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Search Results for " antibiotic "
Targets Recommended: Antibiotic Antibacterial Antibiotic

1121

抑制剂 & 化合物

376

天然产物

4

化合物库

1

TargetMol 试剂盒

6

重组蛋白

48

同位素标记化合物

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Cat. No. Product Name
L4400 抗生素库

692 compounds
692 个具有抗菌活性化合物的独特集合,是医药研究的优良工具库和药物筛选的有效载体;
L4520 抗菌活性库

904 compounds
904 种具有抗菌活性的化合物,是抗菌药物研发的有力工具;
L6500 微生物天然产物库

550 compounds
550 种微生物来源的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
L6820 烟草单体化合物库

747 compounds
747种烟草单体化合物的独特集合,可用于高通量筛选和高内涵筛选

化合物库

抗生素库
Cat.No: L4400
Compounds: 692
抗菌活性库
Cat.No: L4520
Compounds: 904
微生物天然产物库
Cat.No: L6500
Compounds: 550
烟草单体化合物库
Cat.No: L6820
Compounds: 747
Cat. No. Product Name Form Specificity Of Inhibition
C0051 Penicillin-Streptomycin Solution (100×), Sterile

青霉素-链霉素双抗溶液(100×),灭菌

Solution in bottle

TargetMol 试剂盒

青霉素-链霉素双抗溶液(100×),灭菌
Cat.No: C0051
Cat. No. Product Name Target Signaling Pathways
T4084 Sibofimloc

VRT-1353385,Antibiotic-202,Antibiotic 202

Antibacterial; Antibiotic Microbiology/Virology
Sibofimloc (Antibiotic-202) 是一种肠道限制性的,具有口服活性的 FimH 粘附抑制剂,有抗细菌感染活性,被开发用于治疗炎症性肠病的研究。
T26634 Antibiotic A396I

A-396I,Antibiotic A 396I,A 396I,A396I

Others Others
Antibiotic A396I is a biochemical.
T25095 Antibiotic LB 10517

LB 10517,LB10517,Antibiotic LB10517,LB-10517,Antibiotic LB-10517

Others Others
Antibiotic LB 10517 is a catechol-substituted cephalosporin with a broad spectrum of antibacterial.
T0967 Teicoplanin

Antibiotic MDL-507,MDL-507,替考拉宁,Teichomycin

Antibacterial; Antibiotic Microbiology/Virology
Teicoplanin (MDL-507) 是一种半合成的糖肽抗生素, 可用于由革兰氏阳性菌引起的严重感染的相关研究。
T10330 Antibiotic-5d

Antibacterial Microbiology/Virology
Antibiotic-5d 是一种合成的抗菌化合物,对各种革兰氏阳性和革兰氏阴性细菌、真菌和酵母表现出中等的抗菌活性。
T68946 Antibiotic MA 144M1

Others Others
Antibiotic MA 144M1 is an anthracycline glycoside that inhibits the growth of gram-positive bacteria, e.g. Staphyococcus aureaus, Bacillus subtilis and Sarcina lutea, and inhibits the growth of animal tumors such as leukemia L 1210, P 388 and sarcoma 180. It's produced by fermentation of MA 144-producing strains of streptomyces and by the chemical or enzymatic conversion of aclacinomycin A or cinerubin A.
T68945 Antibiotic MA 144M2

Others Others
Antibiotic MA 144M2 is an anthracycline glycoside that inhibits the growth of gram-positive bacteria, e.g. Staphyococcus aureaus, Bacillus subtilis and Sarcina lutea, and inhibits the growth of animal tumors such as leukemia L 1210, P 388 and sarcoma 180. It's produced by fermentation of MA 144-producing strains of streptomyces and by the chemical or enzymatic conversion of aclacinomycin A or cinerubin A.
T24612 Pentachloropseudilin

PClP,Antibiotic A 15104 Y

Myosin; Antibiotic; TGF-beta/Smad Cytoskeletal Signaling; Microbiology/Virology; Stem Cells
Pentachloropseudilin (PClP) 是一种可逆的变构 1 型肌球蛋白抑制剂,具有抗菌活性,抑制 Myo1s 和 5 类肌球蛋白。Pentachloropseudilin 抑制生长因子-β (TGF-β) ,可阻断克氏锥虫对宿主细胞的侵袭。
T25097 Antibiotic tan-592B

TAN592B,Cephabacin F5 hydrochloride,TAN 592B,TAN-592B

Others Others
Antibiotic tan-592B is an antibiotic agent.
T25096 Antibiotic SF 2132

SF2132,SF-2132,SF 2132

Others Others
Antibiotic SF 2132 is a bioactive chemical.
T16073 Micronomicin

小诺霉素,Gentamicin C2b,Antibiotic XK-62-2,Sagamicin

Others; Antibacterial Microbiology/Virology; Others
Micronomicin (Gentamicin C2b) 是一种具有抗菌和杀菌能力的抗生素。
T23740 Antibiotic 273 A2-beta

Others Others
Antibiotic 273 A2-beta is a bioactive chemical.
T16886 Sinefungin

Adenosyl-Ornithine,西奈芬净,A-9145,Antibiotic 32232RP

Others; Histone Methyltransferase; Antibiotic; Antifungal Chromatin/Epigenetic; Microbiology/Virology; Others
Sinefungin (Adenosyl-Ornithine) 是病毒粒子mRNA (鸟嘌呤-7-)-甲基转移酶、 mRNA (核苷-2'-)-甲基转移酶和病毒增殖的有效抑制剂。它还抑制SET7/9,通过抑制H3K4甲基化来改善肾纤维化。
T26633 Antibiotic A 40104A

A 40104A,A40104A,A-40104A

Others Others
Antibiotic A 40104A is an antibiotic.
T25094 Antibiotic K 4

I5B1,I5 B1,K-4,K4,I5-B1

Others Others
Antibiotic K 4 is an inhibitor of angiotensin I converting enzyme produced by Actinomadura spiculosospora.
T23742 Antibiotic YC 17

YC 17,YC-17,YC17

Others Others
Antibiotic YC 17 is a biochemical agent.
T23744 Antibiotic Z-1159-2

Z-1159-2

Others Others
Antibiotic Z-1159-2 is an agent of biochemical.
T23743 Antibiotic Z-1159-1

Z-1159-1

Others Others
Antibiotic Z-1159-1 is an agent of biochemical.
T12092 Monacolin J

Antibiotic MB 530A,Lovastatin diol lactone,辛伐他汀内酯二醇

HMG-CoA Reductase; Autophagy Autophagy; Metabolism
Monacolin J (Antibiotic MB 530A) 是一种胆固醇生物合成抑制剂,抑制 HMG-CoA 还原酶的活性。
T125527 Antibiotic 2158

Others Others
Antibiotic 2158 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125527。
T125208 Antibiotic WB

Others Others
Antibiotic WB 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125208,CAS号为 247919-66-0。
T1910 Ansamitocin P 3'

Maytansinol butyrate,Ansamitocin P-3,安丝菌素P-3,Antibiotic C 15003P3'

Microtubule Associated Cytoskeletal Signaling
Ansamitocin P 3' (Maytansinol butyrate) 是一种具有抗肿瘤活性的抗体-药物偶联细胞毒素。
T125021 Antibiotic Sch 378167

Others Others
Antibiotic Sch 378167 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125021,CAS号为 336108-99-7。
T124135 Antibiotic SB 202742

Others Others
Antibiotic SB 202742 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124135,CAS号为 83173-24-4。
T125547 Antibiotic FF 8181A

Others Others
Antibiotic FF 8181A 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125547,CAS号为 179118-87-7。
T6179 Moxalactam sodium salt

Latamoxef sodium,6059 S,拉氧头孢钠,Moxalactam Disodium,LY-127935,Antibiotic 6059S,Shiomarin,FestamoxinLy

Antibacterial; Antibiotic Microbiology/Virology
Moxalactam sodium salt (LY-127935) 是一种抗生素, 对大肠杆菌和绿脓杆菌有作用。
T126064 Antibiotic PF 1018

Others Others
Antibiotic PF 1018 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T126064。
T73678 Antibiotic DC 81

Others Others
AntibioticDC 81(DC 81)是由链霉菌产生的一种抗肿瘤抗生素,属于吡咯[2,1-c][1,4]苯二氮平(PBD)类。作为一种有效的核酸合成抑制剂,AntibioticDC 81通过识别并与特定DNA序列结合,形成不稳定的共价加合物。
T123925 Antibiotic LL-D253alpha

Others Others
Antibiotic LL-D253alpha 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T123925,CAS号为 92589-99-6。
T124885 Antibiotic LL-P880y

