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Search Results for " angiotensin-converting enzyme (ace) "

Targets Recommended: Angiotensin-converting Enzyme (ACE) RAAS

90

抑制剂 & 化合物

16

天然产物

3

重组蛋白

8

同位素标记化合物

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Cat. No.	Product Name	Target	Signaling Pathways
T7510	Leucylarginylproline	RAAS	Endocrinology/Hormones
	Leucylarginylproline 是一种血管紧张素转换酶抑制剂，IC50=为0.27μM。
T1484	Perindoprilat Perindoprilate,培哚普利	RAAS; MRP; AChR	Endocrinology/Hormones; Immunology/Inflammation; Neuroscience
	Perindoprilat (Perindoprilate) 是一种血管紧张素转换酶抑制剂。
T1489	Fosinopril sodium SQ28555,福辛普利钠	RAAS	Endocrinology/Hormones
	Fosinopril sodium 是一种血管紧张素转换酶（ACE）抑制剂的前药，能够作用于高血压和慢性心力衰竭。
T13865	Resorcinolnaphthalein	RAAS	Endocrinology/Hormones
	Resorcinolnaphthalein 是一种特异性的血管紧张素转换酶 2 激活剂，EC50=19.5 μM。Resorcinolnaphthalein 能够用于高血压和肾纤维化的研究
T16116	MLN-4760	RAAS	Endocrinology/Hormones
	MLN-4760 是选择性的人ACE2抑制剂，IC50=0.44 nM，对人ACE2的选择性是其他相关蛋白的 5000 多倍，包括人睾丸 ACE (IC50，>100 μM) 和牛 carboxypeptidase A (IC50，27 μM)。
T1145	Diminazene Aceturate DIZE	Others; Serine Protease; Parasite	Microbiology/Virology; Others; Proteases/Proteasome
	Diminazene aceturate 是血管紧张素转化酶 2 的激活剂，具有强效抗炎特性。它还是一种抗锥虫药物，适用于牲畜。它主要生化机理是通过与富含腺嘌呤-胸腺嘧啶碱基对的位点发生特异性相互作用，以非插入方式与锥虫动子体 DNA 结合。
T7686	Ramiprilat	RAAS	Endocrinology/Hormones
	Ramiprilat 是 Ramipril 的活性代谢物，是一种口服有活力的血管紧张素转换酶 (ACE) 抑制剂，其 Ki=7 pM。它可用于研究心力衰竭以及高血压。
T1605	Enalapril MK-421,依那普利	RAAS; MRP	Endocrinology/Hormones; Immunology/Inflammation
	Enalapril 是一种血管紧张素转换酶（ACE）抑制剂。
TP1828	N-Acetyl-Ser-Asp-Lys-Pro	RAAS	Endocrinology/Hormones
	N-Acetyl-Ser-Asp-Lys-Pro 通过酶促处理胸腺素 β4 在骨髓细胞中形成。它抑制多能造血干细胞进入细胞周期的 S 期，并防止小鼠中的 Ara-C 致死性。
T7714	Temocapil	Tyrosinase	Proteases/Proteasome
	Temocapil 是一种酪氨酸激酶抑制剂。
T7808	Alacepril Cetapril,阿拉普利,DU-1219	RAAS	Endocrinology/Hormones
	Alacepril (DU-1219) 是一种具有口服活性血管紧张素转换酶 (ACE) 抑制剂，具有长效抗高血压作用。
T7339	Angiotensin (1-7) Ang-(1-7),Angiotensin 1-7,ASP-ARG-VAL-TYR-ILE-HIS-PRO	RAAS; Endogenous Metabolite	Endocrinology/Hormones; Metabolism
	Angiotensin (1-7) (ASP-ARG-VAL-TYR-ILE-HIS-PRO) 是肾素-血管紧张素系统中的内源性七肽。Angiotensin 1-7在心肌细胞中具有抗炎和抗纤维化活性，因此具有心脏保护作用。它能抑制血管紧张素转换酶和释放一氧化氮，是激肽诱导的血管舒张的局部协同调节剂。它阻断 Ang II 诱导的平滑肌细胞增殖和肥大，并显示对内皮的抗血管生成和生长抑制作用。它显示出抗炎活性。
T1645	Ramipril HOE-498,Tritace,雷米普利,Altace,Carasel	Apoptosis; RAAS	Apoptosis; Endocrinology/Hormones
	Ramipril (Altace) 是一种ACE 抑制剂，IC50为5 nM。
T5030	Zofenopril calcium SQ26991,佐芬普利钙,Zofenopril (calcium)	RAAS; Reactive Oxygen Species	Endocrinology/Hormones; Immunology/Inflammation; Metabolism; NF-κB
	Zofenopril calcium (SQ26991) 是一种抗氧化剂和血管紧张素转化酶 (ACE) 抑制剂。
T0180	Benazepril hydrochloride 盐酸贝那普利,CGS 14824A HCl,Benazepril HCl,CGS14824A	RAAS	Endocrinology/Hormones
	Benazepril hydrochloride (CGS 14824A HCl) 是一种血管紧张素转化酶（ACE）抑制剂，能够作用于高血压。
T2679	BMS-265246 BMS265246	CDK	Cell Cycle/Checkpoint
	BMS-265246 是一种有效的选择性 CDK1/2 抑制剂，对 CDK1/cyclin B 和 CDK2/cyclin E 的 IC50分别为6 nM 和9 nM。
