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Search Results for " angiotensin receptor "
Targets Recommended: RAAS Others

161

抑制剂 & 化合物

8

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同位素标记化合物

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Cat. No. Product Name
L7110 抗高血压化合物库

678 compounds
678 种高血压相关的小分子,用于高通量和高内涵筛选;

化合物库

抗高血压化合物库
Cat.No: L7110
Compounds: 678
Cat. No. Product Name Target Signaling Pathways
TP1528 Angiotensin I/II (1-5)

Angiotensin I/II 1-5

RAAS; Others Endocrinology/Hormones; Others
Angiotensin I/II (1-5) 是由血管紧张素 I/II 肽转化而来,有 1-5 个氨基酸组成的多肽。血管紧张素 I 是由肾素对血管紧张素原的作用形成的,血管紧张素 I 可产生血管紧张素 II 。血管紧张素 II 用于高血压、特发性膜性肾病和肾素-血管紧张素系统的研究。
TP1579 Angiotensin I/II (1-6)

Angiotensin I/II 1-6

RAAS; Others Endocrinology/Hormones; Others
Angiotensin I/II (1-6) 是由血管紧张素 I/II 肽转化而来,含有 1-6 个氨基酸的多肽。血管紧张素 I 被血管紧张素转换酶水解,形成具有生物活性的血管紧张素 II。血管紧张素 II 用于高血压、特发性膜性肾病和肾素-血管紧张素系统的研究。
T7577 Angiotensin III, human, mouse

血管紧张素III,Angiotensin III, human, mouse(3TFA)

RAAS Endocrinology/Hormones
Angiotensin III, human, mouse (Angiotensin III, human, mouse(3TFA)) 是一种七肽,是血管紧张素 2 型受体 (AT2R) 激动剂,能够作用于 AT2R (IC50:0.648 nM)及 AT1R (IC50:21.1nM)。
T8560 Angiotensin II human acetate

Ang II acetate,DRVYIHPF acetate,Angiotensin II acetate,血管紧张素II

Apoptosis; RAAS Apoptosis; Endocrinology/Hormones
Angiotensin II human acetate (DRVYIHPF acetate) 是血管收缩剂,是肾素/血管紧张素系统的主要生物活性肽,在调节人类血压中起着核心作用。它刺激交感神经刺激,增加醛固酮生物合成和肾脏活动。它诱导血管平滑肌细胞生长,也诱导细胞凋亡。它通过 LOX-1 依赖的氧化还原敏感途径诱导内皮细胞毛细血管形成。
T7339 Angiotensin (1-7)

Ang-(1-7),Angiotensin 1-7,ASP-ARG-VAL-TYR-ILE-HIS-PRO

RAAS; Endogenous Metabolite Endocrinology/Hormones; Metabolism
Angiotensin (1-7) (ASP-ARG-VAL-TYR-ILE-HIS-PRO) 是肾素-血管紧张素系统中的内源性七肽。Angiotensin 1-7在心肌细胞中具有抗炎和抗纤维化活性,因此具有心脏保护作用。它能抑制血管紧张素转换酶和释放一氧化氮,是激肽诱导的血管舒张的局部协同调节剂。它阻断 Ang II 诱导的平滑肌细胞增殖和肥大,并显示对内皮的抗血管生成和生长抑制作用。它显示出抗炎活性。
TP1929L1 Saralasin acetate(34273-10-4 free base)

RAAS Endocrinology/Hormones
Saralasin acetate(34273-10-4 free base) 是一种非选择性血管紧张素 II 拮抗剂。
T2531 Eprosartan Mesylate

SKF-108566J,甲磺酸依普罗沙坦

RAAS Endocrinology/Hormones
Eprosartan Mesylate (SKF-108566J) 是一种具有选择性、竞争性血管紧张素 II 受体拮抗剂,是具有口服活性的非肽。它结合血管紧张素 II 受体,在大鼠和人类肾上腺皮质膜中的IC50值分别为 9.2 nM 和 3.9 nM,可用作降压剂。
T7354 H-Val-Pro-Pro-OH

RAAS Endocrinology/Hormones
H-Val-Pro-Pro-OH 是一种血管紧张素 I 转化酶(ACE)的抑制剂(IC50:9 μM)。他是一种来源于牛奶的脯氨酸肽衍生物。
T22344 Icatibant Acetate

Bradykinin Receptor GPCR/G Protein
Icatibant acetate 是一种特异性缓激肽 B2 受体拮抗剂,其 IC50=1.07 nM,Ki=0.798 nM。
T1461 Candesartan

CV 11974,坎地沙坦

RAAS Endocrinology/Hormones
Candesartan (CV 11974) 是一种血管紧张素II 受体拮抗剂(IC50:0.26 nM)。
T13376 YS-49

RAAS; Akt; PI3K; Adrenergic Receptor Cytoskeletal Signaling; Endocrinology/Hormones; GPCR/G Protein; Neuroscience; PI3K/Akt/mTOR signaling
YS-49 是一种PI3K/Akt(RhoA 的下游靶标) 的激活剂,可减少 3-甲基胆碱处理的细胞中 RhoA/PTEN 的激活。它是异喹啉化合物生物碱,因能激活心脏β-adrenoceptors 而具有强烈的正性肌力作用。它能通过诱导血红素加氧酶来抑制血管紧张素 II 刺激 VSMC 细胞的增殖。
T5355 Sparsentan

RE-021,DARA-a

RAAS; Endothelin Receptor Endocrinology/Hormones; GPCR/G Protein
Sparsentan (DARA-a) 是一种具有高度选择的血管紧张素 II (Ki:0.8 nM)和内皮素 A 受体(Ki:9.3 nM)的双重拮抗剂。
T6067 PD 123319

(S)-(+)-PD 123319,PD123319

RAAS Endocrinology/Hormones
PD 123319 ((S)-(+)-PD 123319) 是一种血管紧张素 II 受体拮抗剂(IC50:34 nM)。
T7797 Tasosartan

