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Targets Recommended: Nucleoside Antimetabolite/Analog Adrenergic Receptor

381

抑制剂 & 化合物

167

天然产物

1

化合物库

19

重组蛋白

24

同位素标记化合物

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Cat. No. Product Name
L6110 生物碱类天然产物库

500 compounds
500 种生物碱类天然产物的独特集合,可用于高通量筛选和高内涵筛选;

化合物库

生物碱类天然产物库
Cat.No: L6110
Compounds: 500
Cat. No. Product Name Target Signaling Pathways
T21371 Apraclonidine hydrochloride

Iopidine,ALO 2145,Apraclonidina,P-aminoclonidine,4-Aminoclonidine,Apraclonidine HCl,Apraclonidinum

Adrenergic Receptor GPCR/G Protein; Neuroscience
Apraclonidine hydrochloride (ALO 2145) 是一种 α2-肾上腺素能激动剂和弱的 α-1 肾上腺素能受体激动剂。 Apaclonidine hydrochloride 可降低人眼的眼内压,可用于青光眼治疗的研究。
T0378 Oxybuprocaine hydrochloride

Risedronic Acid,Oxybuprocaine HCl,奥布卡因盐酸盐

Sodium Channel Membrane transporter/Ion channel
Oxybuprocaine hydrochloride (Oxybuprocaine HCl) 是可逆的钠通道阻断剂,可防止角膜,结膜和巩膜中疼痛神经的冲动传播。Oxybuprocaine hydrochloride 专用于眼科与耳鼻喉科。
T0141L Cefalonium Dihydrate(5575-21-3 free base)

Cefalonium Dihydrate

Others Others
Cefalonium Dihydrate(5575-21-3 free base) 是第一代头孢菌素类抗生素。
T10858 COH34 analog 1

Others Others
COH34 analog 1 是一种 COH34 氧化类似物,可用于合成具有活性的化合物。
T1483 Citalopram hydrobromide

Lu 10-171,Nitalapram HBr,Bonitrile HBr,XU-62-320,Lu 10-171 HBr,氢溴酸西酞普兰,Citalopram HBr

5-HT Receptor; Serotonin Transporter; Autophagy Autophagy; GPCR/G Protein; Neuroscience
Citalopram hydrobromide (XU-62-320) 是一种选择性 5-羟色胺再摄取抑制剂,可选择性地抑制 CNS 神经元对 5-羟色胺的再摄取,从而增强中枢神经系统中的 5-羟色胺能活性,也具有抗抑郁活性。它抑制兔血小板中 5-HT 的摄取,IC50为 14 nM。
T5046 Haloxyfop

Haloxyfop Acid,(±)-Haloxyfop,吡氟氯禾灵

Others; Acetyl-CoA Carboxylase Metabolism; Others
Haloxyfop (Haloxyfop Acid) 是有效的芳氯氧苯氧丙酸除草剂,广泛应用于阔叶作物的野草。对玉米幼苗叶绿体中乙酰辅酶 A 羧化酶 (EC 6.4.1.2) 具有抑制作用,IC50为 0.5 μM,而对豌豆中该酶无影响。
T2525 Alosetron hydrochloride

Lotronex,盐酸阿洛司琼,GR 68755C,GR 68755,GR 68755X

5-HT Receptor GPCR/G Protein; Neuroscience
Alosetron hydrochloride (GR 68755) 是一种高选择性的 5-HT3 受体拮抗剂,可减轻清醒或麻醉犬直肠扩张的内脏伤害性效应,具有抗炎活性,用于肠易激综合征的研究。它阻断 5HT3 介导的豚鼠肌间和粘膜下神经元的快速去极化,IC50约为 55 nM。
T69984 Ticalopride

5-HT Receptor GPCR/G Protein; Neuroscience
Ticalopride是一种5-HT3 receptor激动剂,可用于治疗消化系统疾病、口颌疾病、耳鼻咽喉疾病,可用于研究神经性贪食症、胃食管反流和肠易激综合征。
T7105 Zinc phthalocyanine

