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Search Results for " bendazol "
Targets Recommended: Dopamine Receptor NO Synthase

20

抑制剂 & 化合物

3

天然产物

9

同位素标记化合物

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Cat. No. Product Name Target Signaling Pathways
T1322 Bendazol

地巴唑,Dibazol,Dibazole

Dopamine Receptor; NO Synthase GPCR/G Protein; Immunology/Inflammation; Neuroscience
Bendazol (Dibazol) 是降压药物,能够提高 NO 合成酶在肾小球和集合小管中的活性。
T0009 Flubendazole

氟苯咪唑,Flumoxanal,Flumoxane,NSC 313680,Fluvermal

Apoptosis; Microtubule Associated; Parasite Apoptosis; Cytoskeletal Signaling; Microbiology/Virology
Flubendazole (Flumoxane) 是用于治疗人类蠕虫感染的驱虫药。它通过抑制微管功能等机制发挥抗癌作用。它诱导p53介导的细胞凋亡,抑制 G2/M 细胞周期。
T6372 Albendazole sulfoxide

Ricobendazole,Albendazole Oxide,阿苯达唑亚砜

Microtubule Associated; Parasite Cytoskeletal Signaling; Microbiology/Virology
Albendazole sulfoxide (Ricobendazole) 是一种驱虫药阿苯达唑的代谢物,有抗寄生虫活性。
T0838 Triclabendazole

三氯苯咪唑,三氯苯达唑,CGA89317

Microtubule Associated; Parasite Cytoskeletal Signaling; Microbiology/Virology
Triclabendazole (CGA89317) 是一种苯并咪唑,与微管蛋白结合,损害细胞内运输机制,且干扰蛋白质的合成。
T6623 Oxibendazole

Apoptosis; Parasite Apoptosis; Microbiology/Virology
Oxibendazole 是一种苯并咪唑驱虫药,用于防止马和一些家养宠物的蛔虫、圆线虫、线虫、蛲虫和肺虫感染。。它可诱导细胞凋亡,具有抗癌和抗炎活性。
T6071 Parbendazole

SKF 29044,帕苯咪唑

Microtubule Associated; Parasite Cytoskeletal Signaling; Microbiology/Virology
Parbendazole (SKF 29044) 是一种有效的 microtubule 重组抑制剂,能够破坏微管蛋白,EC50值为 530 nM,也是广谱驱虫剂。
T3361 Cambendazole

坎苯达唑,Bonlam,MK-905,Novazole

Others Others
Cambendazole (Novazole) 是治疗人类圆线虫病最有效的一种药物。
T38400 Triclabendazole sulfoxide

TCBZ-SO,三氯苯达唑亚砜

BCRP; Parasite Membrane transporter/Ion channel; Microbiology/Virology
Triclabendazole sulfoxide (TCBZ-SO) 是 Triclabendazole 的主要血浆代谢产物。Triclabendazole sulfoxide 具有抗寄生虫活性。Triclabendazole sulfoxide 可以抑制膜转运蛋白ABCG2/BCRP 的活性。
T1141 Fenbendazole

Fenbendazol,苯硫咪唑,芬苯达唑,Phenbendasol,Panacur

Others; HIF/HIF Prolyl-Hydroxylase; Antibiotic; Parasite Chromatin/Epigenetic; Metabolism; Microbiology/Virology; Others
Fenbendazole (Fenbendazol) 是一种广谱苯并咪唑类驱虫剂,对胃肠寄生虫有效。
T37660 5-hydroxy Thiabendazole

Others Others
5-hydroxy Thiabendazole (5-OH TBZ) is a major metabolite of the anthelmintic thiabendazole . Unlike thiabendazole, 5-OH TBZ has no effect on the growth of third-stage A. caninum larvae.
T20960 Luxabendazole

HOE 216V

Others Others
Luxabendazole is a benzimidazole carbamate broad-spectrum anthelmintic agent. It has proved to be effective against immature and adult stages of the major gastrointestinal nematodes, cestodes, and trematodes.
T21226 Albendazole sulfone

Others Others
Albendazole sulfone, a metabolite of Albendazole, is an antibiotic, anthelmintic, and antiparisitic.
T37875 Fenbendazole sulfone

Others Others
Fenbendazole sulfone is a minor metabolite of the anthelmintic fenbendazole . Fenbendazole undergoes oxidation to form oxfendazole, which is further oxidized to form fenbendazole sulfone.
T68947 Etibendazole

