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Search Results for " anti-influenza "
Targets Recommended: Influenza Virus

37

抑制剂 & 化合物

31

天然产物

3

化合物库

2

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Cat. No. Product Name
L1700 抗病毒库

1040 compounds
1040 种具有抗病毒活性的化合物的特有集合,是筛选新型抗病毒药的有效工具;可用于高通量筛选和高内涵筛选;
L1800 抗感染化合物库

2938 compounds
2938 种具有抗感染活性的化合物的特有集合,包括抗细菌、抗真菌、抗巨细胞病毒、抗HIV、抗SARS、抗流感等活性;
L6730 抗病毒中药单体化合物库

268 compounds
268 种具有抗病毒活性的中药单体集合,是药物开发、药理研究的有效工具;

化合物库

抗病毒库
Cat.No: L1700
Compounds: 1040
抗感染化合物库
Cat.No: L1800
Compounds: 2938
抗病毒中药单体化合物库
Cat.No: L6730
Compounds: 268
Cat. No. Product Name Target Signaling Pathways
T72037 Anti-Influenza agent 4

Influenza Virus Microbiology/Virology
Anti-Influenza agent 4 是一种有效且具有选择性的流感病毒 抑制剂,对A/Parma 和 A/Roma 毒株具有抑制作用, EC50 分别为 62 nM 和150 nM。
T9124 Laninamivir octanoate

辛酸拉尼米韦,CS-8958

Influenza Virus Microbiology/Virology
Laninamivir octanoate (CS-8958) 是一种长效流感神经氨酸酶抑制剂,是Laninamivir 的前药, 具有优异的抗流感病毒活性。
T7785 T-1105

Influenza Virus Microbiology/Virology
T-1105 是 T-705 的结构类似物,是一种广谱病毒聚合酶抑制剂,在转化为核糖核苷三磷酸代谢物后抑制 RNA 病毒的聚合酶,有抗病毒活性。
T8333 Aurintricarboxylic acid

ATA,NSC-4056,NSC4056,金精三羧酸,NSC 4056

Apoptosis; P2X Receptor; Influenza Virus; Topoisomerase Apoptosis; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience
Aurintricarboxylic acid (NSC-4056) 是高效的αβ-亚甲基-ATP 敏感选择性P2X1Rs 和P2X3Rs 变构拮抗剂。 它是核糖核酸酶和拓扑异构酶 II 的有效抑制剂,可阻止核酸与酶结合。
T83046 Anti-Influenza agent 5

Influenza Virus Microbiology/Virology
Anti-Influenza agent 5 (Compound IIB-2)为查耳酮类衍生物,具有抑制流感病毒核输出的活性。该化合物能有效抑制对Oseltamivir具有耐药性的病毒株,主要通过阻断流感病毒核蛋白输出作用来抑制病毒复制。
T60778 Anti-Influenza agent 3

Others Others
Anti-Influenza agent 3 (compound 11h) 是有效的抗流感药物,对 MDCK 上皮细胞显示出低细胞毒性。Anti-Influenza agent 3 抑制 M2 WT 和 S31N 离子通道的传导性。Anti-Influenza agent 3 对 A/HK/68 (H3N2, M2-WT) 菌株的 EC50值为 3.29 μM,对 A/WSN/33 (H1N1, M2-S31N) 菌株的 EC50值为 2.45 μM。
T20500 Salcomine

NSC32965,NSC-32965,NSC 32965,双水杨酰胺乙基钴

Influenza Virus Microbiology/Virology
Salcomine (NSC-32965) 具有抗流感病毒活性。
T21339 Peramivir

RWJ270201,BCX 1812,BCX1812,RWJ 270201

Antiviral Immunology/Inflammation
Peramivir (BCX1812) 是一种高选择性的甲型和乙型流感神经氨酸酶抑制剂,具有抗病毒活性和抗细胞因子作用,可用于研究新型冠状病毒和流感病毒感染。
T16914 SP187

UV4,MON-​DNJ

Others; Virus Protease; Influenza Virus Microbiology/Virology; Others
SP187 (MON-​DNJ) 是一种靶向作用于宿主的亚氨基糖。它具有抗丝状病毒感染活性。SP187可用于治疗抗流感和登革热病毒。
T6642 Rimantadine

金刚乙胺,1-Rimantadine

Influenza Virus Microbiology/Virology
Rimantadine (1-Rimantadine) 是一种抗流感病毒药物。
T28443 PPQ-581

