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Targets Recommended: Dopamine Receptor

39

抑制剂 & 化合物

13

天然产物

1

TargetMol 试剂盒

1

重组蛋白

4

同位素标记化合物

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Cat. No. Product Name Form Specificity Of Inhibition
C0052 Penicillin-Streptomycin-Amphotericin B Solution (100×), Sterile

青霉素-链霉素-两性霉素B三抗溶液(100×),灭菌

Solution in bottle

TargetMol 试剂盒

青霉素-链霉素-两性霉素B三抗溶液(100×),灭菌
Cat.No: C0052
Cat. No. Product Name Target Signaling Pathways
T24055 FAUC 213

FAUC213,FAUC-213

Dopamine Receptor GPCR/G Protein; Neuroscience
FAUC 213 是一种具有口服活性的‘、高度选择性的、可透过血脑屏障的多巴胺 D4受体完全拮抗剂,对 hD4.4的 Ki=2.2 nM。它对 D2和 D3受体的活性较低,对于 hD2、hD3的 Ki 分别为 3.4 μM、5.3 μM。它表现出非典型的抗精神病活性。
T1550 Thiamphenicol

甲砜霉素,Dextrosulphenidol,Thiophenicol

Antibacterial; Antibiotic Microbiology/Virology
Thiamphenicol (Dextrosulphenidol) 是 Chloramphenicol 的甲基磺酰基衍生物,是一种广谱抗菌类抗生素。它与 50S 核糖体亚基结合,抑制蛋白质合成并具有抑菌作用 ,特别针对革兰氏阴性,革兰氏阳性需氧和厌氧菌。
T7465 4-Methylbenzylidene camphor

Enzacamene,4-甲基苄亚基樟脑,3-(4-甲基苯亚甲基)樟脑,4-MBC

AChE Neuroscience
4-Methylbenzylidene camphor 是有机的樟脑衍生物,应用于化妆品行业,具有保护皮肤抵抗紫外线(特别是紫外线B 辐射)的能力。
T20525 Chloramphenicol palmitate

Antibacterial; Antibiotic Microbiology/Virology
Chloramphenicol palmitate 是一种广谱抗生素,对革兰氏阳性和革兰氏阴性细菌具有活性。 Chloramphenicol palmitate 可用于在含有氯霉素抗性基因的转化细胞中作为细菌选择剂的研究。
T10311 Amphotericin X1

两性霉素 X1

Others Others
Amphotericin X1 is a derivative of Amphotericin B with good antifungal activity. Amphotericin X1 inhibits Candida albicans 33/079, Cryptococcus neoformans 451, C.parapsilosis 937A, Aspergillus niger 57A and A.fumigatus (MICs: 1 μg/mL, 1 μg/mL, 8 μg/mL, 2
T74079 m-Chloramphenicol

Others Others
m-Chloramphenicol (m-threo-Chloramphenicol) 是 Chloramphenicol 的一种杂质。Chloramphenicol 是一种广谱抗生素,是细菌蛋白质生物合成的有效抑制剂。
T25239 Chloramphenicol stearate

Eusynthomycin,Chloramphenicol monostearate,Madomicetina

Others Others
Chloramphenicol stearate is an antibiotic useful for the therapy of numbers of bacterial infections. This includes an eye ointment to treat conjunctivitis.
TF0050 Amphipol A8-35

Others Others
Amphipol A8-35 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 TF0050,CAS号为 326856-53-5。
T35651 Bromamphenicol

Others Others
Bromamphenicol is a dibrominated derivative of the antibiotic chloramphenicol. It inhibits rat liver mitochondrial and E. coli protein synthesis by 90.6 and 98.8%, respectively, when used at a concentration of 93 μM, and inhibits DNA synthesis in human lymphoblastoid cells by 83% at 1 mM. Bromamphenicol can also bind to the major adhesin subunit DraE from E. coli.
T66682 (1R,3S)-(+)-Camphoric acid

Others Others
(1R,3S)-(+)-Camphoric acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66682,CAS号为 124-83-4。
T65136 Camphorquinone

Others Others
Camphorquinone 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65136,CAS号为 10373-78-1。
T73891 Amphotericin A

Others Others
Amphotericin A 是一种有效的抗真菌抗生素。
T74061 Amphotericin B methyl ester hydrochloride

