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Targets Recommended: cholecystokinin Mitochondrial Metabolism Apoptosis Caspase

479

抑制剂 & 化合物

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Cat. No. Product Name
L5300 线粒体靶向库

812 compounds
812 种具有潜在或确定线粒体靶向活性的化合物,以促进针对线粒体的药物研究;

化合物库

线粒体靶向库
Cat.No: L5300
Compounds: 812
Cat. No. Product Name Target Signaling Pathways
TQ0146 Ac-DEVD-CHO

Apoptosis; Caspase Apoptosis; Proteases/Proteasome
Ac-DEVD-CHO 是一种特异性 Caspase-3 抑制剂(Ki: 230 pM)。Ac-DEVD-CHO在 SLNT 诱导的细胞凋亡中有抑制作用。
TQ0146L Ac-DEVD-CHO acetate

Caspase-3 Inhibitor I,N-acetyl-asp-glu-val-asp-al,Ac-DEVD-CHO acetate (169332-60-9 free base),乙酰基-天冬氨酰-谷氨酰-缬氨酰-天冬氨醛

Caspase Apoptosis; Proteases/Proteasome
Caspase-3 Inhibitor I (N-acetyl-asp-glu-val-asp-al) 是 Caspase-3 的特异性抑制剂。
T41069 CHO-C-PEG2-C-CHO

CHO-C-PEG2-C-CHO

Others Others
CHO-C-PEG2-C-CHO is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.
T21617 MG-115

Z-LL-Nva-CHO

Proteasome Proteases/Proteasome; Ubiquitination
MG-115 (Z-LL-Nva-CHO) 是一种有效且可逆的蛋白酶体抑制剂,对20S 和26S 蛋白酶体的 Ki 值分别为 21 nM 和 35 nM。MG-115 特异性抑制蛋白酶体的胰凝乳蛋白酶样活性,诱导 p53 依赖性细胞凋亡。
T80531 Ac-AAVALLPAVLLALLAP-DEVD-CHO

DEVD-CHO-CPP 32

Caspase Apoptosis; Proteases/Proteasome
DEVD-CHO-CPP 32(Ac-AAVALLPAVLLALLAP-DEVD-CHO)是一种高效且可逆的caspase-3抑制剂。
T80624 Ac-VAD-CHO

Ac-Val-Ala-Asp-CHO

Caspase Apoptosis; Proteases/Proteasome
Ac-VAD-CHO (Ac-Val-Ala-Asp-CHO)是一款caspase抑制剂,能够阻止缺氧细胞内MMP的降解以及细胞色素c的释出。
T39722 CHO-CH2-PEG1-CH2-Boc

CHO-CH2-PEG1-CH2-Boc

Others Others
CHO-CH2-PEG1-CH2-Boc is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.
T78640 Z-LLF-CHO

Z-Leu-Leu-Phe-CHO

Proteasome Proteases/Proteasome; Ubiquitination
Z-LLF-CHO(Z-Leu-Leu-Phe-CHO)为垂体多催化蛋白酶复合物所具有的胰凝乳蛋白酶样活性提供有效抑制,具有Ki值为460 nM。此外,Z-LLF-CHO同样作为NF-κB核转位的抑制剂。
T83205 Ac-DNLD-CHO

Ac-Asp-Asn-Leu-Asp-CHO

Caspase Apoptosis; Proteases/Proteasome
Ac-DNLD-CHO(Ac-Asp-Asn-Leu-Asp-CHO)是一种有效的Caspase-3/7抑制剂,具有较低的IC50(分别为9.89, 245 nM)和Kiapp(分别为0.68、55.7 nM)。该化合物在研究caspase介导的细胞凋亡过程中具有重要应用价值,适用于神经退行性疾病和病毒感染疾病的相关研究。
T2154 MG-132

Z-LLL-al,Z-Leu-Leu-Leu-CHO

Apoptosis; Proteasome; Autophagy Apoptosis; Autophagy; Proteases/Proteasome; Ubiquitination
MG-132 (Z-Leu-Leu-Leu-al) 是一种 26S 蛋白酶体抑制剂 (IC50=100 nM),具有细胞渗透性、可逆性。MG-132 可作为自噬激活剂,可诱导凋亡。
T80735 Z-Gly-Pro-Phe-Leu-CHO

Z-GPFL-CHO

Proteasome Proteases/Proteasome; Ubiquitination
Z-Gly-Pro-Phe-Leu-CHO(Z-GPFL-CHO)是一种具有高选择性和高效率的四肽醛类蛋白酶体抑制剂,优先抑制支链氨基酸(Ki为1.5 µM),对小中性氨基酸的Ki值为2.3 µM,胰凝乳蛋白酶样活性的Ki值为40.5 µM,对肽基-谷氨酰肽水解活性的IC50为3.1 µM。
T78586L Ac-IETD-CHO TFA

Ac-IETD-CHO TFA(191338-86-0 Free base )

Apoptosis; Caspase Apoptosis; Proteases/Proteasome
Ac-IETD-CHO TFA 是一种 granzyme B 和 caspase-8 抑制剂,通过阻断 caspase3 前体裂解抑制 caspase8 活性。Ac-IETD-CHO TFA 抑制 Fas 介导的细胞凋亡(Apoptosis)。
T41236 Z-FY-CHO

Others Others
Z-FY-CHO (Z-Phe-Tyr-CHO) 是一种特异且有效的组织蛋白酶 L (CTSL) 抑制剂。
T36350 Cho-Arg (trifluoroacetate salt)

Others Others
Cho-Arg is a steroid-based cationic lipid that contains a cholesterol skeleton coupled to an L-arginine head group. It forms a complex with plasmid DNA and decreases plasmid DNA migration in an agarose-gel retardant assay at charge ratios greater than or equal to 4. Cho-Arg facilitates transfection of plasmid DNA into H1299 and HeLa cells in the presence or absence of fetal bovine serum, an effect that is reversed by the lipid raft-mediated endocytosis inhibitor methyl-β-cyclodextrin and the cav...
T36368 2H-Cho-Arg (trifluoroacetate salt)

Others Others
2H-Cho-Arg is a steroid-based cationic lipid that contains a 2H-cholesterol skeleton coupled to an L-arginine head group and can be used to facilitate gene transfection. It forms a complex with plasmid DNA (pDNA) and decreases pDNA migration in an electrophoretic mobility shift assay at +/- charge ratios of 4 or higher. 2H-Cho-Arg facilitates transfection of a luciferase gene into H1299 cells, an effect that is reversed by the lipid raft-mediated endocytosis inhibitor methyl-β-cyclodextrin and t...
T29233 Z-LLNle-CHO

Z-LLNle-CHO is a cell permeable inhibitor of gamma-secretase. Z-LLNle-CHO induces apoptosis of human glioblastoma tumor-initiating cells by proteasome inhibition and mitotic arrest response.
T6583 MG-101

ALLN,Ac-LLnL-CHO,Calpain inhibitor I,Calpain inhibitor-1,MG101,钙蛋白酶抑制剂I

Cysteine Protease; Proteasome Proteases/Proteasome; Ubiquitination
MG-101 (Calpain inhibitor I) 是一种有效的半胱氨酸蛋白酶抑制剂,能够抑制钙蛋白酶I (Ki:190 pM),钙蛋白酶II (Ki:220 pM),组织蛋白酶B (Ki:150 pM)和组织蛋白酶L (Ki:500 pM)。
T19883 Ac-YVAD-CHO

L 709049,L-709049,L709049

L 709049是一种生物活性化合物,它是白细胞介素-1β转化酶( Caspase-1)的选择性抑制剂。 Caspase 抑制剂可干扰细胞凋亡的启动,具有多种临床应用前景。
T80513 YVAD-CHO

YVAD-CHO为白细胞介素-1β转换酶(ICE,caspase 1)的抑制剂,能够在一定程度上减缓面神经损伤小鼠运动神经元死亡速率。
T17281 Z-Ile-Leu-aldehyde

Z-IL-CHO,GSI-XII,γ-Secretase inhibitor XII

Others Others
Z-Ile-Leu-aldehyde is an effective and competitive peptide aldehyde inhibitor of γ-secretase and notch.
T38240 2,6-Dichlorodiphenylamine

Antibacterial Microbiology/Virology
2,6-Dichlorodiphenylamine 是双氯芬酸钠的一种结构类似物,显示出抗白色念珠菌活性。2,6-Dichlorodiphenylamine 是非选择性抗炎剂,为COX 的抑制剂,在 CHO 细胞中,对人 COX-1 和 COX-2 的IC50分别为 4 和 1.3 nM。
T80093 IETD-CHO TFA

Caspase Apoptosis; Proteases/Proteasome
IETD-CHO TFA (Caspase-8-IN-1) 是一种高效的 caspase-8 抑制剂。
T80076 Ac-ESMD-CHO

Casein Kinase Metabolism; Stem Cells
Ac-ESMD-CHO是一种抑制caspase-3和caspase-7的化合物。该化合物能有效阻止caspase-3前体肽(CPP32)在Glu-Ser-Met-Asp(ESMD)位点发生的蛋白水解切割作用。
T78586 Ac-​IETD-​CHO

Apoptosis Apoptosis
Ac-IETD-CHO是一种针对granzyme B和caspase 8的有效可逆抑制剂,能够阻止Fas介导的(Apoptosis)、出血和肝衰竭,并且能够抑制细胞毒性T淋巴细胞引发的细胞死亡。
T80467 Boc-AEVD-CHO

Caspase Apoptosis; Proteases/Proteasome
Boc-AEVD-CHO是一种Caspase 8抑制剂,适用于细胞凋亡以及免疫和炎症疾病研究。
T78622 Ac-VDVAD-CHO

Casein Kinase Metabolism; Stem Cells
Ac-VDVAD-CHO为caspase-2/3抑制剂,其IC50值分别为46 nM和15 nM。
T8566 AA92593

Others Others
AA92593 是一种选择性的 OPN4 (melanopsin)竞争性拮抗剂。
T3306 PF-04418948

PF 04418948,PF04418948

Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
PF-04418948 是一种可口服的,选择性的前列腺素EP2受体拮抗剂,IC50为16 nM。
T80537 Ac-AAVALLPAVLLALLAP-LEHD-CHO

Caspase Apoptosis; Proteases/Proteasome
Ac-AAVALLPAVLLALLAP-LEHD-CHO 是半胱天冬酶4、5和9的抑制剂,能够对Neocarzinostatin处理的MCF-7细胞展现保护效果。
T78619 Z-Pro-Pro-CHO

Prolyl Endopeptidase (PREP) Metabolism; Proteases/Proteasome
Z-Pro-Pro-CHO为一种有效的脯氨酰寡肽酶抑制剂,其具有针对人类及曼氏血吸虫脯氨酰寡肽酶的较低半抑制浓度(IC50),分别为0.16 μM和0.01 μM。
T80532 Ac-AAVALLPAVLLALLAP-YVAD-CHO

Caspase Apoptosis; Proteases/Proteasome
Ac-AAVALLPAVLLALLAP-YVAD-CHO为具备细胞穿透能力的caspase-1抑制剂,展现出抗肿瘤活性。
T73852 Ac-YVAD-CHO acetate

Others Others
Ac-YVAD-CHO(L-709049)醋酸盐是一种高效、可逆、特异的四肽白介素1β转化酶(ICE)抑制剂,小鼠和人类的Ki值分别为3.0 nM和0.76 nM。它同时也能抑制caspase-1,从而抑制成熟IL-lβ的产生。
T80536 Ac-AAVALLPAVLLALLAP-LEVD-CHO

Caspase Apoptosis; Proteases/Proteasome
Ac-AAVALLPAVLLALLAP-LEVD-CHO是一caspase-4抑制剂,可穿透细胞膜,并表现出抗肿瘤特性。
T73683 AC-VEID-CHO TFA

AC-VEID-CHO (TFA) 是一种源自多肽的半胱天冬酶抑制剂,针对Caspase-6、Caspase-3和Caspase-7展示出优异的抑制效果,其IC50值分别为16.2 nM、13.6 nM和162.1 nM。该化合物常用于研究阿尔茨海默病、亨廷顿病等神经退行性疾病。
T0432 Diclofenac diethylamine