T6340	Enalaprilat Dihydrate 依那普利拉二水合物,MK-422,MK-422 Dihydrate	RAAS; Autophagy	Autophagy; Endocrinology/Hormones
	Enalaprilat Dihydrate (MK-422 Dihydrate) 是一种有效的血管紧张素转化酶抑制剂，IC50为 1.94 nM。
T3281	Delapril hydrochloride indalapril,地拉普利盐酸盐,Alindapril Hydrochloride,Delapril Hydrochloride,盐酸地拉普利,CV 3317	RAAS	Endocrinology/Hormones
	Delapril hydrochloride (indalapril) 是一种血管紧张素转化酶抑制剂，能够用于心血管疾病的研究。
T5329	Trandolapril	Angiotensin-converting Enzyme (ACE)	Metabolism
	Trandolapril 是 Trandolaprilat 的前体药物。Trandolapril 是一种口服血管紧张素转换酶抑制剂，在高血压和充血性心力衰竭及心肌梗死领域有研究价值。
T6542	Imidapril hydrochloride Novaloc,Imidapril HCl,盐酸咪达普利,Tanapril,TA-6366	RAAS	Endocrinology/Hormones
	Imidapril hydrochloride (Tanapril) 是一种血管紧张素转换酶 (ACE) 抑制剂，具有抗高血压活性。
T0706	Lisinopril dihydrate Lisinopril,Renacor,赖诺普利二水合物,MK-521 (dihydrate)	RAAS; MRP	Endocrinology/Hormones; Immunology/Inflammation
	Lisinopril dihydrate （MK-521) 是一种血管紧张素转化酶抑制剂。Lisinopri dihydrate 能够作用于高血压，充血性心力衰竭和心脏病等。
T6698	Temocapril hydrochloride CS-622 HCl,Acecol,Temocapril HCl,CS-622,盐酸替莫普利	RAAS	Endocrinology/Hormones
	Temocapril hydrochloride (CS-622 HCl) 是血管紧张素转化酶 (ACE) 抑制剂。Temocapril HCl 能够用于充血性心力衰竭、急性心肌梗死、高血压、胰岛素抵抗和肾脏疾病的研究。
T0805	Quinapril hydrochloride CI-906,PD-109452-2,盐酸喹那普利,Quinapril HCl	RAAS	Endocrinology/Hormones
	Quinapril hydrochloride (PD-109452-2) 是一种血管紧张素转化酶(ACE) 抑制剂的原药。
T1484L	Perindopril erbumine 培哚普利叔丁胺,培哚普利叔丁胺盐,S9490-3,Perindopril tert-butylamine salt	Apoptosis; RAAS; MRP	Apoptosis; Endocrinology/Hormones; Immunology/Inflammation
	Perindopril erbumine (S9490-3) 是一种长效血管紧张素转换酶抑制剂。
T1462	Captopril SQ 14225,甲巯丙脯酸,卡托普利,SQ-14534,SA333	RAAS	Endocrinology/Hormones
	Captopril (SA333) 是一种含巯基的，具有口服活性的血管紧张素转换酶(ACE)抑制剂，IC50=0.025 μM，广泛应用于高血压和充血性心力衰竭的研究。Captopril 也是NDM-1抑制剂，IC50=7.9 μM。
T6486	Enalapril Maleate MK-421 Maleate,Renitec Maleate,Glioten Maleate,MK-421 (maleate),Vasotec Maleate,马来酸依那普利	RAAS	Endocrinology/Hormones
	Enalapril Maleate (MK-421 Maleate) 一种是血管紧张素转化酶（ACE）抑制剂。
T6595	Moexipril hydrochloride 莫昔普利盐酸盐,Moexipril HCl,RS-10085,SPM 925,CI-925	Apoptosis; RAAS	Apoptosis; Endocrinology/Hormones
	Moexipril hydrochloride (Moexipril HCl) 是一种有口服活性的，不含巯基的血管紧张素转化酶抑制剂，可治疗高血压和充血性心力衰竭。
T6444	Cilazapril Monohydrate Ro 31-2848 monohydrate,Justor,西拉普利,西拉普利水合物	RAAS	Endocrinology/Hormones
	Cilazapril Monohydrate (Justor) 是一种血管紧张素转化酶抑制剂，能够作用于高血压和充血性心力衰竭的研究。
T25832	Moveltipril Moveltipril calcium,MC-838,Altiopril calcium	RAAS	Endocrinology/Hormones
	Moveltipril (Moveltipril calcium) 是一种强效血管紧张素转换酶(ACE)抑制剂。
T20689	Temocaprilat RNH-5139,RS-5139,RNH 5139,RNH5139,替莫普利,RS5139,RS 5139	Angiotensin-converting Enzyme (ACE)	Metabolism
	Temocaprilat (RS5139) 是一种血管紧张素转换酶 (ACE) 抑制剂。 Temocaprilat 通过缺乏 EHBR 的 cMOAT 有效地从胆汁中排泄，而许多其他 ACE 抑制剂对 cMOAT 的亲和力较低。
T25226	Ceronapril Ceronaprilum,SQ 29852,SQ-29852,SQ29852	RAAS	Endocrinology/Hormones
	Ceronapril (SQ 29852) 是一种具有口服活性和高效性的血管紧张素转换酶 (ACE) 抑制剂(IC50 : 36 nM),可用于研究痴呆和高血压。
T24906L	Tuna AI acetate	Angiotensin-converting Enzyme (ACE)	Metabolism
	Tuna AI acetate 是一种源自金枪鱼肌肉的非竞争性血管紧张素转换酶 (ACE) 抑制剂。
