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 43.9 kDa and the accession number is P30988-1.
TMPH-03097 Beta-elicitin cryptogein Protein, Phytophthora cryptogea, Recombinant (His & Myc)

Beta-elicitin cryptogein,CRY

Phytophthora cryptogea E. coli
Induces local and distal defense responses (incompatible hypersensitive reaction) in plants from the solanaceae and cruciferae families. Elicits leaf necrosis and causes the accumulation of pathogenesis-related proteins. Might interact with the lipidic molecules of the plasma membrane. Beta-elicitin cryptogein Protein, Phytophthora cryptogea, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 17.3 kDa and the accession...
TMPH-00553 Fructose 5-dehydrogenase [NADP(+)] Protein, Erwinia citreus, Recombinant (His & KSI)

Fructose 5-dehydrogenase [NADP(+)],5-ketofructose reductase ...

Erwinia citreus E. coli
Fructose 5-dehydrogenase [NADP(+)] Protein, Erwinia citreus, Recombinant (His & KSI) is expressed in E. coli.
TMPH-00401 LGTase Protein, Citrus unshiu, Recombinant (His & Myc)

Limonoid UDP-glucosyltransferase

Citrus unshiu Baculovirus Insect Cells
LGTase Protein, Citrus unshiu, Recombinant (His & Myc) is expressed in Baculovirus.

重组蛋白

ATP citrate lyase/ACLY Protein, Human, Recombinant (His)
Cat.No: TMPY-02483
Species: Human
Expression System: Baculovirus Insect Cells
Calcitonin receptor Protein, Human, Recombinant (aa 1-153, hFc)
Cat.No: TMPY-00085
Species: Human
Expression System: HEK293 Cells
Procalcitonin/CALCA Protein, Human, Recombinant (His)
Cat.No: TMPY-00066
Species: Human
Expression System: HEK293 Cells
DHAK Protein, Citrobacter freundii, Recombinant (His & SUMO)
Cat.No: TMPH-00400
Species: Citrobacter freundii
Expression System: E. coli
Procalcitonin/CALCA Protein, Human, Recombinant (mFc)
Cat.No: TMPY-04120
Species: Human
Expression System: HEK293 Cells
Citrate synthase Protein, Rickettsia australis, Recombinant (His & Myc)
Cat.No: TMPH-03412
Species: Rickettsia australis
Expression System: E. coli
Isocitrate dehydrogenase/IDH1 Protein, Human, Recombinant (His)
Cat.No: TMPY-02413
Species: Human
Expression System: E. coli
Citrate Synthase Protein, Human, Recombinant (His)
Cat.No: TMPY-04070
Species: Human
Expression System: Baculovirus Insect Cells
Calcitonin receptor Protein, Human, Recombinant (aa 25-154, hFc)
Cat.No: TMPY-00317
Species: Human
Expression System: HEK293 Cells
Beta-elicitin cryptogein Protein, Phytophthora cryptogea, Recombinant (His & Myc)
Cat.No: TMPH-03097
Species: Phytophthora cryptogea
Expression System: E. coli
Fructose 5-dehydrogenase [NADP(+)] Protein, Erwinia citreus, Recombinant (His & KSI)
Cat.No: TMPH-00553
Species: Erwinia citreus
Expression System: E. coli
LGTase Protein, Citrus unshiu, Recombinant (His & Myc)
Cat.No: TMPH-00401
Species: Citrus unshiu
Expression System: Baculovirus Insect Cells
Cat. No. Product Name Target Signaling Pathways
T14687 Deucravacitinib

BMS-986165

Tyrosine Kinases; JAK; IFNAR; Interleukin Angiogenesis; Chromatin/Epigenetic; Immunology/Inflammation; JAK/STAT signaling; Stem Cells; Tyrosine Kinase/Adaptors
Deucravacitinib (BMS-986165) 是一种高选择性、口服生物可利用的变构 TYK2 抑制剂,用于治疗自身免疫性疾病。它通过稳定调节 JH2 结构域来阻断受体介导的 Tyk2 激活,可抑制IL-12/23和 I 型IFN 途径。它选择性结合 TYK2 假激酶 (JH2) 结构域,IC50为1.0 nM。
T11952 Maxacalcitol-D6

Others Others
Maxacalcitol-D6 is a non-calcemic vitamin D3 analog and VDR ligand of VDR-like receptors.Maxacalcitol-D6 is the deuterated form of Maxacalcitol (22-Oxacalcitriol).
TMIJ-0137 Tofacitinib-d3 Citrate