Others Others
PPQ-581 is an anti-influenza agent. PPQ-581 interrupts the crucial RNP trafficking, resulting in influenza replication inhibition, preventing virus-induced cytopathic effects.
T13075L T-705RTP sodium

Others Others
T-705RTP sodium is a selective and GTP-competitive of influenza virus RNA polymerase(IC50 of 0.14 μM and a Ki of 1.52 μM), has potent anti-influenza virus activity.
T13075 T-705RTP

Others Others
T-705RTP is a selective and GTP-competitive of influenza virus RNA polymerase(IC50 of 0.14 μM and a Ki of 1.52 μM), has potent anti-influenza virus activity.
T40267 RdRP-IN-3

Others Others
RdRP-IN-3, a potential anti-influenza drug candidate, functions by inhibiting the activity of RNA-dependent RNA polymerase (RdRp).
T77060 Lesofavumab

Lesofavumab (MHAB5553A) 是一种人 IgG1κ 抗influenza B virus 抗体。
T74614 PROTAC Hemagglutinin Degrader-1

Others Others
PROTACHemagglutinin Degrader-1 (Compound V3) 是一种有效的 PROTAC 流感病毒血凝素 (influenza hemagglutinin(HA)) 降解剂,降解中值浓度为 1.44 μM。PROTACHemagglutinin Degrader-1 具有广谱抗流感病毒活性。
T62059 Influenza A virus-IN-6

Others Others
Influenza A virus-IN-6 (compound 16j) 是有效的选择性甲型流感病毒抑制剂(IC50= 3.88 μM, CC50= 36.64 μM)。Influenza A virus-IN-6 显示出抗 IAV 活性和较低的细胞毒性。
T62888 Influenza A virus-IN-7

Others Others
Influenza A virus-IN-7 (compound 16r) 是一种有效的、口服具有活力的甲型流感病毒抑制剂 (IC50: 3.43 μM, CC50>100 μM)。Influenza A virus-IN-7 具有抗 IAV 作用,细胞毒性低,对病毒 RNA 的转录和复制表现出抑制作用。
T60810 Influenza virus-IN-2

Others Others
Influenza virus-IN-2 (compound 19) 具有抗甲型流感病毒活性,是有效的流感病毒抑制剂,CC50值为 150.85 μM,EC50值为 2.58 μM,。Influenza virus-IN-2 浓度依赖性的抑制 PAN 核酸内切酶,EC50为 489.39 nM。
T60697 Influenza virus-IN-1

Others Others
Influenza virus-IN-1 (compound 14) 具有抗甲型流感病毒活性,它是甲型流感病毒的有效抑制剂,其CC50值 >200 μM,EC50值为 2.46 μM。Influenza virus-IN-1 对 PAN 核酸内切酶显示出浓度依赖性的抑制活性 (EC50 = 312.36 nM)。
T61904 HSP90-IN-14

Others Others
HSP90-IN-14 (compound 4) 是有效的Hsp90 抑制剂(Kd= 0.26μM)。在MDCK 细胞中,HSP90-IN-14 表现出抗流感病毒活性,抗 A/H3N2、A/H1N1 和 B 型流感病毒的EC50分别为 2.6、3.9 和 17 μM。
T61394 Neuraminidase-IN-5

Others Others
Neuraminidase-IN-5 (Compound 5b) 是一种有效的 neuraminidase 抑制剂,IC50为 0.02 μM。神经氨酸酶(NA)是开发抗流感药物的有希望的靶点。Neuraminidase-IN-5 是一种二氢呋喃香豆素衍生物化合物。
T38952 Triperiden

Others Others
Triperiden is a chemical compound that serves as an inhibitor of influenza virus multiplication. Specifically, it exerts its antiviral activity by targeting the haemagglutinin of fowl plague virus (FPV) and inhibiting the conformational change in the haemagglutinin at acid pH. Additionally, Triperiden is classified as an anticholinergic anti-parkinsonism drug.
T74806 HAA-09

Others Others
HAA-09是一种靶向流感PB2_cap结合域的口服抗流感剂。其对甲型流感病毒展示出高效的抗病毒活性,其EC50值达到0.03 μM。同时,HAA-09具有显著的聚合酶抑制效果,IC50值为0.06±0.004 μM。通过阻断病毒复制,HAA-09能有效抑制病毒无引起明显的细胞毒性。
T61509 Neuraminidase-IN-8

Others Others
Neuraminidase-IN-8 (Compound 6d) 是一种有效的神经氨酸酶 (neuraminidase) 抑制剂,其IC50值为 0.027 μM。Neuraminidase-IN-8 具有抗流感活性。
T72717 Anti-IAV agent 1