他索沙坦,WAY-ANA 756

RAAS Endocrinology/Hormones
Tasosartan (WAY-ANA 756) 是长效血管紧张素 II 受体拮抗剂。
T1570 Telmisartan

BIBR 277,替米沙坦

RAAS; Autophagy Autophagy; Endocrinology/Hormones
Telmisartan (BIBR 277) 是一种血管紧张素II 1型受体拮抗剂,能够抑制其活性,IC50值为 9.2 nM。
T0215L Losartan

DuP-753,氯沙坦,洛沙坦

RAAS Endocrinology/Hormones
Losartan (DuP-753) 是一种血管紧张素II 受体拮抗剂,能够与血管紧张素II 竞争性结合AT1受体(IC50:20 nM)。
T6219 Azilsartan Medoxomil

TAK-491,阿齐沙坦酯

RAAS Endocrinology/Hormones
Azilsartan Medoxomil (TAK-491) 是一种具有口服活性的1型血管紧张素II 受体拮抗剂(IC50:0.62 nM)。
T1518 Olmesartan Medoxomil

奥美沙坦酯,CS 866,Benicar

RAAS Endocrinology/Hormones
Olmesartan Medoxomil (Benicar) 是血管紧张素 (angiotensin AT1) 受体选择性抑制剂(IC50:66.2 μM)。
T3461 Losartan Carboxylic Acid

EXP-3174,E-3174

RAAS Endocrinology/Hormones
Losartan Carboxylic Acid (E-3174) 是 Losartan 的活性羧酸代谢产物,是血管紧张素Ⅱ受体 1 型(AT1)拮抗剂。它能够阻断血管紧张素 II 诱导的血管平滑肌细胞反应,可以提高血浆肾素活性,降低平均动脉压。
T2318 Sacubitril/Valsartan

Sacubitril mixture with Valsartan,沙库必曲/缬沙坦,Valsartan,Sacubitril,LCZ696

Apoptosis; RAAS; Neprilysin Apoptosis; Endocrinology/Hormones; Metabolism
Sacubitril/Valsartan (LCZ696),以1:1摩尔比由Valsartan(一种ARB)和Sacubitril(AHU377)组成,为创新口服血管紧张素受体-脑啡肽酶(ARN)双重抑制剂,旨在治疗高血压与心力衰竭。其作用机制包括抑制炎症、氧化应激及细胞凋亡,有助于改善糖尿病心肌病。
T2322 Fimasartan

非马沙坦,BR-A-657,Kanarb

Apoptosis; RAAS Apoptosis; Endocrinology/Hormones
Fimasartan (BR-A-657) 是血管紧张素受体 AT1 非肽类拮抗剂,用于研究高血压和心力衰竭。
T2400 Candesartan Cilexetil

TCV-116,坎地沙坦酯,坎地沙坦西酯

Apoptosis; RAAS Apoptosis; Endocrinology/Hormones
Candesartan Cilexetil (TCV-116) 是一种血管紧张素II 拮抗剂,可用于治疗高血压。
T4431 Olodanrigan

PD-126055,EMA401

RAAS Endocrinology/Hormones
Olodanrigan (EMA401) 是具有口服活性、高选择性及外周受限的血管紧张素 Ⅱ 类型 2 受体(AT2R)拮抗剂。它的缓解疼痛的机制可能是:抑制增强的 AngII/AT2R 诱导的 p38 和 p42/p44 MAPK 激活,进而阻碍 DRG 神经元的过度兴奋性及 DRG 神经元的萌发。它可用于研究神经性疼痛。
T5824 Angiotensin II (3-8), human

Angiotensin IV

RAAS Endocrinology/Hormones
Angiotensin II (3-8), human 是活性稍弱的血管紧张素AT1受体激动剂。
T5964 Olmesartan

CS 088,奥美沙坦,RNH 6270

RAAS Endocrinology/Hormones
Olmesartan (RNH 6270) 是一种血管紧张素 II 受体 (AT1R) 拮抗剂,常用于研究高血压。
T2270 Trans-Tranilast

Tranilast trans-,反式-曲尼司特,反-曲尼司特

RAAS Endocrinology/Hormones
Trans-Tranilast 是抗过敏剂,可用于过敏性鼻炎、支气管哮喘和特应性皮炎的研究。
T6716 Valsartan

Diovan,缬沙坦,Tareg,CGP 48933

RAAS Endocrinology/Hormones
Valsartan (CGP 48933) 是一种血管紧张素 II 受体拮抗剂,有用于高血压和心力衰竭的研究潜力。
T7575 [Sar1, Ile8]-Angiotensin II

[Sar1, Ile8]-Angiotensin II(3TFA)

RAAS; Others Endocrinology/Hormones; Others
[Sar1, Ile8]-Angiotensin II 是一种在血管平滑肌细胞中有多种作用(如正常动脉的收缩,培养的细胞或病变血管的肥大或增生等)的多肽,。
T2690 Tranilast

曲尼司特,MK 341,SB 252218

RAAS; Prostaglandin Receptor Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation
Tranilast (SB 252218) 是一种抗过敏药物,可抑制炎症细胞释放脂质介质和细胞因子,抑制前列腺素 D2 (PGD2)产生,IC50为 0.1 mM。它拮抗血管紧张素 II 并抑制其在血管平滑肌细胞中的生物学作用,具有抗炎和免疫调节作用。
T1057 Azilsartan

TAK-536,阿齐沙坦

RAAS Endocrinology/Hormones
Azilsartan (TAK-536) 是一种高活性的血管紧张素Ⅱ1型受体特异性拮抗剂(IC50:2.6 nM)。
T19930 Nitrosoglutathione