Others Others
Antibiotic LL-P880y 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124885,CAS号为 41206-21-7。
T126422 Antibiotic F01-1358B

Others Others
Antibiotic F01-1358B 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126422,CAS号为 1095602-46-2。
T125813 Antibiotic TAN 1446A

Others Others
Antibiotic TAN 1446A 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125813,CAS号为 148084-27-9。
T125406 Antibiotic Sch 60059

Others Others
Antibiotic Sch 60059 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125406,CAS号为 203061-30-7。
T125507 Antibiotic XR 586

Others Others
Antibiotic XR 586 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125507,CAS号为 185981-24-2。
T125528 Antibiotic ZG 1494alpha

Others Others
Antibiotic ZG 1494alpha 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125528。
T125699 Antibiotic AB 4063B

Others Others
Antibiotic AB 4063B 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125699。
T125403 Antibiotic Sch 60057

Others Others
Antibiotic Sch 60057 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125403,CAS号为 203061-35-2。
T125405 Antibiotic Sch 60065

Others Others
Antibiotic Sch 60065 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125405,CAS号为 203061-31-8。
T126295 Antibiotic JBIR 27

Others Others
Antibiotic JBIR 27 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126295,CAS号为 1172094-65-3。
T124209 Antibiotic L 783277

Others Others
Antibiotic L 783277 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124209,CAS号为 791807-02-8。
T125647 Antibiotic NFAT 133

Others Others
Antibiotic NFAT 133 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125647,CAS号为 165133-85-7。
T125404 Antibiotic Sch 60061

Others Others
Antibiotic Sch 60061 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125404,CAS号为 203061-33-0。
T125657 Antibiotic AB 4015B

Others Others
Antibiotic AB 4015B 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125657。
T125708 Antibiotic F 1839A

Others Others
Antibiotic F 1839A 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125708,CAS号为 159096-43-2。
T124954 Antibiotic AGI-B4

Others Others
Antibiotic AGI-B4 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124954,CAS号为 359828-18-5。
T123922 Antibiotic JM 971B

Others Others
Antibiotic JM 971B 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T123922,CAS号为 92802-16-9。
T125005 Antibiotic LL-D253gamma

Others Others
Antibiotic LL-D253gamma 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125005,CAS号为 34288-35-2。
T21475 Netropsin

Congocidin,Antibiotic T 1384,Antibiotic 1142,Antibiotic T-1384,Sinanomycin,Antibiotic T1384

Others Others
Netropsin is a basic polypeptide isolated from Streptomyces netropsis with antibiotic and antiviral activity. It is strong, specific binding to A-T areas of DNA is useful to genetics research. Netropsin is active against Gram-negative bacteria and Gram-po
T124003 Antibiotic OM 173?2

Others Others
Antibiotic OM 173?2 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124003,CAS号为 88293-10-1。
T25991 Promothiocin A

Antibiotic SF2741A,Antibiotic SF 2741A,Antibiotic SF-2741A

Others Others
Promothiocin A is an antibiotic.

化合物

Sibofimloc
Cat.No: T4084
Synonym: VRT-1353385,Antibiotic-202,Antibiotic 202
Target: Antibacterial, Antibiotic
Antibiotic A396I
Cat.No: T26634
Synonym: A-396I,Antibiotic A 396I,A 396I,A396I
Target: Others
Antibiotic LB 10517
Cat.No: T25095
Synonym: LB 10517,LB10517,Antibiotic LB10517,LB-10517,Antibiotic LB-10517
Target: Others
Teicoplanin
Cat.No: T0967
Synonym: Antibiotic MDL-507,MDL-507,替考拉宁,Teichomycin
Target: Antibacterial, Antibiotic
Antibiotic-5d
Cat.No: T10330
Synonym:
Target: Antibacterial
Antibiotic MA 144M1
Cat.No: T68946
Synonym:
Target: Others
Antibiotic MA 144M2
Cat.No: T68945
Synonym:
Target: Others
Pentachloropseudilin
Cat.No: T24612
Synonym: PClP,Antibiotic A 15104 Y
Target: Myosin, Antibiotic, TGF-beta/Smad
Antibiotic tan-592B
Cat.No: T25097
Synonym: TAN592B,Cephabacin F5 hydrochloride,TAN 592B,TAN-592B
Target: Others
Antibiotic SF 2132
Cat.No: T25096
Synonym: SF2132,SF-2132,SF 2132
Target: Others
Micronomicin
Cat.No: T16073
Synonym: 小诺霉素,Gentamicin C2b,Antibiotic XK-62-2,Sagamicin
Target: Others, Antibacterial
Antibiotic 273 A2-beta
Cat.No: T23740
Synonym:
Target: Others
Sinefungin
Cat.No: T16886
Synonym: Adenosyl-Ornithine,西奈芬净,A-9145,Antibiotic 32232RP
Target: Others, Histone Methyltransferase, Antibiotic, Antifungal
Antibiotic A 40104A
Cat.No: T26633
Synonym: A 40104A,A40104A,A-40104A
Target: Others
Antibiotic K 4
Cat.No: T25094
Synonym: I5B1,I5 B1,K-4,K4,I5-B1
Target: Others
Antibiotic YC 17
Cat.No: T23742
Synonym: YC 17,YC-17,YC17
Target: Others
Antibiotic Z-1159-2
Cat.No: T23744
Synonym: Z-1159-2
Target: Others
Antibiotic Z-1159-1
Cat.No: T23743
Synonym: Z-1159-1
Target: Others
Monacolin J
Cat.No: T12092
Synonym: Antibiotic MB 530A,Lovastatin diol lactone,辛伐他汀内酯二醇
Target: HMG-CoA Reductase, Autophagy
Antibiotic 2158
Cat.No: T125527
Synonym:
Target: Others
Antibiotic WB
Cat.No: T125208
Synonym:
Target: Others
Ansamitocin P 3'
Cat.No: T1910
Synonym: Maytansinol butyrate,Ansamitocin P-3,安丝菌素P-3,Antibiotic C 15003P3'
Target: Microtubule Associated
Antibiotic Sch 378167
Cat.No: T125021
Synonym:
Target: Others
Antibiotic SB 202742
Cat.No: T124135
Synonym:
Target: Others
Antibiotic FF 8181A
Cat.No: T125547
Synonym:
Target: Others
Moxalactam sodium salt
Cat.No: T6179
Synonym: Latamoxef sodium,6059 S,拉氧头孢钠,Moxalactam Disodium,LY-127935,Antibiotic 6059S,Shiomarin,FestamoxinLy
Target: Antibacterial, Antibiotic
Antibiotic PF 1018
Cat.No: T126064
Synonym:
Target: Others
Antibiotic DC 81
Cat.No: T73678
Synonym:
Target: Others
Antibiotic LL-D253alpha
Cat.No: T123925
Synonym:
Target: Others
Antibiotic LL-P880y
Cat.No: T124885
Synonym:
Target: Others
Antibiotic F01-1358B
Cat.No: T126422
Synonym:
Target: Others
Antibiotic TAN 1446A
Cat.No: T125813
Synonym:
Target: Others
Antibiotic Sch 60059
Cat.No: T125406
Synonym:
Target: Others
Antibiotic XR 586
Cat.No: T125507
Synonym:
Target: Others
Antibiotic ZG 1494alpha
Cat.No: T125528
Synonym:
Target: Others
Antibiotic AB 4063B
Cat.No: T125699
Synonym:
Target: Others
Antibiotic Sch 60057
Cat.No: T125403
Synonym:
Target: Others
Antibiotic Sch 60065
Cat.No: T125405
Synonym:
Target: Others
Antibiotic JBIR 27
Cat.No: T126295
Synonym:
Target: Others
Antibiotic L 783277
Cat.No: T124209
Synonym:
Target: Others
Antibiotic NFAT 133
Cat.No: T125647
Synonym:
Target: Others
Antibiotic Sch 60061
Cat.No: T125404
Synonym:
Target: Others
Antibiotic AB 4015B
Cat.No: T125657
Synonym:
Target: Others
Antibiotic F 1839A
Cat.No: T125708
Synonym:
Target: Others
Antibiotic AGI-B4
Cat.No: T124954
Synonym:
Target: Others
Antibiotic JM 971B
Cat.No: T123922
Synonym:
Target: Others
Antibiotic LL-D253gamma
Cat.No: T125005
Synonym:
Target: Others
Netropsin
Cat.No: T21475
Synonym: Congocidin,Antibiotic T 1384,Antibiotic 1142,Antibiotic T-1384,Sinanomycin,Antibiotic T1384
Target: Others
Antibiotic OM 173?2
Cat.No: T124003
Synonym:
Target: Others
Promothiocin A
Cat.No: T25991
Synonym: Antibiotic SF2741A,Antibiotic SF 2741A,Antibiotic SF-2741A
Target: Others
Cat. No. Product Name Target Signaling Pathways
T38097 Antibiotic PF 1052