Others Others
Anti-IAV agent 1-1a) 是一种口服抗甲型流感病毒(IAV)剂,对IAV H1N1及Oseltamivir抗性IAV H1N1的IC50值分别是0.03μM与0.06μM。
T60910 RSV-IN-4

Others Others
RSV-IN-4 (Compound 2) 具有抗 RSV 活性,EC50值为11.76 μM。RSV-IN-4 是呼吸道合胞病毒 (RSV) 和甲流病毒 A (IAV) 的双重抑制剂。
T63233 Neuraminidase-IN-10

Others Others
Neuraminidase-IN-10 是神经氨酸酶 (neuraminidase) 抑制剂,表现出抗流感作用,能够作用于 H1N1 (IC50: 2.6 nM)、H5N1 (IC50: 5.1 nM) 和 H5N8 (IC50: 1.65 nM)。
T61217 RSV-IN-3

Others Others
RSV-IN-3 (Compound 1) 是呼吸道合胞病毒 (RSV) 和流感病毒 A (IAV) 的双重抑制剂。RSV-IN-3 具有抗 RSV 活性 (EC50=32.70 μM)。
T79444 HA-IN-1

Influenza Virus Microbiology/Virology
HA-IN-1(compound 5g)是靶向血凝素(HA)胰蛋白酶切割位点的配体,表现出高亲和力。该化合物能够抑制HA介导的膜融合,并在体内有效降低肺部病毒滴度,展现其作为甲型流感病毒(IAV)抑制剂和抗流感药物的潜力。
T38340 10-Norparvulenone

Others Others
10-Norparvulenone is a fungal metabolite originally isolated fromMicrosphaeropsis.1It decreases viral sialidase activity in, and increases survival of, MDCK cells infected with the mouse-adapted influenza virus A/PR/8/34 when used at a concentration of 1 μg/ml. 1.Fukami, A., Nakamura, T., Kim, Y.P., et al.A new anti-influenza virus antibiotic, 10-norparvulenone from Microsphaeropsis sp. FO-5050J. Antibiot. (Tokyo)53(10)1215-1218(2000)
T60939 Neuraminidase-IN-6

Others Others
Neuraminidase-IN-6 (Compound 5c) 是1,3,4-triazole-3-acetamide 的衍生物。Neuraminidase-IN-6 是神经氨酸酶的有效抑制剂,IC50值为 0.11 μM。神经氨酸酶 (NA) 是抗流感药物开发的理想靶点。
T77158 Diridavumab

Diridavumab为一种针对HA茎的单克隆抗体。它能稳定HA的融合前结构,阻断细胞膜与病毒膜在核内体内因pH变化引起的融合。此抗体主要用于H2流感病毒研究。
T77009 Firivumab

Firivumab (CT-P22; CT120)是一种针对人类IgG1单克隆的抗甲型流感病毒血凝素(Anti-IAV HA)抗体。该抗体能有效中和多种亚型,包括H1N1、H5N1、H6N1、H6N2、H8N4、H8N8、H9N2和H12N7。研究发现,Firivumab在小鼠模型中对H1N1病毒展现出显著的保护效果。
T71291 EICAR

Others Others
EICAR is a drug which acts as an inhibitor of the enzyme IMP dehydrogenase. It is a nucleoside derivative which has both anti-cancer and antiviral effects, and was originally developed for the treatment of leukemia, but was unsuccessful in human clinical trials. It has broad spectrum antiviral effects with activity against vaccinia virus, Semliki forest virus, Junin virus, reovirus, influenza, measles virus and respiratory syncytial virus among others, although it is not active against SARS. T...
T79567 Antiviral agent 35

Influenza Virus Microbiology/Virology
Antiviralagent 35 (compound 4d) 作为一种口服抗流感病毒药物,针对流感病毒复制的早期阶段有效。该化合物能够阻断流感病毒引发的ROS积聚、自噬及细胞凋亡,同时在肺部感染的小鼠模型中,抑制RIG-1通路所介导的炎症响应。Antiviralagent 35展现出低细胞毒性(CC50>800 μM,MDCK细胞)且对H1N1(A/Weiss/43)展现出显著的抗病毒活性,EC50为2.28 μM。
T35686 3-Acetyl Betulinaldehyde

Others Others
3-Acetyl betulinaldehyde is a triterpene and derivative of the cholesterol biosynthesis inhibitor betulin that has been found inA. japonica.1It is an intermediate in the synthesis of 3-acetylbetulinic acid, as well as various lupine and germanicane triterpenes and saponins with anticancer activity.2 1.Tung, N.H., Kwon, H.-J., Kim, J.-H., et al.An anti-influenza component of the bark of Alnus japonicaArch. Pharm. Res.33(3)363-367(2010) 2.Thibeault, D., Gauthier, C., Legault, J., et al.Synthesis a...