酞菁锌,ZnPc

Others Others
Zinc phthalocyanine (ZnPc) 可用于环己烷的光氧化,广泛应用于工业 (催化剂、光导体)和生物医学(光动力疗法、PDT)。
T19999 1-Tetralol, (S)-

(S)-(+)-1,2,3,4-四氢-1-萘酚,(S)-Tetralin-1-ol,(S)-(+)-1,2,3,4-Tetrahydro-1-naphthol,(S)-1-Hydroxytetralin,J330.337C

Others Others
1-Tetralol, (S)- ((S)-1-Hydroxytetralin) 可在细胞实验中用作 AKR1C1 的底物。
T0102 Naloxone hydrochloride

盐酸纳洛酮,Naloxone HCl

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
Naloxone hydrochloride (Naloxone HCl) 是一种特异性、没有激动剂活性的opiate 拮抗剂。它是 mu、delta 和 kappa 阿片受体的竞争性拮抗剂。
T19637 Aluminum phthalocyanine chloride

Phthalocyanine Chloroaluminum,铝酞菁,Chloroaluminum Phthalocyanine

Others Others
Aluminum phthalocyanine chloride (Phthalocyanine Chloroaluminum) 是一种强烈的蓝绿色芳香大环化合物,广泛用于染色。
T0116 Balofloxacin

DNA gyrase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Balofloxacin 是一种具有口服活性的氟喹诺酮类抗生素,可通过干扰 DNA 促旋酶来抑制细菌 DNA 的合成,对革兰氏阴性,革兰氏阳性和厌氧菌具有广谱抗菌活性。它可研究呼吸道,肠道和泌尿道感染。
T27399 Galocitabine

RO 091390,RO-091390,RO091390,RO-09-1390,Neofrutulon

Others Others
Galocitabine (Neofrutulon) 是一种胸苷酸合成酶抑制剂,可能用于治疗癌症。
T6351 MGCD-265 analog

MGCD-265,Glesatinib

Apoptosis; VEGFR; c-Met/HGFR Angiogenesis; Apoptosis; Tyrosine Kinase/Adaptors
MGCD-265 analog (Glesatinib) 是一种口服生物可利用的多靶点酪氨酸激酶抑制剂,具有抗肿瘤活性,对 c-Met 和 VEGFR2 的 IC50 分别为 29 nM 和 10 nM。
T15461 Halopemide

Others; Phospholipase; Dopamine Receptor GPCR/G Protein; Metabolism; Neuroscience; Others
Halopemide 是一种有效的 PLD 抑制剂(对人 PLD1 和 PLD2 的 IC50 = 220 和 310 nM)。 Halopemid 是多巴胺受体的拮抗剂。Halopemid 可用于精神药物研究。
T12770 RR-11a analog

aza-peptide Michael acceptor, 7a

Parasite Microbiology/Virology
RR-11a analog (aza-peptide Michael acceptor, 7a) 是一种天冬酰胺酰内肽酶抑制剂,对阴道毛滴虫中的 AE1、蓖麻硬蜱中的 AE 和曼氏血吸虫中的 AE 的 IC50 分别为 4.5 nM、4.5 nM 和 31 nM。
T25487 Haloperidol decanoate

KD 16,KD-136,KD 136,Neoperidole,Haldol

Others Others
Haloperidol decanoate (KD 16) 是一种典型的抗精神病药物,用作精神分裂症和情绪障碍的维持治疗,配制成用于肌肉注射的酯。
T62606 ALOX15-IN-2

Lipoxygenase Metabolism
ALOX15-IN-2 是一种有效的 ALOX15 亚油酸加氧酶 (linoleate oxygenase) 活性抑制剂,抑制ALOX15 直系同源物亚油酸 (LA) 和花生四烯酸 (AA)进行氧化作用 , IC50 分别为 1.55 和 2.79 μM。
T6529 Halobetasol propionate

