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Cat. No. | Product Name | Form | Specificity Of Inhibition |
---|---|---|---|
C0052 |
Penicillin-Streptomycin-Amphotericin B Solution (100×), Sterile
青霉素-链霉素-两性霉素B三抗溶液(100×),灭菌 |
Solution in bottle |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T24055 |
FAUC 213
FAUC213,FAUC-213 |
Dopamine Receptor | GPCR/G Protein; Neuroscience |
FAUC 213 是一种具有口服活性的‘、高度选择性的、可透过血脑屏障的多巴胺 D4受体完全拮抗剂,对 hD4.4的 Ki=2.2 nM。它对 D2和 D3受体的活性较低,对于 hD2、hD3的 Ki 分别为 3.4 μM、5.3 μM。它表现出非典型的抗精神病活性。 | |||
T1550 |
Thiamphenicol
甲砜霉素,Dextrosulphenidol,Thiophenicol |
Antibacterial; Antibiotic | Microbiology/Virology |
Thiamphenicol (Dextrosulphenidol) 是 Chloramphenicol 的甲基磺酰基衍生物,是一种广谱抗菌类抗生素。它与 50S 核糖体亚基结合,抑制蛋白质合成并具有抑菌作用 ,特别针对革兰氏阴性,革兰氏阳性需氧和厌氧菌。 | |||
T7465 |
4-Methylbenzylidene camphor
Enzacamene,4-甲基苄亚基樟脑,3-(4-甲基苯亚甲基)樟脑,4-MBC |
AChE | Neuroscience |
4-Methylbenzylidene camphor 是有机的樟脑衍生物,应用于化妆品行业,具有保护皮肤抵抗紫外线(特别是紫外线B 辐射)的能力。 | |||
T20525 |
Chloramphenicol palmitate
|
Antibacterial; Antibiotic | Microbiology/Virology |
Chloramphenicol palmitate 是一种广谱抗生素,对革兰氏阳性和革兰氏阴性细菌具有活性。 Chloramphenicol palmitate 可用于在含有氯霉素抗性基因的转化细胞中作为细菌选择剂的研究。 | |||
T10311 |
Amphotericin X1
两性霉素 X1 |
Others | Others |
Amphotericin X1 is a derivative of Amphotericin B with good antifungal activity. Amphotericin X1 inhibits Candida albicans 33/079, Cryptococcus neoformans 451, C.parapsilosis 937A, Aspergillus niger 57A and A.fumigatus (MICs: 1 μg/mL, 1 μg/mL, 8 μg/mL, 2 | |||
T74079 |
m-Chloramphenicol
|
Others | Others |
m-Chloramphenicol (m-threo-Chloramphenicol) 是 Chloramphenicol 的一种杂质。Chloramphenicol 是一种广谱抗生素,是细菌蛋白质生物合成的有效抑制剂。 | |||
T25239 |
Chloramphenicol stearate
Eusynthomycin,Chloramphenicol monostearate,Madomicetina |
Others | Others |
Chloramphenicol stearate is an antibiotic useful for the therapy of numbers of bacterial infections. This includes an eye ointment to treat conjunctivitis. | |||
TF0050 |
Amphipol A8-35
|
Others | Others |
Amphipol A8-35 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 TF0050,CAS号为 326856-53-5。 | |||
T35651 |
Bromamphenicol
|
Others | Others |
Bromamphenicol is a dibrominated derivative of the antibiotic chloramphenicol. It inhibits rat liver mitochondrial and E. coli protein synthesis by 90.6 and 98.8%, respectively, when used at a concentration of 93 μM, and inhibits DNA synthesis in human lymphoblastoid cells by 83% at 1 mM. Bromamphenicol can also bind to the major adhesin subunit DraE from E. coli. | |||
T66682 |
(1R,3S)-(+)-Camphoric acid
|
Others | Others |
(1R,3S)-(+)-Camphoric acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66682,CAS号为 124-83-4。 | |||
T65136 |
Camphorquinone
|
Others | Others |
Camphorquinone 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65136,CAS号为 10373-78-1。 | |||
T73891 |
Amphotericin A
|
Others | Others |
Amphotericin A 是一种有效的抗真菌抗生素。 | |||
T74061 |
Amphotericin B methyl ester hydrochloride
|
Others | Others |