TP1750L	H-Ile-Pro-Pro-OH acetate H-Ile-Pro-Pro-OH acetate(26001-32-1 free base)	Angiotensin-converting Enzyme (ACE)	Metabolism
	H-Ile-Pro-Pro-OH acetate 是一种血管紧张素转换酶抑制剂,为乳源三肽。
T7354	H-Val-Pro-Pro-OH	RAAS	Endocrinology/Hormones
	H-Val-Pro-Pro-OH 是一种血管紧张素 I 转化酶(ACE)的抑制剂(IC50:9 μM)。他是一种来源于牛奶的脯氨酸肽衍生物。
TP1682L	Abz-FR-K(Dnp)-P-OH acetate Abz-FR-K(Dnp)-P-OH acetate (500799-61-1 free base)	Others	Others
	Abz-FR-K(Dnp)-P-OH acetate(500799-61-1 free base) 是一种出色的血管紧张素 I 转换酶 (ACE) 底物，Km 值为 4.0 μM，kcat 值为 210s-1。
TP1920L1	Acein acetate	RAAS	Endocrinology/Hormones
	Acein acetate 是高亲和力血管紧张素转换酶 (ACE) 配体 (Kd = 2.79 nM)。浓度高达 500 nM 时对 ACE 酶活性没有显着影响。增强 NMDA + D-丝氨酸诱导的多巴胺从体外纹状体切片和体内纹状体的释放。
TP1295	Angiotensin I (human, mouse, rat) Angiotensin 1 Human,血管紧张素 1 (人)	Others	Others
	Angiotensin I (human, mouse, rat) 是血管紧张素Ⅱ的前体物质，在血管紧张素转化酶 (ACE) 的参与下裂解成血管紧张素Ⅱ。
TP1404L	Hemorphin-7 acetate(152685-85-3 free base)	Opioid Receptor	Endocrinology/Hormones; GPCR/G Protein; Neuroscience
	Hemorphin-7 acetate(152685-85-3 free base) 是一种 hemorphin 肽，一种源自血红蛋白 β 链的内源性阿片肽。 Hemorphin 肽具有镇痛和抗高血压活性，可激活阿片受体并抑制血管紧张素转换酶 (ACE)。
T27608	Indolapril hydrochloride REV 6000A(SS),CI-907,CI 907,CI907,Indolapril HCl	Others	Others
	Indolapril hydrochloride is a nonsulfhydryl angiotensin converting enzyme (ACE) inhibitor with antihypertensive activity.
T12198	NCX899	Others	Others
	NCX899 shows inhibitory activity against angiotensin-converting enzyme (ACE) activity.
T25254	CL 242817 CL242817,CL-242817	Others	Others
	CL 242817 is an inhibitor of angiotensin converting enzyme (ACE).
T70698	MDL-100173	Others	Others
	MDL-100173 is a dual angiotensin-converting enzyme (ACE)/neutral endopeptidase (NEP) inhibitor.
T20921	Benazepril CGS-14824-A,贝那普利	Others	Others
	Benazepril inhibits the activity of circulating angiotensin-converting enzyme (ACE) in horses.
T62377	Zofenopril	Others	Others
	Zofenopril 是一种 angiotensin-converting enzyme (ACE) 抑制剂 (IC50: 81 μM)。
T13274	Utibapril FPL 63547	Others	Others
	Utibapril is an inhibitor of angiotensin-converting enzyme (ACE) with antihypertensive activities.
T12704	Rentiapril SA-446	RAAS	Endocrinology/Hormones
	Rentiapril is an orally active inhibitor of angiotensin converting enzyme (ACE), with antihypertensive activity.
T68412	Cilazaprilat	Others	Others
	Cilazaprilat is the active metabolite of cilazapril, a pyridazine angiotensin-converting enzyme (ACE) inhibitor with antihypertensive activity.
T28584	Ro 31-8472 Ro-31-8472,Ro 318472	Others	Others
	Ro 31-8472 is an angiotensin-converting enzyme (ACE) inhibitor and an analog of cilazaprilat.
T71028	Lisinopril, epsilon-biotinamidocaproyl-	Others	Others
	Lisinopril, epsilon-biotinamidocaproyl- is an angiotensin converting enzyme (ACE) inhibitor.
T36224	N-Hippuryl-His-Leu (hydrate)
	N-Hippuryl-His-Leu (hydrate) is a synthetic substrate for angiotensin-converting enzyme (ACE) that has been used in the in vitro identification of ACE inhibitors.,