Others Others
Antibiotic PF 1052 is a fungal metabolite originally isolated from Phoma.1,2 It is active against S. aureus, S. parvulus, and C. perfringens (MICs = 3.13, 0.78, and 0.39 μg/ml, respectively), among others.1 It inhibits neutrophil migration in a wound assay using zebrafish larvae expressing GFP-labeled neutrophils, reducing pseudopodia formation and inducing rounding of neutrophils.2 Antibiotic PF 1052 is selective for neutrophil migration over macrophage migration in zebrafish larvae. It also in...
T22262 Ansamitocin p-3

Maytansinol isobutyrate,Antibiotic C 15003P3,NSC292222

Microtubule Associated; ADC Cytotoxin Antibody-drug Conjugate/ADC Related; Cytoskeletal Signaling
Ansamitocin p-3 (Maytansinol isobutyrate) 是一种微管抑制剂,对微管蛋白聚合的 IC50 为 3.4 μM。
T15717 Lasalocid

Lasalocid-A,Antibiotic X-537A,Ionophore X-537A

Antibacterial Microbiology/Virology
Lasalocid (Lasalocid-A) 是一种由链霉菌产生的离子载体抗生素,具有抗菌和寄生虫作用,常添加进饲料中。
T10662L Calcimycin

Antibiotic A-23187,离子载体(钙镁盐混合物),A-23187

Apoptosis; Antibacterial; Antibiotic; Autophagy; Antifungal Apoptosis; Autophagy; Microbiology/Virology
Calcimycin (A-23187) 是抗生素和二价阳离子离子载体。它抑制革兰氏阳性细菌和一些真菌生长,也抑制 ATP 酶的活性并解耦哺乳动物细胞的氧化磷酸化。它通过增加细胞内钙浓度诱导 Ca2+依赖性细胞死亡。
T6512 G-418 disulfate

Geneticin,G418 Sulfate,Antibiotic G-418 sulfate,遗传霉素,Geneticin sulfate

Antibacterial; Antibiotic Microbiology/Virology
G-418 disulfate (Geneticin sulfate) 属于氨基糖苷类抗生素,是一种蛋白质合成的抑制剂,具有真核细胞选择性。G-418 disulfate 通过抑制肽链的延伸来阻断多肽合成。
T6680 Staurosporine

Antibiotic AM-2282,星形孢菌素,AM-2282,CGP 41251,星孢菌素

Apoptosis; PKA; Antibacterial; Antibiotic; Src; PKC; Antifungal Angiogenesis; Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology; Tyrosine Kinase/Adaptors
Staurosporine (AM-2282) 是一种蛋白激酶抑制剂,对 PKC、PKA、c-Fgr、Phosphorylase kinase 和 TAOK2 均有抑制活性 (IC50=6/15/2/3/3000 nM),具有 ATP 竞争性和非选择性。Staurosporine 也可以诱导凋亡。
T5037 Midecamycin

Antibiotic SF-837,Turimycin P3,Medecamycin A1,Rubimycin,麦迪霉素,Platenomycin B1,Espinomycin A

Antibacterial; Antibiotic Microbiology/Virology
Midecamycin (Medecamycin A1) 是乙酰氧基取代的大环内酯类抗生素,对革兰氏阳性和阴性菌有效。
T23741 Antibiotic JI 20A

JI-20 A,BRN 1668513,BRN-1668513,BRN1668513

Others Others
Antibiotic JI 20A is a bioactive chemical.
T15716 Lasalocid sodium

拉沙洛西钠,拉沙里菌素,Ionophore X-537A sodium,Antibiotic X-537A sodium,Lasalocid-A sodium

Antibacterial; Antibiotic; Autophagy Autophagy; Microbiology/Virology
Lasalocid sodium (Lasalocid-A sodium) 是一种抗菌剂。
T26590 Albofungin

Antibiotic P42-1,Antibiotic P42-C

Others Others
Albofungin is a xanthone isolated from A. tumemacerans.
T36417 Nargenicin

Antibiotic 47444

Others Others
Nargenicin is a macrolide antibiotic that selectively inhibits the growth of S. aureus, methicilin resistant S. aureus (MRSA), and M. luteus (MICs = 0.6, 0.3, and 2.5 μg/ml, respectively) over a panel of 11 Gram-positive and Gram-negative bacteria (MICs = >80 μg/ml). [1] It dose-dependently inhibits S. aureus DnaE in the presence of DNase I-activated DNA and E. coli DnaE when used at concentrations of 0.00001-0.1 and 0.01-100 μg/mL, respectively. [2] In murine BV-2 microglial cells, nargenicin (...
T15636 K-252a

Antibiotic K 252a,Antibiotic SF 2370,SF2370

Others Others
K-252a is a staurosporine analog isolated from Nocardiopsis sp. soil fungi. K-252a inhibits protein kinase (IC50: 470 nM, 140 nM, 270 nM, and 1.7 nM for PKC, PKA, Ca2+/calmodulin-dependent kinase type II, and phosphorylase kinase, respectively).
T24253 Kazusamycin A

Antibiotic CL1957B,PD 114721,Antibiotic 81-484

Others Others
Kazusamycin A is a new antitumor antibiotic.
TN7517 Benanomicin B

Antibiotic BU 3608C

Others Others
The compound exhibits excellent antifungal and antiviral activities, including against HIV.
T25563 K 41

K-41,K41,Antibiotic K-41A,37454 RP,Antibiotic A 32887

Others Others
K 41 is a polycyclic polyether antibiotic from Streptomyces hygroscopicus.
TN7525 Parvodicin C2

Antibiotic A40926 B1

Others Others
Parvodicin C2, a glycopeptide antibiotic derived from A. parvosata and part of the parvodicin complex, serves as a component of the A40926 antibiotic complex utilized as a precursor for synthesizing dalbavancin. It exhibits activity against methicillin-sensitive and methicillin-resistant strains of S. aureus, S. epidermidis, S. saprophyticus, S. hemolyticus, and E. faecalis.
T26321 Virustomycin A

Antibiotic AM-2604 A

Others Others
Virustomycin A is an antibiotic.
T24026 Safracin B

Antibiotic Y 16482-alpha,EM 5519,EM-5519,EM5519,Antibiotic EM 5519

Others Others
EM 5519 is an antitumor antibiotic.
T26405 A 201A

Antibiotic 201A,A201A,A-201A

Others Others
A 201A is a nucleoside antibiotic, it is isolated from Streptomyces capreolus.
TN7268 Milbemycin A4

Antibiotic B 41A4,Milbemycin α3

Others Others
Milbemycin A4, a distinguished member of the macrocyclic lactones family featuring a unique spiroketal group, is derived from the fermentation of the soil bacterium Streptomyces hygroscopicus subsp. aureolacrimosus. It acts by enhancing the opening of glutamate and GABA-gated chloride channels, rendering it effective as both a nematocide and insecticide.
T14995 Concanamycin A

Folimycin,Concanamycin,X 4357B,Antibiotic X 4357B

HIV Protease Microbiology/Virology; Proteases/Proteasome
Concanamycin A (Folimycin) 是一种多聚环内酯类抗生素,是选择性空泡状 H+-ATP 酶 (V-ATPase) 和溶酶体酸化抑制剂,可用于研究炎症。Concanamycin A 可增强细胞毒性 T 淋巴细胞对受感染原代细胞的免疫清除,抑制来自 HIV 和猿猴免疫缺陷病毒不同分支的 Nef 等位基因,可用于研究HIV 感染。
T8302 Ceftiofur

Antibacterial; Antibiotic Microbiology/Virology
Ceftiofur 是一种半合成抗生素,对家畜的各种革兰氏阳性和革兰氏阴性菌、好氧菌和厌氧菌均有抗菌活性。
T8641 Vancomycin

Antibacterial; Antibiotic; Autophagy Autophagy; Microbiology/Virology
Vancomycin 是一种糖肽类抗生素,可以通过改变细胞膜的渗透性并选择性地抑制核糖核酸的合成以发挥抗菌活性。Vancomycin 可以用于治疗所有抗生素均无效的严重感染。
T10662 Calcimycin hemicalcium salt

Antibiotic A-23187 hemicalcium salt,A-23187 hemicalcium salt

Others Others
Calcimycin (A-23187) hemicalcium salt is an antibiotic and a unique divalent cation ionophore (like calcium and magnesium). It induces Ca2+-dependent cell death by increasing intracellular calcium concentration.
T2890 Hordenine