S-Nitrosoglutathione,S-亚硝基谷胱甘肽,SNOG,Glutathione thionitrite,GSNO

RAAS; NO Synthase Endocrinology/Hormones; Immunology/Inflammation
Nitrosoglutathione (GSNO) 是一种外源性的 NO 供体,是大鼠酒精脱氢酶III 类同工酶的底物,能够减少脑血管紧张素II 依赖性及非依赖型的 AT1 受体反应。
T1615 Irbesartan

厄贝沙坦,SR-47436,BMS-186295

Apoptosis; RAAS Apoptosis; Endocrinology/Hormones
Irbesartan (SR-47436) 是一种 1 型血管紧张素 II 受体拮抗剂,IC50为1.3 nM。
T0215 Losartan potassium

DuP-753 potassium,洛沙坦钾,氯沙坦钾,MK 954,DuP 753

RAAS Endocrinology/Hormones
Losartan potassium (DuP-753 potassium) 是一种血管紧张素 II 受体 1 型(AT1)拮抗剂,能够与血管紧张素 II 与 AT1 的结合竞争,其 IC50=20 nM。
T3178 BIBS 39

RAAS Endocrinology/Hormones
BIBS 39是新型的非肽类血管紧张素II(AII)受体拮抗剂。
T7616 A 779

RAAS Endocrinology/Hormones
A 779 是一种 G 蛋白偶联受体 Mas 的有效拮抗剂,Mas 受体是Ang1-7 receptor,与传统的AngII 不同。
TP1017L Angiotensin II 5-valine TFA

Angiotensin II 5-valine TFA(58-49-1 free base)

RAAS Endocrinology/Hormones
Angiotensin II 5-valine TFA 是血管紧张素受体的激动剂。
T13390 ZD 7155 hydrochloride

RAAS Endocrinology/Hormones
ZD 7155 hydrochloride 是血管紧张素II 受体1型 (AT1 receptor) 拮抗剂。
T7743 ANGIOTENSIN IV TFA(12676-15-2(free base))

RAAS Endocrinology/Hormones
ANGIOTENSIN IV TFA(12676-15-2(free base)) 是一种不太有效的血管紧张素 AT1 受体激动剂。
T28540 Ripisartan

UP 269-6,UP-2696,UP 2696,UP-269-6,UP269-6

RAAS Endocrinology/Hormones
Ripisartan (UP-269-6) 是一种强效的特异性血管紧张素 II 受体拮抗剂,对血管紧张素 II 介导的交感神经性心动过速反应有抑制作用。
T40220L TRV055 acetate

TRV055 acetate (25849-90-5 Free base)

RAAS Endocrinology/Hormones
TRV055 acetate 是血管紧张素 II 1 型受体的配体,可刺激细胞 Gq 介导的信号传导。
T14337 Buloxibutid

AT2 receptor agonist C21

RAAS Endocrinology/Hormones
Buloxibutid (AT2 receptor agonist C21) 是一种新型且具有选择性小分子 angiotensin II AT2 receptor (血管紧张素 II AT2 受体)激动剂,对 AT2 受体和 AT1 受体的 Ki 值分别为 0.4 nM 和 10 μM。
T24588 Palatrigine

BW-A 256C,BW A256C

Adrenergic Receptor; Angiotensin-converting Enzyme (ACE) GPCR/G Protein; Metabolism; Neuroscience
Palatrigine (BW-A 256C) 是一种具有血管紧张素转换酶抑制和β肾上腺素受体阻断特性的化合物。
T7616L A 779 TFA(159432-28-7 free base)

A 779 3TFA(159432-28-7(free base))

RAAS Endocrinology/Hormones
A 779 TFA 是血管紧张素-(1-7) 受体的有效拮抗剂。
T28009 ME-3221

ME 3221,ME3221

RAAS Endocrinology/Hormones
ME-3221是一种血管紧张素AT1受体拮抗剂,可预防老年中风易发性高血压大鼠的高血压并发症。
T27762 L-162,313

L-162313,L 162,313,L162,313

RAAS Endocrinology/Hormones
L-162,313是一种ANG II受体激动剂,是一种模仿血管紧张素II生物学作用的非肽,可诱导MAP增加。
T2531L Eprosartan

KF-108566J free base,Teveten

RAAS Endocrinology/Hormones
Eprosartan (SKF-108566J free base) 是一种具有选择性和竞争性的非肽类血管紧张素II受体拮抗剂,对AT1受体亚型具有高亲和力,可用作降压剂。Eprosartan 对血管紧张素 II 受体有抑制作用,在大鼠和人类肾上腺皮质膜中的 IC50 值分别为 9.2 nM 和 3.9 nM。
T67848 Valsartan Methyl Ester

RAAS Endocrinology/Hormones
Valsartan Methyl Ester 是一种强效血管紧张素II 受体拮抗剂,IC50=0.06uM。
T28437 Pomisartan

BIBR-363,BIBR 363,BIBR363

RAAS Endocrinology/Hormones
Pomisartan (BIBR-363) 是一种小分子血管紧张素 1 型受体(AT1R)拮抗剂,可用于治疗心血管疾病,研究心脏衰竭和高血压。
T65739 Methyl candesartan

Candesartan Methyl Ester

RAAS Endocrinology/Hormones
Methyl candesartan (Candesartan Methyl Ester) 是一种有效的血管紧张素2受体拮抗剂,可用于研究高血压。
T35834L (Sar¹)-Angiotensin II acetate

RAAS Endocrinology/Hormones
(Sar¹)-Angiotensin II acetate 是血管紧张素 II 的类似物,是血管紧张素 AT1 受体的特异性激动剂。它与富含脑膜的颗粒结合,Kd 为 2.7 nM。它可以刺激胚胎鸡肌细胞中的蛋白质合成和细胞生长。