化合物

Leucylarginylproline

Cat.No: T7510

Target: RAAS

Cat.No: T1484

Synonym: Perindoprilate,培哚普利

Target: RAAS, MRP, AChR

Fosinopril sodium

Cat.No: T1489

Synonym: SQ28555,福辛普利钠

Target: RAAS

Resorcinolnaphthalein

Cat.No: T13865

Target: RAAS

Cat.No: T16116

Target: RAAS

Diminazene Aceturate

Cat.No: T1145

Synonym: DIZE

Target: Others, Serine Protease, Parasite

Cat.No: T7686

Target: RAAS

Cat.No: T1605

Synonym: MK-421,依那普利

Target: RAAS, MRP

N-Acetyl-Ser-Asp-Lys-Pro

Cat.No: TP1828

Target: RAAS

Cat.No: T7714

Target: Tyrosinase

Cat.No: T7808

Synonym: Cetapril,阿拉普利,DU-1219

Target: RAAS

Angiotensin (1-7)

Cat.No: T7339

Synonym: Ang-(1-7),Angiotensin 1-7,ASP-ARG-VAL-TYR-ILE-HIS-PRO

Target: RAAS, Endogenous Metabolite

Cat.No: T1645

Synonym: HOE-498,Tritace,雷米普利,Altace,Carasel

Target: Apoptosis, RAAS

Zofenopril calcium

Cat.No: T5030

Synonym: SQ26991,佐芬普利钙,Zofenopril (calcium)

Target: RAAS, Reactive Oxygen Species

Benazepril hydrochloride

Cat.No: T0180

Synonym: 盐酸贝那普利,CGS 14824A HCl,Benazepril HCl,CGS14824A

Target: RAAS

Cat.No: T2679

Synonym: BMS265246

Target: CDK

Enalaprilat Dihydrate

Cat.No: T6340

Synonym: 依那普利拉二水合物,MK-422,MK-422 Dihydrate

Target: RAAS, Autophagy

Delapril hydrochloride

Cat.No: T3281

Synonym: indalapril,地拉普利盐酸盐,Alindapril Hydrochloride,Delapril Hydrochloride,盐酸地拉普利,CV 3317

Target: RAAS

Cat.No: T5329

Target: Angiotensin-converting Enzyme (ACE)

Imidapril hydrochloride

Cat.No: T6542

Synonym: Novaloc,Imidapril HCl,盐酸咪达普利,Tanapril,TA-6366

Target: RAAS

Lisinopril dihydrate

Cat.No: T0706

Synonym: Lisinopril,Renacor,赖诺普利二水合物,MK-521 (dihydrate)

