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Cat. No. | Product Name | ||
---|---|---|---|
L6750 | 活血化瘀中药单体库 | 580 compounds | |
580种来源于常见活血化瘀中药的单体化合物,是药物开发、药理研究等领域的有效工具。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2S0618 |
β-Elemonic Acid
3-oxo Tirucallic Acid,β-岚香酮酸,Beta-Elemonic acid,3-Oxotirucallenoic Acid,β-榄香酮酸,Elemadienonic Acid |
Apoptosis; Reactive Oxygen Species; COX | Apoptosis; Immunology/Inflammation; Metabolism; Neuroscience; NF-κB |
β-Elemonic Acid (3-Oxotirucallenoic Acid) 是从乳香树中分离得到的一种三萜,具有抗癌和抗炎作用。它抑制脯氨酰内肽酶,诱导细胞凋亡,活性氧和COX-2表达。 | |||
T3248 |
alpha-Boswellic acid
α-Boswellic acid,α-乳香酸 |
Others | Others |
alpha-Boswellic acid 是一种从乳香中提取得到的五环三萜类化合物,具有抗惊厥和抗癌作用。在动物体内,它是预防和减少阿尔茨海默病标志物,可用于阿尔茨海默病的研究。 | |||
TN2448 |
3α-Hydroxy tirucall-7,24-dien-21-oic acid
|
Others | Others |
3α-Hydroxy tirucall-7,24-dien-21-oic acid is a natural product from Boswellia carterii Birdw | |||
TN2457 |
3α-acetoxy-tirucall-7,24-dien-21oic acid
|
Others | Others |
3α-acetoxy-tirucall-7,24-dien-21oic acid is a natural product from Boswellia carterii Birdw | |||
T83340 |
3α-Acetoxyurs-5:12-dien-24-oic acid
|
||
3α-Acetoxyurs-5:12-dien-24-oic acid 为从Boswellia sacra Fluckiger分离所得的一种天然化合物。 | |||
TN1182 |
11-Keto-beta-boswellic acid
11-Keto-beta-boswellic acid,11-酮基-BETA-乳香酸 |
Leukotriene Receptor; NF-κB; Lipoxygenase | GPCR/G Protein; Metabolism; NF-κB |
11-Keto-beta-boswellic acid 是来自乳香的一种五环三萜酸,具有抗炎活性和剂量依赖性心脏保护作用,主要是由于抑制5-脂氧合酶、白三烯、NF-κB 的激活和肿瘤坏死因子 α 的产生。 | |||
T2862 |
Desaminotyrosine
Phloretate,3-(4-Hydroxyphenyl)propanoic acid,Hydro-p-coumaric acid,对羟基苯丙酸,3-(4-Hydroxyphenyl)propionic acid,Phloretic acid,根皮酸 |
Others; Influenza Virus; Endogenous Metabolite | Metabolism; Microbiology/Virology; Others |
Desaminotyrosine (3-(4-Hydroxyphenyl)propionic acid) 是一种与微生物相关的代谢物,通过增强 I 型干扰素信号传导来预防流感。 | |||
TN2450 |
Acetyl 11α-methoxy-β-boswellic Acid
|
Others | Others |
Acetyl 11α-methoxy-β-boswellic Acid是从乳香树脂中提取到的三萜类化合物。 | |||
TWS1563 |
Incensole
|
Others | Others |
Incensole 是一种 14-membered 二萜类化合物,分离自烯属植物的香精油和乳香树脂中。它能够激活脑中离子通道,并可以缓解焦虑或抑郁,从而显示出抗炎和抗抑郁的特性。 | |||
TN1255 |
3-O-Acetyl-11-hydroxy-beta-boswellic acid
|
Lipoxygenase | Metabolism |
3-O-Acetyl-11-hydroxy-beta-boswellic acid 是 5-脂氧合酶抑制剂。 | |||
TN1097 |
β-Boswellic acid
Beta-boswellic acid,β-乳香酸 |
Lipoxygenase; DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism |
β-Boswellic acid (Beta-boswellic acid) 是从乳香的树胶脂中分离出来的一种天然产物。它是 5-脂氧合酶(5-LO) 产物形成的非还原型抑制剂,其直接与 5-LO 相互作用或阻断其易位。具有抗癌、抗肿瘤和抗高血脂活性。 | |||
T5S1569 |
AKBA
乙酰基-11-酮基-beta-乳香酸,3-O-Acetyl-11-keto-β-boswellic acid,3-O-Acetyl-11-keto-beta-boswellic acid,Acetyl-11-keto-β-boswellic acid |
Others; Reactive Oxygen Species; HIF/HIF Prolyl-Hydroxylase; Endogenous Metabolite | Chromatin/Epigenetic; Immunology/Inflammation; Metabolism; NF-κB; Others |
AKBA (3-O-Acetyl-11-keto-beta-boswellic acid) 是一种从乳香中分离的天然成分,是新颖的 Nrf2 的活化剂。 | |||
TN1257 |
3-O-Acetyl-α-boswellic acid
3-O-Acetyl-alpha-boswellic acid,α-Boswellic acid acetate,乙酰基-ALPHA-乳香酸 |
Prostaglandin Receptor | GPCR/G Protein; Immunology/Inflammation |
3-O-Acetyl-α-boswellic acid (α-Boswellic acid acetate) 能够抑制 T 细胞功能,具有很强的抗炎作用。 | |||
TN1258 |
3-Acetyl-beta-boswellic acid
3-O-Acetyl-beta-boswellic acid,3-乙酰基-BETA-乳香酸 |
DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
3-Acetyl-beta-boswellic acid 是一种乳香酸,分离自乳香锯缘胶树脂。 | |||
TN4463 |
Lupeolic acid
|
COX; Prostaglandin Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Lupeolic acid has anti-inflammatory activity. | |||
TN1988 |
Nephthenol
|
Others | Others |
Nephthenol shows antiproliferative activity against the cell lines HUVEC and K-562 and for cytotoxicity against the cell line HeLa. | |||
TN1764 |
Incensole acetate
|
TNF; NF-κB | Apoptosis; NF-κB |
Incensole acetate is a novel anti-inflammatory compound that inhibits NF-κB activation. |