Apoptosis; COX Apoptosis; Immunology/Inflammation; Neuroscience
Diclofenac diethylamine 是非选择性抗炎剂,通过活化 caspase 级联反应来诱导神经干细胞凋亡。它是一种COX 抑制剂,在 CHO 细胞中,对人COX-1和COX-2的IC50值分别为 4 和 1.3 nM。它对绵羊COX-1和COX-2的IC50值分别为 5.1 μM 和0.84 μM。
T1671 Mirabegron

YM178,米拉贝隆

Adrenergic Receptor GPCR/G Protein; Neuroscience
Mirabegron (YM178) 是选择性的肾上腺素受体激动剂,EC50=22.4 nM。
T9927 Panitumumab

EGFR Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Panitumumab 是一种重组全人源 IgG2 单克隆抗体,可与表皮生长因子(EGFR)结合,具有抗肿瘤活性。
T8991 BMS986187

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
BMS986187 是一种有效的δ-阿片受体选择性正变构调节剂 (PAM),其 EC50= 0.03 μM,pKB= 6.02 (~1 μM)。BMS986187 对 μ 受体无明显 PAM 活性 (EC50=3 μM)。
T2667 PIK-75

Apoptosis; DNA-PK; PI3K Apoptosis; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
PIK75 是一种可逆的DNA-PK 和p110α-选择性的抑制剂,抑制 DNA-PK、p110α 和 p110γ,IC50分别为 2、5.8 和 76 nM。它诱导凋亡,抑制 p110α 效果比抑制 p110β 高 200 多倍,p110β的IC50为 1.3 μM。
T6470 Diclofenac Potassium

双氯芬酸钾,CGP-45840B,Cataflam,Voltfast

Apoptosis; Others; COX Apoptosis; Immunology/Inflammation; Neuroscience; Others
Diclofenac Potassium (CGP-45840B) 是一种非甾体抗炎药,用于减轻炎症并在某些情况下作为镇痛剂减轻疼痛。它通过活化 caspase 级联反应来诱导神经干细胞凋亡。它是一种COX 抑制剂,在 CHO 细胞中,对人 COX-1 和 COX-2 的IC50值分别为 4 和 1.3 nM。它对绵羊 COX-1 和 COX-2 的IC50值分别为 5.1 μM 和0.84 μM。
T1555 Diclofenac sodium

GP 45840,双氯芬酸钠

Apoptosis; COX Apoptosis; Immunology/Inflammation; Neuroscience
Diclofenac sodium (GP 45840) 是一种非选择性抗炎剂,是 COX 抑制剂,在 CHO 细胞中,对人 COX-1 和 COX-2 的 IC50值分别为 4 和 1.3 nM。它对绵羊 COX-1 和 COX-2 的 IC50值分别为 5.1 μM,0.84 μM。它通过活化 caspase 级联反应来诱导神经干细胞凋亡。
T0196 Diclofenac

双氯芬酸,奥尔芬,Diclofenacum,Voltaren

Apoptosis; COX Apoptosis; Immunology/Inflammation; Neuroscience
Diclofenac (Diclofenacum) 是一种具有抗炎活性的非甾体苯乙酸衍生物,是 COX 抑制剂,在 CHO 细胞中,对人 COX-1 和 COX-2 的 IC50值分别为 4 和 1.3 nM。它对绵羊 COX-1 和 COX-2 的 IC50值分别为 5.1 μM,0.84 μM。它通过活化 caspase 级联反应来诱导神经干细胞凋亡。
T1566 Aripiprazole

阿立哌唑,OPC-14597

5-HT Receptor GPCR/G Protein; Neuroscience
Aripiprazole (OPC-14597) 是血清素受体 5-HT1A 和多巴胺 D2 受体的部分激动剂,还用作突触后拮抗剂和血清素受体 5-HT2A 的拮抗剂。
T6905 Netupitant

Ro 67-31898/000,奈妥吡坦,CID 6451149

Neurokinin receptor GPCR/G Protein; Neuroscience
Netupitant (CID 6451149) 是一种高效选择性、可口服的神经激肽 1 受体 (NK1) 拮抗剂,具有止吐作用,在 CHO 细胞中对 hNK1的 Ki 值为 0.95 nM。
T6140 SB-334867 free base

SB334867A free base,SB-334867,SB 334867,SB334867

OX Receptor GPCR/G Protein; Neuroscience
SB-334867 free base (SB334867A free base) 是一种选择性 orexin-1(OX1) 受体拮抗剂,对 OX2有选择性,pKb 为7.4,对 5-HT2B、5-HT2C 的选择性是 100 倍,pKi 值分别为 5.4 和 5.3。它减少乙醇消耗,还抑制吗啡诱导的体内运动活动敏感性的获得。
T23386 SR 142948

Neurotensin Receptor GPCR/G Protein
SR 142948 是一种神经降压素 (NT) 受体拮抗剂。
T2287 PIK-75 hydrochloride

PIK-75 HCl,2-甲基-5-硝基苯磺酸 [(6-溴咪唑并[1,2-a]吡啶-3-基)亚甲基]甲基肼盐酸盐,PIK-75

Apoptosis; DNA-PK; PI3K Apoptosis; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
PIK-75 hydrochloride (PIK-75 HCl) 是一种可逆的 DNA-PK 和 p110α-选择性抑制剂,抑制 DNA-PK,p110α和 p110γ,可诱导凋亡。
TP2500 Cholecystokinin (26-33) free acid

CCK (26-33) free acid

cholecystokinin GPCR/G Protein
Cholecystokinin (26-33) free acid 是胆囊收缩素 (CCK) 的一部分, 是脊椎动物中枢神经系统中存在的 CCKB 型受体的高选择性配体,可诱导大鼠轻度味觉厌恶条件反射。
T35941 DC-Chol hydrochloride

Cholesteryl 3β-N-(dimethylaminoethyl)carbamate hydrochloride,DC-Chol (hydrochloride),DC-Cholesterol hydrochloride,​Cholesteryl 3β-N-(dimethylaminoethyl)carbamate

Beta Amyloid Neuroscience
DC-Chol hydrochloride(DC-Cholesterol hydrochloride) 在适当的实验条件下能抑制 Aβ40 纤维的形成且以剂量依赖性的方式显著抑制氧化hCT的淀粉样蛋白形成。DC-Chol hydrochloride可诱导改善和平衡的免疫力,能够促进乙型肝炎疫苗的研究。
T2227 Hemicholinium 3

半胆碱基-3,Hemicholinium-3,Hemicholine

Others; AChE Neuroscience; Others
Hemicholinium 3 是一种竞争性的、高亲和力的胆碱转运蛋白 (HACU) 抑制剂,Ki=25 nM。它是一种神经肌肉阻滞剂,能够抑制乙酰胆碱 (ACh)的合成和释放。它抑制Epibatidine 诱发的收缩和 [3H] 乙酰胆碱释放,IC50分别为 897 nM 和 693 nM。

化合物

Ac-DEVD-CHO
Cat.No: TQ0146
Synonym:
Target: Apoptosis, Caspase
Ac-DEVD-CHO acetate
Cat.No: TQ0146L
Synonym: Caspase-3 Inhibitor I,N-acetyl-asp-glu-val-asp-al,Ac-DEVD-CHO acetate (169332-60-9 free base),乙酰基-天冬氨酰-谷氨酰-缬氨酰-天冬氨醛
Target: Caspase
CHO-C-PEG2-C-CHO
Cat.No: T41069
Synonym: CHO-C-PEG2-C-CHO
Target: Others
MG-115
Cat.No: T21617
Synonym: Z-LL-Nva-CHO
Target: Proteasome
Ac-AAVALLPAVLLALLAP-DEVD-CHO
Cat.No: T80531
Synonym: DEVD-CHO-CPP 32
Target: Caspase
Ac-VAD-CHO
Cat.No: T80624
Synonym: Ac-Val-Ala-Asp-CHO
Target: Caspase
CHO-CH2-PEG1-CH2-Boc
Cat.No: T39722
Synonym: CHO-CH2-PEG1-CH2-Boc
Target: Others
Z-LLF-CHO
Cat.No: T78640
Synonym: Z-Leu-Leu-Phe-CHO
Target: Proteasome
Ac-DNLD-CHO
Cat.No: T83205
Synonym: Ac-Asp-Asn-Leu-Asp-CHO
Target: Caspase
MG-132
Cat.No: T2154
Synonym: Z-LLL-al,Z-Leu-Leu-Leu-CHO
Target: Apoptosis, Proteasome, Autophagy
Z-Gly-Pro-Phe-Leu-CHO
Cat.No: T80735
Synonym: Z-GPFL-CHO
Target: Proteasome
Ac-IETD-CHO TFA
Cat.No: T78586L
Synonym: Ac-IETD-CHO TFA(191338-86-0 Free base )
Target: Apoptosis, Caspase
Z-FY-CHO
Cat.No: T41236
Synonym:
Target: Others
Cho-Arg (trifluoroacetate salt)
Cat.No: T36350
Synonym:
Target: Others
2H-Cho-Arg (trifluoroacetate salt)
Cat.No: T36368
Synonym:
Target: Others
Z-LLNle-CHO
Cat.No: T29233
Synonym:
Target:
MG-101
Cat.No: T6583
Synonym: ALLN,Ac-LLnL-CHO,Calpain inhibitor I,Calpain inhibitor-1,MG101,钙蛋白酶抑制剂I
Target: Cysteine Protease, Proteasome
Ac-YVAD-CHO
Cat.No: T19883
Synonym: L 709049,L-709049,L709049
Target:
YVAD-CHO
Cat.No: T80513
Synonym:
Target:
Z-Ile-Leu-aldehyde
Cat.No: T17281
Synonym: Z-IL-CHO,GSI-XII,γ-Secretase inhibitor XII
Target: Others
2,6-Dichlorodiphenylamine
Cat.No: T38240
Synonym:
Target: Antibacterial
IETD-CHO TFA
Cat.No: T80093
Synonym:
Target: Caspase
Ac-ESMD-CHO
Cat.No: T80076
Synonym:
Target: Casein Kinase
Ac-​IETD-​CHO
Cat.No: T78586
Synonym:
Target: Apoptosis
Boc-AEVD-CHO
Cat.No: T80467
Synonym:
Target: Caspase
Ac-VDVAD-CHO
Cat.No: T78622
Synonym:
Target: Casein Kinase
AA92593
Cat.No: T8566
Synonym:
Target: Others
PF-04418948
Cat.No: T3306
Synonym: PF 04418948,PF04418948
Target: Prostaglandin Receptor
Ac-AAVALLPAVLLALLAP-LEHD-CHO
Cat.No: T80537
Synonym:
Target: Caspase
Z-Pro-Pro-CHO
Cat.No: T78619
Synonym:
Target: Prolyl Endopeptidase (PREP)
Ac-AAVALLPAVLLALLAP-YVAD-CHO
Cat.No: T80532
Synonym:
Target: Caspase
Ac-YVAD-CHO acetate
Cat.No: T73852
Synonym:
Target: Others
Ac-AAVALLPAVLLALLAP-LEVD-CHO
Cat.No: T80536
Synonym:
Target: Caspase
AC-VEID-CHO TFA
Cat.No: T73683
Synonym:
Target:
Diclofenac diethylamine
Cat.No: T0432
Synonym:
Target: Apoptosis, COX
Mirabegron
Cat.No: T1671
Synonym: YM178,米拉贝隆
Target: Adrenergic Receptor
Panitumumab
Cat.No: T9927
Synonym:
Target: EGFR
BMS986187
Cat.No: T8991
Synonym:
Target: Opioid Receptor
PIK-75
Cat.No: T2667
Synonym:
Target: Apoptosis, DNA-PK, PI3K
Diclofenac Potassium
Cat.No: T6470
Synonym: 双氯芬酸钾,CGP-45840B,Cataflam,Voltfast
Target: Apoptosis, Others, COX
Diclofenac sodium
Cat.No: T1555
Synonym: GP 45840,双氯芬酸钠
Target: Apoptosis, COX
Diclofenac
Cat.No: T0196
Synonym: 双氯芬酸,奥尔芬,Diclofenacum,Voltaren
Target: Apoptosis, COX
Aripiprazole
Cat.No: T1566
Synonym: 阿立哌唑,OPC-14597
Target: 5-HT Receptor
Netupitant
Cat.No: T6905
Synonym: Ro 67-31898/000,奈妥吡坦,CID 6451149
Target: Neurokinin receptor
SB-334867 free base
Cat.No: T6140
Synonym: SB334867A free base,SB-334867,SB 334867,SB334867
Target: OX Receptor
SR 142948
Cat.No: T23386
Synonym:
Target: Neurotensin Receptor
PIK-75 hydrochloride
Cat.No: T2287
Synonym: PIK-75 HCl,2-甲基-5-硝基苯磺酸 [(6-溴咪唑并[1,2-a]吡啶-3-基)亚甲基]甲基肼盐酸盐,PIK-75
Target: Apoptosis, DNA-PK, PI3K
Cholecystokinin (26-33) free acid
Cat.No: TP2500
Synonym: CCK (26-33) free acid
Target: cholecystokinin
DC-Chol hydrochloride
Cat.No: T35941
Synonym: Cholesteryl 3β-N-(dimethylaminoethyl)carbamate hydrochloride,DC-Chol (hydrochloride),DC-Cholesterol hydrochloride,​Cholesteryl 3β-N-(dimethylaminoethyl)carbamate
Target: Beta Amyloid
Hemicholinium 3
Cat.No: T2227
Synonym: 半胆碱基-3,Hemicholinium-3,Hemicholine
Target: Others, AChE
Cat. No. Product Name Target Signaling Pathways
T5214 Cholesteryl linoleate