Target: RAAS, MRP

Temocapril hydrochloride

Cat.No: T6698

Synonym: CS-622 HCl,Acecol,Temocapril HCl,CS-622,盐酸替莫普利

Target: RAAS

Quinapril hydrochloride

Cat.No: T0805

Synonym: CI-906,PD-109452-2,盐酸喹那普利,Quinapril HCl

Target: RAAS

Perindopril erbumine

Cat.No: T1484L

Synonym: 培哚普利叔丁胺,培哚普利叔丁胺盐,S9490-3,Perindopril tert-butylamine salt

Target: Apoptosis, RAAS, MRP

Cat.No: T1462

Synonym: SQ 14225,甲巯丙脯酸,卡托普利,SQ-14534,SA333

Target: RAAS

Enalapril Maleate

Cat.No: T6486

Synonym: MK-421 Maleate,Renitec Maleate,Glioten Maleate,MK-421 (maleate),Vasotec Maleate,马来酸依那普利

Target: RAAS

Moexipril hydrochloride

Cat.No: T6595

Synonym: 莫昔普利盐酸盐,Moexipril HCl,RS-10085,SPM 925,CI-925

Target: Apoptosis, RAAS

Cilazapril Monohydrate

Cat.No: T6444

Synonym: Ro 31-2848 monohydrate,Justor,西拉普利,西拉普利水合物

Target: RAAS

Cat.No: T25832

Synonym: Moveltipril calcium,MC-838,Altiopril calcium

Target: RAAS

Cat.No: T20689

Synonym: RNH-5139,RS-5139,RNH 5139,RNH5139,替莫普利,RS5139,RS 5139

Target: Angiotensin-converting Enzyme (ACE)

Cat.No: T25226

Synonym: Ceronaprilum,SQ 29852,SQ-29852,SQ29852

Target: RAAS

Tuna AI acetate

Cat.No: T24906L

Target: Angiotensin-converting Enzyme (ACE)

H-Ile-Pro-Pro-OH acetate

Cat.No: TP1750L

Synonym: H-Ile-Pro-Pro-OH acetate(26001-32-1 free base)

Target: Angiotensin-converting Enzyme (ACE)

H-Val-Pro-Pro-OH

Cat.No: T7354

Target: RAAS

Abz-FR-K(Dnp)-P-OH acetate

Cat.No: TP1682L

Synonym: Abz-FR-K(Dnp)-P-OH acetate (500799-61-1 free base)

Target: Others

Acein acetate

Cat.No: TP1920L1

Target: RAAS

Angiotensin I (human, mouse, rat)

Cat.No: TP1295

Synonym: Angiotensin 1 Human,血管紧张素 1 (人)

Target: Others

Hemorphin-7 acetate(152685-85-3 free base)

Cat.No: TP1404L

Target: Opioid Receptor

Indolapril hydrochloride

Cat.No: T27608

Synonym: REV 6000A(SS),CI-907,CI 907,CI907,Indolapril HCl

Target: Others

Cat.No: T12198

Target: Others

Cat.No: T25254

Synonym: CL242817,CL-242817

Target: Others

Cat.No: T70698

Target: Others

Cat.No: T20921

Synonym: CGS-14824-A,贝那普利

Target: Others

Cat.No: T62377

Target: Others

Cat.No: T13274

Synonym: FPL 63547

Target: Others

Cat.No: T12704

Synonym: SA-446

Target: RAAS

Cat.No: T68412

Target: Others

Cat.No: T28584

Synonym: Ro-31-8472,Ro 318472

Target: Others

Lisinopril, epsilon-biotinamidocaproyl-

Cat.No: T71028

Target: Others

N-Hippuryl-His-Leu (hydrate)