Others Others
Etibendazole is a microtubule inhibitor.
T23922 Cyclobendazole

R 17,147,Ciclobendazol,Ciclobendazole,CC 2481,R 17147

Others Others
Cyclobendazole is a antihelmintic agent.
T40928 2-Aminoflubendazole

Others Others
2-Aminoflubendazole, a metabolite of benzimidazoles (BZ), belongs to a class of drugs effective against fungi, protozoa, and helminths.
T29458 5-Hydroxymebendazole

R 19167,R19167,R-19167

Others Others
5-Hydroxymebendazole is a biochemical.
T32834 Lobendazole

SK&F 24529,SKF 24529,NSC-42044,NSC42044,NSC 42044

Others Others
Lobendazole is a metabolite of thiophanate.
T32109 Hybendazole hydrochloride

AT-1921,AT1921,AT 1921,Hybendazole HCl

Others Others
Hybendazole hydrochloride is a bio-active chemical.
T20528 Mebendazole-amine

R 18986,R-18986,G1029,R18986,G 1029,G-1029

Others Others
R-18986 is a biochemical substance.

化合物

Bendazol
Cat.No: T1322
Synonym: 地巴唑,Dibazol,Dibazole
Target: Dopamine Receptor, NO Synthase
Flubendazole
Cat.No: T0009
Synonym: 氟苯咪唑,Flumoxanal,Flumoxane,NSC 313680,Fluvermal
Target: Apoptosis, Microtubule Associated, Parasite
Albendazole sulfoxide
Cat.No: T6372
Synonym: Ricobendazole,Albendazole Oxide,阿苯达唑亚砜
Target: Microtubule Associated, Parasite
Triclabendazole
Cat.No: T0838
Synonym: 三氯苯咪唑,三氯苯达唑,CGA89317
Target: Microtubule Associated, Parasite
Oxibendazole
Cat.No: T6623
Synonym:
Target: Apoptosis, Parasite
Parbendazole
Cat.No: T6071
Synonym: SKF 29044,帕苯咪唑
Target: Microtubule Associated, Parasite
Cambendazole
Cat.No: T3361
Synonym: 坎苯达唑,Bonlam,MK-905,Novazole
Target: Others
Triclabendazole sulfoxide
Cat.No: T38400
Synonym: TCBZ-SO,三氯苯达唑亚砜
Target: BCRP, Parasite
Fenbendazole
Cat.No: T1141
Synonym: Fenbendazol,苯硫咪唑,芬苯达唑,Phenbendasol,Panacur
Target: Others, HIF/HIF Prolyl-Hydroxylase, Antibiotic, Parasite
5-hydroxy Thiabendazole
Cat.No: T37660
Synonym:
Target: Others
Luxabendazole
Cat.No: T20960
Synonym: HOE 216V
Target: Others
Albendazole sulfone
Cat.No: T21226
Synonym:
Target: Others
Fenbendazole sulfone
Cat.No: T37875
Synonym:
Target: Others
Etibendazole
Cat.No: T68947
Synonym:
Target: Others
Cyclobendazole
Cat.No: T23922
Synonym: R 17,147,Ciclobendazol,Ciclobendazole,CC 2481,R 17147
Target: Others
2-Aminoflubendazole
Cat.No: T40928
Synonym:
Target: Others
5-Hydroxymebendazole
Cat.No: T29458
Synonym: R 19167,R19167,R-19167
Target: Others
Lobendazole
Cat.No: T32834
Synonym: SK&F 24529,SKF 24529,NSC-42044,NSC42044,NSC 42044
Target: Others
Hybendazole hydrochloride
Cat.No: T32109
Synonym: AT-1921,AT1921,AT 1921,Hybendazole HCl
Target: Others
Mebendazole-amine
Cat.No: T20528
Synonym: R 18986,R-18986,G1029,R18986,G 1029,G-1029
Target: Others
Cat. No. Product Name Target Signaling Pathways
T1155 Mebendazole

甲苯达唑,甲苯咪唑,Telmin,Mebenvet,Vermox,Pantelmin

Apoptosis; Microtubule Associated; Parasite Apoptosis; Cytoskeletal Signaling; Microbiology/Virology
Mebendazole (Mebenvet) 是一种 hedgehog 抑制剂,用作驱虫药。
T1152 Albendazole

SKF-62979,阿苯达唑

HIF/HIF Prolyl-Hydroxylase; Microtubule Associated; Antibiotic; Parasite Chromatin/Epigenetic; Cytoskeletal Signaling; Metabolism; Microbiology/Virology
Albendazole (SKF-62979) 是一种广谱抗寄生虫剂,具有高效,低宿主毒性的特点。 它用于研究人类和动物的胃肠道寄生虫。
T0938 Thiabendazole