CE(18:2(9Z,12Z)),Cholesterol Linoleate,Linoleic Acid cholesteryl ester,胆甾烯基亚油酸酯

Others; Endogenous Metabolite Metabolism; Others
Cholesteryl linoleate 是低密度脂蛋白和动脉粥样硬化病变中主要的胆固醇酯。它存在于 LDL 中的胆固醇酯,利用 LDL 受体相关蛋白转移到表达 15-脂氧合酶的巨噬细胞和 CHO 细胞的质膜,被氧化形成胆固醇亚油酸氢过氧化物。
T2968 Hyodeoxycholic acid

NSC 60672,猪去氧胆酸,α-Hyodeoxycholic Acid,HDCA

FXR; Endogenous Metabolite; GPCR19 GPCR/G Protein; Metabolism
Hyodeoxycholic acid (NSC 60672) 是由肠道菌群在小肠中形成的次级胆汁酸,是TGR5(GPCR19)的激动剂, CHO 细胞中的EC50=31.6 µM。它已用于研究高胆固醇血症的治疗。
T7628 3b-Hydroxy-5-cholenoic acid

Endogenous Metabolite Metabolism
3b-Hydroxy-5-cholenoic acid 是内源性的单羟基胆酸的一种,大量崔乃在于患有肝胆管状发育不全的儿童体内。
TN2215 Taurochenodeoxycholic acid sodium

牛磺鹅去氧胆酸钠盐,Sodium taurochenodeoxycholate,牛磺鹅去氧胆酸钠

Apoptosis; Endogenous Metabolite Apoptosis; Metabolism
Taurochenodeoxycholic acid sodium (Sodium taurochenodeoxycholate) 是动物胆汁酸的主要生物活性物质之一。它可诱导细胞凋亡,具有抗炎和免疫调节作用。
T3742 3-Methylcatechol

3-甲基苯邻二酚,3-Methylpyrocatechol,2,3-Toluenediol,3-甲基邻苯二酚,2,3-dihydroxytoluene

Others Others
3-Methylcatechol (2,3-Toluenediol) 是由 Pseudomonas putidaMC2 产生,能够用作化学合成中的分子砌块。
T19124 3-​Oxocholic acid

3-Ketocholic acid

Endogenous Metabolite Metabolism
3-​Oxocholic acid(3-Ketocholic acid) 是胆汁酸的代谢产物,也是产气荚膜梭菌在肠道中由胆汁降解的主要产物。33-​Oxocholic acid 是一种主要存在于哺乳动物的胆汁中类固醇酸。
TN2349 Taurodeoxycholate sodium salt

Sodium taurodeoxylate,牛磺脱氧胆酸钠

Endogenous Metabolite Metabolism
Taurodeoxycholate sodium salt (Sodium taurodeoxylate) 是胆盐相关的阴离子洗涤剂,用于分离膜蛋白,包括线粒体内膜蛋白。它还可以抑制各种炎症反应。
T40646 Lipoteichoic acid

Complement System Immunology/Inflammation
Lipoteichoic acid 是 Staphylococcus aureus 细胞壁的聚合物,通过诱导 C3 和抑制 CD55 来激活补体系统,通过 IGF-1 途径减少脂肪沉积。
T6805 Choline bitartrate

2,3,4-trihydroxy-4-oxobutanoate,2-hydroxyethyl(trimethyl)azanium,酒石酸氢胆碱

Others; AChR Neuroscience; Others
Choline bitartrate (2-hydroxyethyl(trimethyl)azanium) 是一种存在于食物中的营养胆碱,可影响肝脏疾病、动脉粥样硬化和神经系统疾病等疾病。它是神经递质乙酰胆碱的前体,作为甲基供体参与各种代谢过程和脂质代谢。
T6751 Acetylcholine iodide

Acetylcolina

Others Others
Acetylcholine iodide (Acetylcolina) 是一种在中枢和外周神经系统中常见的神经递质。
TN3651 Cichoriin

Others Others
Cichoriin 对SARS-CoV-2有明显活性,是治疗重症COVID-19的潜在候选物质。
T4717 25-Hydroxycholesterol

25-羟基胆固醇,25-羟基胆甾醇

Others; Endogenous Metabolite; HMG-CoA Reductase Metabolism; Others
25-Hydroxycholesterol 是胆固醇的代谢产物,由巨噬细胞响应 Toll 样受体激活而分泌。它有效抑制 B 细胞产生 IgA,EC50约为 65 nM。
T5240 Cholestenone

胆甾烯酮,4-胆甾烯-3-酮,(+)-4-Cholesten-3-one

Others; Endogenous Metabolite Metabolism; Others
Cholestenone 是胆固醇的中间氧化产物,主要在肝脏中代谢。它能够会导致细胞长期功能缺陷。它在膜中具有很高的流动性,会影响胆固醇的翻转和外排。
T2962 5α-Cholestan-3β-ol

Dihydrocholesterol,Zymostanol,5α-Cholestanol,5alpha-Cholestanol,NSC 18188,Beta-Cholestanol,二氢胆甾醇

Others; Endogenous Metabolite Metabolism; Others
Dihydrocholesterol 是衍生化的类固醇化合物的一种,抑制胆固醇吸收。
TJA2398 Taurodeoxycholic acid sodium hydrate

Sodium taurodeoxycholate monohydrate,Taurodeoxychloic Acid sodium hydrate,Taurohyodeoxycholic acid sodium salt,牛磺猪去氧胆酸

Apoptosis; Caspase Apoptosis; Proteases/Proteasome
Taurodeoxycholic acid sodium hydrate (Sodium taurodeoxycholate monohydrate) 通过阻断钙介导的凋亡通路和 Caspase-12的活化来阻止细胞凋亡。它可用于原发性胆汁性肝硬化、胰岛素抵抗、淀粉样变性、囊性纤维化、胆汁淤积和肌萎缩侧索硬化症。
T2S0142 4-Hydroxylonchocarpin

异补骨脂色烯查耳酮,Isobavachromene

Others Others
Isobavachromene is a natural product from Psoralea corylifolia
T5077 Deoxycholic acid sodium salt

脱氧胆酸钠,Sodium deoxycholate,Sodium Desoxycholate

Endogenous Metabolite; GPCR19 GPCR/G Protein; Metabolism
Deoxycholic acid sodium salt (Sodium deoxycholate) 是 G 蛋白偶联胆汁酸受体TGR5的激活剂。
T9510 1,2-Distearoyl-sn-glycero-3-phosphorylcholine

DSPC,L-ALPHA-PHOSPHATIDYLCHOLINE, DISTEAROYL,1,2-Distearoyl-sn-glycero-3-PC,二硬脂酰磷脂酰胆碱

Others Others
1,2-Distearoyl-sn-glycero-3-phosphorylcholine (L-ALPHA-PHOSPHATIDYLCHOLINE, DISTEAROYL) 是一种脂质纳米颗粒(LNP) 系统中的脂质成分,可用于合成脂质体。
T4136 Lapachol

Bethabarra wood,CI75490,黄钟花醌,Greenhartin,Tecomin

Others; Influenza Virus; Antibacterial; Parasite; Antifungal Microbiology/Virology; Others
Lapachol (CI75490) 是从Tabebuia avellanedae 中分离得到的一种萘醌。它具有具有抗菌、抗炎、镇痛、抗肿瘤和抗生素特性。
T4727 Taurolithocholic acid sodium salt

牛磺石胆酸钠,Sodium taurolithocholate

Others; Calcium Channel Membrane transporter/Ion channel; Metabolism; Others
Taurolithocholic acid sodium salt (Sodium taurolithocholate) 是抑胆剂和 Ca2+激动剂,可抑制放射性配体与毒蕈碱 M1 结合。
T75319 Taurodeoxycholic acid

Taurodeoxychloic acid

Apoptosis; Calcium Channel; Caspase Apoptosis; Membrane transporter/Ion channel; Metabolism; Proteases/Proteasome
Taurodeoxycholic acid (Taurodeoxychloic acid) 是脱氧胆酸的胆汁酸牛磺酸共轭物,是一种人体代谢物,可稳定线粒体膜,减少自由基形成。Taurodeoxycholic acid 通过阻断钙介导的凋亡通路以及 Caspase-12 激活来抑制凋亡 (apoptosis)。Taurodeoxycholic acid具有神经保护活性,可用于研究 3-硝基丙酸诱导或稳定遗传的亨廷顿舞蹈病 (HD) 。
T1317 Cinchonidine

奎宁树,α-Quinidine,辛可尼丁,L-Cinchonidine

5-HT Receptor; Serotonin Transporter; Parasite GPCR/G Protein; Microbiology/Virology; Neuroscience
Cinchonidine (L-Cinchonidine) 是在金鸡纳和角蒿中发现的一种生物碱,有抗疟活性。 它是用于有机化学中不对称合成的砌块,是血清素转运蛋白的弱抑制剂。
TQ0274 27-Hydroxycholesterol

27-羟基胆固醇,5,25R-胆甾烯-3BETA,26-二醇,25(R)-27-hydroxy Cholesterol

Estrogen/progestogen Receptor; Liver X Receptor Endocrinology/Hormones; Metabolism
27-Hydroxycholesterol (25(R)-27-hydroxy Cholesterol) 是一种有效的、选择性的雌激素受体调节剂和肝X 受体激动剂。
T6S0659 Rhynchophylline

钩藤碱,Rhynchophyllin,Rhyncophylline,Mitrinermine,Mitrinermin

Calcium Channel; NF-κB Membrane transporter/Ion channel; Metabolism; NF-κB
Rhynchophylline (Mitrinermine) 是一种生物碱类化合物,从钩藤中分离得到,具有很高的生物活性,被广泛用于抗炎、神经保护等方面的研究。
T4713 Phosphorylcholine chloride calcium salt tetrahydrate

Phosphocholine chloride calcium salt tet,胆碱磷酸氯化钙四水,CalciuM Phosphorylcholine Tetrahydrate

Others; Endogenous Metabolite Metabolism; Others
Phosphorylcholine chloride calcium salt tetrahydrate (Phosphocholine chloride calcium salt tet) 是内源性代谢产物的一种。
T5072 Glycocholic acid hydrate

Others; Endogenous Metabolite Metabolism; Others
Glycocholic acid hydrate 是内源性代谢产物的一种。
T8712 1-Palmitoyl-sn-glycero-3-phosphocholine

1-十六酰-SN-丙三醇-磷酸胆碱,1-Hexadecanoyl-sn-glycero-3-phosphocholine

Others Others
1-Palmitoyl-sn-glycero-3-phosphocholine (1-Hexadecanoyl-sn-glycero-3-phosphocholine) 是一种用于荧光探针设计的磷酸胆碱。
T10085 20(S)-Hydroxycholesterol