卤贝他索丙酸酯,Halobetasol Propionate,Ulobetasol propionate,BMY-30056,卤倍他索丙酸酯,CGP-14458

Phospholipase Metabolism
Halobetasol propionate (BMY-30056) 是一种在皮肤外使用的合成类固醇,具有抗炎,止痒和收缩血管的活性。
T0348 Labetalol hydrochloride

盐酸拉贝洛尔,Sch-15719W,AH-5158 hydrochloride,Labetalol HCl,柳胺苄心定

Adrenergic Receptor GPCR/G Protein; Neuroscience
Labetalol hydrochloride (Sch-15719W) 是混合的α/β肾上腺素能拮抗剂,可用于研究高血压。
T9436 BenzeneazoMalononitrile

Others Others
BenzeneazoMalononitrile 能抑制多种类型细胞的生长,包括治疗细胞;也还被证明可以抑制几种酶的活性,包括那些参与药物代谢的酶;还被证明可以抑制几种激素的活性,包括那些与血糖水平调节有关的激素。
T21355 6-Chloro-1-tetralone

6-Chloro-α-Tetralone,5-CHLORO-L-INDOMONE,6-chloro-3;5-CHLORO-1-INDOMONE,5-CHLORO-1-INDOMONE,6-chloro-3

Others Others
6-Chloro-1-tetralone (6-chloro-3;5-Chloro-1-Indomone) 是合成药物化合物的重要中间体。
T2542 Prucalopride

R-93877,普芦卡必利,普卡必利

5-HT Receptor GPCR/G Protein; Neuroscience
Prucalopride (R-93877) 是一种选择性、高亲和力的 5-HT4A/4B 受体激动剂,Ki 为2.5和 8 nM。它对 5-HT4A/4B 受体的选择性是其他 5-HT 受体亚型的 290 倍以上。
T30027 Amosulalol

Adrenergic Receptor GPCR/G Protein; Neuroscience
Amosulalol 是一种 α 和 β 肾上腺素能受体拮抗剂。
T20950 MK-8245 analog

MK-8245-analog,MK 8245 analog

Others Others
MK-8245 analog 是 MK-8245 的类似物,MK-8245 是一种肝脏靶向的硬脂酰辅酶 A 去饱和酶 (SCD) 抑制剂。它可用于治疗血脂异常和糖尿病。
T7103 idalopirdine

Lu AE58054

5-HT Receptor GPCR/G Protein; Neuroscience
Idalopirdine (Lu AE58054) 是一种选择性的5-HT6 受体拮抗剂,Ki 为 0.83 nM。
T4538 palovarotene

Ro 3300074,R 667,帕罗伐汀

Retinoid Receptor; Autophagy Autophagy; Metabolism
Palovarotene (Ro 3300074) 是核视网膜酸受体γ 的激动剂。
T7944 VPS34 inhibitor 1 (Compound 19, PIK-III analogue)

PIK-III analogue

PI3K PI3K/Akt/mTOR signaling
VPS34 inhibitor 1 (Compound 19, PIK-III analogue) (PIK-III analogue) 是一种有效的选择性 VPS34抑制剂( IC50 : 15 nM)。
T16022 Arhalofenate

JNJ 39659100,芳卤芬酯,4-氯-ALPHA-[3-(三氟甲基)苯氧基]苯乙酸 2-(乙酰基氨基)乙酯,MBX 102

PPAR DNA Damage/DNA Repair; Metabolism
Arhalofenate (JNJ 39659100) 是一种选择性的(PPAR)-γ部分激动剂,用于研究 2 型糖尿病。
T40437L Caloxin 2A1 acetate

Proton pump Membrane transporter/Ion channel
Caloxin 2A1 acetate 是细胞外质膜 Ca2+-ATPase (PMCA) 肽的抑制剂。 Caloxin 2A1 acetate 抑制 140-kDa 酸稳定酰基磷酸盐的 Ca2+ 依赖性形成。
T3355 Naloxegol oxalate