化合物

Angiotensin I/II (1-5)
Cat.No: TP1528
Synonym: Angiotensin I/II 1-5
Target: RAAS, Others
Angiotensin I/II (1-6)
Cat.No: TP1579
Synonym: Angiotensin I/II 1-6
Target: RAAS, Others
Angiotensin III, human, mouse
Cat.No: T7577
Synonym: 血管紧张素III,Angiotensin III, human, mouse(3TFA)
Target: RAAS
Angiotensin II human acetate
Cat.No: T8560
Synonym: Ang II acetate,DRVYIHPF acetate,Angiotensin II acetate,血管紧张素II
Target: Apoptosis, RAAS
Angiotensin (1-7)
Cat.No: T7339
Synonym: Ang-(1-7),Angiotensin 1-7,ASP-ARG-VAL-TYR-ILE-HIS-PRO
Target: RAAS, Endogenous Metabolite
Saralasin acetate(34273-10-4 free base)
Cat.No: TP1929L1
Synonym:
Target: RAAS
Eprosartan Mesylate
Cat.No: T2531
Synonym: SKF-108566J,甲磺酸依普罗沙坦
Target: RAAS
H-Val-Pro-Pro-OH
Cat.No: T7354
Synonym:
Target: RAAS
Icatibant Acetate
Cat.No: T22344
Synonym:
Target: Bradykinin Receptor
Candesartan
Cat.No: T1461
Synonym: CV 11974,坎地沙坦
Target: RAAS
YS-49
Cat.No: T13376
Synonym:
Target: RAAS, Akt, PI3K, Adrenergic Receptor
Sparsentan
Cat.No: T5355
Synonym: RE-021,DARA-a
Target: RAAS, Endothelin Receptor
PD 123319
Cat.No: T6067
Synonym: (S)-(+)-PD 123319,PD123319
Target: RAAS
Tasosartan
Cat.No: T7797
Synonym: 他索沙坦,WAY-ANA 756
Target: RAAS
Telmisartan
Cat.No: T1570
Synonym: BIBR 277,替米沙坦
Target: RAAS, Autophagy
Losartan
Cat.No: T0215L
Synonym: DuP-753,氯沙坦,洛沙坦
Target: RAAS
Azilsartan Medoxomil
Cat.No: T6219
Synonym: TAK-491,阿齐沙坦酯
Target: RAAS
Olmesartan Medoxomil
Cat.No: T1518
Synonym: 奥美沙坦酯,CS 866,Benicar
Target: RAAS
Losartan Carboxylic Acid
Cat.No: T3461
Synonym: EXP-3174,E-3174
Target: RAAS
Sacubitril/Valsartan
Cat.No: T2318
Synonym: Sacubitril mixture with Valsartan,沙库必曲/缬沙坦,Valsartan,Sacubitril,LCZ696
Target: Apoptosis, RAAS, Neprilysin
Fimasartan
Cat.No: T2322
Synonym: 非马沙坦,BR-A-657,Kanarb
Target: Apoptosis, RAAS
Candesartan Cilexetil
Cat.No: T2400
Synonym: TCV-116,坎地沙坦酯,坎地沙坦西酯
Target: Apoptosis, RAAS
Olodanrigan
Cat.No: T4431
Synonym: PD-126055,EMA401
Target: RAAS
Angiotensin II (3-8), human
Cat.No: T5824
Synonym: Angiotensin IV
Target: RAAS
Olmesartan
Cat.No: T5964
Synonym: CS 088,奥美沙坦,RNH 6270
Target: RAAS
Trans-Tranilast
Cat.No: T2270
Synonym: Tranilast trans-,反式-曲尼司特,反-曲尼司特
Target: RAAS
Valsartan
Cat.No: T6716
Synonym: Diovan,缬沙坦,Tareg,CGP 48933
Target: RAAS
[Sar1, Ile8]-Angiotensin II
Cat.No: T7575
Synonym: [Sar1, Ile8]-Angiotensin II(3TFA)
Target: RAAS, Others
Tranilast
Cat.No: T2690
Synonym: 曲尼司特,MK 341,SB 252218
Target: RAAS, Prostaglandin Receptor
Azilsartan
Cat.No: T1057
Synonym: TAK-536,阿齐沙坦
Target: RAAS
Nitrosoglutathione
Cat.No: T19930
Synonym: S-Nitrosoglutathione,S-亚硝基谷胱甘肽,SNOG,Glutathione thionitrite,GSNO
Target: RAAS, NO Synthase
Irbesartan
Cat.No: T1615
Synonym: 厄贝沙坦,SR-47436,BMS-186295
Target: Apoptosis, RAAS
Losartan potassium
Cat.No: T0215
Synonym: DuP-753 potassium,洛沙坦钾,氯沙坦钾,MK 954,DuP 753
Target: RAAS
BIBS 39
Cat.No: T3178
Synonym:
Target: RAAS
A 779
Cat.No: T7616
Synonym:
Target: RAAS
Angiotensin II 5-valine TFA
Cat.No: TP1017L
Synonym: Angiotensin II 5-valine TFA(58-49-1 free base)
Target: RAAS
ZD 7155 hydrochloride
Cat.No: T13390
Synonym:
Target: RAAS
ANGIOTENSIN IV TFA(12676-15-2(free base))
Cat.No: T7743
Synonym:
Target: RAAS
Ripisartan
Cat.No: T28540
Synonym: UP 269-6,UP-2696,UP 2696,UP-269-6,UP269-6
Target: RAAS
TRV055 acetate
Cat.No: T40220L
Synonym: TRV055 acetate (25849-90-5 Free base)
Target: RAAS
Buloxibutid
Cat.No: T14337
Synonym: AT2 receptor agonist C21
Target: RAAS
Palatrigine
Cat.No: T24588
Synonym: BW-A 256C,BW A256C
Target: Adrenergic Receptor, Angiotensin-converting Enzyme (ACE)
A 779 TFA(159432-28-7 free base)
Cat.No: T7616L
Synonym: A 779 3TFA(159432-28-7(free base))
Target: RAAS
ME-3221
Cat.No: T28009
Synonym: ME 3221,ME3221
Target: RAAS
L-162,313
Cat.No: T27762
Synonym: L-162313,L 162,313,L162,313
Target: RAAS
Eprosartan
Cat.No: T2531L
Synonym: KF-108566J free base,Teveten
Target: RAAS
Valsartan Methyl Ester
Cat.No: T67848
Synonym:
Target: RAAS
Pomisartan
Cat.No: T28437
Synonym: BIBR-363,BIBR 363,BIBR363
Target: RAAS
Methyl candesartan
Cat.No: T65739
Synonym: Candesartan Methyl Ester
Target: RAAS
(Sar¹)-Angiotensin II acetate
Cat.No: T35834L
Synonym:
Target: RAAS
Cat. No. Product Name Target Signaling Pathways
T7040 Angiotensin II human