Tofacitinib-d3 Citrate 是 Tofacitinib Citrate 的氘代化合物。Tofacitinib Citrate 的 CAS 号为 540737-29-9。Tofacitinib citrate是JAK1/2/3抑制剂,IC50分别为112,20 和 1 nM。它具有抗菌,抗真菌和抗病毒活性。
TMID-0242 Capecitabine-d11

Capecitabine-d11 是 Capecitabine 的氘代化合物。Capecitabine 的 CAS 号为 154361-50-9。Capecitabine 是一种可口服的前药,可由胸苷磷酸化酶催化转变为其活性代谢物 Fluorouracil。
TMIJ-0267 Upadacitinib-15N-d2

Upadacitinib-15N-d2 是 Upadacitinib 的 15N 和氘代化合物。Upadacitinib 的 CAS 号为 1310726-60-3。Upadacitinib 是高效选择性的,具有口服活性的JAK1抑制剂,IC50为43 nM,可用于多种自身免疫性疾病的研究。它对 JAK1 的选择性约为 JAK2 的 74 倍。
T70394 Deucravacitinib HCl

Deucravacitinib HCl is a Highly Potent and Selective Allosteric Inhibitor of TYK2. BMS-986165 Blocks Il-12, IL-23 and type I Interferon Signaling and Provides for Robust Efficacy in Preclinical Models of Inflammatory Bowel Disease. MS-986165 potently binds to the Tyk2 pseudokinase domain (Ki = 0.02 nM), and is highly selective against a panel of 265 kinases and pseudokinases. The compound potently inhibited IL-23-, IL-12-, and Type I interferon-driven cellular signaling and transcriptional resp...
TMIH-0615 Zuclomiphene-d4 Citrate

cis-Clomiphene-d4 Citrate

Zuclomiphene-d4 Citrate 是 Zuclomiphene Citrate 的氘代化合物。Zuclomiphene Citrate 的 CAS 号为 14158-66-8。
TMIH-0159 Citalopram-d6

Citalopram-d6 是 Citalopram 的氘代化合物。Citalopram 的 CAS 号为 59729-33-8。Citalopram (Lu 10-171) 是一种具有口服活性的、选择性的血清素再摄取抑制剂 (SSRI),是一种选择性5-羟色胺再摄取抑制剂,是一种 S(+)-对映体 (Escitalopram) 和 R(-)-对映体的外消旋混合物。Citalopram 具有抗抑郁活性,可增强血清素能神经传递,可用于研究老年痴呆。
T12363 Paricalcitol-D6

Others Others
Paricalcitol-D6 is the deuterated form of Paricalcitol, which is used for the prevention and treatment of secondary hyperparathyroidism (excessive secretion of parathyroid hormone) associated with chronic renal failure.
T11934 Macitentan-d4

Macitentan D4,ACT-064992 D4

Endothelin Receptor GPCR/G Protein
Macitentan-d4 (ACT-064992 D4) 是一种 Macitentan 氘代物,可被当作非多肽 ETA 和 ETB  (内皮素受体)双拮抗剂。Macitentan-d4 比 Macitentan 毒性更低,半衰期更长,可用于研究由内皮素受体介导介导的疾病。
T19088 13-cis Acitretin D3

Isoacitretin D3,13-​cis Acitretin D3

Others Others
13-cis Acitretin D3 (Isoacitretin D3) is a deuterium-labeled 13-cis Acitretin. 13-cis Acitretin is the metabolite of Acitretin after chronic administration. Acitretin is a second-generation, systemic retinoid.
TMIH-0373 N-Desmethyl citalopram-d4 Oxalate

N-Desmethyl citalopram-d4 Oxalate 是 N-Desmethyl citalopram Oxalate 的氘代化合物。
T10351 Aprocitentan D4

ACT-132577 D4

Others Others
Aprocitentan D4 (ACT-132577 D4) is a deuterium-labeled Aprocitentan. Aprocitentan is a major and pharmacologically active metabolite of Macitentan. Aprocitentan is a dual ETA/ETB antagonist (IC50s: 3.4 nM and 987 nM; pA2s: 6.7 and 5.5).
TMIH-0158 Citalopram-d6 Oxalate

Citalopram-d6 Oxalate 是 Citalopram Oxalate 的氘代化合物。Citalopram Oxalate 的 CAS 号为 207559-01-1。
TMIH-0211 EN Clomiphene-d4 Citrate

EN Clomiphene-d4 Citrate 是 EN Clomiphene Citrate 的氘代化合物。
TMIH-0157 Citalopram-d4 Oxalate

