Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6205 |
AT7519
|
Apoptosis; GSK-3; CDK | Apoptosis; Cell Cycle/Checkpoint; PI3K/Akt/mTOR signaling; Stem Cells |
AT7519 是一种CDK 抑制剂,对 CDK1,CDK2,CDK4-CDK6 以及 CDK9 的IC50值分别为 210,47,100,13,170 和 <10 nM。 | |||
T1778 |
AT7519 Hydrochloride
AT7519 HCl,AT 7519 hydrochloride salt |
Apoptosis; GSK-3; CDK | Apoptosis; Cell Cycle/Checkpoint; PI3K/Akt/mTOR signaling; Stem Cells |
AT7519 Hydrochloride (AT7519 HCl) 是一种多CDK 抑制剂,对 CDK1、CDK2、CDK4-CDK6 以及 CDK9 的IC50值分别为 210、47、100、13、170 和 <10 nM。 | |||
T22590 |
AT7519 TFA
AT7519 trifluoroacetate |
Others | Others |
AT7519 is a kinase inhibitor (IC50: 0.19, 0.044, 0.51, 0.067, 0.66 and 0.018 μM for CDK1/cyclinB, CDK2/CyclinA, CDK2/Cyclin E, CDk4/CyclinD1, CDK6/Cyclin D3, CDk5/p35). | |||
T68411 |
AT-7519M
|
Others | Others |
AT-7519M is a small molecule inhibitor of cyclin-dependent kinases 1, 2, 4, 5, and 9 with in vitro activity against lymphoid malignancies. | |||
T83652 |
Cyclin K degrader 1
|
Others | Others |
Cyclin K degrader 1 是 Cyclin K 降解剂。Cyclin K degrader 1是由AT-7519转变而来的降解剂,对 Cyclin K 降解活性较弱,但不会导致降解亲和力持续下降。 |