DRVYIHPF,Angiotensin II,Hypertensin II,血管紧张素Ⅱ,Ang II,血管紧张素II

Apoptosis; RAAS Apoptosis; Endocrinology/Hormones
Angiotensin II human (Ang II) 是一种生物活性肽,一种血管收缩剂。Angiotensin II 可以与 AT1R 和 AT2R 相互作用,调节人类血压,刺激交感神经,增加醛固酮生物合成和肾脏活动。
T5S0106 Peimisine

贝母辛,Ebeiensine

RAAS; AChR Endocrinology/Hormones; Neuroscience
Peimisine (Ebeiensine) 非竞争性拮抗气管平滑肌 M 受体,抑制 Ach 引起的平滑肌收缩。它兴奋 β 受体和拮抗内钙释放,促进一氧化氮释放,可舒张气管平滑肌,有平喘作用。
T2836 Isorhamnetin

3-methylquercetin,3'-Methylquercetin,Isorhamnetol,异鼠李素,3'-Methoxyquercetin

MEK; PI3K; Endogenous Metabolite MAPK; Metabolism; PI3K/Akt/mTOR signaling
Isorhamnetin (3-methylquercetin) 是从中草药沙棘中提取的一种类黄酮,可通过抑制MEK1和PI3K 来抑制皮肤癌。
T37298 Spinacine

Endogenous Metabolite Metabolism
Spinacine 是人内源性代谢产物。
TN4860 Pueroside B

COX; PPAR DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Neuroscience
Pueroside B may can treat coronary heart disease, it can interact with two or more targets[peroxisome proliferator activated receptor γ (PPAR-γ), angiotensin-converting enzyme (ACE), hydroxymethylglutaryl coenzyme A receptor (HMGR), cyclooxygenase-2 (COX2
T38593 1-Methyl-2-[(6Z,9Z)-6,9-pentadecadienyl]-4(1H)-quinolone

Others Others
Methyl-2-[(6Z,9Z)-6,9-pentadecadienyl]-4(1H)-quinolone9, a quinolone alkaloid derived from Evodia rutaecarpa, is a potent antagonist of the angiotensin II receptor, displaying an IC50 value of 48.2 μM.
TN1061 Ganoderol B

Androgen Receptor Endocrinology/Hormones
Ganoderol B is a potent β ±-glucosidase and angiotensin-converting enzyme inhibitor, with an IC(50) of β ±-glucosidase is 119.8 uM. It may be useful in prostate cancer and benign prostatic hyperplasia (BPH) therapy through suppressing the function of andr
T75697 1-Methyl-2-[(4Z,7Z)-4,7-tridecadienyl]-4(1H)-quinolone

Others Others
1-Methyl-2-[(4Z,7Z)-4,7-tridecadienyl]-4(1H)-quinolone,为喹诺酮类生物碱,作用为二酰基甘油酰基转移酶抑制剂与血管紧张素II受体阻断剂,其IC50值依次为20.1 μM与34.1 μM。此化合物亦展现对幽门螺杆菌的有效抗活性,MIC值达10 μg/mL。

天然产物

Angiotensin II human
Cat.No: T7040
Synonym: DRVYIHPF,Angiotensin II,Hypertensin II,血管紧张素Ⅱ,Ang II,血管紧张素II
Target: Apoptosis, RAAS
Peimisine
Cat.No: T5S0106
Synonym: 贝母辛,Ebeiensine
Target: RAAS, AChR
Isorhamnetin
Cat.No: T2836
Synonym: 3-methylquercetin,3'-Methylquercetin,Isorhamnetol,异鼠李素,3'-Methoxyquercetin
Target: MEK, PI3K, Endogenous Metabolite
Spinacine
Cat.No: T37298
Synonym:
Target: Endogenous Metabolite
Pueroside B
Cat.No: TN4860
Synonym:
Target: COX, PPAR
1-Methyl-2-[(6Z,9Z)-6,9-pentadecadienyl]-4(1H)-quinolone
Cat.No: T38593
Synonym:
Target: Others
Ganoderol B
Cat.No: TN1061
Synonym:
Target: Androgen Receptor
1-Methyl-2-[(4Z,7Z)-4,7-tridecadienyl]-4(1H)-quinolone
Cat.No: T75697
Synonym:
Target: Others
Cat. No. Product Name Species Expression System
TMPH-02268 AGTR2 Protein, Human, Recombinant (His & SUMO)

AT2 receptor,Angiotensin II type-2 rec...

Human E. coli
Receptor for angiotensin II. Cooperates with MTUS1 to inhibit ERK2 activation and cell proliferation.
TMPH-02267 AGTRAP Protein, Human, Recombinant (His & Myc & SUMO)

ATRAP,AT1 receptor-associated protein,Type-1 an...