Antibacterial; Antibiotic Microbiology/Virology
Hordenine 是一种植物中发现的苯乙胺生物碱,可抑制 cAMP 产生起到抑制黑色素生成的作用。
T1381 Milbemycin oxime

Others; Antibiotic; Parasite Microbiology/Virology; Others
Milbemycin oxime 是一种大环内酯,具有广谱抗寄生虫活性。它由 Milbemycin A4 和 A3 组成。它可结合谷氨酸门控的氯离子通道,可作用于肠道线虫,肺和心脏蠕虫。
T8063 Cephapirin Benzathine

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Cephapirin Benzathine 是头孢哌啶的苄硫醚盐形式,是一种广谱抗生素。
T3S0137 Bavachalcone

Antibacterial; Antibiotic Microbiology/Virology
Bavachalcone 是从补骨脂中分离的化合物,广泛用于中药,具有抗生素和抗癌等活性。
T21328 Carubicin

carminomycin,Carminomycin I,Carminomicin I,Antibiotic R 588A,Demethyldaunomycin

Others Others
Carubicin is an anthracycline antineoplastic antibiotic isolated from the bacterium Actinomadura carminata. Carubicin intercalates into DNA and interacts with topoisomerase II, thereby inhibiting DNA replication and repair and RNA and protein synthesis.
T6803 Chaetocin

毛壳素

Histone Methyltransferase; Antibacterial; Antibiotic Chromatin/Epigenetic; Microbiology/Virology
Chaetocin 特异性抑制组蛋白甲基转移酶(HMT) SU(VAR)3-9,IC50值为0.6 μM。它还可抑制硫氧还蛋白还原酶,IC50值为4 μM。
T13815 Penicillic acid

Apoptosis; Caspase; Antibacterial; Antibiotic Apoptosis; Microbiology/Virology; Proteases/Proteasome
Penicillic acid,一种由多种Aspergillus和Penicillium物种合成的polyketide mycotoxin,通过阻碍caspase-8的自我处理作用,抑制Fas ligand引发的apoptosis。此外,体外研究表明,Penicillic acid在rat alveolar macrophages中显示出cytotoxic特性。
TQ0260 Cerulenin

Antibiotic; Antifungal; Fatty Acid Synthase Metabolism; Microbiology/Virology
Cerulenin 是广泛使用的天然脂肪酸合成酶抑制剂。它是由真菌Cephalosporium caeruleus 产生的。它抑制拓扑异构酶I 催化活性并增强 SN-38 诱导的细胞凋亡。它具有抗真菌和抗肿瘤活性。
T25622 Lankacidins

Bundlin A,Lankacidin C,Antibiotic T-2636 C,NSC 145118,Lankacidin

Others Others
Lankacidins is an antitumor antibiotic of the macrolide tetraenes family from Streptomyces.
T10815 Cinnamoylglycine

Endogenous Metabolite Metabolism
Cinnamoylglycine 是肉桂酸和的甘氨酸结合物,是人体尿液代谢物。它被用作的尿液标志物,能够作为在抗生素研究期之后定殖耐药性的标志物。
T0444 Econazole

(±)-Econazol,益康唑

Antibiotic; Antifection; Antifungal Microbiology/Virology
Econazole ((±)-Econazol) 是一种咪唑衍生物,是一种抗真菌剂。
T7868 Farnesol

法呢醇,里哪醇

Endogenous Metabolite; Antibacterial; Antibiotic Metabolism; Microbiology/Virology
Farnesol 是一种半萜醇,能够调节细胞间的通讯,有抑菌活性。
T1029 Aztreonam

SQ-26,776,氨曲南

Antibacterial; Antibiotic Microbiology/Virology
Aztreonam (SQ-26,776) 是单环β-内酰胺抗生素,与青霉素结合蛋白3有较高亲和力。
T8062 Cefazedone

Refosporen,头孢西酮

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Cefazedone (Refosporen) 是一种具有抗革兰氏阳性和革兰氏阴性菌活性的时间依赖性头孢菌素抗生素。
T6S0141 Corylin

补骨脂异黄酮,补骨脂宁

Antibacterial; Antibiotic; STAT JAK/STAT signaling; Microbiology/Virology; Stem Cells
Corylin 是一种从补骨脂中分离的生物活性化合物,有抗生素或抗癌作用。
T1257 Bestatin

Ubenimex,乌苯美司

Others; Aminopeptidase; Antibacterial; Antibiotic; LTR Immunology/Inflammation; Metabolism; Microbiology/Virology; Others
Bestatin (Ubenimex) 是 CD13 (Aminopeptidase N)/APN 和 leukotriene A4 hydrolase 抑制剂,可用于癌症研究。
T21498 Phleomycin

DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Phleomycin 是在链霉菌中发现的,引起 DNA 切割的抗癌糖肽抗生素之一。 它类似于博来霉素,它结合并插入 DNA 以破坏双螺旋的完整性。
T0709 Natamycin

纳他霉素,Pimaricin

Estrogen/progestogen Receptor; Endogenous Metabolite; Antibiotic; Antifungal Endocrinology/Hormones; Metabolism; Microbiology/Virology
Natamycin (Pimaricin) 是由数个链霉菌菌株生产的大环内酯类抗生素,可通过抑制氨基酸和葡萄糖跨质膜的运输来抑制真菌生长。它是一种食品防腐剂,在农业中作抗真菌剂。它可研究真菌性角膜炎。
T3S0209 Vincristine

ERK; p38 MAPK; NF-κB; Akt; JNK; mTOR Cytoskeletal Signaling; MAPK; NF-κB; PI3K/Akt/mTOR signaling
Vincristine 属于生物碱类天然产物,可与微管蛋白结合并抑制微管的形成,从而抑制肿瘤细胞的有丝分裂。Vincristine 可用作微管去稳定剂,用于研究治疗血液系统肿瘤,如白血病和淋巴瘤以及儿童肉瘤的相关研究。
T14854 Caerulomycin A

浅蓝霉素,Cerulomycin,Caerulomycin

Antifungal Microbiology/Virology
Caerulomycin A (Caerulomycin) 是抗真菌和抗细菌化合物,能够诱导 T 细胞的产生。它能够抑制 IFN-γ 诱导的 STAT1 通路,从而增强 TGF-β-Smad3 信号通路。它可用于自身免疫病的研究。
T8504 Dianemycin

Nanchangmycin (free acid)

Antibacterial; Antibiotic Microbiology/Virology
Dianemycin (Nanchangmycin (free acid)) 由Streptomyces nanchangensis 产生的一种聚醚抗生素,抑制革兰氏阳性菌。它也是一种针对 Zika 病毒的广谱抗病毒药物。
TN1722 Hamamelitannin

Antifection Microbiology/Virology
Hamamelitannin 是分离自 Hamamelis virginiana 树皮的一种多酚,是群体感应抑制剂。它通过影响肽聚糖生物合成和 eDNA 释放增加金黄色葡萄球菌生物膜的抗生素敏感性。
T1022 Hygromycin B

潮霉素B,Hygrovetine

ribosome; Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Hygromycin B (Hygrovetine) 是一种氨基糖苷类抗生素,通过干扰易位并导致 70S 核糖体的错误翻译来抑制蛋白质合成。Hygromycin B 可用于筛选转染 hph 或 hyg 抗性基因的原核或者真核细胞。
T4004 Concanavalin A

Apoptosis Apoptosis
Concanavalin A 是 Ca2+/Mn2+依赖性和甘露糖/葡萄糖结合植物凝集素。它能够促使程序性细胞死亡。
T16542 Piromidic acid

吡咯酸,吡乙酸三氮萘

Antibacterial; Antibiotic Microbiology/Virology
Piromidic acid 是一种抗菌剂。它对革兰氏阴性菌和葡萄球菌具有活性,可研究肠道,泌尿和胆道感染。
T8019 Sorbic acid

Anti-infection; Endogenous Metabolite; Antibacterial; Antibiotic; Antifungal Metabolism; Microbiology/Virology
Sorbic acid 是一种高效安全无毒的食品防腐剂。它可抑制大多数霉菌,酵母和某些细菌。
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天然产物