化合物

Anti-Influenza agent 4
Cat.No: T72037
Synonym:
Target: Influenza Virus
Laninamivir octanoate
Cat.No: T9124
Synonym: 辛酸拉尼米韦,CS-8958
Target: Influenza Virus
T-1105
Cat.No: T7785
Synonym:
Target: Influenza Virus
Aurintricarboxylic acid
Cat.No: T8333
Synonym: ATA,NSC-4056,NSC4056,金精三羧酸,NSC 4056
Target: Apoptosis, P2X Receptor, Influenza Virus, Topoisomerase
Anti-Influenza agent 5
Cat.No: T83046
Synonym:
Target: Influenza Virus
Anti-Influenza agent 3
Cat.No: T60778
Synonym:
Target: Others
Salcomine
Cat.No: T20500
Synonym: NSC32965,NSC-32965,NSC 32965,双水杨酰胺乙基钴
Target: Influenza Virus
Peramivir
Cat.No: T21339
Synonym: RWJ270201,BCX 1812,BCX1812,RWJ 270201
Target: Antiviral
SP187
Cat.No: T16914
Synonym: UV4,MON-​DNJ
Target: Others, Virus Protease, Influenza Virus
Rimantadine
Cat.No: T6642
Synonym: 金刚乙胺,1-Rimantadine
Target: Influenza Virus
PPQ-581
Cat.No: T28443
Synonym:
Target: Others
T-705RTP sodium
Cat.No: T13075L
Synonym:
Target: Others
T-705RTP
Cat.No: T13075
Synonym:
Target: Others
RdRP-IN-3
Cat.No: T40267
Synonym:
Target: Others
Lesofavumab
Cat.No: T77060
Synonym:
Target:
PROTAC Hemagglutinin Degrader-1
Cat.No: T74614
Synonym:
Target: Others
Influenza A virus-IN-6
Cat.No: T62059
Synonym:
Target: Others
Influenza A virus-IN-7
Cat.No: T62888
Synonym:
Target: Others
Influenza virus-IN-2
Cat.No: T60810
Synonym:
Target: Others
Influenza virus-IN-1
Cat.No: T60697
Synonym:
Target: Others
HSP90-IN-14
Cat.No: T61904
Synonym:
Target: Others
Neuraminidase-IN-5
Cat.No: T61394
Synonym:
Target: Others
Triperiden
Cat.No: T38952
Synonym:
Target: Others
HAA-09
Cat.No: T74806
Synonym:
Target: Others
Neuraminidase-IN-8
Cat.No: T61509
Synonym:
Target: Others
Anti-IAV agent 1
Cat.No: T72717
Synonym:
Target: Others
RSV-IN-4
Cat.No: T60910
Synonym:
Target: Others
Neuraminidase-IN-10
Cat.No: T63233
Synonym:
Target: Others
RSV-IN-3
Cat.No: T61217
Synonym:
Target: Others
HA-IN-1
Cat.No: T79444
Synonym:
Target: Influenza Virus
10-Norparvulenone
Cat.No: T38340
Synonym:
Target: Others
Neuraminidase-IN-6
Cat.No: T60939
Synonym:
Target: Others
Diridavumab
Cat.No: T77158
Synonym:
Target:
Firivumab
Cat.No: T77009
Synonym:
Target:
EICAR
Cat.No: T71291
Synonym:
Target: Others
Antiviral agent 35
Cat.No: T79567
Synonym:
Target: Influenza Virus
3-Acetyl Betulinaldehyde
Cat.No: T35686
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
TN2331 Eleutheroside B1

刺五加苷B1

Influenza Virus Microbiology/Virology
Eleutheroside B1是具有广谱抗人流感病毒的一种香豆素。它抑制多种趋化因子基因和流感病毒核蛋白基因的 mRNA 表达。它具有抗病毒、抗流感和抗炎活性,且细胞毒性小。
T2738 Dehydroandrographolide

NOS; Influenza Virus Immunology/Inflammation; Microbiology/Virology
Dehydroandrographolide 是从草药穿心莲中提取的一种天然产物。它通过使 iNOS 失活来降低 LPS 诱导的急性肺损伤中的氧化应激,有抗感染活性。
T2982 Xanthone