20α-Hydroxycholesterol

Smo Stem Cells
20(S)-Hydroxycholesterol (20α-Hydroxycholesterol) 是平滑 (smo) 癌蛋白的变构激活剂。
T19189 Allocholic acid

Others Others
Allocholic acid 是一种胆汁酸,在脊椎动物中发现,在肝脏再生和致癌过程中会重新出现,也是成熟嗅觉系统的特定性刺激物。
T8714 1-Stearoyl-sn-glycero-3-phosphocholine

1-硬脂酰-SN-甘油-3-磷酰胆碱,1-stearoyl-lysophosphatidylcholine,L-ALPHA-LYSOPHOSPHATIDYLCHOLINE, STEAROY

Others Others
1-Stearoyl-sn-glycero-3-phosphocholine (L-ALPHA-LYSOPHOSPHATIDYLCHOLINE, STEAROY) 是一种用于脂质代谢研究的化学物质。
T2965 Deoxycholic acid

Cholorebic,去氧胆酸,脱氧胆酸,Deoxycholate,Desoxycholic acid,Cholanoic Acid,Cholerebic

Endogenous Metabolite; GPCR19 GPCR/G Protein; Metabolism
Deoxycholic acid (Cholanoic Acid) 是 G 蛋白偶联胆汁酸受体 TGR5的激活剂。
TN7235 4-methoxylonchocarpin

TNF; NF-κB Apoptosis; NF-κB
4-methoxylonchocarpin 是从Abrus precatorius 的根中分离出来的以一种有效的抗炎化合物。4-methoxylonchocarpin 通过抑制LPS 与巨噬细胞的TLR4结合来抑制NF-κB 激活TNF 表达,抑制TNBS 引起的小鼠结肠炎。
T13505 3α,12β-Dihydroxycholanoic acid

Lagodeoxycholic acid

Endogenous Metabolite Metabolism
3α,12β-Dihydroxycholanoic acid (Lagodeoxycholic acid) 是一种广泛存在于动物体内的胆汁酸。
T0760 Cholesterol

Cholesterin,Cholesteryl alcohol,胆固醇

Estrogen Receptor/ERR; MRP; Endogenous Metabolite; ROR Endocrinology/Hormones; Immunology/Inflammation; Metabolism
Cholesterol (Cholesteryl alcohol) 属于天然产物,是哺乳动物中的主要固醇,是一种雌激素相关受体 α (ERRα) 的激动剂。Cholesterol 广泛存在于动物的细胞膜,也是合成几种重要荷尔蒙及胆酸的材料。
T5352 GLYCODEOXYCHOLIC ACID

Others; Endogenous Metabolite Metabolism; Others
Glycodeoxycholic Acid 是内源性代谢产物的一种,是一种存在于黑链霉菌、布氏锥虫和隐单胞菌中的天然产物,可诱导阻塞性胆汁淤积症患者的肝细胞坏死和自噬。
T2744 Methyl Cholate

胆酸甲酯,Cholic acid methyl ester

Others Others
Methyl Cholate 是胆酸的甲酯形式。其中胆酸是一种由肝脏产生的主要胆汁酸,由胆固醇合成。Methyl Cholate 具有抗炎抗肿瘤活性。
T31964 Glycolithocholic acid

Lithocholic acid glycine conjugate,甘氨石胆酸,Lithocholylglycine

Endogenous Metabolite Metabolism
Glycolithocholic acid (Lithocholic acid glycine conjugate) 属于内源性代谢产物,是甘氨酸结合的次级胆汁酸。它可用于诊断非酒精性脂肪性肝炎,溃疡性结肠炎和原发性硬化性胆管炎。
T2963 Cholic Acid

Cholanic acid,胆汁酸,Cholate,Colalin

Endogenous Metabolite Metabolism
Cholic Acid (Cholate) 是肝脏产生的主要胆汁酸,与牛磺酸或甘氨酸缀合,有助于脂肪吸收和胆固醇排泄。
TN7024 Hyocholic acid

Others Others
Hyocholic acid 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN7024,CAS号为 547-75-1。
T8092 Taurohyodeoxycholic acid sodium salt

Sodium taurohyodeoxycholate hydrate

Caspase Apoptosis; Proteases/Proteasome
Taurohyodeoxycholic acid sodium salt (Sodium taurohyodeoxycholate hydrate) 通过阻断钙介导的细胞凋亡途径以及 Caspase-12 活化来防止细胞凋亡
T74293 Allolithocholic acid

Others Others
Allolithocholic acid 是一种类固醇酸,在正常血清和粪便中可发现。该化合物促进脂肪与甾醇在肠道及肝脏的排泄、吸收与运输。
TN5173 Trichorabdal A

Antifection Microbiology/Virology
Trichorabdal A 是一种二萜化合物,分离自 Rabdosia trichocarpa,抗肿瘤作用强大。
T8040 Cholesterol myristate

胆甾烯基豆蔻酸酯,Cholesteryl myristate,胆固醇肉豆蔻酸,Cholesteryl tetradecanoate

Others; Potassium Channel; GABA Receptor; Endogenous Metabolite; AChR Membrane transporter/Ion channel; Metabolism; Neuroscience; Others
Cholesterol myristate (Cholesteryl myristate) 是粗吻海龙中的一种类固醇,可与多种离子通道结合,例如nAChR、GABAA 受体和内向整流钾离子通道。
T22293 Chondroitine sulfate

Chondroitine sulfate (From cattle)

Others Others
Chondroitine sulfate 是软骨的重要结构成分,已被用作治疗关节不适的膳食补充剂。
T1039 Choline chloride

Biocolina,Biocoline,Hepacholine,氯化胆碱

AChR Neuroscience
Choline chloride (Biocoline) 是一种必需营养素,可激活 α7 烟碱受体,具有抗炎、镇痛的活性。对动脉粥样硬化、神经系统疾病和肝脏疾病等具有影响。
T19161 7α-Hydroxycholesterol

Others Others
7α-Hydroxycholesterol 是一种由酶促氧化和非酶促氧化形成的胆固醇氧化物,可用作脂质过氧化的生物标志物。
T2202 Lithocholic acid

3α-Hydroxy-5β-cholanic acid,石胆酸

Apoptosis; Others; FXR; Endogenous Metabolite; Autophagy Apoptosis; Autophagy; Metabolism; Others
Lithocholic acid (3α-Hydroxy-5β-cholanic acid) 是由鹅去氧胆酸盐通过细菌作用形成的胆汁酸,通常与甘氨酸或牛磺酸结合,被用作利胆剂。 它作为清洁剂溶解脂肪以供吸收,并且本身被吸收。
T5234 Glycoursodeoxycholic acid

Ursodeoxycholylglycine,甘氨熊胆酸,GUDCA

Others; Endogenous Metabolite Metabolism; Others
Glycoursodeoxycholic acid (Ursodeoxycholylglycine) 是一种酰基甘氨酸和胆汁酸-甘氨酸缀合物,是熊去氧胆酸的代谢物。
T4779 4-Methylcatechol

p-Methylcatechol,3,4-二羟基甲苯,Homocatechol,4-methylbenzene-1,2-diol,3,4-Dihydroxytoluene

Others; Endogenous Metabolite Metabolism; Others
4-Methylcatechol (3,4-Dihydroxytoluene) 是 p-toluate 的代谢物,它是 Catechol 2,3-Dioxygenase 的自杀性底物抑制剂。
T1221 Acetylcholine chloride

ACh chloride,Pilofrin,氯化乙酰胆碱

Calcium Channel; Endogenous Metabolite; AChR Membrane transporter/Ion channel; Metabolism; Neuroscience
Acetylcholine chloride (Pilofrin) 是一种神经递质,是胆碱能激动剂,通过刺激烟碱乙酰胆碱受体调节多巴胺能神经元活性,在体外抑制 p53 突变肽的聚集。
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天然产物