Amphotericin B methyl ester hydrochloride 是多烯类抗生素 Amphotericin B (A634250) 的甲酯衍生物。Amphotericin B methyl ester hydrochloride 是胆固醇结合物,具有显著的抗真菌活性。Amphotericin B methyl ester hydrochloride 干扰HIV-1颗粒的产生,抑制HIV-1的复制。 | |||
T72093 |
Thiamphenicol glycinate hydrochloride
甲砜霉素甘氨酸酯盐酸盐 |
Others | Others |
Thiamphenicol glycinate hydrochloride 是一种广谱抗菌剂,可用于呼吸道感染的研究。 | |||
T64105 |
Voriconazole camphorsulfonate
|
Others | Others |
Voriconazole (UK-109496) camphorsulfonate 是一种二代广谱的三唑类抗真菌 (antifungal) 化合物,对真菌麦角甾醇的生物合成表现出抑制作用。Voriconazole camphorsulfonate 能够抑制由真菌细胞色素 P450 酶介导的 14-α-羊毛甾醇去甲基化作用,表现出抗真菌效果。 | |||
T34895 |
Tocamphyl
Tocanfil,Biliphorin,Gallogen |
Others | Others |
Tocamphyl is a cholagogic agent that stimulates pancreatic exocrine and bile flow when administered in the duodenum. | |||
T30475 |
Bismuth camphocarbonate
Bi-Valeas,Solmuth,Cardyl,Rectobismutina,Angimuth |
Others | Others |
Bismuth camphocarbonate is used for herpes zoster. | |||
T20401 |
(-)-Isopinocampheol
l-Isopinocampheol |
Others | Others |
(-)-Isopinocampheol is a monoterpene and a component of several plant essential oils. It showed dual viricidal activity against herpes simplex virus 1. | |||
T66968 |
(1S)-(+)-Camphor-10-sulphonic acid
|
Others | Others |
(1S)-(+)-Camphor-10-sulphonic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66968,CAS号为 3144-16-9。 | |||
T65673 |
(+)-10,2-Camphorsultam
|
Others | Others |
(+)-10,2-Camphorsultam 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65673,CAS号为 108448-77-7。 | |||
T71810 |
Thiamphenicol palmitate
|
Others | Others |
Thiamphenicol palmitate is a Prodrug of Thiamphenicol, inhibiting the 50S subunit of the bacterial ribosome and protein translation. | |||
T10309 |
Amphethinile
Amphetinile,CRC 82-07 |
Others | Others |
Amphethinile is an anti-tubulin agent. The Ka of Amphethinile with tubulin is 1.3 μM. | |||
T71443 |
Amphidinolide D
|
Others | Others |
Amphidinolide D is a powerful activator of actomyosin ATPase enhances skeletal muscle contraction. | |||
T30037 |
Amphidinolide C
|
Others | Others |
Amphidinolide C is a potent cytotoxic 25-membered macrolide from marine dinoflagellate Amphidinium sp. | |||
T30036 |
Amphenidone
|
Others | Others |
Amphenidone is a Tranquilizer. | |||
T30038 |
Amphidinolide F
|
Others | Others |
Amphidinolide F is a new cytotoxic macrolide | |||
T25083 |
Amphotalide
RP 6171,RP-6171,RP6171,Schistomide |
Others | Others |
Amphotalide is an anthelminthic agent. | |||
T24401 |
L-erythro-Chloramphenicol
L(+)-erythro-Chloramphenicol |
Others | Others |
L-erythro-Chloramphenicol functions as a potent inhibitor of electron transport. | |||
T131515 |
Picroside II (Amphicoside)
|
Others | Others |
Picroside II (Amphicoside) 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T131515。 | |||
T30041 |
Amphoglucamine
|
Others | Others |
Amphoglucamine is used in the combined chemotherapy of viral diseases. | |||
T65131 |
(+/-)-10-Camphorsulfonic Acid
|
Others | Others |