Genicide,呫吨酮,氧杂蒽酮,Xanthenone,Benzophenone oxide

Apoptosis; Others; Influenza Virus; Antibacterial; Antifungal Apoptosis; Microbiology/Virology; Others
Xanthone (Xanthenone) 是一种从山竹果中分离得到的天然产物,具有抗炎,抗氧化,抗肿瘤,抗过敏,抗细菌,抗真菌和抗病毒活性。在癌变的不同阶段可控制细胞分裂和生长,凋亡,炎症和转移。
T2957 Arctigenin

牛蒡苷元,牛蒡子苷元,(-)-Arctigenin

Apoptosis; MMP; Influenza Virus; Autophagy Apoptosis; Autophagy; Microbiology/Virology; Proteases/Proteasome
Arctigenin ((-)-Arctigenin) 是一种存在于牛蒡中的木脂素,具有抗氧化、抗肿瘤、抗炎和抗病毒活性。它可研究代谢紊乱和中枢神经系统功能障碍。
T13229 Tunicamycin

Influenza Virus; Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Tunicamycin 是一种抗生素的混合物,通过阻断 GlcNAc 磷酸转移酶 (GPT),抑制 N-连接糖基化。Tunicamycin 具有抗肿瘤活性,还具有抗细菌、抗真菌和抗病毒活性。
T6569 Mimosine

Leucenine,NSC 69188,含羞草素,Leucenol,L-Mimosine

Others Others
Mimosine (Leucenol) 是一种酪氨酸类似物,具有抗癌和抗炎等活性。它可通过其强大的铁结合活性作为抗氧化剂,是一种 Fe(III) 螯合剂。它作用于人类白血病细胞,通过金属离子螯合、线粒体激活和诱导活性氧产生来诱导细胞凋亡。
T5S2059 Glaucine

Calcium Channel; Dopamine Receptor; Influenza Virus; Adrenergic Receptor; PDE GPCR/G Protein; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience
Glaucine 是从海罂粟中分离的一种生物碱,具有镇咳、抗炎和支气管扩张作用。它是具有口服活性的磷酸二酯酶 4 选择性抑制剂。它还是非选择性的 α-肾上腺素受体拮抗剂,具有抗氧化和抗病毒活性。
T26288 Clovamide

trans-Clovamide,N-trans-Caffeoy-L-dopa

Apoptosis; Influenza Virus; ROS; Antibacterial Apoptosis; Immunology/Inflammation; Microbiology/Virology
Clovamide (trans-Clovamide) 是一种天然存在的咖啡酰结合物,具有抗菌、抗炎、抗氧化和神经保护作用。它是一种极好的活性氧和氧自由基清除剂。
T3376 Cynaroside

朝蓟糖甙,Luteoloside,Luteolin 7-β-D-Glucopyranoside,Luteolin 7-O-Glucoside,Luteolin 7-O-β-D-glucoside,木犀草苷,Luteolin 7-glucoside

Others; Influenza Virus; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others
Cynaroside (Luteolin 7-O-Glucoside) 是一个抗氧化类黄酮。它还是一种流感依赖 RNA 的RNA 聚合酶抑制剂,IC50为 32 nM。
TN2353 8-Hydroxyapigenin

Isoscutellarein

Antioxidant; Influenza Virus Microbiology/Virology; oxidation-reduction
8-Hydroxyapigenin (Isoscutellarein) 是从植物黄芩中提取的黄铜类化合物,具有抗炎抗氧和抗流感病毒的活性。
TN3120 5-Hydroxy-7-acetoxy-8-methoxyflavone

Histone Demethylase; Antiviral Chromatin/Epigenetic; Immunology/Inflammation
5-Hydroxy-7-acetoxy-8-methoxyflavone 是一种类黄酮化合物,可以抑制脂质过氧化,可能具有抗流感病毒活性。
T75675 Nepasaikosaponin K

Antiviral Immunology/Inflammation
Nepasaikosaponin K 是一种从柴胡根中分离出来小分子化合物,具有抗流感和抗病毒活性,可用于研究病毒感染。
TN2166 Rupestonic acid

ERK; p38 MAPK; Influenza Virus; Nrf2 Immunology/Inflammation; MAPK; Microbiology/Virology
Rupestonic acid 是青蒿 Artemisia rupestris L. 中的一种化合物,Artemisia rupestris L. 是一种著名的治疗感冒的维吾尔族传统药物。 Rupestonic acid 具有抗流感病毒活性。
T0875 Acetylcysteine