Human E. coli
Appears to be a negative regulator of type-1 angiotensin II receptor-mediated signaling by regulating receptor internalization as well as mechanism of receptor desensitization such as phosphorylation. Induces also a decrease in cell proliferation and angiotensin II-stimulated transcriptional activity.
TMPH-01739 NLRP3 Protein, Human, Recombinant (His)

PYRIN-containing APAF1-like protein 1,Caterpiller protein 1....

Human E. coli
NLRP3 Protein, Human, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 27.7 kDa and the accession number is Q96P20.
TMPY-02869 MMP-12 Protein, Human, Recombinant (catalytic domain)

HME,ME,MMP-12,MME,matrix metallopeptidase 12

Human E. coli
Matrix metalloproteinases (MMPs) are a family of zinc-dependent endopeptidases that degrade components of the extracellular matrix (ECM) and play essential roles in various physiological processes such as morphogenesis, differentiation, angiogenesis, and tissue remodeling, as well as pathological processes including inflammation, arthritis, cardiovascular diseases, pulmonary diseases, and tumor invasion. Macrophage Metalloelastase, also known as Matrix metalloproteinase-12, Macrophage elastase, ...
TMPK-00438 SARS-COV-2 Spike S Trimer Protein (His & Avi)

COVID-19,S protein,S glycoprotein,Spike glycoprotein

SARS-CoV-2 HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays key parts in the induction of neutralizing-antibody and T-cell responses, as well as protective immunity. SARS-COV-2 Spike S Trimer Protein (His & Avi) is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weight is 136.6 kDa and the accession number i...
TMPK-00908 SARS Spike S1 Protein (hFc & Avi)

Spike protein S1,S1 protein,Spike,S1 protein,S glycoprotein ...

SARS HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays key parts in the induction of neutralizing-antibody and T-cell responses, as well as protective immunity. SARS Spike S1 Protein (hFc & Avi) is expressed in HEK293 mammalian cells with C-hFc-Avi tag. The predicted molecular weight is 100.6 kDa and the accession number is P59594.
TMPK-00913 SARS Spike S1 Protein (His & Avi), Biotinylated

Spike protein S1,S glycoprotein Subunit1,S1 protein,Spike,S1...

SARS HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays key parts in the induction of neutralizing-antibody and T-cell responses, as well as protective immunity. SARS Spike S1 Protein (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weight is 75.9 kDa and the accession number ...
TMPK-00440 SARS-COV-2 Spike S1 Protein (His & Avi), Biotinylated

S1 protein,S glycoprotein Subunit1,Spike,S1 protein,Spike pr...

SARS-CoV-2 HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays key parts in the induction of neutralizing-antibody and T-cell responses, as well as protective immunity. SARS-COV-2 Spike S1 Protein (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weight is 77.9 kDa and the accession n...
TMPK-00909 SARS Spike S1 Protein (hFc & Avi), Biotinylated

Spike protein S1,S glycoprotein Subunit1,Spike,S1 protein,S1...

SARS HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays key parts in the induction of neutralizing-antibody and T-cell responses, as well as protective immunity. SARS Spike S1 Protein (hFc & Avi), Biotinylated is expressed in HEK293 mammalian cells with C-hFc-Avi tag. The predicted molecular weight is 100.6 kDa and the accession number...
TMPK-00432 SARS-COV-2 Spike S1 Protein (hFc & Avi)

Spike protein S1,S glycoprotein Subunit1,S1 protein,Spike,S1...

SARS-CoV-2 HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays key parts in the induction of neutralizing-antibody and T-cell responses, as well as protective immunity. SARS-COV-2 Spike S1 Protein (hFc & Avi) is expressed in HEK293 mammalian cells with C-hFc-Avi tag. The predicted molecular weight is 102.6 kDa and the accession number is A0A6...
TMPK-00434 SARS-COV-2 Spike RBD Protein (hFc & Avi), Biotinylated

S protein RBD,S glycoprotein RBD,Spike protein RBD

SARS-CoV-2 HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays key parts in the induction of neutralizing-antibody and T-cell responses, as well as protective immunity. SARS-COV-2 Spike RBD Protein (hFc & Avi), Biotinylated is expressed in HEK293 mammalian cells with C-hFc-Avi tag. The predicted molecular weight is 51.7 kDa and the accession ...
TMPK-00911 SARS Spike RBD Protein (His & Avi)

S protein RBD,Spike protein RBD,S glycoprotein RBD

SARS HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays key parts in the induction of neutralizing-antibody and T-cell responses, as well as protective immunity. SARS Spike RBD Protein (His & Avi) is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weight is 27.9 kDa and the accession number is P59594.
TMPK-00439 SARS-COV-2 Spike RBD Protein (His & Avi), Biotinylated

S protein RBD,S glycoprotein RBD,Spike protein RBD

SARS-CoV-2 HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays key parts in the induction of neutralizing-antibody and T-cell responses, as well as protective immunity. SARS-COV-2 Spike RBD Protein (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weight is 27 kDa and the accession nu...
TMPK-00912 SARS Spike RBD Protein (His & Avi), Biotinylated

S glycoprotein RBD,S protein RBD,Spike protein RBD

SARS HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays key parts in the induction of neutralizing-antibody and T-cell responses, as well as protective immunity. SARS Spike RBD Protein (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weight is 27.9 kDa and the accession number...
TMPK-00442 SARS-COV-2 (Omicron B.1.1.529) Spike S Trimer Protein (His & Avi), Biotinylated

S glycoprotein,COVID-19,S protein,Spike glycoprotein

SARS-CoV-2 HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays key parts in the induction of neutralizing-antibody and T-cell responses, as well as protective immunity. SARS-COV-2 (Omicron B.1.1.529) Spike S Trimer Protein (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weight is 13...
TMPK-00441 SARS-COV-2 Spike S Trimer Protein (His & Avi), Biotinylated

Spike glycoprotein,S glycoprotein,S protein,COVID-19

SARS-CoV-2 HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays key parts in the induction of neutralizing-antibody and T-cell responses, as well as protective immunity. SARS-COV-2 Spike S Trimer Protein (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weight is 136.6 kDa and the acce...
TMPK-00443 SARS-COV-2 (Omicron B.1.1.529) Spike S1 Protein (His & Avi), Biotinylated

Spike,S1 protein,S glycoprotein Subunit1,S1 protein,Spike pr...

