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Cat. No.	Product Name	Target	Signaling Pathways
T50022	BRD4 Inhibitor 30	Others	Others
	4-(2-fluorophenyl)-2,3-dihydro-1,3-thiazol-2-one 是一种噻唑-2-酮类化合物，被发现具有抗炎、抗细菌、抗真菌和抗肿瘤等活性。
T16154	MS417 GTPL7512	Epigenetic Reader Domain; HIV Protease	Chromatin/Epigenetic; Microbiology/Virology; Proteases/Proteasome
	MS417 (GTPL7512) 是一种 BET 特异性 BRD4 抑制剂，与 BRD4-BD1 和 BRD4-BD2 结合，Kd 值分别为 36.1和25.4 nM，IC50值分别为 30和46 nM。它对 CBP BRD 的选择性较低，IC50值为 32.7 μM。
T1854	MS436	Epigenetic Reader Domain	Chromatin/Epigenetic
	MS436 是溴结构域抑制剂，作用于 BRD4 BrD1的Ki 为 30 到 50 nM 之间，比作用于 BrD2 选择性高 10 倍。
T38381	CAY17c	Others	Others
	CAY17c is an inhibitor of bromodomain-containing protein 4 (BRD4; IC50= 0.71 μM), as well as class I histone deacetylases (HDACs; IC50s = 0.046, 0.058, 0.075, and 0.167 μM for HDAC1, -2, -3, and -8, respectively) and class IIb HDACs (IC50s = 0.073 and 0.923 μM for HDAC6 and HDAC10, respectively).1It is selective for these enzymes over BRD2, -3, and -T (IC50s = >20 μM for all), as well as over HDAC4, -5, -7, -9, and -11 (IC50s = >10 μM for all). CAY17c inhibits the proliferation of HCT116, SW620,...