20
3
9
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1322 |
Bendazol
地巴唑,Dibazol,Dibazole |
Dopamine Receptor; NO Synthase | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Bendazol (Dibazol) 是降压药物,能够提高 NO 合成酶在肾小球和集合小管中的活性。 | |||
T0009 |
Flubendazole
氟苯咪唑,Flumoxanal,Flumoxane,NSC 313680,Fluvermal |
Apoptosis; Microtubule Associated; Parasite | Apoptosis; Cytoskeletal Signaling; Microbiology/Virology |
Flubendazole (Flumoxane) 是用于治疗人类蠕虫感染的驱虫药。它通过抑制微管功能等机制发挥抗癌作用。它诱导p53介导的细胞凋亡,抑制 G2/M 细胞周期。 | |||
T6372 |
Albendazole sulfoxide
Ricobendazole,Albendazole Oxide,阿苯达唑亚砜 |
Microtubule Associated; Parasite | Cytoskeletal Signaling; Microbiology/Virology |
Albendazole sulfoxide (Ricobendazole) 是一种驱虫药阿苯达唑的代谢物,有抗寄生虫活性。 | |||
T0838 |
Triclabendazole
三氯苯咪唑,三氯苯达唑,CGA89317 |
Microtubule Associated; Parasite | Cytoskeletal Signaling; Microbiology/Virology |
Triclabendazole (CGA89317) 是一种苯并咪唑,与微管蛋白结合,损害细胞内运输机制,且干扰蛋白质的合成。 | |||
T6623 |
Oxibendazole
|
Apoptosis; Parasite | Apoptosis; Microbiology/Virology |
Oxibendazole 是一种苯并咪唑驱虫药,用于防止马和一些家养宠物的蛔虫、圆线虫、线虫、蛲虫和肺虫感染。。它可诱导细胞凋亡,具有抗癌和抗炎活性。 | |||
T6071 |
Parbendazole
SKF 29044,帕苯咪唑 |
Microtubule Associated; Parasite | Cytoskeletal Signaling; Microbiology/Virology |
Parbendazole (SKF 29044) 是一种有效的 microtubule 重组抑制剂,能够破坏微管蛋白,EC50值为 530 nM,也是广谱驱虫剂。 | |||
T3361 |
Cambendazole
坎苯达唑,Bonlam,MK-905,Novazole |
Others | Others |
Cambendazole (Novazole) 是治疗人类圆线虫病最有效的一种药物。 | |||
T38400 |
Triclabendazole sulfoxide
TCBZ-SO,三氯苯达唑亚砜 |
BCRP; Parasite | Membrane transporter/Ion channel; Microbiology/Virology |
Triclabendazole sulfoxide (TCBZ-SO) 是 Triclabendazole 的主要血浆代谢产物。Triclabendazole sulfoxide 具有抗寄生虫活性。Triclabendazole sulfoxide 可以抑制膜转运蛋白ABCG2/BCRP 的活性。 | |||
T1141 |
Fenbendazole
Fenbendazol,苯硫咪唑,芬苯达唑,Phenbendasol,Panacur |
Others; HIF/HIF Prolyl-Hydroxylase; Antibiotic; Parasite | Chromatin/Epigenetic; Metabolism; Microbiology/Virology; Others |
Fenbendazole (Fenbendazol) 是一种广谱苯并咪唑类驱虫剂,对胃肠寄生虫有效。 | |||
T37660 |
5-hydroxy Thiabendazole
|
Others | Others |
5-hydroxy Thiabendazole (5-OH TBZ) is a major metabolite of the anthelmintic thiabendazole . Unlike thiabendazole, 5-OH TBZ has no effect on the growth of third-stage A. caninum larvae. | |||
T20960 |
Luxabendazole
HOE 216V |
Others | Others |
Luxabendazole is a benzimidazole carbamate broad-spectrum anthelmintic agent. It has proved to be effective against immature and adult stages of the major gastrointestinal nematodes, cestodes, and trematodes. | |||
T21226 |
Albendazole sulfone
|
Others | Others |
Albendazole sulfone, a metabolite of Albendazole, is an antibiotic, anthelmintic, and antiparisitic. | |||
T37875 |
Fenbendazole sulfone
|
Others | Others |
Fenbendazole sulfone is a minor metabolite of the anthelmintic fenbendazole . Fenbendazole undergoes oxidation to form oxfendazole, which is further oxidized to form fenbendazole sulfone. | |||
T68947 |
Etibendazole
|
Others | Others |
Etibendazole is a microtubule inhibitor. | |||
T23922 |
Cyclobendazole
R 17,147,Ciclobendazol,Ciclobendazole,CC 2481,R 17147 |
Others | Others |
Cyclobendazole is a antihelmintic agent. | |||
T40928 |
2-Aminoflubendazole
|
Others | Others |
2-Aminoflubendazole, a metabolite of benzimidazoles (BZ), belongs to a class of drugs effective against fungi, protozoa, and helminths. | |||