Cholesteryl linoleate
Cat.No: T5214
Synonym: CE(18:2(9Z,12Z)),Cholesterol Linoleate,Linoleic Acid cholesteryl ester,胆甾烯基亚油酸酯
Target: Others, Endogenous Metabolite
Hyodeoxycholic acid
Cat.No: T2968
Synonym: NSC 60672,猪去氧胆酸,α-Hyodeoxycholic Acid,HDCA
Target: FXR, Endogenous Metabolite, GPCR19
3b-Hydroxy-5-cholenoic acid
Cat.No: T7628
Synonym:
Target: Endogenous Metabolite
Taurochenodeoxycholic acid sodium
Cat.No: TN2215
Synonym: 牛磺鹅去氧胆酸钠盐,Sodium taurochenodeoxycholate,牛磺鹅去氧胆酸钠
Target: Apoptosis, Endogenous Metabolite
3-Methylcatechol
Cat.No: T3742
Synonym: 3-甲基苯邻二酚,3-Methylpyrocatechol,2,3-Toluenediol,3-甲基邻苯二酚,2,3-dihydroxytoluene
Target: Others
3-​Oxocholic acid
Cat.No: T19124
Synonym: 3-Ketocholic acid
Target: Endogenous Metabolite
Taurodeoxycholate sodium salt
Cat.No: TN2349
Synonym: Sodium taurodeoxylate,牛磺脱氧胆酸钠
Target: Endogenous Metabolite
Lipoteichoic acid
Cat.No: T40646
Synonym:
Target: Complement System
Choline bitartrate
Cat.No: T6805
Synonym: 2,3,4-trihydroxy-4-oxobutanoate,2-hydroxyethyl(trimethyl)azanium,酒石酸氢胆碱
Target: Others, AChR
Acetylcholine iodide
Cat.No: T6751
Synonym: Acetylcolina
Target: Others
Cichoriin
Cat.No: TN3651
Synonym:
Target: Others
25-Hydroxycholesterol
Cat.No: T4717
Synonym: 25-羟基胆固醇,25-羟基胆甾醇
Target: Others, Endogenous Metabolite, HMG-CoA Reductase
Cholestenone
Cat.No: T5240
Synonym: 胆甾烯酮,4-胆甾烯-3-酮,(+)-4-Cholesten-3-one
Target: Others, Endogenous Metabolite
5α-Cholestan-3β-ol
Cat.No: T2962
Synonym: Dihydrocholesterol,Zymostanol,5α-Cholestanol,5alpha-Cholestanol,NSC 18188,Beta-Cholestanol,二氢胆甾醇
Target: Others, Endogenous Metabolite
Taurodeoxycholic acid sodium hydrate
Cat.No: TJA2398
Synonym: Sodium taurodeoxycholate monohydrate,Taurodeoxychloic Acid sodium hydrate,Taurohyodeoxycholic acid sodium salt,牛磺猪去氧胆酸
Target: Apoptosis, Caspase
4-Hydroxylonchocarpin
Cat.No: T2S0142
Synonym: 异补骨脂色烯查耳酮,Isobavachromene
Target: Others
Deoxycholic acid sodium salt
Cat.No: T5077
Synonym: 脱氧胆酸钠,Sodium deoxycholate,Sodium Desoxycholate
Target: Endogenous Metabolite, GPCR19
1,2-Distearoyl-sn-glycero-3-phosphorylcholine
Cat.No: T9510
Synonym: DSPC,L-ALPHA-PHOSPHATIDYLCHOLINE, DISTEAROYL,1,2-Distearoyl-sn-glycero-3-PC,二硬脂酰磷脂酰胆碱
Target: Others
Lapachol
Cat.No: T4136
Synonym: Bethabarra wood,CI75490,黄钟花醌,Greenhartin,Tecomin
Target: Others, Influenza Virus, Antibacterial, Parasite, Antifungal
Taurolithocholic acid sodium salt
Cat.No: T4727
Synonym: 牛磺石胆酸钠,Sodium taurolithocholate
Target: Others, Calcium Channel
Taurodeoxycholic acid
Cat.No: T75319
Synonym: Taurodeoxychloic acid
Target: Apoptosis, Calcium Channel, Caspase
Cinchonidine
Cat.No: T1317
Synonym: 奎宁树,α-Quinidine,辛可尼丁,L-Cinchonidine
Target: 5-HT Receptor, Serotonin Transporter, Parasite
27-Hydroxycholesterol
Cat.No: TQ0274
Synonym: 27-羟基胆固醇,5,25R-胆甾烯-3BETA,26-二醇,25(R)-27-hydroxy Cholesterol
Target: Estrogen/progestogen Receptor, Liver X Receptor
Rhynchophylline
Cat.No: T6S0659
Synonym: 钩藤碱,Rhynchophyllin,Rhyncophylline,Mitrinermine,Mitrinermin
Target: Calcium Channel, NF-κB
Phosphorylcholine chloride calcium salt tetrahydrate
Cat.No: T4713
Synonym: Phosphocholine chloride calcium salt tet,胆碱磷酸氯化钙四水,CalciuM Phosphorylcholine Tetrahydrate
Target: Others, Endogenous Metabolite
Glycocholic acid hydrate
Cat.No: T5072
Synonym:
Target: Others, Endogenous Metabolite
1-Palmitoyl-sn-glycero-3-phosphocholine
Cat.No: T8712
Synonym: 1-十六酰-SN-丙三醇-磷酸胆碱,1-Hexadecanoyl-sn-glycero-3-phosphocholine
Target: Others
20(S)-Hydroxycholesterol
Cat.No: T10085
Synonym: 20α-Hydroxycholesterol
Target: Smo
Allocholic acid
Cat.No: T19189
Synonym:
Target: Others
1-Stearoyl-sn-glycero-3-phosphocholine
Cat.No: T8714
Synonym: 1-硬脂酰-SN-甘油-3-磷酰胆碱,1-stearoyl-lysophosphatidylcholine,L-ALPHA-LYSOPHOSPHATIDYLCHOLINE, STEAROY
Target: Others
Deoxycholic acid
Cat.No: T2965
Synonym: Cholorebic,去氧胆酸,脱氧胆酸,Deoxycholate,Desoxycholic acid,Cholanoic Acid,Cholerebic
Target: Endogenous Metabolite, GPCR19
4-methoxylonchocarpin
Cat.No: TN7235
Synonym:
Target: TNF, NF-κB
3α,12β-Dihydroxycholanoic acid
Cat.No: T13505
Synonym: Lagodeoxycholic acid
Target: Endogenous Metabolite
Cholesterol
Cat.No: T0760
Synonym: Cholesterin,Cholesteryl alcohol,胆固醇
Target: Estrogen Receptor/ERR, MRP, Endogenous Metabolite, ROR
GLYCODEOXYCHOLIC ACID
Cat.No: T5352
Synonym:
Target: Others, Endogenous Metabolite
Methyl Cholate
Cat.No: T2744
Synonym: 胆酸甲酯,Cholic acid methyl ester
Target: Others
Glycolithocholic acid
Cat.No: T31964
Synonym: Lithocholic acid glycine conjugate,甘氨石胆酸,Lithocholylglycine
Target: Endogenous Metabolite
Cholic Acid
Cat.No: T2963
Synonym: Cholanic acid,胆汁酸,Cholate,Colalin
Target: Endogenous Metabolite
Hyocholic acid
Cat.No: TN7024
Synonym:
Target: Others
Taurohyodeoxycholic acid sodium salt
Cat.No: T8092
Synonym: Sodium taurohyodeoxycholate hydrate
Target: Caspase
Allolithocholic acid
Cat.No: T74293
Synonym:
Target: Others
Trichorabdal A
Cat.No: TN5173
Synonym:
Target: Antifection
Cholesterol myristate
Cat.No: T8040
Synonym: 胆甾烯基豆蔻酸酯,Cholesteryl myristate,胆固醇肉豆蔻酸,Cholesteryl tetradecanoate
Target: Others, Potassium Channel, GABA Receptor, Endogenous Metabolite, AChR
Chondroitine sulfate
Cat.No: T22293
Synonym: Chondroitine sulfate (From cattle)
Target: Others
Choline chloride
Cat.No: T1039
Synonym: Biocolina,Biocoline,Hepacholine,氯化胆碱
Target: AChR
7α-Hydroxycholesterol
Cat.No: T19161
Synonym:
Target: Others
Lithocholic acid
Cat.No: T2202
Synonym: 3α-Hydroxy-5β-cholanic acid,石胆酸
Target: Apoptosis, Others, FXR, Endogenous Metabolite, Autophagy
Glycoursodeoxycholic acid
Cat.No: T5234
Synonym: Ursodeoxycholylglycine,甘氨熊胆酸,GUDCA
Target: Others, Endogenous Metabolite
4-Methylcatechol
Cat.No: T4779
Synonym: p-Methylcatechol,3,4-二羟基甲苯,Homocatechol,4-methylbenzene-1,2-diol,3,4-Dihydroxytoluene
Target: Others, Endogenous Metabolite
Acetylcholine chloride
Cat.No: T1221
Synonym: ACh chloride,Pilofrin,氯化乙酰胆碱
Target: Calcium Channel, Endogenous Metabolite, AChR
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Cat. No. Product Name Species Expression System
TMPY-01693 Butyrylcholinesterase Protein, Human, Recombinant (His)

CHE1,E1,butyrylcholinesterase,CHE2

Human HEK293 Cells
Butyrylcholinesterase Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 66.5 kDa and the accession number is P06276.
TMPY-03006 CHODL Protein, Rat, Recombinant (hFc)

chondrolectin

Rat HEK293 Cells
CHODL Protein, Rat, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 48.9 kDa and the accession number is D3ZI86.
TMPY-04905 Zika virus (ZIKV) (strain Zika SPH2016) ZIKV-E (Stem/anchor domain of flavivirus envelope glycoprotein E) protein (Fc)

ZIKV HEK293 Cells
Zika virus (ZIKV) (strain Zika SPH2016) ZIKV-E (Stem/anchor domain of flavivirus envelope glycoprotein E) protein (Fc) is expressed in HEK293 mammalian cells with Fc tag. The predicted molecular weight is 36.7 kDa and the accession number is ALU33341.1.
TMPY-02941 CHODL Protein, Rat, Recombinant (His)

chondrolectin

Rat HEK293 Cells
CHODL Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 23.3 kDa and the accession number is D3ZI86.
TMPY-02408 CHODL Protein, Mouse, Recombinant (His)

3110074E07Rik,MT75,PRED12,chondrolectin

Mouse HEK293 Cells
CHODL Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 23.4 kDa and the accession number is EDK98299.1.
TMPK-01188 CHODL Protein, Human, Recombinant (hFc)

PRED12,C21orf68,CHODL,MT75,Chondrolectin,3...

Human HEK293 Cells
chondrolectin (CHODL) is commonly overexpressed in the majority of lung cancers, indicating a possible correlation between CHODL and metastasis of lung cancer cells. the expression of CHODL is significantly decreased in HCC clinical samples and in HCC cell lines. Overexpression of CHODL in SMMC7721 cells with a lentiviral vector increased SMMC7721 cell migration and invasion.
TMPH-03234 Acetylcholinesterase Protein, Rat, Recombinant (His)

AChE,EC:3.1.1.7

Rat E. coli
Terminates signal transduction at the neuromuscular junction by rapid hydrolysis of the acetylcholine released into the synaptic cleft. Acetylcholinesterase Protein, Rat, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 68.9 kDa and the accession number is P37136.
TMPH-03702 MTA/SAH nucleosidase Protein, Vibrio cholerae serotype O1, Recombinant (His & Myc)

5'-deoxyadenosine nucleosidase,5'-methylthioadenosine nucleo...

Vibrio cholerae E. coli
Catalyzes the irreversible cleavage of the glycosidic bond in both 5'-methylthioadenosine (MTA) and S-adenosylhomocysteine (SAH/AdoHcy) to adenine and the corresponding thioribose, 5'-methylthioribose and S-ribosylhomocysteine, respectively. Also cleaves 5'-deoxyadenosine, a toxic by-product of radical S-adenosylmethionine (SAM) enzymes, into 5-deoxyribose and adenine. MTA/SAH nucleosidase Protein, Vibrio cholerae serotype O1, Recombinant (His & Myc) is expressed in E. coli expression system wit...
TMPH-03703 Zot Protein, Vibrio cholerae serotype O1, Recombinant (His)

Zona occludens toxin,Zonular occludens toxin,zot

Vibrio cholerae E. coli
Increases the permeability of the small intestine mucosa by affecting the structure of intercellular tight junctions (zonula occludens). Zot Protein, Vibrio cholerae serotype O1, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 48.4 kDa and the accession number is P38442.
TMPH-00390 MOMP Protein, Chlamydia trachomatis, Recombinant (His & Myc)

ompA,Major outer membrane porin, serovar B

Chlamydia trachomatis E. coli
In elementary bodies (EBs, the infectious stage, which is able to survive outside the host cell) provides the structural integrity of the outer envelope through disulfide cross-links with the small cysteine-rich protein and the large cysteine-rich periplasmic protein. It has been described in publications as the Sarkosyl-insoluble COMC (Chlamydia outer membrane complex), and serves as the functional equivalent of peptidoglycan.; Permits diffusion of specific solutes through the outer membrane. M...
TMPH-02413 Lymphocytic choriomeningitis virus (LCMV) (strain Armstrong) GPC Protein (His & SUMO)

GPC,Pre-glycoprotein polyprotein GP complex

LCMV E. coli
Lymphocytic choriomeningitis virus (LCMV) (strain Armstrong) GPC Protein (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 42.4 kDa and the accession number is P09991.
TMPH-03644 Hydrophobin-2/HFB2 Protein, Trichoderma reesei, Recombinant (His & SUMOstar)

Hydrophobin-2,hfb2,Hydrophobin II

Hypocrea jecorina P. pastoris (Yeast)
Responsible for spore hydrophobicity and protection. Hydrophobin-2/HFB2 Protein, Trichoderma reesei, Recombinant (His & SUMOstar) is expressed in yeast with N-6xHis-SUMOSTAR tag. The predicted molecular weight is 23.2 kDa and the accession number is P79073.
TMPY-00647 Chorionic Gonadotropin/CGA Protein, Human, Recombinant (His)

CG-α,FSH alpha,glycoprotein hormones, alpha polypeptide,FSHA...

Human HEK293 Cells
Chorionic Gonadotropin/CGA Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 11.6 kDa and the accession number is P01215.
TMPY-02923 Chorionic Gonadotropin/CGA Protein, Human, Recombinant (mFc)

HCG,GPHa,CG-ALPHA,glycoprotein hormones, alpha polypeptide,g...

Human HEK293 Cells
Chorionic Gonadotropin/CGA Protein, Human, Recombinant (mFc) is expressed in HEK293 mammalian cells with mFc tag. The predicted molecular weight is 36.6 kDa and the accession number is P01215.
TMPY-01742 Acetylcholinesterase Protein, Mouse, Recombinant (His)

Acre,Chrne,acetylcholinesterase (Yt blood group)

Mouse HEK293 Cells
Acetylcholinesterase, also known as ACHE, is an enzyme that degrades (through its hydrolytic activity) the neurotransmitter acetylcholine, producing choline and an acetate group. Acetylcholinesterase plays a crucial role in nerve impulse transmission at cholinergic synapses by rapid hydrolysis of the neurotransmitter acetylcholine (ACh). ACHE appears to be a potential therapeutic target at muscle injuries including organophosphate myopathy. It is an externally oriented membrane-bound enzyme and ...
TMPH-03182 DTE Protein, Pseudomonas cichorii, Recombinant (His & Myc)

Ketose 3-epimerase,D-ribulose 3-epimerase,DTE,D-tagatose 3-e...

Pseudomonas cichorii E. coli
Catalyzes the epimerization of various ketoses at the C(3) position. It is able to interconvert D-tagatose and D-ribulose to D-sorbose and D-xylulose, respectively. The enzyme is also able to accept other ketopentoses such as D-psicose with lower efficiency. DTE Protein, Pseudomonas cichorii, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 40.1 kDa and the accession number is O50580.
TMPH-00220 Adrenodoxin, mitochondrial Protein, Bovine, Recombinant (His)

Hepato-ferredoxin,FDX1,Ferredoxin-1,Adrenodoxin, mitocho...