N-Acetylcysteine,乙酰半胱氨酸,N-Acetyl-L-cysteine,LNAC,NAC,N-Acetyl Cysteine,易咳净

Apoptosis; TNF; Ferroptosis; Influenza Virus; Reactive Oxygen Species; ROS; Endogenous Metabolite Apoptosis; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
Acetylcysteine (NAC) 是半胱氨酸的 N-乙酰衍生物,是一种 ROS 抑制剂和粘液溶解剂。Acetylcysteine 可诱导细胞凋亡,可用于减少粘液的厚度,还具有抗流感病毒活性。
TN1051 1-Caffeoylquinic acid

金银花,1-咖啡酰奎宁酸

NF-κB NF-κB
1-Caffeoylquinic acid 是一种有效的NF-κB 抑制剂,对 p105 的 RH 结构域显示高结合亲和力,Ki= 0.002 μM,结合能为 1.50 Kcal/mol。它抑制PD-1/PD-L1相互作用。它具有抗氧化应激能力。
T4S2126 Ginkgetin

银杏双黄酮,银杏素

Apoptosis; Wnt/beta-catenin; COX; STAT; Autophagy Apoptosis; Autophagy; Cytoskeletal Signaling; Immunology/Inflammation; JAK/STAT signaling; Neuroscience; Stem Cells
Ginkgetin 是从银杏叶中分离得到的一种双黄酮,具有抗肿瘤、抗炎、神经保护、抗真菌的作用。它也是 Wnt 信号抑制剂,IC50值为 5.92 μM。
T27380 FR-198248

Others Others
FR-198248, a new anti-influenza agent, shows antiinfluenza virus activity in Madin-Darby canine kidney (MDCK) cells in vitro.
TN1066 Filixic acid ABA

Influenza Virus Microbiology/Virology
Filixic acid ABA exhibits inhibitory effects on neuraminidase of influenza virus H5N1 with IC50 as 29.57 ± 2.48 μM, it may have anti-influenza virus activity.
TN5005 Shegansu B

Influenza Virus Microbiology/Virology
Shegansu B exhibits significant in vitro anti-influenza viral activity in MDCK cells.
TN1506 Clemastanin B

直铁线莲宁B,落叶松树脂醇苷B

Influenza Virus Microbiology/Virology
Clemastanin B has antioxidant and anti-inflammatory activities, it exerts its anti-influenza activity by inhibiting the virus multiplication, prophylaxsis and blocking the virus attachment.
TN3461 Asebotin

Influenza Virus Microbiology/Virology
Asebotin shows anti-influenza A virus activity, it also possesses potent antiviral activity (100% inhibition at the concentration of 1 ug /mL) against highly pathogenic avian influenza strain H5N1. Asebotin can inhibit the proliferation of murine B cells.
T8521 Gnetin D

Gnetin D exhibits significant in vitro anti-influenza viral activity in MDCK cells, with IC(50) values from 0.67 to 11.99 ug/mL.
T36734 Methyl brevifolincarboxylate

Others Others
Methyl brevifolincarboxylate (Brevifolincarboxylic acid methyl ester) is a potent influenza virus PB2 cap-binding inhibitor. Methyl brevifolincarboxylate exhibits inhibitory activity against influenza virus A/Puerto Rico/8/34 (H1N1) and A/Aichi/2/68 (H3N2) with IC50s of 27.16 μM and 33.41 μM. Anti-oxidant activity[1][2]. Methyl brevifolincarboxylate exhibits significant DPPH radical scavenging activity with an IC50 value of 8.9 μM. [1]. Wu QY, et al. Chromatographic fingerprint and the simultane...
TN2311 Wulignan A1

五脂素 A1

Antifection Microbiology/Virology
Wulignan A1 exhibits activity against leukemia P-388 in vitro; it also may have anti-influenza virus H1N1 and H1N1-TR (a Tamiflu drug resistant virus strain) activities.
TN6204 Santin

5,7-Dihydroxy-3,6,4'-trimethoxyflavone

Influenza Virus Microbiology/Virology
Santin (5,7-Dihydroxy-3,6,4'-trimethoxyflavone) 是从桦树芽中提取的黄酮类化合物,具有抗增殖、抗流感和抗癌活性。 Santin 可用于有关抗 IAV 药物的研究。
TN2176 Sanggenol A

Influenza Virus; Antifection Microbiology/Virology
Sanggenol A 抑制甲型流感病毒和肺炎球菌神经氨酸酶,因此可作为双重作用的抗感染试剂。
TN4392 Koaburaside