Others Others
Amphotericin B methyl ester hydrochloride 是多烯类抗生素 Amphotericin B (A634250) 的甲酯衍生物。Amphotericin B methyl ester hydrochloride 是胆固醇结合物,具有显著的抗真菌活性。Amphotericin B methyl ester hydrochloride 干扰HIV-1颗粒的产生,抑制HIV-1的复制。
T72093 Thiamphenicol glycinate hydrochloride

甲砜霉素甘氨酸酯盐酸盐

Others Others
Thiamphenicol glycinate hydrochloride 是一种广谱抗菌剂,可用于呼吸道感染的研究。
T64105 Voriconazole camphorsulfonate

Others Others
Voriconazole (UK-109496) camphorsulfonate 是一种二代广谱的三唑类抗真菌 (antifungal) 化合物,对真菌麦角甾醇的生物合成表现出抑制作用。Voriconazole camphorsulfonate 能够抑制由真菌细胞色素 P450 酶介导的 14-α-羊毛甾醇去甲基化作用,表现出抗真菌效果。
T34895 Tocamphyl

Tocanfil,Biliphorin,Gallogen

Others Others
Tocamphyl is a cholagogic agent that stimulates pancreatic exocrine and bile flow when administered in the duodenum.
T30475 Bismuth camphocarbonate

Bi-Valeas,Solmuth,Cardyl,Rectobismutina,Angimuth

Others Others
Bismuth camphocarbonate is used for herpes zoster.
T20401 (-)-Isopinocampheol

l-Isopinocampheol

Others Others
(-)-Isopinocampheol is a monoterpene and a component of several plant essential oils. It showed dual viricidal activity against herpes simplex virus 1.
T66968 (1S)-(+)-Camphor-10-sulphonic acid

Others Others
(1S)-(+)-Camphor-10-sulphonic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66968,CAS号为 3144-16-9。
T65673 (+)-10,2-Camphorsultam

Others Others
(+)-10,2-Camphorsultam 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65673,CAS号为 108448-77-7。
T71810 Thiamphenicol palmitate

Others Others
Thiamphenicol palmitate is a Prodrug of Thiamphenicol, inhibiting the 50S subunit of the bacterial ribosome and protein translation.
T10309 Amphethinile

Amphetinile,CRC 82-07

Others Others
Amphethinile is an anti-tubulin agent. The Ka of Amphethinile with tubulin is 1.3 μM.
T71443 Amphidinolide D

Others Others
Amphidinolide D is a powerful activator of actomyosin ATPase enhances skeletal muscle contraction.
T30037 Amphidinolide C

Others Others
Amphidinolide C is a potent cytotoxic 25-membered macrolide from marine dinoflagellate Amphidinium sp.
T30036 Amphenidone

Others Others
Amphenidone is a Tranquilizer.
T30038 Amphidinolide F

Others Others
Amphidinolide F is a new cytotoxic macrolide
T25083 Amphotalide

RP 6171,RP-6171,RP6171,Schistomide

Others Others
Amphotalide is an anthelminthic agent.
T24401 L-erythro-Chloramphenicol

L(+)-erythro-Chloramphenicol

Others Others
L-erythro-Chloramphenicol functions as a potent inhibitor of electron transport.
T131515 Picroside II (Amphicoside)

Others Others
Picroside II (Amphicoside) 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T131515。
T30041 Amphoglucamine

Others Others
Amphoglucamine is used in the combined chemotherapy of viral diseases.
T65131 (+/-)-10-Camphorsulfonic Acid

Others Others
(+/-)-10-Camphorsulfonic Acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65131,CAS号为 5872-08-2。
T30040 Amphocil

Amphotericin B cholesteryl sulfate

Others Others
Amphocil is used to treat patients with invasive fungal infection.
T10310 Amphotericin B methyl ester

Others Others
Amphotericin B methyl ester is the derivative of the antibiotic Amphotericin B. Amphotericin B methyl ester is the cholesterol-binding compound that possesses significant antifungal activity. It disrupts HIV-1 particle production and potently inhibits HIV
T66944 (1R)-(-)-10-Camphorsulfonic acid

Others Others
(1R)-(-)-10-Camphorsulfonic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66944,CAS号为 35963-20-3。
T30039 Amphimedine

Others Others
Amphimedine is a Pyridoacridine Marine Alkaloid.
T20818 Propetamphos

Deadmag,Safrotin S 200

Others Others
Propetamphos, an organophosphate pesticide, can effectively control cockroaches, flies, mosquitoes, and other pests. It is also effective for cattle lice.
T65662 (1S)-(+)-(10-Camphorsulfonyl)oxaziridine