Cat.No: T36224

Cat. No.	Product Name	Target	Signaling Pathways
T5S0106	Peimisine 贝母辛,Ebeiensine	RAAS; AChR	Endocrinology/Hormones; Neuroscience
	Peimisine (Ebeiensine) 非竞争性拮抗气管平滑肌 M 受体，抑制 Ach 引起的平滑肌收缩。它兴奋 β 受体和拮抗内钙释放，促进一氧化氮释放，可舒张气管平滑肌，有平喘作用。
T13299	Vicenin 3 维采宁-3,维采宁 3	RAAS	Endocrinology/Hormones
	Vicenin 3来源于广金钱草的地上部分。Vicenin 3是血管紧张素转换酶抑制剂，IC50=46.91 μM。
T8270	Deserpidine 地舍平,Harmonyl	RAAS	Endocrinology/Hormones
	Deserpidine (Harmonyl) 是从 Rauwolfia canescens 的根中分离的生物碱。Deserpidine 与 Reserpine 相关。Deserpidine 是竞争性血管紧张素转化酶抑制剂，可以被用作抗高血压药以及镇定剂。Deserpidine 还减少了肾上腺皮质血管紧张素 II 诱导的醛固酮分泌。
T5796	Plantainoside D Isoplantamajoside,车前草苷D	RAAS; PKC	Chromatin/Epigenetic; Cytoskeletal Signaling; Endocrinology/Hormones
	Plantainoside D (Isoplantamajoside) 可以抑制 ACE ，IC50=2.17 mM。Plantainoside D 也是IKK-β抑制剂。
T21418	Lisinopril Linopril,赖诺普利,Zestril,Prinivil,Lisipril	RAAS	Endocrinology/Hormones
	Lisinopril (Prinivil) 是一种血管紧张素转化酶抑制剂，能够作用于高血压，充血性心力衰竭和心脏病等。
T3851	Vicenin 2 Vicenin -2,维采宁 2,新西兰牡荆苷	RAAS	Endocrinology/Hormones
	Vicenin 2 来源于广金钱草 (Desmodium styracifolium) 的地上部分。Vicenin 2 是一种血管紧张素转换酶 (ACE) 抑制剂，IC50=43.83 μM。
T3753	Sinapinic Acid Sinapic acid,芥子酸,Synapoic acid	Apoptosis; RAAS; Reactive Oxygen Species; HDAC	Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Endocrinology/Hormones; Immunology/Inflammation; Metabolism; NF-κB
	Sinapinic Acid (Synapoic acid) 是从 Hydnophytum formicarumJack. 根中分离到的酚类，是HDAC 抑制剂，对ACE-I 的活性也有抑制作用。它有抗肿瘤活性，诱导肿瘤细胞凋亡，具有抗氧化、抗糖尿病的作用。
T6627	Phosphoramidon Disodium Phosphoramidon Disodium Salt,磷酰胺二钠	RAAS; Neprilysin; Others	Endocrinology/Hormones; Metabolism; Others
	Phosphoramidon Disodium (Phosphoramidon Disodium Salt) Salt 是一种金属蛋白酶 (metalloprotease) 抑制剂。Phosphoramidon Disodium Salt 抑制内皮素转化酶 (ECE) ，中性肽内切酶 (NEP) 和血管紧张素转换酶 (ACE) 的IC50分别为 3.5 ，0.034 和 78 μM。
TN2295	Vicenin-1 Vicenin -1	Antioxidant; Angiotensin-converting Enzyme (ACE)	Metabolism; oxidation-reduction
	Vicenin-1 (Vicenin -1) 是一种来自豆科植物胡卢巴种子中分离出来的类黄酮糖苷，具有强大的抗炎和抗氧化活性，抑制血管紧张素转换酶 (ACE) 。
TN1464	Camellianin A	Apoptosis; RAAS	Apoptosis; Endocrinology/Hormones
	Camellianin A 是从 A. nitida 和茶叶中提取得到的类黄酮列化合物，具有抗癌活性，抑制血管紧张素转换酶 (ACE) 活性，促进 Hep G2 和 MCF-7 细胞凋亡。Camellianin A 可预防CCl4-通过施加抗氧化应激、抗炎和抗细胞凋亡诱导肝损伤。
T38481	Camellianin B	Others	Others
	Camellianin B, a flavonoid compound and metabolite of Camellianin A, exhibits antioxidant properties and acts as an angiotensin converting enzyme (ACE) inhibitor.
TN5645	Isomartynoside
	Isomartynoside has inhibition against the angiotensin converting enzyme (ACE) activities, the IC 50 value is 505±26.7μg/ml, it may have antihypertensive effect. Isomartynoside also shows obvious anti-fatigue activity.
TN4860	Pueroside B	COX; PPAR	DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Neuroscience
	Pueroside B may can treat coronary heart disease, it can interact with two or more targets[peroxisome proliferator activated receptor γ (PPAR-γ), angiotensin-converting enzyme (ACE), hydroxymethylglutaryl coenzyme A receptor (HMGR), cyclooxygenase-2 (COX2
TN4431	Leucosceptoside A	RAAS; PKC	Chromatin/Epigenetic; Cytoskeletal Signaling; Endocrinology/Hormones
	Leucosceptoside A shows inhibitory activity against PKCalpha with the IC50 value of 19.0 microM; it also exhibits strong inhibitory capacity against α-glucosidase. Leucosceptoside A has antihypertensive effect, it shows angiotensin converting enzyme (ACE)
T79958	Isocrenatoside	Angiotensin-converting Enzyme (ACE)	Metabolism
	Isocrenatoside (compound 6)为环状八肽，具有ACE抑制活性。该化合物可通过乙醇提取Microtoena prainiana茎部分离纯化。研究显示，1 mg/mL浓度下，Isocrenatoside的ACE抑制效率高达99.3%。
TN1104	Cyanidin 3-sambubioside chloride Cyanidin-3-O-sambubioside chloride	RAAS; Antioxidant; NO Synthase	Endocrinology/Hormones; Immunology/Inflammation; oxidation-reduction
	Cyanidin 3-sambubioside chloride (Cyanidin-3-O-sambubioside chloride) 是一种从植物中提取的花青素，是一种 NO和 H274Y 突变的抑制剂，对流感神经氨酸酶具有抑制作用。Cyanidin 3-sambubioside chloride 具有抗氧化，抗血管生成和抗病毒活性，抑制血管紧张素转换酶 (ACE) 的活性，可用于研究病毒感染和心血管疾病。