SARS-CoV-2 HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays key parts in the induction of neutralizing-antibody and T-cell responses, as well as protective immunity. SARS-COV-2 (Omicron B.1.1.529) Spike S1 Protein (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weight is 77.94 kD...
TMPK-00444 SARS-COV-2 Spike S1 NTD Protein (His & Flag)

S1 protein NTD,Spike glycoprotein Subunit1 NTD,S glycoprotei...

SARS-CoV-2 HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays key parts in the induction of neutralizing-antibody and T-cell responses, as well as protective immunity. SARS-COV-2 Spike S1 NTD Protein (His & Flag) is expressed in HEK293 mammalian cells with C-His-Flag tag. The predicted molecular weight is 35 kDa and the accession number is A...
TMPK-00910 SARS Spike S1 Protein (His & Avi)

S1 protein,S glycoprotein Subunit1,Spike protein S1,Spike,S1...

SARS HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays key parts in the induction of neutralizing-antibody and T-cell responses, as well as protective immunity. SARS Spike S1 Protein (His & Avi) is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weight is 75.9 kDa and the accession number is P59594.
TMPK-00437 SARS-COV-2 Spike RBD Protein (His & Avi)

S glycoprotein RBD,Spike protein RBD,S protein RBD

SARS-CoV-2 HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays key parts in the induction of neutralizing-antibody and T-cell responses, as well as protective immunity. SARS-COV-2 Spike RBD Protein (His & Avi) is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weight is 27 kDa and the accession number is A0A6G7...
TMPK-00433 SARS-COV-2 Spike S1 Protein (hFc & Avi), Biotinylated

S1 protein,Spike,S1 protein,Spike protein S1,S glycoprotein ...

SARS-CoV-2 HEK293 Cells
The spike protein (S) of coronavirus (CoV) attaches the virus to its cellular receptor, angiotensin-converting enzyme 2 (ACE2). A defined receptor-binding domain (RBD) on S mediates this interaction.The S protein plays key parts in the induction of neutralizing-antibody and T-cell responses, as well as protective immunity. SARS-COV-2 Spike S1 Protein (hFc & Avi), Biotinylated is expressed in HEK293 mammalian cells with C-hFc-Avi tag. The predicted molecular weight is 102.6 kDa and the accession ...
TMPY-06885 SARS-CoV-2 XBB.1.16 (Omicron) Spike S1+S2 trimer Protein (ECD, His)

The spike (S) glycoprotein of coronaviruses contains protrusions that will only bind to certain receptors on the host cell. Known receptors bind S1 are ACE2, angiotensin-converting enzyme 2; DPP4, dipeptidyl peptidase-4; APN, aminopeptidase N; CEACAM, carcinoembryonic antigen-related cell adhesion molecule 1; Sia, sialic acid; O-ac Sia, O-acetylated sialic acid. The spike is essential for both host specificity and viral infectivity. The term 'peplomer' is typically used to refer to a grouping of...
TMPH-02274 JAK2 Protein, Human, Recombinant (His)

JAK2,Janus kinase 2,Tyrosine-protein kinase JAK2

Human E. coli
Non-receptor tyrosine kinase involved in various processes such as cell growth, development, differentiation or histone modifications. Mediates essential signaling events in both innate and adaptive immunity. In the cytoplasm, plays a pivotal role in signal transduction via its association with type I receptors such as growth hormone (GHR), prolactin (PRLR), leptin (LEPR), erythropoietin (EPOR), thrombopoietin (THPO); or type II receptors including IFN-alpha, IFN-beta, IFN-gamma and multiple int...

重组蛋白

AGTR2 Protein, Human, Recombinant (His & SUMO)
Cat.No: TMPH-02268
Species: Human
Expression System: E. coli
AGTRAP Protein, Human, Recombinant (His & Myc & SUMO)
Cat.No: TMPH-02267
Species: Human
Expression System: E. coli
NLRP3 Protein, Human, Recombinant (His)
Cat.No: TMPH-01739
Species: Human
Expression System: E. coli
MMP-12 Protein, Human, Recombinant (catalytic domain)
Cat.No: TMPY-02869
Species: Human
Expression System: E. coli
SARS-COV-2 Spike S Trimer Protein (His & Avi)
Cat.No: TMPK-00438
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS Spike S1 Protein (hFc & Avi)
Cat.No: TMPK-00908
Species: SARS
Expression System: HEK293 Cells
SARS Spike S1 Protein (His & Avi), Biotinylated
Cat.No: TMPK-00913
Species: SARS
Expression System: HEK293 Cells
SARS-COV-2 Spike S1 Protein (His & Avi), Biotinylated
Cat.No: TMPK-00440
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS Spike S1 Protein (hFc & Avi), Biotinylated
Cat.No: TMPK-00909
Species: SARS
Expression System: HEK293 Cells
SARS-COV-2 Spike S1 Protein (hFc & Avi)
Cat.No: TMPK-00432
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-COV-2 Spike RBD Protein (hFc & Avi), Biotinylated
Cat.No: TMPK-00434
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS Spike RBD Protein (His & Avi)
Cat.No: TMPK-00911
Species: SARS
Expression System: HEK293 Cells
SARS-COV-2 Spike RBD Protein (His & Avi), Biotinylated
Cat.No: TMPK-00439
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS Spike RBD Protein (His & Avi), Biotinylated
Cat.No: TMPK-00912
Species: SARS
Expression System: HEK293 Cells
SARS-COV-2 (Omicron B.1.1.529) Spike S Trimer Protein (His & Avi), Biotinylated
Cat.No: TMPK-00442
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-COV-2 Spike S Trimer Protein (His & Avi), Biotinylated
Cat.No: TMPK-00441
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-COV-2 (Omicron B.1.1.529) Spike S1 Protein (His & Avi), Biotinylated
Cat.No: TMPK-00443
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-COV-2 Spike S1 NTD Protein (His & Flag)
Cat.No: TMPK-00444
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS Spike S1 Protein (His & Avi)
Cat.No: TMPK-00910
Species: SARS
Expression System: HEK293 Cells
SARS-COV-2 Spike RBD Protein (His & Avi)
Cat.No: TMPK-00437
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-COV-2 Spike S1 Protein (hFc & Avi), Biotinylated
Cat.No: TMPK-00433
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 XBB.1.16 (Omicron) Spike S1+S2 trimer Protein (ECD, His)
Cat.No: TMPY-06885
Species:
Expression System:
JAK2 Protein, Human, Recombinant (His)
Cat.No: TMPH-02274
Species: Human
Expression System: E. coli
Cat. No. Product Name Target Signaling Pathways
T11870 Losartan D4