Others Others
(1S)-(+)-(10-Camphorsulfonyl)oxaziridine 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65662,CAS号为 104322-63-6。
T84892 D-Amphetamine hemisulfate

Dextroamphetamine

Others Others
D-Amphetamine sulfate, a central nervous system (CNS) stimulant, acts on monoamine transporters to increase noradrenaline, dopamine, and serotonin levels in synapses. Additionally, it serves as an antagonist to the α7 nicotinic acetylcholine receptor (nAChR).
T124427 Camphans?ure (+)-

Others Others
Camphans?ure (+)- 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124427,CAS号为 67111-66-4。

化合物

FAUC 213
Cat.No: T24055
Synonym: FAUC213,FAUC-213
Target: Dopamine Receptor
Thiamphenicol
Cat.No: T1550
Synonym: 甲砜霉素,Dextrosulphenidol,Thiophenicol
Target: Antibacterial, Antibiotic
4-Methylbenzylidene camphor
Cat.No: T7465
Synonym: Enzacamene,4-甲基苄亚基樟脑,3-(4-甲基苯亚甲基)樟脑,4-MBC
Target: AChE
Chloramphenicol palmitate
Cat.No: T20525
Synonym:
Target: Antibacterial, Antibiotic
Amphotericin X1
Cat.No: T10311
Synonym: 两性霉素 X1
Target: Others
m-Chloramphenicol
Cat.No: T74079
Synonym:
Target: Others
Chloramphenicol stearate
Cat.No: T25239
Synonym: Eusynthomycin,Chloramphenicol monostearate,Madomicetina
Target: Others
Amphipol A8-35
Cat.No: TF0050
Synonym:
Target: Others
Bromamphenicol
Cat.No: T35651
Synonym:
Target: Others
(1R,3S)-(+)-Camphoric acid
Cat.No: T66682
Synonym:
Target: Others
Camphorquinone
Cat.No: T65136
Synonym:
Target: Others
Amphotericin A
Cat.No: T73891
Synonym:
Target: Others
Amphotericin B methyl ester hydrochloride
Cat.No: T74061
Synonym:
Target: Others
Thiamphenicol glycinate hydrochloride
Cat.No: T72093
Synonym: 甲砜霉素甘氨酸酯盐酸盐
Target: Others
Voriconazole camphorsulfonate
Cat.No: T64105
Synonym:
Target: Others
Tocamphyl
Cat.No: T34895
Synonym: Tocanfil,Biliphorin,Gallogen
Target: Others
Bismuth camphocarbonate
Cat.No: T30475
Synonym: Bi-Valeas,Solmuth,Cardyl,Rectobismutina,Angimuth
Target: Others
(-)-Isopinocampheol
Cat.No: T20401
Synonym: l-Isopinocampheol
Target: Others
(1S)-(+)-Camphor-10-sulphonic acid
Cat.No: T66968
Synonym:
Target: Others
(+)-10,2-Camphorsultam
Cat.No: T65673
Synonym:
Target: Others
Thiamphenicol palmitate
Cat.No: T71810
Synonym:
Target: Others
Amphethinile
Cat.No: T10309
Synonym: Amphetinile,CRC 82-07
Target: Others
Amphidinolide D
Cat.No: T71443
Synonym:
Target: Others
Amphidinolide C
Cat.No: T30037
Synonym:
Target: Others
Amphenidone
Cat.No: T30036
Synonym:
Target: Others
Amphidinolide F
Cat.No: T30038
Synonym:
Target: Others
Amphotalide
Cat.No: T25083
Synonym: RP 6171,RP-6171,RP6171,Schistomide
Target: Others
L-erythro-Chloramphenicol
Cat.No: T24401
Synonym: L(+)-erythro-Chloramphenicol
Target: Others
Picroside II (Amphicoside)
Cat.No: T131515
Synonym:
Target: Others
Amphoglucamine
Cat.No: T30041
Synonym:
Target: Others
(+/-)-10-Camphorsulfonic Acid
Cat.No: T65131
Synonym:
Target: Others
Amphocil
Cat.No: T30040
Synonym: Amphotericin B cholesteryl sulfate
Target: Others
Amphotericin B methyl ester
Cat.No: T10310
Synonym:
Target: Others
(1R)-(-)-10-Camphorsulfonic acid
Cat.No: T66944
Synonym:
Target: Others
Amphimedine
Cat.No: T30039
Synonym:
Target: Others
Propetamphos
Cat.No: T20818
Synonym: Deadmag,Safrotin S 200
Target: Others
(1S)-(+)-(10-Camphorsulfonyl)oxaziridine
Cat.No: T65662
Synonym:
Target: Others
D-Amphetamine hemisulfate
Cat.No: T84892
Synonym: Dextroamphetamine
Target: Others
Camphans?ure (+)-
Cat.No: T124427
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T8258 Chloramphenicol succinate sodium

