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Cat. No. Product Name Target Signaling Pathways
T3289 Amifostine

氨磷汀,Ethyol,WR2721,Gammaphos

Others; HIF/HIF Prolyl-Hydroxylase Chromatin/Epigenetic; Metabolism; Others
Amifostine (Ethyol) 是一种广谱细胞保护剂和辐射防护剂,具有清除自由基的作用。它可选择性保护正常组织免受放射线和化学疗法造成的损害。它是有效的 HIF-α1和 p53诱导剂,可降低肾脏毒性并具有抗血管生成作用。
T6381 Amifostine trihydrate

Ethyol trihydrate,WR2721,三水氨磷汀,Amifostine

Others; HIF/HIF Prolyl-Hydroxylase Chromatin/Epigenetic; Metabolism; Others
Amifostine trihydrate (WR2721) 是一种广谱细胞保护剂和辐射防护剂。它可选择性保护正常组织免受放射线和化学疗法造成的损害。它是有效的HIF-α1和p53诱导剂。它通过清除氧衍生的自由基来保护细胞免受损伤。它可降低肾脏毒性并具有抗血管生成作用。
T37538 Amifostine thiol

WR-1065

p53 Apoptosis
Amifostine thiol (WR-1065) 是放射保护剂,可保护 DNA 免受快速中子诱导的链断裂。Amifostine thiol 以剂量依赖性方式改善 (P<0.001) 6-OHDA 诱导的僵滞,通过 JNK 依赖的信号通路激活 p53。
TQ0133 Amifostine thiol dihydrochloride

WR 1065,硫代乙基氨基乙基胺盐酸盐

p53 Apoptosis
Amifostine thiol dihydrochloride (WR 1065) 可通过 JNK 依赖性信号通路激活 p53。它还可以保护正常组织免受某些抗癌药物的毒性作用。
T3289L Amifostine Hydrate

Others Others
Amifostine Hydrate is a radiation protective agent that induces splenic vasodilation and blocks autonomic ganglion.
T3289L2 Amifostine sodium

WR-2721 sodium,WR2721 sodium,WR 2721 sodium

Others Others
Amifostine sodium is a phosphorothioate proposed as a radiation-protective agent. It causes splenic vasodilation and may block autonomic ganglia.

化合物

Amifostine
Cat.No: T3289
Synonym: 氨磷汀,Ethyol,WR2721,Gammaphos
Target: Others, HIF/HIF Prolyl-Hydroxylase
Amifostine trihydrate
Cat.No: T6381
Synonym: Ethyol trihydrate,WR2721,三水氨磷汀,Amifostine
Target: Others, HIF/HIF Prolyl-Hydroxylase
Amifostine thiol
Cat.No: T37538
Synonym: WR-1065
Target: p53
Amifostine thiol dihydrochloride
Cat.No: TQ0133
Synonym: WR 1065,硫代乙基氨基乙基胺盐酸盐
Target: p53
Amifostine Hydrate
Cat.No: T3289L
Synonym:
Target: Others
Amifostine sodium
Cat.No: T3289L2
Synonym: WR-2721 sodium,WR2721 sodium,WR 2721 sodium
Target: Others
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