Bovine E. coli
Essential for the synthesis of various steroid hormones. Participates in the reduction of mitochondrial cytochrome P450 for steroidogenesis. Transfers electrons from adrenodoxin reductase to CYP11A1, a cytochrome P450 that catalyzes cholesterol side-chain cleavage to produce pregnenolone, the precursor of most steroid hormones. Does not form a ternary complex with adrenodoxin reductase and CYP11A1 but shuttles between the two enzymes to transfer electrons. Adrenodoxin, mitochondrial Protein, Bov...
TMPY-04586 Chorionic Gonadotropin/CGA Protein, Human, Recombinant

FSH alpha,glycoprotein hormones, alpha polypeptide,LHA,CG-AL...

Human HEK293 Cells
Chorionic Gonadotropin/CGA Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 10.2 kDa and the accession number is P01215.
TMPJ-00744 Toxin B Protein, Vibriocholerae, Recombinant

Cholera enterotoxin γ chain,Choleragenoid,...

Vibrio cholerae E. coli
Cholera toxin is protein complex secreted by the bacterium Vibrio cholerae. It is responsible for the massive, watery diarrhea characteristic of cholera infection. Cholera enterotoxin subunit B (CTXB) pentameric ring directs the A subunit to its target by binding to the GM1 gangliosides present on the surface of the intestinal epithelial cells. It can bind five GM1 gangliosides. It has no toxic activity by itself.
TMPH-03614 DNA photolyase Protein, Synechococcus sp., Recombinant (His & Myc & SUMO)

DNA photolyase,Deoxyribodipyrimidine photo-lyase,phr,phrA,Ph...

Synechococcus E. coli
Involved in repair of UV radiation-induced DNA damage. Catalyzes the light-dependent monomerization (300-600 nm) of cyclobutyl pyrimidine dimers (in cis-syn configuration), which are formed between adjacent bases on the same DNA strand upon exposure to ultraviolet radiation. DNA photolyase Protein, Synechococcus sp., Recombinant (His & Myc & SUMO) is expressed in E. coli expression system with N-10xHis-SUMO and C-Myc tag. The predicted molecular weight is 74.3 kDa and the accession number is P05...
TMPH-00026 Catechol 1,2-dioxygenase Protein, Acinetobacter baylyi, Recombinant (His)

Equinatoxin-2,EqTII,DELTA-AITX-Aeq1a,Equinatoxin II,DELTA-ac...

Actinia equina E. coli
Catechol 1,2-dioxygenase Protein, Acinetobacter baylyi, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 23.9 kDa and the accession number is P61914.
TMPH-00017 acpS Protein, Acholeplasma laidlawii, Recombinant (His & Myc)

Holo-ACP synthase,Holo-[acyl-carrier-protein] synthase,acpS,...

Acholeplasma laidlawii E. coli
Transfers the 4'-phosphopantetheine moiety from coenzyme A to a Ser of acyl-carrier-protein. acpS Protein, Acholeplasma laidlawii, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 20.9 kDa and the accession number is A9NHV3.
TMPH-00389 OmcB Protein, Chlamydia trachomatis, Recombinant (His & SUMO)

Large cysteine-rich periplasmic protein OmcB,Cysteine-rich o...

Chlamydia trachomatis E. coli
In elementary bodies (EBs, the infectious stage, which is able to survive outside the host cell) provides the structural integrity of the outer envelope through disulfide cross-links with the small cysteine-rich protein and the major outer membrane protein. It has been described in publications as the Sarkosyl-insoluble COMC (Chlamydia outer membrane complex), and serves as the functional equivalent of peptidoglycan. OmcB Protein, Chlamydia trachomatis, Recombinant (His & SUMO) is expressed in E...
TMPH-00392 Small-CRP Protein, Chlamydia trachomatis, Recombinant (His & SUMO)

omcA,Small cysteine-rich outer membrane protein OmcA,9 kDa c...

Chlamydia trachomatis E. coli
In elementary bodies (EBs, the infectious stage, which is able to survive outside the host cell) provides the structural integrity of the outer envelope through disulfide cross-links with the large cysteine-rich periplasmic protein and the major outer membrane porin. It has been described in publications as the Sarkosyl-insoluble COMC (Chlamydia outer membrane complex), and serves as the functional equivalent of peptidoglycan. Small-CRP Protein, Chlamydia trachomatis, Recombinant (His & SUMO) is...
TMPH-02244 Trichohyalin Protein, Human, Recombinant (His & Myc)

TCHH,Trichohyalin

Human E. coli
Intermediate filament-associated protein that associates in regular arrays with keratin intermediate filaments (KIF) of the inner root sheath cells of the hair follicle and the granular layer of the epidermis. It later becomes cross-linked to KIF by isodipeptide bonds. It may serve as scaffold protein, together with involucrin, in the organization of the cell envelope or even anchor the cell envelope to the KIF network. It may be involved in its own calcium-dependent postsynthetic processing dur...
TMPH-03615 Ribonuclease J Protein, Synechocystis sp., Recombinant (His & SUMO)

rnj,Ribonuclease J

Synechocystis E. coli
An RNase that has 5'-3' exonuclease and possibly endoonuclease activity. Involved in maturation of rRNA and in some organisms also mRNA maturation and/or decay. Ribonuclease J Protein, Synechocystis sp., Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 86.4 kDa and the accession number is P54123.
TMPH-03605 CHOD Protein, Streptomyces sp., Recombinant (GST)

choA,Cholesterol isomerase,CHOD,<...

Streptomyces E. coli
Bifunctional enzyme that catalyzes the oxidation of the 3-beta-hydroxy group of cholesterol and the isomerization of the double bond of the resulting product. CHOD Protein, Streptomyces sp., Recombinant (GST) is expressed in E. coli expression system with N-GST tag. The predicted molecular weight is 81.9 kDa and the accession number is P12676.
TMPH-03645 Alpha-TCS Protein, Trichosanthes kirilowii, Recombinant (His)

rRNA N-glycosidase,EC:3.2.2.22,Ribosome-inactivating protein...

Trichosanthes kirilowii E. coli
Inactivates eukaryotic 60S ribosomal subunits. Alpha-TCS Protein, Trichosanthes kirilowii, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 30.8 kDa and the accession number is P09989.
TMPH-03057 Chorismate synthase Protein, Neurospora crassa, Recombinant (His)

B7F21.10,NCU05420,aro-2,5-enolpyruvylshikimate-3-phosphate p...

Neurospora crassa E. coli
Bifunctional enzyme that possesses chorismate synthase and intrinsic flavin reductase activity, it uses NADPH to reduce FMN.
TMPH-02412 Lymphocytic choriomeningitis virus (LCMV) (strain WE) GPC Protein (His & Myc)

Pre-glycoprotein polyprotein GP complex,GPC

LCMV E. coli
Lymphocytic choriomeningitis virus (LCMV) (strain WE) GPC Protein (His & Myc) is expressed in E. coli expression system with N-6xHis and C-Myc tag. The predicted molecular weight is 30.9 kDa and the accession number is P07399.
TMPH-00393 pGP3-D Protein, Chlamydia trachomatis, Recombinant (His)

Proteins P-6/P-7,Virulence plasmid protein pGP3-D

Chlamydia trachomatis P. pastoris (Yeast)
pGP3-D Protein, Chlamydia trachomatis, Recombinant (His) is expressed in yeast with N-10xHis tag. The predicted molecular weight is 30.3 kDa and the accession number is P0CE18.
TMPH-03613 NblA Protein, Synechococcus elongatus, Recombinant (His & Myc)

nblA,Phycobilisome degradation protein NblA

Synechococcus elongatus E. coli
Involved in phycobilisome (PBS) degradation during nutrient deprivation. May mark the PBS for degradation by covalent association with PBS components or may disrupt the PBS via ionic interactions. NblA Protein, Synechococcus elongatus, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 14.5 kDa and the accession number is P35087.
TMPY-02309 CHODL Protein, Mouse, Recombinant (hFc)

3110074E07Rik,chondrolectin,MT75,PRED12

Mouse HEK293 Cells
CHODL Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 48.9 kDa and the accession number is EDK98299.1.
TMPY-01596 Butyrylcholinesterase Protein, Mouse, Recombinant (His)

C730038G20Rik,butyrylcholinesterase

Mouse HEK293 Cells
Butyrylcholinesterase Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 66.7 kDa and the accession number is Q03311.
TMPH-00388 Chaperonin GroEL Protein, Chlamydia trachomatis, Recombinant (His & SUMO)

Cpn60,mopA,60 kDa chaperonin,Chaperonin-60,Chaperonin GroEL,...

Chlamydia trachomatis E. coli
Together with its co-chaperonin GroES, plays an essential role in assisting protein folding. The GroEL-GroES system forms a nano-cage that allows encapsulation of the non-native substrate proteins and provides a physical environment optimized to promote and accelerate protein folding. Chaperonin GroEL Protein, Chlamydia trachomatis, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 74.0 kDa and the accession number is P0C0...
TMPH-03068 OV16 Protein, Onchocerca volvulus, Recombinant (His)

OV16,OV-16 antigen

Onchocerca volvulus E. coli
OV16 Protein, Onchocerca volvulus, Recombinant (His) is expressed in E. coli.
TMPH-00391 MOMP Protein, Chlamydia trachomatis serovar L2, Recombinant (His & SUMO)

ompA,Major outer membrane porin

Chlamydia trachomatis serovar L2 E. coli
In elementary bodies (EBs, the infectious stage, which is able to survive outside the host cell) provides the structural integrity of the outer envelope through disulfide cross-links with the small cysteine-rich protein and the large cysteine-rich periplasmic protein. It has been described in publications as the Sarkosyl-insoluble COMC (Chlamydia outer membrane complex), and serves as the functional equivalent of peptidoglycan.; Permits diffusion of specific solutes through the outer membrane. M...
TMPH-00265 Ferrochelatase, mitochondrial Protein, Bovine, Recombinant (His & Myc & SUMO)

Ferrochelatase, mitochondrial,Protoheme ferro-lyase...

Bovine E. coli
Catalyzes the ferrous insertion into protoporphyrin IX. Ferrochelatase, mitochondrial Protein, Bovine, Recombinant (His & Myc & SUMO) is expressed in E. coli expression system with N-10xHis-SUMO and C-Mycd tag. The predicted molecular weight is 58.1 kDa and the accession number is P22600.
TMPH-00394 pGP3-D Protein, Chlamydia trachomatis, Recombinant (E. coli, His)

Proteins P-6/P-7,Virulence plasmid protein pGP3-D

Chlamydia trachomatis E. coli
pGP3-D Protein, Chlamydia trachomatis, Recombinant (E. coli, His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 31.9 kDa and the accession number is P0CE18.
TMPH-00757 Reticuline oxidase Protein, Eschscholzia californica, Recombinant (His)

BBE1,Tetrahydroprotoberberine synthase,Berberine bridge-form...

Eschscholzia californica E. coli
Essential to the formation of benzophenanthridine alkaloids in the response of plants to pathogenic attack. Catalyzes the stereospecific conversion of the N-methyl moiety of (S)-reticuline into the berberine bridge carbon of (S)-scoulerine.
TMPY-01010 NGF Protein, Human, Recombinant

Beta-NGF,神经生长因子,β-NGF,NGFB,nerve growth factor (β polypeptid...

Human CHO Cells
NGF Protein, Human, Recombinant is expressed in CHO mammalian cells. The predicted molecular weight is 13.2 kDa and the accession number is P01138.
TMPY-03565 Mannan Binding Lectin/MBL2 Protein, Human, Recombinant

MBPD,MBP-C,mannose-binding lectin (protein C) 2, soluble,COL...

Human CHO Cells
Mannan Binding Lectin/MBL2 Protein, Human, Recombinant is expressed in CHO mammalian cells. The predicted molecular weight is 24 kDa and the accession number is P11226.
TMPY-03145 IFN-beta Protein, Human, Recombinant

IFN-β,interferon, β1, fibroblast,IFNB,IFB,IFF,Interferon β,I...

Human CHO Cells
IFN-beta Protein, Human, Recombinant is expressed in CHO mammalian cells. The predicted molecular weight is 20 kDa and the accession number is P01574.
TMPY-00467 NKG2D/CD314 Protein, Human, Recombinant (hFc)

D12S2489E,killer cell lectin-like receptor subfamily K, memb...