Chloramphenicol sodium succinate,琥珀酸钠氯霉素,氯霉素琥珀酸钠

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Chloramphenicol succinate sodium 是 Chloramphenicol 的前药,具有血液学毒性。它是琥珀酸脱氢酶的竞争底物和抑制剂。
TMS2262 (-)-CAMPHOR

L-Camphor,左旋樟脑

Others Others
(-)-CAMPHOR (L-Camphor) 是樟脑的手性中间体,在食品中用作风味添加剂和甜味剂。
T7959 (+)-ISOPINOCAMPHEOL

Others Others
(+)-ISOPINOCAMPHEOL 是一种天然产物。
T20191 (-)-Camphoric acid

(-)-樟脑酸,L-Camphoric acid,Camphoric acid, (-)-

GluR Neuroscience
(-)-Camphoric acid (L-Camphoric acid) 是一种活性较低的樟脑酸对映异构体,樟脑酸可诱导 GluR 表达。
T1205 Chloramphenicol

Chlornitromycin,Levomycetin,Chloromycetin,氯霉素

ribosome; HIF/HIF Prolyl-Hydroxylase; Antibacterial; Antibiotic Chromatin/Epigenetic; Metabolism; Microbiology/Virology
Chloramphenicol (Chloromycetin) 是一种广谱抗生素,有效抑制细菌蛋白质生物合成。它主要作用于细菌 70S 核糖体的 50S 亚基,对肽基转移酶有活性,抑制肽键的形成。
T1067 Amphotericin B

NSC 527017,两性霉素B

Antibiotic; Antifungal Microbiology/Virology
Amphotericin B (NSC-527017) 是一种多烯类抗真菌剂,对许多真菌物种具有广谱活性。Amphotericin B 不可逆地结合麦角甾醇,破坏细胞膜完整性,从而起到抗真菌活性。
T0882 (+)-Camphor

D-(+)-Camphor,D-Camphor,(+)-樟脑,(1R)-(+)-Camphor

Antibacterial; TRP/TRPV Channel Membrane transporter/Ion channel; Microbiology/Virology
(+)-Camphor (D-Camphor) 是一种食品添加剂,在医学上可用作防腐剂。
T2952 Camphor

樟脑,(±)-Camphor,Bornan-2-one,2-Camphanone,2-Bornanone,Formosa

Influenza Virus; TRP/TRPV Channel Membrane transporter/Ion channel; Microbiology/Virology
Camphor (2-Camphanone) 是一种双环单萜酮,广泛存在于植物中,尤其是樟脑。 它是一种激动剂,局部用作皮肤止痒剂和抗感染剂,具有抗病毒,镇咳和抗癌活性。
T82002 Juniper camphor

Juniper camphor为倍半萜烯类化合物,可通过分馏樟脑蓝油的高沸点馏分进行分离。
T25240 Chloramphenicol succinate

Paraxin succinate,Kemicetine succinate,CPSA

Others Others
Chloramphenicol succinate is an inactive precursor of chloramphenicol. It is used for parenteral administration of chloramphenicol.
TN7563 Chloramphenicol Acetate

Others Others
Chloramphenicol acetate, an acetylated and inactive derivative of chloramphenicol, is synthesized in E. coli and S. aureus through the action of the inducible enzyme chloramphenicol acetyltransferase, utilizing acetyl coenzyme A (acetyl-CoA), to impart resistance to chloramphenicol. This compound exhibits no antibiotic activity against S. sonnei in turbidimetric assays.
TN4667 Norcamphor

Others Others
Norcamphor 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4667,CAS号为 497-38-1。
T38588 Amphotericin B trihydrate

Others Others
Amphotericin B trihydrate, a polyene antibiotic, is derived from Streptomyces nodosus fermenter cultures. It exhibits antileishmanial properties.