2-(4-Thiazolyl)benzimidazole,噻菌灵

Microtubule Associated; Mitochondrial Metabolism; Parasite Cytoskeletal Signaling; Metabolism; Microbiology/Virology
Thiabendazole (2-(4-Thiazolyl)benzimidazole) 是具有驱虫特性的苯并咪唑衍生物。

天然产物

Mebendazole
Cat.No: T1155
Synonym: 甲苯达唑,甲苯咪唑,Telmin,Mebenvet,Vermox,Pantelmin
Target: Apoptosis, Microtubule Associated, Parasite
Albendazole
Cat.No: T1152
Synonym: SKF-62979,阿苯达唑
Target: HIF/HIF Prolyl-Hydroxylase, Microtubule Associated, Antibiotic, Parasite
Thiabendazole
Cat.No: T0938
Synonym: 2-(4-Thiazolyl)benzimidazole,噻菌灵
Target: Microtubule Associated, Mitochondrial Metabolism, Parasite
Cat. No. Product Name Target Signaling Pathways
TMIJ-0484 Thiabendazole NH-d6

Thiabendazole NH-d6 是 Thiabendazole NH 的氘代化合物。Thiabendazole NH 的 CAS 号为 148-79-8。Thiabendazole 是具有驱虫特性的苯并咪唑衍生物。
T71055 Albendazole-d7

Albendazole-d7 is intended for use as an internal standard for the quantification of albendazole by GC- or LC-MS. Albendazole is an orally bioavailable benzimidazole anthelmintic that is active against a variety of helminths, including liver flukes, tapeworms, and roundworms. It eliminates Trichostrongylus in the fourth stomach of cattle and sheep when orally administered at doses ranging from 2.5 to 10 mg/kg as well as other species in the fourth stomach and the small and large intestine. Alben...
T19184 Albendazole sulfoxide D3

Albendazole oxide D3,Ricobendazole D3

Others Others
Albendazole sulfoxide D3 is deuterium-labeled Albendazole sulfoxide. Albendazole sulfoxide is a broad-spectrum anthelmintic.
TMIH-0570 Thiabendazole-d4

Thiabendazole-d4 是 Thiabendazole 的氘代化合物。
TMIJ-0295 Flubendazole-d3 (methyl-d3)

Flubendazole-d3 (methyl-d3) 是 Flubendazole 的氘代化合物。Flubendazole 的 CAS 号为 31430-15-6。Flubendazole 是用于治疗人类蠕虫感染的驱虫药。它通过抑制微管功能等机制发挥抗癌作用。它诱导p53介导的细胞凋亡,抑制 G2/M 细胞周期。
T19183 Albendazole-d3

Albendazole D3

Others Others
Albendazole D3 is the deuterium-labeled Albendazole. Albendazole is used as a drug indicated for the treatment of a variety of worm infestations.
TMIJ-0471 Mebendazole-d3

Mebendazole-d3 是 Mebendazole 的氘代化合物。Mebendazole 的 CAS 号为 31431-39-7。Mebendazole是一种hedgehog抑制剂,用作驱虫药。
TMIJ-0307 Fenbendazole-d3

Fenbendazole-d3 是 Fenbendazole 的氘代化合物。Fenbendazole 的 CAS 号为 43210-67-9。Fenbendazole是一种广谱苯并咪唑类驱虫剂,对胃肠寄生虫有效。
TMIH-0077 Albendazole sulfone-d3

Albendazole sulfone-d3 是 Albendazole sulfone 的氘代化合物。

同位素标记化合物

Thiabendazole NH-d6
Cat.No: TMIJ-0484
Synonym:
Target:
Albendazole-d7
Cat.No: T71055
Synonym:
Target:
Albendazole sulfoxide D3
Cat.No: T19184
Synonym: Albendazole oxide D3,Ricobendazole D3
Target: Others
Thiabendazole-d4
Cat.No: TMIH-0570
Synonym:
Target:
Flubendazole-d3 (methyl-d3)
Cat.No: TMIJ-0295
Synonym:
Target:
Albendazole-d3
Cat.No: T19183
Synonym: Albendazole D3
Target: Others
Mebendazole-d3
Cat.No: TMIJ-0471
Synonym:
Target:
Fenbendazole-d3
Cat.No: TMIJ-0307
Synonym:
Target:
Albendazole sulfone-d3
Cat.No: TMIH-0077
Synonym:
Target:
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