Antibiotic PF 1052
Cat.No: T38097
Synonym:
Target: Others
Ansamitocin p-3
Cat.No: T22262
Synonym: Maytansinol isobutyrate,Antibiotic C 15003P3,NSC292222
Target: Microtubule Associated, ADC Cytotoxin
Lasalocid
Cat.No: T15717
Synonym: Lasalocid-A,Antibiotic X-537A,Ionophore X-537A
Target: Antibacterial
Calcimycin
Cat.No: T10662L
Synonym: Antibiotic A-23187,离子载体(钙镁盐混合物),A-23187
Target: Apoptosis, Antibacterial, Antibiotic, Autophagy, Antifungal
G-418 disulfate
Cat.No: T6512
Synonym: Geneticin,G418 Sulfate,Antibiotic G-418 sulfate,遗传霉素,Geneticin sulfate
Target: Antibacterial, Antibiotic
Staurosporine
Cat.No: T6680
Synonym: Antibiotic AM-2282,星形孢菌素,AM-2282,CGP 41251,星孢菌素
Target: Apoptosis, PKA, Antibacterial, Antibiotic, Src, PKC, Antifungal
Midecamycin
Cat.No: T5037
Synonym: Antibiotic SF-837,Turimycin P3,Medecamycin A1,Rubimycin,麦迪霉素,Platenomycin B1,Espinomycin A
Target: Antibacterial, Antibiotic
Antibiotic JI 20A
Cat.No: T23741
Synonym: JI-20 A,BRN 1668513,BRN-1668513,BRN1668513
Target: Others
Lasalocid sodium
Cat.No: T15716
Synonym: 拉沙洛西钠,拉沙里菌素,Ionophore X-537A sodium,Antibiotic X-537A sodium,Lasalocid-A sodium
Target: Antibacterial, Antibiotic, Autophagy
Albofungin
Cat.No: T26590
Synonym: Antibiotic P42-1,Antibiotic P42-C
Target: Others
Nargenicin
Cat.No: T36417
Synonym: Antibiotic 47444
Target: Others
K-252a
Cat.No: T15636
Synonym: Antibiotic K 252a,Antibiotic SF 2370,SF2370
Target: Others
Kazusamycin A
Cat.No: T24253
Synonym: Antibiotic CL1957B,PD 114721,Antibiotic 81-484
Target: Others
Benanomicin B
Cat.No: TN7517
Synonym: Antibiotic BU 3608C
Target: Others
K 41
Cat.No: T25563
Synonym: K-41,K41,Antibiotic K-41A,37454 RP,Antibiotic A 32887
Target: Others
Parvodicin C2
Cat.No: TN7525
Synonym: Antibiotic A40926 B1
Target: Others
Virustomycin A
Cat.No: T26321
Synonym: Antibiotic AM-2604 A
Target: Others
Safracin B
Cat.No: T24026
Synonym: Antibiotic Y 16482-alpha,EM 5519,EM-5519,EM5519,Antibiotic EM 5519
Target: Others
A 201A
Cat.No: T26405
Synonym: Antibiotic 201A,A201A,A-201A
Target: Others
Milbemycin A4
Cat.No: TN7268
Synonym: Antibiotic B 41A4,Milbemycin α3
Target: Others
Concanamycin A
Cat.No: T14995
Synonym: Folimycin,Concanamycin,X 4357B,Antibiotic X 4357B
Target: HIV Protease
Ceftiofur
Cat.No: T8302
Synonym:
Target: Antibacterial, Antibiotic
Vancomycin
Cat.No: T8641
Synonym:
Target: Antibacterial, Antibiotic, Autophagy
Calcimycin hemicalcium salt
Cat.No: T10662
Synonym: Antibiotic A-23187 hemicalcium salt,A-23187 hemicalcium salt
Target: Others
Hordenine
Cat.No: T2890
Synonym:
Target: Antibacterial, Antibiotic
Milbemycin oxime
Cat.No: T1381
Synonym:
Target: Others, Antibiotic, Parasite
Cephapirin Benzathine
Cat.No: T8063
Synonym:
Target: Others, Antibacterial, Antibiotic
Bavachalcone
Cat.No: T3S0137
Synonym:
Target: Antibacterial, Antibiotic
Carubicin
Cat.No: T21328
Synonym: carminomycin,Carminomycin I,Carminomicin I,Antibiotic R 588A,Demethyldaunomycin
Target: Others
Chaetocin
Cat.No: T6803
Synonym: 毛壳素
Target: Histone Methyltransferase, Antibacterial, Antibiotic
Penicillic acid
Cat.No: T13815
Synonym:
Target: Apoptosis, Caspase, Antibacterial, Antibiotic
Cerulenin
Cat.No: TQ0260
Synonym:
Target: Antibiotic, Antifungal, Fatty Acid Synthase
Lankacidins
Cat.No: T25622
Synonym: Bundlin A,Lankacidin C,Antibiotic T-2636 C,NSC 145118,Lankacidin
Target: Others
Cinnamoylglycine
Cat.No: T10815
Synonym:
Target: Endogenous Metabolite
Econazole
Cat.No: T0444
Synonym: (±)-Econazol,益康唑
Target: Antibiotic, Antifection, Antifungal
Farnesol
Cat.No: T7868
Synonym: 法呢醇,里哪醇
Target: Endogenous Metabolite, Antibacterial, Antibiotic
Aztreonam
Cat.No: T1029
Synonym: SQ-26,776,氨曲南
Target: Antibacterial, Antibiotic
Cefazedone
Cat.No: T8062
Synonym: Refosporen,头孢西酮
Target: Others, Antibacterial, Antibiotic
Corylin
Cat.No: T6S0141
Synonym: 补骨脂异黄酮,补骨脂宁
Target: Antibacterial, Antibiotic, STAT
Bestatin
Cat.No: T1257
Synonym: Ubenimex,乌苯美司
Target: Others, Aminopeptidase, Antibacterial, Antibiotic, LTR
Phleomycin
Cat.No: T21498
Synonym:
Target: DNA/RNA Synthesis, Antibacterial, Antibiotic
Natamycin
Cat.No: T0709
Synonym: 纳他霉素,Pimaricin
Target: Estrogen/progestogen Receptor, Endogenous Metabolite, Antibiotic, Antifungal
Vincristine
Cat.No: T3S0209
Synonym:
Target: ERK, p38 MAPK, NF-κB, Akt, JNK, mTOR
Caerulomycin A
Cat.No: T14854
Synonym: 浅蓝霉素,Cerulomycin,Caerulomycin
Target: Antifungal
Dianemycin
Cat.No: T8504
Synonym: Nanchangmycin (free acid)
Target: Antibacterial, Antibiotic
Hamamelitannin
Cat.No: TN1722
Synonym:
Target: Antifection
Hygromycin B
Cat.No: T1022
Synonym: 潮霉素B,Hygrovetine
Target: ribosome, Antibacterial, Antibiotic, Antifungal
Concanavalin A
Cat.No: T4004
Synonym:
Target: Apoptosis
Piromidic acid
Cat.No: T16542
Synonym: 吡咯酸,吡乙酸三氮萘
Target: Antibacterial, Antibiotic
Sorbic acid
Cat.No: T8019
Synonym:
Target: Anti-infection, Endogenous Metabolite, Antibacterial, Antibiotic, Antifungal
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Cat. No. Product Name Species Expression System
TMPY-00672 Azurocidin/CAP37 Protein, Human, Recombinant (His)

AZU,NAZC,azurocidin 1,hHBP,AZAMP,HUMAZUR,CAP37,HBP,AZU1

Human HEK293 Cells
Azurocidin (AZU1), also known as heparin-binding protein (HBP) or cationic antimicrobial protein 37 (CAP37), is an azurophil granule antibiotic protein, with monocyte chemotactic and antibacterial activity. The Azurophil granules, specialized lysosomes of the neutrophil, contain at least 10 proteins implicated in the killing of microorganisms. Azurocidin is a member of the serine protease family that includes Cathepsin G, neutrophil elastase (NE), and proteinase 3 (PR3), however, Azurocidin is n...
TMPH-00639 Hygromycin-B 4-O-kinase Protein, E. coli, Recombinant (His)

Hygromycin B phosphotransferase,hph,Hygromycin-B kinase,Hygr...

E. coli E. coli
The aminoglycoside phosphotransferases achieve inactivation of their antibiotic substrates by phosphorylation. Only phosphorylates hygromycin and closely related compounds such as demethyl analogs and destomycin.
TMPH-00027 Aculeacin-A acylase Protein, Actinoplanes utahensis, Recombinant (His & SUMO)

Aculeacin-A acylase

Actinoplanes utahensis E. coli
Catalyzes the hydrolysis of the palmitoyl moiety of the antifungal antibiotic, aculeacin-A, giving a hexapeptide moiety and a long chain fatty acid. Aculeacin-A acylase Protein, Actinoplanes utahensis, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 35.1 kDa and the accession number is P29958.
TMPJ-00611 SFP Protein, B.subtilis, Recombinant (His)

Surfactin synthase-activating enzyme,sfp,lpa-8,4'-phosphopan...