天然产物

Chloramphenicol succinate sodium
Cat.No: T8258
Synonym: Chloramphenicol sodium succinate,琥珀酸钠氯霉素,氯霉素琥珀酸钠
Target: Others, Antibacterial, Antibiotic
(-)-CAMPHOR
Cat.No: TMS2262
Synonym: L-Camphor,左旋樟脑
Target: Others
(+)-ISOPINOCAMPHEOL
Cat.No: T7959
Synonym:
Target: Others
(-)-Camphoric acid
Cat.No: T20191
Synonym: (-)-樟脑酸,L-Camphoric acid,Camphoric acid, (-)-
Target: GluR
Chloramphenicol
Cat.No: T1205
Synonym: Chlornitromycin,Levomycetin,Chloromycetin,氯霉素
Target: ribosome, HIF/HIF Prolyl-Hydroxylase, Antibacterial, Antibiotic
Amphotericin B
Cat.No: T1067
Synonym: NSC 527017,两性霉素B
Target: Antibiotic, Antifungal
(+)-Camphor
Cat.No: T0882
Synonym: D-(+)-Camphor,D-Camphor,(+)-樟脑,(1R)-(+)-Camphor
Target: Antibacterial, TRP/TRPV Channel
Camphor
Cat.No: T2952
Synonym: 樟脑,(±)-Camphor,Bornan-2-one,2-Camphanone,2-Bornanone,Formosa
Target: Influenza Virus, TRP/TRPV Channel
Juniper camphor
Cat.No: T82002
Synonym:
Target:
Chloramphenicol succinate
Cat.No: T25240
Synonym: Paraxin succinate,Kemicetine succinate,CPSA
Target: Others
Chloramphenicol Acetate
Cat.No: TN7563
Synonym:
Target: Others
Norcamphor
Cat.No: TN4667
Synonym:
Target: Others
Amphotericin B trihydrate
Cat.No: T38588
Synonym:
Target: Others
Cat. No. Product Name Species Expression System
TMPY-02300 BIN1 Protein, Human, Recombinant (His)

AMPHL,bridging integrator 1,AMPH2,SH3P9

Human E. coli
Amphiphysin 2, also named bridging integrator-1 (BIN1) or SH3P9, Amphiphysin2/BIN1 is a crescent-shaped N-BAR protein playing a key role in forming deeply invaginated tubes in muscle T-tubules, has been recently implicated in rare and common diseases affecting different tissues and physiological functions. BIN1 downregulation is linked to cancer progression and also correlates with ventricular cardiomyopathy and arrhythmia preceding heart failure. Increased BIN1 expression is linked to increased...

重组蛋白

BIN1 Protein, Human, Recombinant (His)
Cat.No: TMPY-02300
Species: Human
Expression System: E. coli
Cat. No. Product Name Target Signaling Pathways
TMIJ-0011 Chloramphenicol-d5

Chloramphenicol-d5 是 Chloramphenicol 的氘代化合物。Chloramphenicol 的 CAS 号为 56-75-7。Chloramphenicol 是一种广谱抗生素,有效抑制细菌蛋白质生物合成。它主要作用于细菌 70S 核糖体的 50S 亚基,对肽基转移酶有活性,抑制肽键的形成。
TMIJ-0034 ent-Thiamphenicol-d3

ent-Thiamphenicol-d3 是 ent-Thiamphenicol 的氘代化合物。ent-Thiamphenicol 的 CAS 号为 19934-71-5。ent-Thiamphenicol 是抗微生物化合物 Thiamphenicol 的对映体类似物。
TMIJ-0022 Thiamphenicol-Methyl-d3

Thiamphenicol-Methyl-d3 是 Thiamphenicol 的氘代化合物。Thiamphenicol 的 CAS 号为 15318-45-3。Thiamphenicol是 Chloramphenicol 的甲基磺酰基衍生物,是一种广谱抗菌类抗生素。它与 50S 核糖体亚基结合,抑制蛋白质合成并具有抑菌作用 ,特别针对革兰氏阴性,革兰氏阳性需氧和厌氧菌。
TMIJ-0075 Amphotericin-d3

Amphotericin-d3 是 Amphotericin 的氘代化合物。Amphotericin 的 CAS 号为 1397-89-3。Amphotericin B是一种抗真菌剂,对许多真菌物种具有广谱活性。

同位素标记化合物

Chloramphenicol-d5
Cat.No: TMIJ-0011
Synonym:
Target:
ent-Thiamphenicol-d3
Cat.No: TMIJ-0034
Synonym:
Target:
Thiamphenicol-Methyl-d3
Cat.No: TMIJ-0022
Synonym:
Target:
Amphotericin-d3
Cat.No: TMIJ-0075
Synonym:
Target:
TargetMol Loading
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