IL Receptor; TNF; Influenza Virus Apoptosis; Immunology/Inflammation; Microbiology/Virology
Koaburaside exhibits antioxidant activity with an IC50 value of 9.0μM, it shows weak inhibitory activity against influenza A neuraminidase. Koaburaside may have anti-allergic inflammatory activity, it can suppress histamine release from mast cells.
TN1347 8-Prenylkaempferol

去甲脱水淫羊藿黄素

p38 MAPK; NF-κB; PI3K MAPK; NF-κB; PI3K/Akt/mTOR signaling
8-Prenylkaempferol is an effective agent for attenuating pro-inflammatory NO induction, it may be an anti-inflammatory agent for suppressing influenza A virus-induced RANTES production acts by blocking PI3K-mediated transcriptional activation of NF-κB and
T73465 Goitrin

L-5-Vinyl-2-thiooxazolidone,(S)-Goitrin,(S)-Goitrin ; L-5-Vinyl-2-thiooxazolidone

Others Others
Goitrin ((S)-Goitrin) 为芥子油苷-黑芥子酶反应产物,有效抑制甲状腺过氧化物酶并阻碍碘在甲状腺的利用。此外,该化合物亦展现出对抗流感病毒(H1N1)的活性。
TN4108 Ganoderic acid Z

Antifection Microbiology/Virology
The binding affinities of ganoderic acid DM and ganoderic acid Z (ΔGbind, -16.83 and-10.99 kcal mol-1) are comparable to that of current commercial drug oseltamivir (-23.62 kcal mol-1);Ganoderic acid DM is a potential source of anti-influenza ingredient, with novel binding pattern and advantage over oseltamivir, it has steric hindrance on the 150 cavity of N1 protein, and exerts activities across the H274Y and N294S mutations, is the attractive candidates of novel neuraminidase (NA) inhibitors....
TN1104 Cyanidin 3-sambubioside chloride

Cyanidin-3-O-sambubioside chloride

RAAS; Antioxidant; NO Synthase Endocrinology/Hormones; Immunology/Inflammation; oxidation-reduction
Cyanidin 3-sambubioside chloride (Cyanidin-3-O-sambubioside chloride) 是一种从植物中提取的花青素,是一种 NO和 H274Y 突变的抑制剂,对流感神经氨酸酶具有抑制作用。Cyanidin 3-sambubioside chloride 具有抗氧化,抗血管生成和抗病毒活性,抑制血管紧张素转换酶 (ACE) 的活性,可用于研究病毒感染和心血管疾病。

