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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2373 |
Vipadenant
CEB-4520,BIIB-014 |
Adenosine Receptor | GPCR/G Protein; Neuroscience |
Vipadenant (CEB-4520) 是一种腺苷受体拮抗剂,抑制 A2A 和 A1 活性的 Ki 值分别为 1.3 和 68 nM。 | |||
T28654 |
Sabcomeline hydrochloride
BCI224,BRL-55473,BCI-224,CEB-2424,SB-202026A,Sabcomeline HCl |
Others | Others |
Sabcomeline is a selective M1 receptor partial agonist. | |||
T3715 |
Acebilustat
阿西鲁司特,CTX-4430 |
Aminopeptidase; LTR | Immunology/Inflammation; Metabolism |
Acebilustat (CTX-4430) 是一种具有口服活性的白三烯 A4 水解酶抑制剂,可用于炎症研究。 | |||
T10977 |
DCEBIO
|
Potassium Channel | Membrane transporter/Ion channel |
DCEBIO 是1-EBIO 的衍生物,是 T84 结肠细胞中Cl-分泌的极有效的激活剂。DCEBIO 通过激活 hIK1 K+通道和顶端膜的 Cl-传导促进 Cl-的分泌。 | |||
T5167 |
Cebranopadol
西博帕多,GRT6005 |
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
Cebranopadol (GRT6005) 是镇痛 NOP 和阿片受体激动剂,对人 NOP、μ-阿片 (MOP)、κ-阿片 (KOP) 和 δ-阿片 (DOP) 受体的 Ki 值分别为 0.9、0.7、2.6 和 18 nM。 | |||
T1012 |
Acebutolol hydrochloride
盐酸醋丁洛尔,Acebutolol HCl |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Acebutolol hydrochloride (Acebutolol HCl) 是一种 β-肾上腺素受体拮抗剂,用于研究高血压、心绞痛和心律失常。 | |||
T23604 |
Acebrochol
|
Others | Others |
Acebrochol is a neuroactive steroid. It may act as a sedative and hypnotic, by the mechanism of altering ligand-gated ion channels and cell surface receptors. | |||
T25881 |
Novocebrin
D8955,D-8955,D 8955 |
Others | Others |
Novocebrin is a central nervous system activator. | |||
T15155 |
Docebenone
AA 861 |
Others | Others |
Docebenone is a selective and orally active inhibitor of 5-LO. | |||
T21021 |
Deacyl acebutolol
Acetolol,M,B 17127 |
Others | Others |
Deacyl acebutolol is the major metabolite of Acebutolol. | |||
T64272 |
MTL-CEBPA
|
Others | Others |
MTL-CEPBA 是一种靶向 C/EBPα 上调的小活化 RNA,表现出抗炎和抗癌效果。 | |||
T23605 |
Aceburic acid
|
Others | Others |
Aceburic acid is the acetyl ester of gamma-hydroxybutyrate. | |||
T10749 |
Cebranopadol ((1α,4α)stereoisomer)
GRT6005 (1α,4α)stereoisomer |
Others | Others |
Cebranopadol ((1α,4α)stereoisomer) is a stereoisomer of cebranopadol which is a potent ORL-1 agonist. |
Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPY-03604 |
VAMP3 Protein, Human, Recombinant (His)
vesicle-associated membrane protein 3,CEB |
Human | E. coli |
VAMP3, also known as cellubrevin, is a member of the vesicle-associated membrane protein (VAMP)/synaptobrevin family. Synaptobrevins/VAMPs, syntaxins, and the 25-kD synaptosomal-associated protein are the main components of a protein complex involved in the docking and/or fusion of synaptic vesicles with the presynaptic membrane. Because of VAMP3 gene's high homology to other known VAMPs, its broad tissue distribution, and its subcellular localization, VAMP3 was shown to be the human equivalent ... | |||
TMPY-03794 |
CEBP gamma Protein, Human, Recombinant (His)
CCAAT/enhancer binding protein (C/EBP), gamma,GPE1BP,CEB... |
Human | E. coli |
CEBPG, also known as CEBP gamma, is a transcription factor which belongs to the CEBP family. Members of this family regulate viral and cellular CCAAT/enhancer element-mediated transcription. CEBP proteins contain the bZIP region, which is characterized by two motifs in the C-terminal half of the protein: a basic region involved in DNA binding and a leucine zipper motif involved in dimerization. CEBPG binds to the enhancer element PRE-I of the IL-4 gene. It Might change the DNA-binding specificit... | |||
TMPH-01067 |
CEBPD Protein, Human, Recombinant (His & Myc)
Nuclear factor NF-IL6-beta,CCAAT/enhancer-binding protein de... |
Human | E. coli |
Transcription activator that recognizes two different DNA motifs: the CCAAT homology common to many promoters and the enhanced core homology common to many enhancers. Important transcription factor regulating the expression of genes involved in immune and inflammatory responses. Transcriptional activator that enhances IL6 transcription alone and as heterodimer with CEBPB. CEBPD Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The pred... |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T10229 |
Acebutolol D7
|
Others | Others |
Acebutolol D7 is a deuterium-labeled Acebutolol. Acebutolol is a selective antagonist of the β1 adrenergic receptor used in the treatment of angina pectoris, hypertension, and cardiac arrhythmias. |