T29458 |
5-Hydroxymebendazole
R 19167,R19167,R-19167 |
Others | Others |
5-Hydroxymebendazole is a biochemical. | |||
T32834 |
Lobendazole
SK&F 24529,SKF 24529,NSC-42044,NSC42044,NSC 42044 |
Others | Others |
Lobendazole is a metabolite of thiophanate. | |||
T32109 |
Hybendazole hydrochloride
AT-1921,AT1921,AT 1921,Hybendazole HCl |
Others | Others |
Hybendazole hydrochloride is a bio-active chemical. | |||
T20528 |
Mebendazole-amine
R 18986,R-18986,G1029,R18986,G 1029,G-1029 |
Others | Others |
R-18986 is a biochemical substance. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1155 |
Mebendazole
甲苯达唑,甲苯咪唑,Telmin,Mebenvet,Vermox,Pantelmin |
Apoptosis; Microtubule Associated; Parasite | Apoptosis; Cytoskeletal Signaling; Microbiology/Virology |
Mebendazole (Mebenvet) 是一种 hedgehog 抑制剂,用作驱虫药。 | |||
T1152 |
Albendazole
SKF-62979,阿苯达唑 |
HIF/HIF Prolyl-Hydroxylase; Microtubule Associated; Antibiotic; Parasite | Chromatin/Epigenetic; Cytoskeletal Signaling; Metabolism; Microbiology/Virology |
Albendazole (SKF-62979) 是一种广谱抗寄生虫剂,具有高效,低宿主毒性的特点。 它用于研究人类和动物的胃肠道寄生虫。 | |||
T0938 |
Thiabendazole
2-(4-Thiazolyl)benzimidazole,噻菌灵 |
Microtubule Associated; Mitochondrial Metabolism; Parasite | Cytoskeletal Signaling; Metabolism; Microbiology/Virology |
Thiabendazole (2-(4-Thiazolyl)benzimidazole) 是具有驱虫特性的苯并咪唑衍生物。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TMIJ-0484 |
Thiabendazole NH-d6
|
||
Thiabendazole NH-d6 是 Thiabendazole NH 的氘代化合物。Thiabendazole NH 的 CAS 号为 148-79-8。Thiabendazole 是具有驱虫特性的苯并咪唑衍生物。 | |||
T71055 |
Albendazole-d7
|
||
Albendazole-d7 is intended for use as an internal standard for the quantification of albendazole by GC- or LC-MS. Albendazole is an orally bioavailable benzimidazole anthelmintic that is active against a variety of helminths, including liver flukes, tapeworms, and roundworms. It eliminates Trichostrongylus in the fourth stomach of cattle and sheep when orally administered at doses ranging from 2.5 to 10 mg/kg as well as other species in the fourth stomach and the small and large intestine. Alben... | |||
T19184 |
Albendazole sulfoxide D3
Albendazole oxide D3,Ricobendazole D3 |
Others | Others |
Albendazole sulfoxide D3 is deuterium-labeled Albendazole sulfoxide. Albendazole sulfoxide is a broad-spectrum anthelmintic. | |||
TMIH-0570 |
Thiabendazole-d4
|
||
Thiabendazole-d4 是 Thiabendazole 的氘代化合物。 | |||
TMIJ-0295 |
Flubendazole-d3 (methyl-d3)
|
||
Flubendazole-d3 (methyl-d3) 是 Flubendazole 的氘代化合物。Flubendazole 的 CAS 号为 31430-15-6。Flubendazole 是用于治疗人类蠕虫感染的驱虫药。它通过抑制微管功能等机制发挥抗癌作用。它诱导p53介导的细胞凋亡,抑制 G2/M 细胞周期。 | |||
T19183 |
Albendazole-d3
Albendazole D3 |
Others | Others |
Albendazole D3 is the deuterium-labeled Albendazole. Albendazole is used as a drug indicated for the treatment of a variety of worm infestations. | |||
TMIJ-0471 |
Mebendazole-d3
|
||
Mebendazole-d3 是 Mebendazole 的氘代化合物。Mebendazole 的 CAS 号为 31431-39-7。Mebendazole是一种hedgehog抑制剂,用作驱虫药。 | |||
TMIJ-0307 |
Fenbendazole-d3
|
||
Fenbendazole-d3 是 Fenbendazole 的氘代化合物。Fenbendazole 的 CAS 号为 43210-67-9。Fenbendazole是一种广谱苯并咪唑类驱虫剂,对胃肠寄生虫有效。 | |||
TMIH-0077 |
Albendazole sulfone-d3
|
||
Albendazole sulfone-d3 是 Albendazole sulfone 的氘代化合物。 |