(+/-)-10-Camphorsulfonic Acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65131,CAS号为 5872-08-2。 | |||
T30040 |
Amphocil
Amphotericin B cholesteryl sulfate |
Others | Others |
Amphocil is used to treat patients with invasive fungal infection. | |||
T10310 |
Amphotericin B methyl ester
|
Others | Others |
Amphotericin B methyl ester is the derivative of the antibiotic Amphotericin B. Amphotericin B methyl ester is the cholesterol-binding compound that possesses significant antifungal activity. It disrupts HIV-1 particle production and potently inhibits HIV | |||
T66944 |
(1R)-(-)-10-Camphorsulfonic acid
|
Others | Others |
(1R)-(-)-10-Camphorsulfonic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T66944,CAS号为 35963-20-3。 | |||
T30039 |
Amphimedine
|
Others | Others |
Amphimedine is a Pyridoacridine Marine Alkaloid. | |||
T20818 |
Propetamphos
Deadmag,Safrotin S 200 |
Others | Others |
Propetamphos, an organophosphate pesticide, can effectively control cockroaches, flies, mosquitoes, and other pests. It is also effective for cattle lice. | |||
T65662 |
(1S)-(+)-(10-Camphorsulfonyl)oxaziridine
|
Others | Others |
(1S)-(+)-(10-Camphorsulfonyl)oxaziridine 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65662,CAS号为 104322-63-6。 | |||
T84892 |
D-Amphetamine hemisulfate
Dextroamphetamine |
Others | Others |
D-Amphetamine sulfate, a central nervous system (CNS) stimulant, acts on monoamine transporters to increase noradrenaline, dopamine, and serotonin levels in synapses. Additionally, it serves as an antagonist to the α7 nicotinic acetylcholine receptor (nAChR). | |||
T124427 |
Camphans?ure (+)-
|
Others | Others |
Camphans?ure (+)- 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124427,CAS号为 67111-66-4。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T8258 |
Chloramphenicol succinate sodium
Chloramphenicol sodium succinate,琥珀酸钠氯霉素,氯霉素琥珀酸钠 |
Others; Antibacterial; Antibiotic | Microbiology/Virology; Others |
Chloramphenicol succinate sodium 是 Chloramphenicol 的前药,具有血液学毒性。它是琥珀酸脱氢酶的竞争底物和抑制剂。 | |||
TMS2262 |
(-)-CAMPHOR
L-Camphor,左旋樟脑 |
Others | Others |
(-)-CAMPHOR (L-Camphor) 是樟脑的手性中间体,在食品中用作风味添加剂和甜味剂。 | |||
T7959 |
(+)-ISOPINOCAMPHEOL
|
Others | Others |
(+)-ISOPINOCAMPHEOL 是一种天然产物。 | |||
T20191 |
(-)-Camphoric acid
(-)-樟脑酸,L-Camphoric acid,Camphoric acid, (-)- |
GluR | Neuroscience |
(-)-Camphoric acid (L-Camphoric acid) 是一种活性较低的樟脑酸对映异构体,樟脑酸可诱导 GluR 表达。 | |||
T1205 |
Chloramphenicol
Chlornitromycin,Levomycetin,Chloromycetin,氯霉素 |
ribosome; HIF/HIF Prolyl-Hydroxylase; Antibacterial; Antibiotic | Chromatin/Epigenetic; Metabolism; Microbiology/Virology |
Chloramphenicol (Chloromycetin) 是一种广谱抗生素,有效抑制细菌蛋白质生物合成。它主要作用于细菌 70S 核糖体的 50S 亚基,对肽基转移酶有活性,抑制肽键的形成。 | |||
T1067 |
Amphotericin B
NSC 527017,两性霉素B |
Antibiotic; Antifungal | Microbiology/Virology |
Amphotericin B (NSC-527017) 是一种多烯类抗真菌剂,对许多真菌物种具有广谱活性。Amphotericin B 不可逆地结合麦角甾醇,破坏细胞膜完整性,从而起到抗真菌活性。 | |||
T0882 |
(+)-Camphor
D-(+)-Camphor,D-Camphor,(+)-樟脑,(1R)-(+)-Camphor |