Citalopram-d4 Oxalate 是 Citalopram Oxalate 的氘代化合物。Citalopram Oxalate 的 CAS 号为 207559-01-1。
TMIJ-0190 Gemcitabine EP Impurity C-13C-15N2

Gemcitabine EP Impurity C-13C-15N2 是 Gemcitabine EP Impurity C 的 13C 和 15 N 的标记化合物。
TMIJ-0153 Dapagliflozin-13C6 (glucitol-13C6)

Dapagliflozin-13C6 (glucitol-13C6) 是 Dapagliflozin 的 13C 的标记化合物。Dapagliflozin 的 CAS 号为 461432-26-8。Dapagliflozin竞争性的葡萄糖协同转运蛋白2 (SGLT2) 抑制剂,可促进尿液中葡萄糖的排泄,在糖尿病 (DM) 研究中具有价值。Dapagliflozin 诱导HIF1表达并减轻肾脏 IR 损伤。
TMIJ-0261 Baricitinib-d5

Baricitinib-d5 是 Baricitinib 的氘代化合物。Baricitinib 的 CAS 号为 1187594-09-7。Baricitinib 是一种选择性,可口服的JAK1和JAK2抑制剂,IC50分别为5.9 nM 和 5.7 nM,具有潜在的抗炎、免疫调节和抗肿瘤活性。
T10663 Calcitriol-d6

Calcitriol D6,骨化三醇 D6

Others Others
Calcitriol D6 is the deuterated form of Calcitriol, which is the hormonally active form of vitamin D. Calcitriol is the active metabolite of vitamin D3 that activates the vitamin D receptor.
T19305 Eldecalcitol-d6

Others Others
Eldecalcitol is an orally active analogue of active vitamin D used in the treatment of osteoporosis. Eldecalcitol-d6 is the deuterium labeled Eldecalcitol.
TMIH-0383 N-Despropyl Macitentan-d4

N-Despropyl Macitentan-d4 是 N-Despropyl Macitentan 的氘代化合物。N-Despropyl Macitentan 的 CAS 号为 1103522-45-7。Aprocitentan 是一种 Macitentan 的主要活性代谢物。它是ETA/ETB的双重拮抗剂,其pA2值分别为 6.7 和 5.5,IC50分别为 3.4 nM 和 987 nM。

同位素标记化合物

Deucravacitinib
Cat.No: T14687
Synonym: BMS-986165
Target: Tyrosine Kinases, JAK, IFNAR, Interleukin
Maxacalcitol-D6
Cat.No: T11952
Synonym:
Target: Others
Tofacitinib-d3 Citrate
Cat.No: TMIJ-0137
Synonym:
Target:
Capecitabine-d11
Cat.No: TMID-0242
Synonym:
Target:
Upadacitinib-15N-d2
Cat.No: TMIJ-0267
Synonym:
Target:
Deucravacitinib HCl
Cat.No: T70394
Synonym:
Target:
Zuclomiphene-d4 Citrate
Cat.No: TMIH-0615
Synonym: cis-Clomiphene-d4 Citrate
Target:
Citalopram-d6
Cat.No: TMIH-0159
Synonym:
Target:
Paricalcitol-D6
Cat.No: T12363
Synonym:
Target: Others
Macitentan-d4
Cat.No: T11934
Synonym: Macitentan D4,ACT-064992 D4
Target: Endothelin Receptor
13-cis Acitretin D3
Cat.No: T19088
Synonym: Isoacitretin D3,13-​cis Acitretin D3
Target: Others
N-Desmethyl citalopram-d4 Oxalate
Cat.No: TMIH-0373
Synonym:
Target:
Aprocitentan D4
Cat.No: T10351
Synonym: ACT-132577 D4
Target: Others
Citalopram-d6 Oxalate
Cat.No: TMIH-0158
Synonym:
Target:
EN Clomiphene-d4 Citrate
Cat.No: TMIH-0211
Synonym:
Target:
Citalopram-d4 Oxalate
Cat.No: TMIH-0157
Synonym:
Target:
Gemcitabine EP Impurity C-13C-15N2
Cat.No: TMIJ-0190
Synonym:
Target:
Dapagliflozin-13C6 (glucitol-13C6)
Cat.No: TMIJ-0153
Synonym:
Target:
Baricitinib-d5
Cat.No: TMIJ-0261
Synonym:
Target:
Calcitriol-d6
Cat.No: T10663
Synonym: Calcitriol D6,骨化三醇 D6
Target: Others
Eldecalcitol-d6
Cat.No: T19305
Synonym:
Target: Others
N-Despropyl Macitentan-d4
Cat.No: TMIH-0383
Synonym:
Target:
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