NKTR-118,NKTR-118 oxalate,AZ 13337019,AZ-13337019 oxalate

P450 Metabolism
Naloxegol oxalate (NKTR-118) 是一种外周选择性 opioid 样物质拮抗剂,用于治疗 opioid 样物质引起的便秘。
T67851 rac Desmethyl Citalopram Hydrochloride

5-HT Receptor GPCR/G Protein; Neuroscience
rac Desmethyl Citalopram Hydrochloride 是一种5-羟色胺摄取抑制剂,IC50值为0.013μM。
T22936 Idalopirdine Hydrochloride

Lu AE58054盐酸盐,Lu AE58054 Hydrochloride,Idalopirdine HCl

5-HT Receptor GPCR/G Protein; Neuroscience
Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) 是一种选择性的5-HT6 受体拮抗剂,Ki 为 0.83 nM。
T2401 Alogliptin Benzoate

苯甲酸阿格列汀,SYR 322,Alogliptin(SYR-322)benzoate

Ferroptosis; Proteasome; DPP-4 Apoptosis; Proteases/Proteasome; Ubiquitination
Alogliptin Benzoate (SYR 322) 是一种有效且特异性的 DPP-4 抑制剂 ,IC50值小于 10 nM,其选择性比 DPP-8/9 高 10,000 倍以上,可用于研究 2 型糖尿病。
T4384 Halofenozide

Others Others
Halofenozide 是一种新的昆虫生长调节剂 (IGR),具有苯甲酰肼结构,也是一种蜕皮激素 (ecdysteroid) 激动剂。可模拟天然昆虫蜕皮激素 20-羟基蜕皮激素的作用,
T60221 Tabernanthalog

TBG

5-HT Receptor GPCR/G Protein; Neuroscience
Tabernanthalog (TBG) 是一种5-HT2A 激动剂。在啮齿类动物中,Tabernanthalog 已被发现可促进结构神经可塑性并产生抗抑郁作用。
T6040 Aloxistatin

E64d,Loxistatin,阿洛司他丁,E64c ethyl ester

SARS-CoV; Cysteine Protease Microbiology/Virology; Proteases/Proteasome
Aloxistatin (E64d) 是一种不可逆的、可透过膜的溶酶体和细胞溶质半胱氨酸蛋白酶抑制剂,能够抑制完整血小板中的钙蛋白酶活性。它是一种半胱氨酸蛋白酶抑制剂,具有血小板聚集抑制活性。
T0141 Cephalonium

头孢洛宁,Cefalonium

Others Others
Cephalonium (Cefalonium) 是第一代头孢菌素类抗生素。
T7666 Valorphin TFA(144313-54-2(free base))

Valorphin TFA(144313-54-2(free bas))

Others Others
Valorphin TFA(144313-54-2(free base)) 是具有 opioid 类镇痛活性的二氢戊酸的半合成衍生物。
TP1215L Abaloparatide acetate(247062-33-5 free base)

Others Others
Abaloparatide acetate(247062-33-5 free base) 是一种甲状旁腺激素受体 1 PTHR1 类似物,是 PTHR1 信号通路的有效和选择性激活剂。
T35326 Labetalone hydrochloride

Labetalone hydrochloride,Benzoic amide

Others; Adrenergic Receptor GPCR/G Protein; Neuroscience; Others
Labetalone hydrochloride 是一种口服有效的肾上腺素能受体阻断药物,对 α 和 β 受体部位都有竞争性拮抗作用。
T0954 Halothane

Narcotane,氟烷,Anestan

Potassium Channel; Chloride channel; GABA Receptor; NMDAR Membrane transporter/Ion channel; Neuroscience
Halothane (Anestan) 可以减弱内皮依赖性舒张作用。
T0025 Haloperidol

Aloperidin,氟哌啶醇,Serenace,Haldol

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
Haloperidol (Serenace) 是一种安定药,是一种dopamine D2 receptor 拮抗剂。
T6921 ONO-4059 analog