天然产物

Cat.No: T5S0106

Synonym: 贝母辛,Ebeiensine

Target: RAAS, AChR

Cat.No: T13299

Synonym: 维采宁-3,维采宁 3

Target: RAAS

Cat.No: T8270

Synonym: 地舍平,Harmonyl

Target: RAAS

Plantainoside D

Cat.No: T5796

Synonym: Isoplantamajoside,车前草苷D

Target: RAAS, PKC

Cat.No: T21418

Synonym: Linopril,赖诺普利,Zestril,Prinivil,Lisipril

Target: RAAS

Cat.No: T3851

Synonym: Vicenin -2,维采宁 2,新西兰牡荆苷

Target: RAAS

Cat.No: T3753

Synonym: Sinapic acid,芥子酸,Synapoic acid

Target: Apoptosis, RAAS, Reactive Oxygen Species, HDAC

Phosphoramidon Disodium

Cat.No: T6627

Synonym: Phosphoramidon Disodium Salt,磷酰胺二钠

Target: RAAS, Neprilysin, Others

Cat.No: TN2295

Synonym: Vicenin -1

Target: Antioxidant, Angiotensin-converting Enzyme (ACE)

Cat.No: TN1464

Target: Apoptosis, RAAS

Cat.No: T38481

Target: Others

Cat.No: TN5645

Cat.No: TN4860

Target: COX, PPAR

Leucosceptoside A

Cat.No: TN4431

Target: RAAS, PKC

Cat.No: T79958

Target: Angiotensin-converting Enzyme (ACE)

Cyanidin 3-sambubioside chloride

Cat.No: TN1104

Synonym: Cyanidin-3-O-sambubioside chloride

Target: RAAS, Antioxidant, NO Synthase

Species：

Expression System：

Tag：

Cat. No.	Product Name	Species	Expression System
TMPJ-00386	ACE2/ACEH Protein, Human, Recombinant (HEK293, His & Avi), Biotinylated Metalloprotease MPROT15,ACEH,Angiotensin-<...	Human	HEK293 Cells
	Angiotensin-Converting Enzyme 2 (ACE-2) is an integral membrane protein and a zinc metalloprotease of the ACE family, the ACE family includes somatic and germinal ACE. ACE-2 cleaves angiotensins I and II as a carboxypeptidase, ACE-2 converts angiotensin I to angiotensin 1-9, and angiotensin II to angiotensin 1-7. ACE-2 is also able to hydrolyze apelin-13 and dynorphin-13 with high efficiency. ACE-2 can be high expressed in testis, kidney and heart, in colon, small intestine and ovary at moderate...
TMPH-03081	ACE2 Protein, Paguma larvata, Recombinant (hFc) EC:3.4.17.23,Angiotensin-converting en...	Paguma larvata	HEK293 Cells
	ACE2 Protein, Paguma larvata, Recombinant (hFc) is expressed in HEK293 mammalian cells with C-hFc tag. The predicted molecular weight is 112.7 kDa and the accession number is Q56NL1.
TMPY-02574	Chymase 1 Protein, Human, Recombinant (His) MCT1,chymase 1, mast cell,chymase,CYH	Human	Baculovirus Insect Cells
	The STR polymorphism in the CMA1 gene is associated with asthma and that this association is even stronger with atopic asthma. CMA1 and IL-4 in atopic asthma and for IL-4 in atopy in general. The local angiotensin II system (LAS) has numerous functions, including the regulation of growth and differentiation in the gastrointestinal tract. Angiotensin II (AngII) may be generated by angiotensin-I-converting enzyme (ACE) or mast cell chymase (CMA1) and plays an important role in inflammatory process...