Antibacterial; TRP/TRPV Channel | Membrane transporter/Ion channel; Microbiology/Virology |
(+)-Camphor (D-Camphor) 是一种食品添加剂,在医学上可用作防腐剂。 | |||
T2952 |
Camphor
樟脑,(±)-Camphor,Bornan-2-one,2-Camphanone,2-Bornanone,Formosa |
Influenza Virus; TRP/TRPV Channel | Membrane transporter/Ion channel; Microbiology/Virology |
Camphor (2-Camphanone) 是一种双环单萜酮,广泛存在于植物中,尤其是樟脑。 它是一种激动剂,局部用作皮肤止痒剂和抗感染剂,具有抗病毒,镇咳和抗癌活性。 | |||
T82002 |
Juniper camphor
|
||
Juniper camphor为倍半萜烯类化合物,可通过分馏樟脑蓝油的高沸点馏分进行分离。 | |||
T25240 |
Chloramphenicol succinate
Paraxin succinate,Kemicetine succinate,CPSA |
Others | Others |
Chloramphenicol succinate is an inactive precursor of chloramphenicol. It is used for parenteral administration of chloramphenicol. | |||
TN7563 |
Chloramphenicol Acetate
|
Others | Others |
Chloramphenicol acetate, an acetylated and inactive derivative of chloramphenicol, is synthesized in E. coli and S. aureus through the action of the inducible enzyme chloramphenicol acetyltransferase, utilizing acetyl coenzyme A (acetyl-CoA), to impart resistance to chloramphenicol. This compound exhibits no antibiotic activity against S. sonnei in turbidimetric assays. | |||
TN4667 |
Norcamphor
|
Others | Others |
Norcamphor 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4667,CAS号为 497-38-1。 | |||
T38588 |
Amphotericin B trihydrate
|
Others | Others |
Amphotericin B trihydrate, a polyene antibiotic, is derived from Streptomyces nodosus fermenter cultures. It exhibits antileishmanial properties. |
Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPY-02300 |
BIN1 Protein, Human, Recombinant (His)
AMPHL,bridging integrator 1,AMPH2,SH3P9 |
Human | E. coli |
Amphiphysin 2, also named bridging integrator-1 (BIN1) or SH3P9, Amphiphysin2/BIN1 is a crescent-shaped N-BAR protein playing a key role in forming deeply invaginated tubes in muscle T-tubules, has been recently implicated in rare and common diseases affecting different tissues and physiological functions. BIN1 downregulation is linked to cancer progression and also correlates with ventricular cardiomyopathy and arrhythmia preceding heart failure. Increased BIN1 expression is linked to increased... |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TMIJ-0011 |
Chloramphenicol-d5
|
||
Chloramphenicol-d5 是 Chloramphenicol 的氘代化合物。Chloramphenicol 的 CAS 号为 56-75-7。Chloramphenicol 是一种广谱抗生素,有效抑制细菌蛋白质生物合成。它主要作用于细菌 70S 核糖体的 50S 亚基,对肽基转移酶有活性,抑制肽键的形成。 | |||
TMIJ-0034 |
ent-Thiamphenicol-d3
|
||
ent-Thiamphenicol-d3 是 ent-Thiamphenicol 的氘代化合物。ent-Thiamphenicol 的 CAS 号为 19934-71-5。ent-Thiamphenicol 是抗微生物化合物 Thiamphenicol 的对映体类似物。 | |||
TMIJ-0022 |
Thiamphenicol-Methyl-d3
|
||
Thiamphenicol-Methyl-d3 是 Thiamphenicol 的氘代化合物。Thiamphenicol 的 CAS 号为 15318-45-3。Thiamphenicol是 Chloramphenicol 的甲基磺酰基衍生物,是一种广谱抗菌类抗生素。它与 50S 核糖体亚基结合,抑制蛋白质合成并具有抑菌作用 ,特别针对革兰氏阴性,革兰氏阳性需氧和厌氧菌。 | |||
TMIJ-0075 |
Amphotericin-d3
|
||
Amphotericin-d3 是 Amphotericin 的氘代化合物。Amphotericin 的 CAS 号为 1397-89-3。Amphotericin B是一种抗真菌剂,对许多真菌物种具有广谱活性。 |