Human CHO Cells
NKG2D/CD314 Protein, Human, Recombinant (hFc) is expressed in CHO mammalian cells with hFc tag. The predicted molecular weight is 46.5 kDa and the accession number is A0A024RAP8.
TMPY-02638 TGF beta 1 Protein, Human/Rhesus/Cynomolgus/Canine, Recombinant

transforming growth factor, beta 1,转化生长因子,transforming growt...

Human,Rhesus,Cynomolgus,Canine CHO Cells
TGF beta 1 Protein, Human/Rhesus/Cynomolgus/Canine, Recombinant is expressed in CHO mammalian cells. The predicted molecular weight is 12.8 kDa and the accession number is A0A499FJK2.
TMPY-01714 IFN gamma Protein, Human, Recombinant

IFI,interferon, γ,IFN γ,IFG,IFN gamma,interferon, gamma,干扰素,...

Human CHO Cells
IFN gamma Protein, Human, Recombinant is expressed in CHO mammalian cells. The predicted molecular weight is 16.7 kDa and the accession number is A0A7R8GUN6.
TMPY-03142 IL-27 Protein, Human, Recombinant (His)

IL27p28,IL-27,白介素,IL27A,interleukin 27,p28,白细胞介素,IL-27A,IL30

Human CHO Cells
IL-27 Protein, Human, Recombinant (His) is expressed in CHO mammalian cells with His tag. The predicted molecular weight is 56 kDa and the accession number is NP_005746.2&NP_663634.2.
TMPY-01993 IL-13 Protein, Human, Recombinant

IL-13,P600,interleukin 13,ALRH,白介素,白细胞介素

Human CHO Cells
IL-13 Protein, Human, Recombinant is expressed in CHO mammalian cells. The predicted molecular weight is 12.5 kDa and the accession number is AAK53823.1.
TMPY-02327 HGF Protein, Human, Recombinant

SF,hepatocyte growth factor (hepapoietin A,HGFB,F-TCF,F-TCFB...

Human CHO Cells
HGF Protein, Human, Recombinant is expressed in CHO mammalian cells. The predicted molecular weight is 79.7 kDa and the accession number is P14210-1.
TMPY-03626 R-Spondin 1/RSPO1 Protein, Human, Recombinant

RSPO,R-spondin 1,CRISTIN3

Human CHO Cells
R-Spondin 1/RSPO1 Protein, Human, Recombinant is expressed in CHO mammalian cells. The predicted molecular weight is 26.8 kDa and the accession number is Q2MKA7-1.
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重组蛋白

Butyrylcholinesterase Protein, Human, Recombinant (His)
Cat.No: TMPY-01693
Species: Human
Expression System: HEK293 Cells
CHODL Protein, Rat, Recombinant (hFc)
Cat.No: TMPY-03006
Species: Rat
Expression System: HEK293 Cells
Zika virus (ZIKV) (strain Zika SPH2016) ZIKV-E (Stem/anchor domain of flavivirus envelope glycoprotein E) protein (Fc)
Cat.No: TMPY-04905
Species: ZIKV
Expression System: HEK293 Cells
CHODL Protein, Rat, Recombinant (His)
Cat.No: TMPY-02941
Species: Rat
Expression System: HEK293 Cells
CHODL Protein, Mouse, Recombinant (His)
Cat.No: TMPY-02408
Species: Mouse
Expression System: HEK293 Cells
CHODL Protein, Human, Recombinant (hFc)
Cat.No: TMPK-01188
Species: Human
Expression System: HEK293 Cells
Acetylcholinesterase Protein, Rat, Recombinant (His)
Cat.No: TMPH-03234
Species: Rat
Expression System: E. coli
MTA/SAH nucleosidase Protein, Vibrio cholerae serotype O1, Recombinant (His & Myc)
Cat.No: TMPH-03702
Species: Vibrio cholerae
Expression System: E. coli
Zot Protein, Vibrio cholerae serotype O1, Recombinant (His)
Cat.No: TMPH-03703
Species: Vibrio cholerae
Expression System: E. coli
MOMP Protein, Chlamydia trachomatis, Recombinant (His & Myc)
Cat.No: TMPH-00390
Species: Chlamydia trachomatis
Expression System: E. coli
Lymphocytic choriomeningitis virus (LCMV) (strain Armstrong) GPC Protein (His & SUMO)
Cat.No: TMPH-02413
Species: LCMV
Expression System: E. coli
Hydrophobin-2/HFB2 Protein, Trichoderma reesei, Recombinant (His & SUMOstar)
Cat.No: TMPH-03644
Species: Hypocrea jecorina
Expression System: P. pastoris (Yeast)
Chorionic Gonadotropin/CGA Protein, Human, Recombinant (His)
Cat.No: TMPY-00647
Species: Human
Expression System: HEK293 Cells
Chorionic Gonadotropin/CGA Protein, Human, Recombinant (mFc)
Cat.No: TMPY-02923
Species: Human
Expression System: HEK293 Cells
Acetylcholinesterase Protein, Mouse, Recombinant (His)
Cat.No: TMPY-01742
Species: Mouse
Expression System: HEK293 Cells
DTE Protein, Pseudomonas cichorii, Recombinant (His & Myc)
Cat.No: TMPH-03182
Species: Pseudomonas cichorii
Expression System: E. coli
Adrenodoxin, mitochondrial Protein, Bovine, Recombinant (His)
Cat.No: TMPH-00220
Species: Bovine
Expression System: E. coli
Chorionic Gonadotropin/CGA Protein, Human, Recombinant
Cat.No: TMPY-04586
Species: Human
Expression System: HEK293 Cells
Toxin B Protein, Vibriocholerae, Recombinant
Cat.No: TMPJ-00744
Species: Vibrio cholerae
Expression System: E. coli
DNA photolyase Protein, Synechococcus sp., Recombinant (His & Myc & SUMO)
Cat.No: TMPH-03614
Species: Synechococcus
Expression System: E. coli
Catechol 1,2-dioxygenase Protein, Acinetobacter baylyi, Recombinant (His)
Cat.No: TMPH-00026
Species: Actinia equina
Expression System: E. coli
acpS Protein, Acholeplasma laidlawii, Recombinant (His & Myc)
Cat.No: TMPH-00017
Species: Acholeplasma laidlawii
Expression System: E. coli
OmcB Protein, Chlamydia trachomatis, Recombinant (His & SUMO)
Cat.No: TMPH-00389
Species: Chlamydia trachomatis
Expression System: E. coli
Small-CRP Protein, Chlamydia trachomatis, Recombinant (His & SUMO)
Cat.No: TMPH-00392
Species: Chlamydia trachomatis
Expression System: E. coli
Trichohyalin Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-02244
Species: Human
Expression System: E. coli
Ribonuclease J Protein, Synechocystis sp., Recombinant (His & SUMO)
Cat.No: TMPH-03615
Species: Synechocystis
Expression System: E. coli
CHOD Protein, Streptomyces sp., Recombinant (GST)
Cat.No: TMPH-03605
Species: Streptomyces
Expression System: E. coli
Alpha-TCS Protein, Trichosanthes kirilowii, Recombinant (His)
Cat.No: TMPH-03645
Species: Trichosanthes kirilowii
Expression System: E. coli
Chorismate synthase Protein, Neurospora crassa, Recombinant (His)
Cat.No: TMPH-03057
Species: Neurospora crassa
Expression System: E. coli
Lymphocytic choriomeningitis virus (LCMV) (strain WE) GPC Protein (His & Myc)
Cat.No: TMPH-02412
Species: LCMV
Expression System: E. coli
pGP3-D Protein, Chlamydia trachomatis, Recombinant (His)
Cat.No: TMPH-00393
Species: Chlamydia trachomatis
Expression System: P. pastoris (Yeast)
NblA Protein, Synechococcus elongatus, Recombinant (His & Myc)
Cat.No: TMPH-03613
Species: Synechococcus elongatus
Expression System: E. coli
CHODL Protein, Mouse, Recombinant (hFc)
Cat.No: TMPY-02309
Species: Mouse
Expression System: HEK293 Cells
Butyrylcholinesterase Protein, Mouse, Recombinant (His)
Cat.No: TMPY-01596
Species: Mouse
Expression System: HEK293 Cells
Chaperonin GroEL Protein, Chlamydia trachomatis, Recombinant (His & SUMO)
Cat.No: TMPH-00388
Species: Chlamydia trachomatis
Expression System: E. coli
OV16 Protein, Onchocerca volvulus, Recombinant (His)
Cat.No: TMPH-03068
Species: Onchocerca volvulus
Expression System: E. coli
MOMP Protein, Chlamydia trachomatis serovar L2, Recombinant (His & SUMO)
Cat.No: TMPH-00391
Species: Chlamydia trachomatis serovar L2
Expression System: E. coli
Ferrochelatase, mitochondrial Protein, Bovine, Recombinant (His & Myc & SUMO)
Cat.No: TMPH-00265
Species: Bovine
Expression System: E. coli
pGP3-D Protein, Chlamydia trachomatis, Recombinant (E. coli, His)
Cat.No: TMPH-00394
Species: Chlamydia trachomatis
Expression System: E. coli
Reticuline oxidase Protein, Eschscholzia californica, Recombinant (His)
Cat.No: TMPH-00757
Species: Eschscholzia californica
Expression System: E. coli
NGF Protein, Human, Recombinant
Cat.No: TMPY-01010
Species: Human
Expression System: CHO Cells
Mannan Binding Lectin/MBL2 Protein, Human, Recombinant
Cat.No: TMPY-03565
Species: Human
Expression System: CHO Cells
IFN-beta Protein, Human, Recombinant
Cat.No: TMPY-03145
Species: Human
Expression System: CHO Cells
NKG2D/CD314 Protein, Human, Recombinant (hFc)
Cat.No: TMPY-00467
Species: Human
Expression System: CHO Cells
TGF beta 1 Protein, Human/Rhesus/Cynomolgus/Canine, Recombinant
Cat.No: TMPY-02638
Species: Human,Rhesus,Cynomolgus,Canine
Expression System: CHO Cells
IFN gamma Protein, Human, Recombinant
Cat.No: TMPY-01714
Species: Human
Expression System: CHO Cells
IL-27 Protein, Human, Recombinant (His)
Cat.No: TMPY-03142
Species: Human
Expression System: CHO Cells
IL-13 Protein, Human, Recombinant
Cat.No: TMPY-01993
Species: Human
Expression System: CHO Cells
HGF Protein, Human, Recombinant
Cat.No: TMPY-02327
Species: Human
Expression System: CHO Cells
R-Spondin 1/RSPO1 Protein, Human, Recombinant
Cat.No: TMPY-03626
Species: Human
Expression System: CHO Cells
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Cat. No. Product Name Target Signaling Pathways
TMIH-0552 Tauroursodeoxycholic Acid-d4 Sodium Salt

Tauroursodeoxycholic Acid-d4 Sodium Salt 是 Tauroursodeoxycholic Acid Sodium Salt 的氘代化合物。Tauroursodeoxycholic Acid Sodium Salt 的 CAS 号为 14605-22-2。Tauroursodeoxycholate,又称 ursodoxicoltaurine,是一种高度亲水性的三级胆汁酸,在人体内以低浓度产生。Tauroursodeoxycholate 是 ursodeoxycholic acid 更亲水的形式,而 ursodeoxycholic acid 是人类体内自然产生的更丰富的胆汁酸。Tauroursodeoxycholate 正在研究用于几种疾病,如原发性胆汁性肝硬化(PBC)、胰岛素抵抗、淀粉样变性、囊性纤维化、胆汁淤滞和肌萎缩性侧索硬化症。
TMIH-0145 Chenodeoxycholic Acid-d4

Chenodeoxycholic Acid-d4 是 Chenodeoxycholic Acid 的氘代化合物。
TMIH-0148 Cholic acid-d4

Cholic acid-d4 是 Cholic acid 的氘代化合物。
TMIJ-0197 Tauroursodeoxycholic-2,2,3,4,4-d5 Acid