氯沙坦 D4,DuP-753 D4

Others Others
Losartan D4, the deuterium-labeled version of Losartan, functions as an angiotensin II receptor antagonist. It inhibits the interaction between angiotensin II and AT1 receptors by competing for binding, achieving an IC50 value of 20 nM.
T11675 Irbesartan-d4

厄贝沙坦 D4,SR-47436 D4,BMS-186295 D4

Others Others
Irbesartan D4, a deuterium-labeled variant of Irbesartan, is a highly potent and specific antagonist of the angiotensin II type 1 (AT1) receptor.
T11869 Losartan (D4 Carboxylic Acid)

E-3174 D4,氯沙坦羧酸 D4,EXP-3174 D4

Others Others
Losartan D4 Carboxylic Acid is the deuterium labeled Losartan, which is an angiotensin II receptor antagonist.
TMIJ-0185 Telmisartan-13C-d3

Telmisartan-13C-d3 是 Telmisartan 的 13C 和氘代化合物。Telmisartan 的 CAS 号为 144701-48-4。Telmisartan 是一种血管紧张素II 1型受体拮抗剂,能够抑制其活性,IC50值为 9.2 nM。
T10440 Azilsartan-d5

TAK-536 D5

Others Others
Azilsartan (TAK-536) D5 is the deuterium-labeled Azilsartan. Azilsartan is a specific antagonist of the angiotensin II type 1 receptor.
T12300 Olmesartan-d4

RNH-6270 D4,奥美沙坦 D4

Others Others
Olmesartan D4 is the deuterium labeled Olmesartan. Olmesartan is an antagonist of angiotensin II receptor (AT1R) used to treat high blood pressure.
T10670 Candesartan-d4

坎地沙坦 D4,CV-11974 D4

Others Others
Candesartan D4 is the deuterium labeled Candesartan. Candesartan is an antagonist of angiotensin II receptor.
T13282 Valsartan-d9

CGP-48933 D9,缬沙坦 D9

Others Others
Valsartan D9 is a deuterium-labeled valsartan. Valsartan is an antagonist of the angiotensin II receptor and for the treatment of high blood pressure and heart failure.
TMIJ-0131 rac-Valsartan-d9

rac-Valsartan-d9 是 rac-Valsartan 的氘代化合物。rac-Valsartan 的 CAS 号为 137862-53-4。Valsarta 是一种血管紧张素 II 受体拮抗剂,有用于高血压和心力衰竭的研究潜力。
TMID-0241 Olmesartan-d6 Acid

Olmesartan-d6 Acid 是 Olmesartan Acid 的氘代化合物。Olmesartan Acid 的 CAS 号为 144689-24-7。Olmesartan 是一种血管紧张素II受体 (AT1R) 拮抗剂,常用于研究高血压。
TMIJ-0317 Nadolol-d9 (Mixture of Diastereomers)

Nadolol-d9 (Mixture of Diastereomers) 是 Nadolol 的氘代化合物。Nadolol 的 CAS 号为 42200-33-9。Nadolol 是一种有机阴离子转运多肽 1A2 (OATP1A2) 的底物,是一种非选择性的、具有口服活性的 β-肾上腺素受体 (β-adrenergic receptors) 阻滞剂,可用于高血压,心绞痛和血管性头痛的研究。

同位素标记化合物

Losartan D4
Cat.No: T11870
Synonym: 氯沙坦 D4,DuP-753 D4
Target: Others
Irbesartan-d4
Cat.No: T11675
Synonym: 厄贝沙坦 D4,SR-47436 D4,BMS-186295 D4
Target: Others
Losartan (D4 Carboxylic Acid)
Cat.No: T11869
Synonym: E-3174 D4,氯沙坦羧酸 D4,EXP-3174 D4
Target: Others
Telmisartan-13C-d3
Cat.No: TMIJ-0185
Synonym:
Target:
Azilsartan-d5
Cat.No: T10440
Synonym: TAK-536 D5
Target: Others
Olmesartan-d4
Cat.No: T12300
Synonym: RNH-6270 D4,奥美沙坦 D4
Target: Others
Candesartan-d4
Cat.No: T10670
Synonym: 坎地沙坦 D4,CV-11974 D4
Target: Others
Valsartan-d9
Cat.No: T13282
Synonym: CGP-48933 D9,缬沙坦 D9
Target: Others
rac-Valsartan-d9
Cat.No: TMIJ-0131
Synonym:
Target:
Olmesartan-d6 Acid
Cat.No: TMID-0241
Synonym:
Target:
Nadolol-d9 (Mixture of Diastereomers)
Cat.No: TMIJ-0317
Synonym:
Target:
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