Bacillus subtilis E. coli
The Bacillus subtilis enzyme Sfp, required for production of the lipoheptapeptide antibiotic surfactin, posttranslationally phosphopantetheinylates a serine residue in each of the seven peptidyl carrier protein domains of the first three subunits (SrfABC) of surfactin synthetase to yield docking sites for amino acid loading and peptide bond formation.
TMPY-01812 Enoyl-ACP Reductase Protein, E. coli, Recombinant (His)

b1288,JW1281,gts,ECK1283,qmeA,envM

E. coli E. coli
Enoyl-ACP reductase, also known as NADH-dependent enoyl-ACP reductase and FABI, is a cell inner membrane and peripheral membrane protein which belongs to theshort-chain dehydrogenases/reductases (SDR) family and FabI subfamily. Microorganisms produce many kinds of antibiotics which function in an antagonistic capacity in nature where they have much competition. Bacterial FAS provides essential fatty acids for use in the assembly of key cellular components. Among them, FABI is an enoyl-ACP...
TMPY-01679 LCN1 Protein, Human, Recombinant (His)

TLC,MGC71975,TP,VEGP,Lipocalin 1,PMFA

Human HEK293 Cells
Lipocalin-1, also known as Von Ebner gland protein, VEG protein, Tear Prealbumin, VEGP, Tear lipocalin, and LCN1 is a secreted protein that belongs to the calycin superfamily and Lipocalin family. Human Lipocalin-1 / VEGP was originally described as a major protein of human tear fluid, which was thought to be tear specific. Lipocalin-1 / VEGP is identical to lingual von Ebner's gland protein and is also produced in the prostate, nasal mucosa, and tracheal mucosa. Homologous proteins have been fo...

重组蛋白

Azurocidin/CAP37 Protein, Human, Recombinant (His)
Cat.No: TMPY-00672
Species: Human
Expression System: HEK293 Cells
Hygromycin-B 4-O-kinase Protein, E. coli, Recombinant (His)
Cat.No: TMPH-00639
Species: E. coli
Expression System: E. coli
Aculeacin-A acylase Protein, Actinoplanes utahensis, Recombinant (His & SUMO)
Cat.No: TMPH-00027
Species: Actinoplanes utahensis
Expression System: E. coli
SFP Protein, B.subtilis, Recombinant (His)
Cat.No: TMPJ-00611
Species: Bacillus subtilis
Expression System: E. coli
Enoyl-ACP Reductase Protein, E. coli, Recombinant (His)
Cat.No: TMPY-01812
Species: E. coli
Expression System: E. coli
LCN1 Protein, Human, Recombinant (His)
Cat.No: TMPY-01679
Species: Human
Expression System: HEK293 Cells
Cat. No. Product Name Target Signaling Pathways
T13026 Sulfadimethoxypyrimidine D4

Others Others
Sulfadimethoxypyrimidine D4, a deuterium-labeled version of Sulfadimethoxypyrimidine, is a sulfonamide antibiotic characterized by its broad-spectrum antibacterial effectiveness.
T11853 Linezolid-d3

Linezolid D3,PNU-100766 D3

Others Others
Linezolid D3, a deuterium-labeled version of Linezolid, is a synthetic antibiotic designed to halt the initiation of bacterial protein synthesis.
T13035 Sulfathiazole-d4

Others Others
Sulfathiazole D4 is a deuterium labeled Sulfathiazole. Sulfathiazole used as a short-acting sulfonamide antibiotic.
T13031 Sulfamethoxazole-d4

Ro 4-2130 D4,磺胺甲恶唑 D4

Others Others
Sulfamethoxazole D4 is a deuterium labeled Sulfamethoxazole (Ro 4-2130). Sulfamethoxazole is a sulfonamide bacteriostatic antibiotic.
T10306 Amoxicillin D4

Amoxycillin D4

Others Others
Amoxicillin D4 (Amoxycillin D4) is a deuterium-labeled Amoxicillin. Amoxicillin is an antibiotic with broad-spectrum antimicrobial activity.
T13024 Sulfadimethoxine-d4

Sulphadimethoxine D4

Others Others
Sulfadimethoxine D4 is a deuterium labeled Sulfadimethoxine (Sulphadimethoxine). Sulfadimethoxine is a sulfonamide antibiotic used to treat many infections.
TMID-0271 Miloxacin-d3

Miloxacin-d3 是 Miloxacin 的氘代化合物。Miloxacin 的 CAS 号为 37065-29-5。
TMID-0004 Ampicillin-d5

Ampicillin-d5 是 Ampicillin 的氘代化合物。Ampicillin 的 CAS 号为 69-53-4。Ampicillin是一种广谱、半合成的β-内酰胺类青霉素抗生素,具有杀菌活性。
TMIJ-0037 Sarafloxacin-d8 Hydrochloride

Sarafloxacin-d8 Hydrochloride 是 Sarafloxacin Hydrochloride 的氘代化合物。Sarafloxacin Hydrochloride 的 CAS 号为 91296-87-6。Sarafloxacin hydrochloride是一种抗菌化合物。
TMID-0293 Acetylisovaleryltylosin-d3 Tartrate

Acetylisovaleryltylosin-d3 Tartrate 是 Acetylisovaleryltylosin Tartrate 的氘代化合物。Acetylisovaleryltylosin Tartrate 的 CAS 号为 63428-13-7。Tylvalosin tartrate是一种对革兰氏阳性细菌具有抗性的大环内酯类抗生素。
TMID-0079 Norfloxacin-d8

Norfloxacin-d8 是 Norfloxacin 的氘代化合物。Norfloxacin 的 CAS 号为 70458-96-7。Norfloxacin是广谱抗生素,能通过结合DNA旋转酶抑制革兰氏阳性和阴性菌。
TMIJ-0111 Azithromycin-13C-d3

Azithromycin-13C-d3 是 Azithromycin 的 13C 和氘代化合物。Azithromycin 的 CAS 号为 83905-01-5。Azithromycin是一种常用于细菌感染研究的大环内酯抗生素。
TMIJ-0297 Acetylsulfamethoxazole-d4

Acetylsulfamethoxazole-d4 是 Acetylsulfamethoxazole 的氘代化合物。Acetylsulfamethoxazole 的 CAS 号为 21312-10-7。N4-Acetylsulfamethoxazole 是磺胺甲恶唑的一种代谢物。Sulfamethoxazole 属于磺胺类抗菌素,可用于细菌感染。
TMIH-0154 Ciprofloxacin-d8

Ciprofloxacin-d8 是 Ciprofloxacin 的氘代化合物。Ciprofloxacin 的 CAS 号为 85721-33-1。Ciprofloxacin是一种有高抗菌活性的氟喹诺酮类抗生素。
TMID-0080 Amikacin-d5

Amikacin-d5 是 Amikacin 的氘代化合物。Amikacin 的 CAS 号为 37517-28-5。Amikacin 是半合成的卡那霉素类似物,对革兰氏阴性菌 (包括庆大霉素和妥布霉素耐药菌株) 具有广谱活性,有耳毒性和肾毒性。
TMIH-0530 Sulbactam-d2

Sulbactam-d2 是 Sulbactam 的氘代化合物。Sulbactam 的 CAS 号为 68373-14-8。Sulbactam是一种竞争性、不可逆的 β-内酰胺酶抑制剂,抑制耐多药不动杆菌-鲍曼不动杆菌复合物。它具有抗菌活性。
TMIJ-0109 Erythromycin Ethylsuccinate-13C-d3

Erythromycin Ethylsuccinate-13C-d3 是 Erythromycin Ethylsuccinate 的 13C 和氘代化合物。Erythromycin Ethylsuccinate 的 CAS 号为 1264-62-6。Erythromycin Ethylsuccinate是一种由红链霉菌产生的大环内酯类抗生素,有潜力用于多种细菌感染。它具有抗HIV-1病毒活性。
T36537 Nitrofurantoin-13C3

Nitrofurantoin-13C3

Nitrofurantoin-13C3is intended for use as an internal standard for the quantification of nitrofurantoin by GC- or LC-MS. Nitrofurantoin is a nitrofuran antibiotic.1In vivo, nitrofurantoin (25-100 mg/kg) reducesE. colireplication and abscess formation in the renal medulla of infected rats in a dose-dependent manner. It prevents kidney and bladder infection in rats following bladder inoculation with clinical isolates ofP. mirabilis. Nitrofurantoin also prevents alkalization of urine, as well as ca...
TMIJ-0011 Chloramphenicol-d5