Tauroursodeoxycholic-2,2,3,4,4-d5 Acid 是 Tauroursodeoxycholic Acid 的氘代化合物。Tauroursodeoxycholic Acid 的 CAS 号为 14605-22-2。Tauroursodeoxycholate,又称 ursodoxicoltaurine,是一种高度亲水性的三级胆汁酸,在人体内以低浓度产生。Tauroursodeoxycholate 是 ursodeoxycholic acid 更亲水的形式,而 ursodeoxycholic acid 是人类体内自然产生的更丰富的胆汁酸。Tauroursodeoxycholate 正在研究用于几种疾病,如原发性胆汁性肝硬化(PBC)、胰岛素抵抗、淀粉样变性、囊性纤维化、胆汁淤滞和肌萎缩性侧索硬化症。
TMID-0058 Glycocholic acid-d4

Glycocholic acid-d4 是 Glycocholic acid 的氘代化合物。Glycocholic acid 的 CAS 号为 475-31-0。Glycocholic acid 是一种胆汁酸,具有抗肿瘤活性,能够靶向作用于耐药泵和非耐药泵通路。
TMIJ-0332 Taurolithocholic Acid-d5 Sodium Salt (Major)

Taurolithocholic Acid-d5 Sodium Salt (Major) 是 Taurolithocholic Acid Sodium Salt 的氘代化合物。Taurolithocholic Acid Sodium Salt 的 CAS 号为 6042-32-6。Taurolithocholic acid sodium salt 是抑胆剂和Ca2+激动剂,可抑制放射性配体与毒蕈碱 M1 结合。
TMIH-0182 Deoxycholic-2,2,4,4-d4 Acid

Deoxycholic-2,2,4,4-d4 Acid 是 Deoxycholic-2,2,4,4 Acid 的氘代化合物。
TMIJ-0198 Taurochenodeoxycholic Acid-d5 Sodium Salt

Taurochenodeoxycholic Acid-d5 Sodium Salt 是 Taurochenodeoxycholic Acid Sodium Salt 的氘代化合物。Taurochenodeoxycholic Acid Sodium Salt 的 CAS 号为 6009-98-9。Taurochenodeoxycholic acid sodium 是动物胆汁酸的主要生物活性物质之一。它可诱导细胞凋亡,具有抗炎和免疫调节作用。
TMIJ-0199 Tauroursodeoxycholic-d4 Acid

Tauroursodiol-d4

Tauroursodeoxycholic-d4 Acid 是 Tauroursodeoxycholic Acid 的氘代化合物。Tauroursodeoxycholic Acid 的 CAS 号为 14605-22-2。Tauroursodeoxycholate,又称 ursodoxicoltaurine,是一种高度亲水性的三级胆汁酸,在人体内以低浓度产生。Tauroursodeoxycholate 是 ursodeoxycholic acid 更亲水的形式,而 ursodeoxycholic acid 是人类体内自然产生的更丰富的胆汁酸。Tauroursodeoxycholate 正在研究用于几种疾病,如原发性胆汁性肝硬化(PBC)、胰岛素抵抗、淀粉样变性、囊性纤维化、胆汁淤滞和肌萎缩性侧索硬化症。
TMID-0294 Taurodeoxycholic Acid-d4 Sodium Salt

Taurodeoxycholic Acid-d4 Sodium Salt 是 Taurodeoxycholic Acid Sodium Salt 的氘代化合物。Taurodeoxycholic Acid Sodium Salt 的 CAS 号为 1180-95-6。Taurodeoxycholate sodium salt 是胆盐相关的阴离子洗涤剂,用于分离膜蛋白,包括线粒体内膜蛋白。它还可以抑制各种炎症反应。
TMID-0224 Cholesterol-d6

Cholesterol-d6 是 Cholesterol 的氘代化合物。Cholesterol 的 CAS 号为 57-88-5。Cholesterol 是哺乳动物中的主要固醇,占质膜结构成分的 20-25%。Cholesterol 在确定膜的流动性和渗透性特征以及转运蛋白和信号蛋白的功能中起着重要作用。Cholesterol 还是内源性雌激素相关受体 α 激动剂。
TMID-0225 Cholesterol-d6-1

Cholesterol-d6-1 是 Cholesterol 的氘代化合物。Cholesterol 的 CAS 号为 57-88-5。Cholesterol 是哺乳动物中的主要固醇,占质膜结构成分的 20-25%。Cholesterol 在确定膜的流动性和渗透性特征以及转运蛋白和信号蛋白的功能中起着重要作用。Cholesterol 还是内源性雌激素相关受体 α 激动剂。
T33348 Methyl-d9-choline

J2.078.736H

Methyl -D9- choline is an isotopically labeled choline tracer.
TMIH-0590 Ursodeoxycholic Acid-d4

Ursodeoxycholic Acid-d4 是 Ursodeoxycholic Acid 的氘代化合物。
TMIH-0257 Glycoursodeoxycholic Acid-d4

Glycoursodeoxycholic Acid-d4 是 Glycoursodeoxycholic Acid 的氘代化合物。Glycoursodeoxycholic Acid 的 CAS 号为 64480-66-6。Glycoursodeoxycholic acid 是一种酰基甘氨酸和胆汁酸-甘氨酸缀合物,是熊去氧胆酸的代谢物。
TMIH-0286 Isochenodeoxycholic Acid-d4

Isochenodeoxycholic Acid-d4 是 Isochenodeoxycholic Acid 的氘代化合物。Isochenodeoxycholic Acid 的 CAS 号为 566-24-5。
TMID-0223 Cholesterol-d7

Cholesterol-d7 是 Cholesterol 的氘代化合物。Cholesterol 的 CAS 号为 57-88-5。Cholesterol 是哺乳动物中的主要固醇,占质膜结构成分的 20-25%。Cholesterol 在确定膜的流动性和渗透性特征以及转运蛋白和信号蛋白的功能中起着重要作用。Cholesterol 还是内源性雌激素相关受体 α 激动剂。
TMIH-0254 Glycochenodeoxycholic Acid-d4

Glycochenodeoxycholic Acid-d4 是 Glycochenodeoxycholic Acid 的氘代化合物。
TMIH-0149 Choline-d4 Chloride

Choline-d4 Chloride 是 Choline Chloride 的氘代化合物。
TMID-0226 Cholesterol-d4

Cholesterol-d4 是 Cholesterol 的氘代化合物。Cholesterol 的 CAS 号为 57-88-5。Cholesterol 是哺乳动物中的主要固醇,占质膜结构成分的 20-25%。Cholesterol 在确定膜的流动性和渗透性特征以及转运蛋白和信号蛋白的功能中起着重要作用。Cholesterol 还是内源性雌激素相关受体 α 激动剂。
TMIJ-0304 Lithocholic Acid-d4

Lithocholic Acid-d4 是 Lithocholic Acid 的氘代化合物。Lithocholic Acid 的 CAS 号为 434-13-9。Lithocholic acid是由鹅去氧胆酸盐通过细菌作用形成的胆汁酸,通常与甘氨酸或牛磺酸结合,被用作利胆剂。 它作为清洁剂溶解脂肪以供吸收,并且本身被吸收。
TMID-0232 Choline-d13 Bromide (N,N,N-trimethyl-d9; 1,1,2,2-d4)

Choline-d13 Bromide (N,N,N-trimethyl-d9; 1,1,2,2-d4) 是 Choline Bromide 的氘代化合物。Choline Bromide 的 CAS 号为 1927-06-6。
TMID-0052 Taurocholic Acid-d4 Sodium

Taurocholic Acid-d4 Sodium 是 Taurocholic Acid Sodium 的氘代化合物。Taurocholic Acid Sodium 的 CAS 号为 145-42-6。Sodium taurocholate hydrate 具有显著的生物学效应,例如通过上调 VEGF-A 的表达抑制肝动脉结扎所致的胆道损伤。对免疫系统具有一定的调节作用。
TMIH-0255 Glycolithocholic-2,2,4,4-d4 Acid

Glycolithocholic-2,2,4,4-d4 Acid 是 Glycolithocholic-2,2,4,4 Acid 的氘代化合物。
TMID-0161 5-alpha-Cholestane-2,2,4,4-d4

5-alpha-Cholestane-2,2,4,4-d4 是 5-alpha-Cholestane 的氘代化合物。5-alpha-Cholestane 的 CAS 号为 481-21-0。5α-Cholestane 属于一类称为胆甾烷类固醇的有机化合物。
T11655 Indomethacin-D4

Indometacin-D4,吲哚美辛-D4

CDK Cell Cycle/Checkpoint
Indomethacin-D4 is a deuterium labeled Indomethacin. Indomethacin is a potent and nonselective inhibitor of COX1 and COX2, with IC50s of 18 nM and 26 nM for human COX-1 and COX-2, respectively, in CHO cells.
TMIJ-0127 Diclofenac-d4

Diclofenac-d4 是 Diclofenac 的氘代化合物。Diclofenac 的 CAS 号为 15307-86-5。Diclofenac 是一种具有抗炎活性的非甾体苯乙酸衍生物,是COX抑制剂,在 CHO 细胞中,对人 COX-1 和 COX-2 的IC50值分别为 4 和 1.3 nM。它对绵羊 COX-1 和 COX-2 的IC50值分别为 5.1 μM,0.84 μM。它通过活化 caspase 级联反应来诱导神经干细胞凋亡。

同位素标记化合物

Tauroursodeoxycholic Acid-d4 Sodium Salt
Cat.No: TMIH-0552
Synonym:
Target:
Chenodeoxycholic Acid-d4
Cat.No: TMIH-0145
Synonym:
Target:
Cholic acid-d4
Cat.No: TMIH-0148
Synonym:
Target:
Tauroursodeoxycholic-2,2,3,4,4-d5 Acid
Cat.No: TMIJ-0197
Synonym:
Target:
Glycocholic acid-d4
Cat.No: TMID-0058
Synonym:
Target:
Taurolithocholic Acid-d5 Sodium Salt (Major)
Cat.No: TMIJ-0332
Synonym:
Target:
Deoxycholic-2,2,4,4-d4 Acid
Cat.No: TMIH-0182
Synonym:
Target:
Taurochenodeoxycholic Acid-d5 Sodium Salt
Cat.No: TMIJ-0198
Synonym:
Target:
Tauroursodeoxycholic-d4 Acid
Cat.No: TMIJ-0199
Synonym: Tauroursodiol-d4
Target:
Taurodeoxycholic Acid-d4 Sodium Salt
Cat.No: TMID-0294
Synonym:
Target:
Cholesterol-d6
Cat.No: TMID-0224
Synonym:
Target:
Cholesterol-d6-1
Cat.No: TMID-0225
Synonym:
Target:
Methyl-d9-choline
Cat.No: T33348
Synonym: J2.078.736H
Target:
Ursodeoxycholic Acid-d4
Cat.No: TMIH-0590
Synonym:
Target:
Glycoursodeoxycholic Acid-d4
Cat.No: TMIH-0257
Synonym:
Target:
Isochenodeoxycholic Acid-d4
Cat.No: TMIH-0286
Synonym:
Target:
Cholesterol-d7
Cat.No: TMID-0223
Synonym:
Target:
Glycochenodeoxycholic Acid-d4
Cat.No: TMIH-0254
Synonym:
Target:
Choline-d4 Chloride
Cat.No: TMIH-0149
Synonym:
Target:
Cholesterol-d4
Cat.No: TMID-0226
Synonym:
Target:
Lithocholic Acid-d4
Cat.No: TMIJ-0304
Synonym:
Target:
Choline-d13 Bromide (N,N,N-trimethyl-d9; 1,1,2,2-d4)
Cat.No: TMID-0232
Synonym:
Target:
Taurocholic Acid-d4 Sodium
Cat.No: TMID-0052
Synonym:
Target:
Glycolithocholic-2,2,4,4-d4 Acid
Cat.No: TMIH-0255
Synonym:
Target:
5-alpha-Cholestane-2,2,4,4-d4
Cat.No: TMID-0161
Synonym:
Target:
Indomethacin-D4
Cat.No: T11655
Synonym: Indometacin-D4,吲哚美辛-D4
Target: CDK
Diclofenac-d4
Cat.No: TMIJ-0127
Synonym:
Target:
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