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Cat. No. Product Name Target Signaling Pathways
T84917 CDK-IN-11

Others Others
CDK-IN-11,一种杂环化合物,可促进心肌细胞成熟。
T10743 CDK9-IN-11

CDK Cell Cycle/Checkpoint
CDK9-IN-11 是一种有效的CDK9抑制剂,可作为 PROTAC CDK9 Degrader-1 的配体。
T1785 Palbociclib

PD 0332991,帕博西尼,帕布昔利布

CDK Cell Cycle/Checkpoint
Palbociclib (PD 0332991) 是一种 CDK 抑制剂,抑制 CDK4 和 CDK6 (IC50=11/16 nM),具有口服活性。Palbociclib 具有抗肿瘤活性,有用于 ER 阳性和 HER2 阴性乳腺癌的研究潜力。
T10745 CDK9-IN-7

CDK Cell Cycle/Checkpoint
CDK9-IN-7 (compound 21e) 是一种高效选择性的,具有口服活性的 CDK9/cyclin T 抑制剂 (IC50=11 nM),与抑制其他 CDK 相比更有效 (CDK4/cyclinD=148 nM; CDK6/cyclinD=145 nM)。CDK9-IN-7 具有抗癌活性并没有明显的毒性。CDK9-IN-7 诱导非小细胞肺癌 (NSCLC) 细胞凋亡,在 G2 期阻滞细胞周期,并具有抑制非小细胞肺癌干细胞特性。
T69196 AG-012986

Others Others
AG-012986 is a multitargeted cyclin-dependent kinase (CDK) inhibitor active against CDK1, CDK2, CDK4/6, CDK5, and CDK9, with selectivity over a diverse panel of non-CDK kinases. AG-012986 showed antiproliferative activities in vitro with IC(50)s of <100 nmol/L in 14 of 18 tumor cell lines. In vivo, significant antitumor efficacy induced by AG-012986 was seen (tumor growth inhibition, >83.1%) in 10 of 11 human xenograft tumor models. AG-012986 also showed dose-dependent retinoblastoma Ser(795) hy...
T69197 AG-012986 HCl

Others Others
AG-012986 HCl is a multitargeted cyclin-dependent kinase (CDK) inhibitor active against CDK1, CDK2, CDK4/6, CDK5, and CDK9, with selectivity over a diverse panel of non-CDK kinases. AG-012986 HCl showed antiproliferative activities in vitro with IC(50)s of <100 nmol/L in 14 of 18 tumor cell lines. In vivo, significant antitumor efficacy induced by AG-012986 HCl was seen (tumor growth inhibition, >83.1%) in 10 of 11 human xenograft tumor models. AG-012986 HCl also showed dose-dependent retinoblas...

化合物

CDK-IN-11
Cat.No: T84917
Synonym:
Target: Others
CDK9-IN-11
Cat.No: T10743
Synonym:
Target: CDK
Palbociclib
Cat.No: T1785
Synonym: PD 0332991,帕博西尼,帕布昔利布
Target: CDK
CDK9-IN-7
Cat.No: T10745
Synonym:
Target: CDK
AG-012986
Cat.No: T69196
Synonym:
Target: Others
AG-012986 HCl
Cat.No: T69197
Synonym:
Target: Others
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