Chloramphenicol-d5 是 Chloramphenicol 的氘代化合物。Chloramphenicol 的 CAS 号为 56-75-7。Chloramphenicol 是一种广谱抗生素,有效抑制细菌蛋白质生物合成。它主要作用于细菌 70S 核糖体的 50S 亚基,对肽基转移酶有活性,抑制肽键的形成。
TMID-0234 Penicillin G-d5 potassium salt

Penicillin G-d5 potassium salt 是 Penicillin G potassium salt 的氘代化合物。Penicillin G potassium salt 的 CAS 号为 113-98-4。Benzylpenicillin potassium是青霉素家族的一种速效抗生素。
TMIH-0418 Ozenoxacin-d3

Ozenoxacin-d3 是 Ozenoxacin 的氘代化合物。Ozenoxacin 的 CAS 号为 245765-41-7。Ozenoxacin是一种新型喹诺酮类抗生素,能够抵抗大多数从在皮肤和软组织感染中分离的微生物。
TMID-0195 Levofloxacin-d8

Levofloxacin-d8 是 Levofloxacin 的氘代化合物。Levofloxacin 的 CAS 号为 100986-85-4。Levofloxacin是合成的氟喹诺酮类抗生素,有抑制细菌DNA旋转酶的超螺旋活性的作用,能阻止DNA复制。
TMIJ-0184 Cefditoren-d3

Cefditoren-d3 是 Cefditoren 的氘代化合物。Cefditoren 的 CAS 号为 104146-53-4。
TMIJ-0158 Sitafloxacin-d4

Sitafloxacin-d4 是 Sitafloxacin 的氘代化合物。Sitafloxacin 的 CAS 号为 127254-12-0。Sitafloxacin (Sitafloxacin anhydrous) 是一种具有口服活性的氟喹诺酮类抗生素,具有广谱的抗菌活性。Sitafloxacin 可用于研究呼吸道感染和尿路感染。
TMIH-0300 Levofloxacin-d3

Levofloxacin-d3 是 Levofloxacin 的氘代化合物。Levofloxacin 的 CAS 号为 100986-85-4。Levofloxacin是合成的氟喹诺酮类抗生素,有抑制细菌DNA旋转酶的超螺旋活性的作用,能阻止DNA复制。
TMIJ-0022 Thiamphenicol-Methyl-d3

Thiamphenicol-Methyl-d3 是 Thiamphenicol 的氘代化合物。Thiamphenicol 的 CAS 号为 15318-45-3。Thiamphenicol是 Chloramphenicol 的甲基磺酰基衍生物,是一种广谱抗菌类抗生素。它与 50S 核糖体亚基结合,抑制蛋白质合成并具有抑菌作用 ,特别针对革兰氏阴性,革兰氏阳性需氧和厌氧菌。
TMID-0283 Vancomycin-13C-d3

Vancomycin-13C-d3 是 Vancomycin 的 13C 和氘代化合物。Vancomycin 的 CAS 号为 1404-90-6。Vancomycin 是一种抗生素,用于通过阻止细菌生长来治疗严重的细菌感染。它还改变细胞膜的渗透性并选择性地抑制核糖核酸的合成。
TMID-0284 Vancomycin-d12 TFA

Vancomycin-d12 TFA 是 Vancomycin TFA 的氘代化合物。Vancomycin TFA 的 CAS 号为 1404-90-6。Vancomycin 是一种抗生素,用于通过阻止细菌生长来治疗严重的细菌感染。它还改变细胞膜的渗透性并选择性地抑制核糖核酸的合成。
TMIJ-0520 (1E,13E) Tilmicosin-d3

(1E,13E) Tilmicosin-d3 是 Tilmicosin 的氘代化合物。Tilmicosin 的 CAS 号为 108050-54-0。Tilmicosin是一种抗生素,可研究曼氏杆菌和巴氏杆菌相关的牛羊呼吸系统疾病。
TMID-0227 Rifabutin-d7

Rifabutin-d7 是 Rifabutin 的氘代化合物。Rifabutin 的 CAS 号为 72559-06-9。Rifabutin是半合成的安莎霉素抗生素,抑制 DNA 依赖性 RNA 聚合酶,有抗分枝杆菌作用。
TMIJ-0281 Lincomycin-d3

Lincomycin-d3 是 Lincomycin 的氘代化合物。Lincomycin 的 CAS 号为 7179-49-9。Lincomycin hydrochloride monohydrate 是一种窄谱抗生素, 具有与红霉素相似的效力, 对革兰氏阳性球菌的作用效果很好, 主要抑制细菌细胞蛋白质的合成。
TMID-0194 Ofloxacin-d8

Ofloxacin-d8 是 Ofloxacin 的氘代化合物。Ofloxacin 的 CAS 号为 82419-36-1。Ofloxacin是可抑制细菌DNA旋转酶的一种氟喹诺酮类抗生素。
T37250 Cefazolin-13C2,15N

Cefazolin-13C2,15N

Cefazolin-13C2,15N is intended for use as an internal standard for the quantification of cefazolin by GC- or LC-MS. Cefazolin is a broad-spectrum cephalosporin antibiotic that is active in vitro against various Gram-positive and Gram-negative bacteria (MICs = 0.2-12.5 μg/ml). It also inhibits the growth of clinical isolates of S. aureus, E. coli, P. mirabilis, and K. pneumoniae (MICs = 0.1-25 μg/ml). In vivo, cefazolin protects against S. aureus, E. coli, and P. mirabilis infection in mice (ED50...
TMIJ-0179 Faropenem-d7 Sodium Salt

Faropenem-d7 Sodium Salt 是 Faropenem Sodium Salt 的氘代化合物。Faropenem Sodium Salt 的 CAS 号为 122547-49-3。Faropenem sodium 是一种口服生物可利用的青霉烯类抗生素,能有效杀灭结核分枝杆菌,治疗结核病和社区获得性肺炎。
TMIJ-0288 Danofloxacin-d3

Danofloxacin-d3 是 Danofloxacin 的氘代化合物。Danofloxacin 的 CAS 号为 112398-08-0。Danofloxacin free base 是一种具有口服活性第三代氟喹诺酮抗菌剂,对大多数革兰氏阴性和革兰氏阳性细菌,支原体和衣原体物种具有广谱的活性,并通过抑制细菌的 DNA 回转酶发挥抗菌作用。它可用于牛,猪和鸡呼吸道疾病的研究。
TMIJ-0181 Clindamycin-13C-d3

Clindamycin-13C-d3 是 Clindamycin 的 13C 和氘代化合物。Clindamycin 的 CAS 号为 18323-44-9。Clindamycin 从细菌核糖体中解离肽基-tRNA,破坏细菌蛋白质合成。 它是一种半合成广谱抗生素,由母体化合物林可霉素化学修饰而成。
TMIJ-0340 Lincomycin-13C-d3

Lincomycin-13C-d3 是 Lincomycin 的 13C 和氘代化合物。Lincomycin 的 CAS 号为 7179-49-9。Lincomycin hydrochloride monohydrate 是一种窄谱抗生素, 具有与红霉素相似的效力, 对革兰氏阳性球菌的作用效果很好, 主要抑制细菌细胞蛋白质的合成。
TMID-0084 Tigecycline-d9

Tigecycline-d9 是 Tigecycline 的氘代化合物。Tigecycline 的 CAS 号为 220620-09-7。Tigecycline是甘氨酰环素抗生素,对Acinetobacter baumannii(A. baumannii) 的 MIC50和 MIC90分别为 1 和 2 mg/L。它对E. coli(MG1655 菌株) 的平均抑制浓度 (MIC) 约 125 ng/ mL。
T71984 Enrofloxacin-d5

Enrofloxacin-d5 is intended for use as an internal standard for the quantification of enrofloxacin by GC- or LC-MS. Enrofloxacin is a fluoroquinolone antibiotic. It is active against panels of Campylobacter, E. coli, and Salmonella isolates (mean MIC50s = 0.06, 0.5, and 0.03 µg/ml, respectively). It is also active against equine isolates of L. intracellularis (MICs = 0.125-0.5 µg/ml). Enrofloxacin inhibits bacterial DNA gyrase. In vivo, enrofloxacin (10 mg/kg) increases survival in a mouse model...
TMID-0292 Tylosin-d3

Tylosin-d3 是 Tylosin 的氘代化合物。Tylosin 的 CAS 号为 1401-69-0。Tylosin 是一种兽医用大环内酯类抗生素,是Streptomyces fradiae的产物。它对革兰氏阳性菌具有高抗菌活性。它是饲料添加剂用于促进动物生长。它被用于治疗家禽、猪和牛的细菌性痢疾和呼吸道疾病。
TMIJ-0026 2-NP-AMOZ-d5