天然产物

Eleutheroside B1
Cat.No: TN2331
Synonym: 刺五加苷B1
Target: Influenza Virus
Dehydroandrographolide
Cat.No: T2738
Synonym:
Target: NOS, Influenza Virus
Xanthone
Cat.No: T2982
Synonym: Genicide,呫吨酮,氧杂蒽酮,Xanthenone,Benzophenone oxide
Target: Apoptosis, Others, Influenza Virus, Antibacterial, Antifungal
Arctigenin
Cat.No: T2957
Synonym: 牛蒡苷元,牛蒡子苷元,(-)-Arctigenin
Target: Apoptosis, MMP, Influenza Virus, Autophagy
Tunicamycin
Cat.No: T13229
Synonym:
Target: Influenza Virus, Antibacterial, Antibiotic, Antifungal
Mimosine
Cat.No: T6569
Synonym: Leucenine,NSC 69188,含羞草素,Leucenol,L-Mimosine
Target: Others
Glaucine
Cat.No: T5S2059
Synonym:
Target: Calcium Channel, Dopamine Receptor, Influenza Virus, Adrenergic Receptor, PDE
Clovamide
Cat.No: T26288
Synonym: trans-Clovamide,N-trans-Caffeoy-L-dopa
Target: Apoptosis, Influenza Virus, ROS, Antibacterial
Cynaroside
Cat.No: T3376
Synonym: 朝蓟糖甙,Luteoloside,Luteolin 7-β-D-Glucopyranoside,Luteolin 7-O-Glucoside,Luteolin 7-O-β-D-glucoside,木犀草苷,Luteolin 7-glucoside
Target: Others, Influenza Virus, DNA/RNA Synthesis
8-Hydroxyapigenin
Cat.No: TN2353
Synonym: Isoscutellarein
Target: Antioxidant, Influenza Virus
5-Hydroxy-7-acetoxy-8-methoxyflavone
Cat.No: TN3120
Synonym:
Target: Histone Demethylase, Antiviral
Nepasaikosaponin K
Cat.No: T75675
Synonym:
Target: Antiviral
Rupestonic acid
Cat.No: TN2166
Synonym:
Target: ERK, p38 MAPK, Influenza Virus, Nrf2
Acetylcysteine
Cat.No: T0875
Synonym: N-Acetylcysteine,乙酰半胱氨酸,N-Acetyl-L-cysteine,LNAC,NAC,N-Acetyl Cysteine,易咳净
Target: Apoptosis, TNF, Ferroptosis, Influenza Virus, Reactive Oxygen Species, ROS, Endogenous Metabolite
1-Caffeoylquinic acid
Cat.No: TN1051
Synonym: 金银花,1-咖啡酰奎宁酸
Target: NF-κB
Ginkgetin
Cat.No: T4S2126
Synonym: 银杏双黄酮,银杏素
Target: Apoptosis, Wnt/beta-catenin, COX, STAT, Autophagy
FR-198248
Cat.No: T27380
Synonym:
Target: Others
Filixic acid ABA
Cat.No: TN1066
Synonym:
Target: Influenza Virus
Shegansu B
Cat.No: TN5005
Synonym:
Target: Influenza Virus
Clemastanin B
Cat.No: TN1506
Synonym: 直铁线莲宁B,落叶松树脂醇苷B
Target: Influenza Virus
Asebotin
Cat.No: TN3461
Synonym:
Target: Influenza Virus
Gnetin D
Cat.No: T8521
Synonym:
Target:
Methyl brevifolincarboxylate
Cat.No: T36734
Synonym:
Target: Others
Wulignan A1
Cat.No: TN2311
Synonym: 五脂素 A1
Target: Antifection
Santin
Cat.No: TN6204
Synonym: 5,7-Dihydroxy-3,6,4'-trimethoxyflavone
Target: Influenza Virus
Sanggenol A
Cat.No: TN2176
Synonym:
Target: Influenza Virus, Antifection
Koaburaside
Cat.No: TN4392
Synonym:
Target: IL Receptor, TNF, Influenza Virus
8-Prenylkaempferol
Cat.No: TN1347
Synonym: 去甲脱水淫羊藿黄素
Target: p38 MAPK, NF-κB, PI3K
Goitrin
Cat.No: T73465
Synonym: L-5-Vinyl-2-thiooxazolidone,(S)-Goitrin,(S)-Goitrin ; L-5-Vinyl-2-thiooxazolidone
Target: Others
Ganoderic acid Z
Cat.No: TN4108
Synonym:
Target: Antifection
Cyanidin 3-sambubioside chloride
Cat.No: TN1104
Synonym: Cyanidin-3-O-sambubioside chloride
Target: RAAS, Antioxidant, NO Synthase
Cat. No. Product Name Species Expression System
TMPY-02219 Influenza A H1N1 (A/Puerto Rico/8/34/Mount Sinai) Non-structural/NS1 Protein (His)

NS1 Protein

H1N1 E. coli
The NS1 Influenza protein is created by the internal protein-encoding, linear negative-sense, single-stranded RNA, NS gene segment and which also codes for the nuclear export protein or NEP, formerly referred to as the NS2 protein, which mediates the export of vRNPs. The non-structural (NS1) protein is found in Influenzavirus A, Influenzavirus B, and Influenzavirus C. The non-structural (NS1) protein of the highly pathogenic avian H5N1 viruses circulating in poultry and waterfowl in Southeast As...
TMPJ-00527 SP-D Protein, Human, Recombinant (His)

Lung Surfactant Protein D,SFTP4,COLEC7,SFTPD,PSP-D,SP-D,Pulm...

Human HEK293 Cells
Surfactant Pulmonary-Associated Protein D (SP-D) is a 43 kDa member of the collectin family of innate immune modulators. Its principal components consist of a collagen-like region and a C-terminal carbohydrate recognition domain (CRD), a structure that places it in a subset of pattern recognition proteins termed defense collagens. SP-D is constitutively secreted by alveolar lining cells and epithelium associated with tubular structures and induced in cardiac smooth muscle and endothelial cells. ...

重组蛋白

Influenza A H1N1 (A/Puerto Rico/8/34/Mount Sinai) Non-structural/NS1 Protein (His)
Cat.No: TMPY-02219
Species: H1N1
Expression System: E. coli
SP-D Protein, Human, Recombinant (His)
Cat.No: TMPJ-00527
Species: Human
Expression System: HEK293 Cells
TargetMol Loading
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