Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T26800 |
BIBO3304
BIBO-3304,BIBO 3304 |
Others | Others |
BIBO3304 is a selective NPY Y1 receptor antagonist (IC50 values are 0.38 and 0.72 nM at human and rat receptors respectively). BIBO3304 inhibits NPY- and fasting-induced feeding in vivo following central administration. | |||
T10539 |
BIBO3304 TFA
|
Neuropeptide Y Receptor | GPCR/G Protein; Neuroscience |
BIBO3304 TFA 是一种可口服的、选择性的神经肽 Y(NPY) Y1受体高效拮抗剂,对人和大鼠 Y1 受体均具有高亲和力,IC50分别为 0.38 和 0.72 nM。 | |||
T84889 |
BIBO3304 diTFA
|
Others | Others |
BIBO3304 (diTFA) 是口服有效、选择性的神经肽Y(NPY)Y1受体高效拮抗剂。对人类及大鼠Y1受体具高亲和力,IC50值分别为0.38和0.72 nM。BIBO3304 (diTFA) 通过Wnt/β-catenin信号通路促进骨肌腱愈合。 |