2-NP-AMOZ-d5 是 2-NP-AMOZ 的氘代化合物。2-NP-AMOZ 的 CAS 号为 183193-59-1。2-NP-AMOZ 是 AMOZ 的 2-硝基苯基衍生物,AMOZ 是抗生素呋喃他酮的代谢产物。2-NP-AMOZ 专门作为蛋白质结合 AMOZ 检测的可靠工具。
TMIJ-0327 Cefpodoxime-d3 Acid

Cefpodoxime-d3 Acid 是 Cefpodoxime Acid 的氘代化合物。Cefpodoxime Acid 的 CAS 号为 80210-62-4。Cefpodoxime (free acid) 是一种口服的第三代头孢菌素抗生素。除铜绿假单胞菌、肠球菌和脆弱拟杆菌外,它对大多数革兰氏阳性和革兰氏阴性微生物均有效。
TMIJ-0170 Cefdinir-13C-15N2

Cefdinir-13C-15N2 是 Cefdinir 的 13C 和 15 N 的标记化合物。Cefdinir 的 CAS 号为 91832-40-5。Cefdinir是头孢菌素类中的一种半合成广谱抗生素,对几种革兰氏阴性和革兰氏阳性细菌引起的感染有效。它可研究耳,鼻窦,喉咙和皮肤的常见细菌感染。
TMID-0290 Cefpodoxime proxetil-d3

Cefpodoxime proxetil-d3 是 Cefpodoxime proxetil 的氘代化合物。Cefpodoxime proxetil 的 CAS 号为 87239-81-4。Cefpodoxime Proxetil 是一种口服的广谱型抗生素。它与青霉素结合蛋白结合,抑制肽聚糖的合成,干扰细菌细胞壁的生物合成。
TMID-0286 Rifaximin-d6

Rifaximin-d6 是 Rifaximin 的氘代化合物。Rifaximin 的 CAS 号为 80621-81-4。Rifaximin是一种胃肠道选择性抗生素,与细菌 DNA 依赖性 RNA 聚合酶的 β 亚基结合,抑制细菌 RNA 合成。与革兰氏阴性菌(MIC:8-50 毫克/毫升)相比,它对革兰氏阳性菌株(MIC:0.03-5 毫克/毫升)的敏感性更高。
TMIJ-0287 Meropenem-d6-1

Meropenem-d6-1 是 Meropenem-1 的氘代化合物。Meropenem-1 的 CAS 号为 96036-03-2。Meropenem是一种具有广谱抗菌活性的碳青霉烯抗生素,对敏感和耐药的淋病奈瑟氏球菌,流感嗜血杆菌和杜克氏杆菌的 MIC 值分别为 0.02-0.06 mg/mL,0.03-0.12 mg/mL 和 0.015-0.12 mg/mL。
T36021 Flumequine-13C3

Flumequine-13C3

Flumequine-13C3is intended for use as an internal standard for the quantification of flumequine by GC- or LC-MS. Flumequine is a fluoroquinolone antibiotic.1It is active againstS. aureus, S. pyogenes, B. subtilis, E. coli, P. aeruginosa, S. faecalis, andK. pneumoniae(MICs = 1-100 μg/ml). Flumequine is also active against field isolates of B. hyodysenteriae (MICs = 6.25-200 μg/ml).2It inhibits DNA gyrase, disrupting supercoiling of bacterial DNA to block transcription and replication.3In vivo, fl...
T71293 Nifuroxazide-d4

Nifuroxazide-d4 is intended for use as an internal standard for the quantification of nifuroxazide by GC- or LC-MS. Nifuroxazide is a nitrofuran antibiotic. It is active against strains of the enteropathogenic bacteria C. jejuni, Salmonella, Y. enterocolitica, Shigella, and E. coli. It inhibits quorum sensing and virulence factor production in P. aeruginosa. Nifuroxazide inhibits STAT3 activity in a reporter assay and decreases viability of U266 and INA-6 myeloma cells, which have constitutive S...

同位素标记化合物

Sulfadimethoxypyrimidine D4
Cat.No: T13026
Synonym:
Target: Others
Linezolid-d3
Cat.No: T11853
Synonym: Linezolid D3,PNU-100766 D3
Target: Others
Sulfathiazole-d4
Cat.No: T13035
Synonym:
Target: Others
Sulfamethoxazole-d4
Cat.No: T13031
Synonym: Ro 4-2130 D4,磺胺甲恶唑 D4
Target: Others
Amoxicillin D4
Cat.No: T10306
Synonym: Amoxycillin D4
Target: Others
Sulfadimethoxine-d4
Cat.No: T13024
Synonym: Sulphadimethoxine D4
Target: Others
Miloxacin-d3
Cat.No: TMID-0271
Synonym:
Target:
Ampicillin-d5
Cat.No: TMID-0004
Synonym:
Target:
Sarafloxacin-d8 Hydrochloride
Cat.No: TMIJ-0037
Synonym:
Target:
Acetylisovaleryltylosin-d3 Tartrate
Cat.No: TMID-0293
Synonym:
Target:
Norfloxacin-d8
Cat.No: TMID-0079
Synonym:
Target:
Azithromycin-13C-d3
Cat.No: TMIJ-0111
Synonym:
Target:
Acetylsulfamethoxazole-d4
Cat.No: TMIJ-0297
Synonym:
Target:
Ciprofloxacin-d8
Cat.No: TMIH-0154
Synonym:
Target:
Amikacin-d5
Cat.No: TMID-0080
Synonym:
Target:
Sulbactam-d2
Cat.No: TMIH-0530
Synonym:
Target:
Erythromycin Ethylsuccinate-13C-d3
Cat.No: TMIJ-0109
Synonym:
Target:
Nitrofurantoin-13C3
Cat.No: T36537
Synonym: Nitrofurantoin-13C3
Target:
Chloramphenicol-d5
Cat.No: TMIJ-0011
Synonym:
Target:
Penicillin G-d5 potassium salt
Cat.No: TMID-0234
Synonym:
Target:
Ozenoxacin-d3
Cat.No: TMIH-0418
Synonym:
Target:
Levofloxacin-d8
Cat.No: TMID-0195
Synonym:
Target:
Cefditoren-d3
Cat.No: TMIJ-0184
Synonym:
Target:
Sitafloxacin-d4
Cat.No: TMIJ-0158
Synonym:
Target:
Levofloxacin-d3
Cat.No: TMIH-0300
Synonym:
Target:
Thiamphenicol-Methyl-d3
Cat.No: TMIJ-0022
Synonym:
Target:
Vancomycin-13C-d3
Cat.No: TMID-0283
Synonym:
Target:
Vancomycin-d12 TFA
Cat.No: TMID-0284
Synonym:
Target:
(1E,13E) Tilmicosin-d3
Cat.No: TMIJ-0520
Synonym:
Target:
Rifabutin-d7
Cat.No: TMID-0227
Synonym:
Target:
Lincomycin-d3
Cat.No: TMIJ-0281
Synonym:
Target:
Ofloxacin-d8
Cat.No: TMID-0194
Synonym:
Target:
Cefazolin-13C2,15N
Cat.No: T37250
Synonym: Cefazolin-13C2,15N
Target:
Faropenem-d7 Sodium Salt
Cat.No: TMIJ-0179
Synonym:
Target:
Danofloxacin-d3
Cat.No: TMIJ-0288
Synonym:
Target:
Clindamycin-13C-d3
Cat.No: TMIJ-0181
Synonym:
Target:
Lincomycin-13C-d3
Cat.No: TMIJ-0340
Synonym:
Target:
Tigecycline-d9
Cat.No: TMID-0084
Synonym:
Target:
Enrofloxacin-d5
Cat.No: T71984
Synonym:
Target:
Tylosin-d3
Cat.No: TMID-0292
Synonym:
Target:
2-NP-AMOZ-d5
Cat.No: TMIJ-0026
Synonym:
Target:
Cefpodoxime-d3 Acid
Cat.No: TMIJ-0327
Synonym:
Target:
Cefdinir-13C-15N2
Cat.No: TMIJ-0170
Synonym:
Target:
Cefpodoxime proxetil-d3
Cat.No: TMID-0290
Synonym:
Target:
Rifaximin-d6
Cat.No: TMID-0286
Synonym:
Target:
Meropenem-d6-1
Cat.No: TMIJ-0287
Synonym:
Target:
Flumequine-13C3
Cat.No: T36021
Synonym: Flumequine-13C3
Target:
Nifuroxazide-d4
Cat.No: T71293
Synonym:
Target:
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