重组蛋白

ACE2/ACEH Protein, Human, Recombinant (HEK293, His & Avi), Biotinylated

Cat.No: TMPJ-00386

Species: Human

Expression System: HEK293 Cells

ACE2 Protein, Paguma larvata, Recombinant (hFc)

Cat.No: TMPH-03081

Species: Paguma larvata

Expression System: HEK293 Cells

Chymase 1 Protein, Human, Recombinant (His)

Cat.No: TMPY-02574

Species: Human

Expression System: Baculovirus Insect Cells

Cat. No.	Product Name	Target	Signaling Pathways
T11193	Enalaprilat-d5 sodium MK-422 D5 Sodium Salt,依那普利拉钠 D5,Enalaprilat D5 Sodium Salt	Others	Others
	Enalaprilat D5 Sodium Salt is the deuterium labeled Enalaprilat, which is an angiotensin-converting enzyme (ACE) inhibitor.
T11192	Enalapril D5 maleate MK-421 D5 maleate,马来酸依那普利D5	Others	Others
	Enalapril D5 maleate is deuterium labeled Enalapril, which is an angiotensin converting enzyme (ACE) inhibitor.
T11194	Enalaprilat D5 MK-422 D5,依那普利拉 D5	Others	Others
	Enalaprilat D5 is the deuterium labeled Enalaprilat, which is an angiotensin-converting enzyme (ACE) inhibitor.
T13196	Trandolaprilate D5 Trandolaprilat D5,RU 44403 D5	Others	Others
	Trandolaprilate D5 is a deuterium-labeled Trandolaprilate. Trandolaprilate is an inhibitor of angiotensin-converting enzyme (ACE).
T13195	Trandolapril D5 RU44570 D5	Others	Others
	Trandolapril D5 is a deuterium labeled Trandolapril. Trandolapril is an orally active inhibitor of angiotensin converting enzyme (ACE) for hypertension and congestive heart failure (CHF).
T71065	Quinapril-d5
	Quinapril-d5 is intended for use as an internal standard for the quantification of quinapril by GC- or LC-MS. Quinapril is a prodrug form of the angiotensin converting enzyme (ACE) inhibitor quinaprilat. In vivo, quinapril reduces mean arterial pressure in renal hypertensive and spontaneously hypertensive rats. It inhibits angiotensin I-induced pressor responses in normotensive rats and dogs. Quinapril prevents left ventricular heart failure in CHF 14.6 cardiomyopathic hamsters. Formulations con...
TMIJ-0253	Benazepril-d5 HCl
	Benazepril-d5 HCl 是 Benazepril HCl 的氘代化合物。Benazepril HCl 的 CAS 号为 86541-74-4。Benazepril hydrochloride 是一种血管紧张素转化酶（ACE）抑制剂，能够作用于高血压。
T70883	Moexipril-d5
	Moexipril-d5 intended for use as an internal standard for the quantification of moexipril by GC- or LC-MS. Moexipril is a prodrug form of the angiotensin converting enzyme (ACE) inhibitor moexiprilat. It is converted to moexiprilat in vivo by side chain ester hydrolysis. Moexipril inhibits ACE in a cell-free assay (IC50 = 2.7 µM for the rabbit enzyme). It also inhibits phosphodiesterase 4 (IC50s = 38, 160, and 230 µM for PDE4B2, PDE4A5 and PDE4D5, respectively). Moexipril (0.1-30 mg/kg per day) ...

同位素标记化合物

Enalaprilat-d5 sodium

Cat.No: T11193

Synonym: MK-422 D5 Sodium Salt,依那普利拉钠 D5,Enalaprilat D5 Sodium Salt

Target: Others

Enalapril D5 maleate

Cat.No: T11192

Synonym: MK-421 D5 maleate,马来酸依那普利D5

Target: Others

Cat.No: T11194

Synonym: MK-422 D5,依那普利拉 D5

Target: Others

Trandolaprilate D5

Cat.No: T13196

Synonym: Trandolaprilat D5,RU 44403 D5

Target: Others

Trandolapril D5

Cat.No: T13195

Synonym: RU44570 D5

Target: Others

Cat.No: T71065

Benazepril-d5 HCl

Cat.No: TMIJ-0253

Cat.No: T70883

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