ONO-4059 analogue,ONO-WG-307,GS-4059 analog

Apoptosis; BTK Angiogenesis; Apoptosis; Tyrosine Kinase/Adaptors
ONO-4059 analog (ONO-WG-307) 是 ONO-4059 的类似物,ONO-4059 是一种高效、选择性的口服 BTK 抑制剂,IC50 为 23.9 nM。
T2058 Palosuran

ACT-058362

GPR Endocrinology/Hormones; GPCR/G Protein
Palosuran (ACT-058362) 是人类 UT 受体的新型强效特异性拮抗剂,对表达人重组受体的 CHO 细胞膜的IC50值为 3.6 nM。它可改善糖尿病大鼠的胰腺和肾脏功能。
T11265 Faropenem daloxate

法罗培南酯,Faropenem medoxil

Antibacterial; Antibiotic Microbiology/Virology
Faropenem daloxate (Faropenem medoxil) 是β-内酰胺类口服抗生素。
T2518 ARRY-380 (analog )

HER2-Inhibitor-1,ARRY380,ARRY-380 analog

EGFR; HER Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
ARRY-380 analog (HER2-Inhibitor-1) 是EGFR (ErbB1)的抑制剂。
T2480 Apabetalone

RVX-208,RVX000222,阿帕他隆

Epigenetic Reader Domain; HIV Protease Chromatin/Epigenetic; Microbiology/Virology; Proteases/Proteasome
Apabetalone (RVX000222) 是一种 BET 溴结构域抑制剂,用于研究治疗糖尿病、动脉粥样硬化和冠状动脉疾病。
T5839 Phosalone

Parasite Microbiology/Virology
Phosalone 是一种有机磷酸盐化学品,通常用作杀虫剂和杀螨剂。

化合物

Apraclonidine hydrochloride
Cat.No: T21371
Synonym: Iopidine,ALO 2145,Apraclonidina,P-aminoclonidine,4-Aminoclonidine,Apraclonidine HCl,Apraclonidinum
Target: Adrenergic Receptor
Oxybuprocaine hydrochloride
Cat.No: T0378
Synonym: Risedronic Acid,Oxybuprocaine HCl,奥布卡因盐酸盐
Target: Sodium Channel
Cefalonium Dihydrate(5575-21-3 free base)
Cat.No: T0141L
Synonym: Cefalonium Dihydrate
Target: Others
COH34 analog 1
Cat.No: T10858
Synonym:
Target: Others
Citalopram hydrobromide
Cat.No: T1483
Synonym: Lu 10-171,Nitalapram HBr,Bonitrile HBr,XU-62-320,Lu 10-171 HBr,氢溴酸西酞普兰,Citalopram HBr
Target: 5-HT Receptor, Serotonin Transporter, Autophagy
Haloxyfop
Cat.No: T5046
Synonym: Haloxyfop Acid,(±)-Haloxyfop,吡氟氯禾灵
Target: Others, Acetyl-CoA Carboxylase
Alosetron hydrochloride
Cat.No: T2525
Synonym: Lotronex,盐酸阿洛司琼,GR 68755C,GR 68755,GR 68755X
Target: 5-HT Receptor
Ticalopride
Cat.No: T69984
Synonym:
Target: 5-HT Receptor
Zinc phthalocyanine
Cat.No: T7105
Synonym: 酞菁锌,ZnPc
Target: Others
1-Tetralol, (S)-
Cat.No: T19999
Synonym: (S)-(+)-1,2,3,4-四氢-1-萘酚,(S)-Tetralin-1-ol,(S)-(+)-1,2,3,4-Tetrahydro-1-naphthol,(S)-1-Hydroxytetralin,J330.337C
Target: Others
Naloxone hydrochloride
Cat.No: T0102
Synonym: 盐酸纳洛酮,Naloxone HCl
Target: Opioid Receptor
Aluminum phthalocyanine chloride
Cat.No: T19637
Synonym: Phthalocyanine Chloroaluminum,铝酞菁,Chloroaluminum Phthalocyanine
Target: Others
Balofloxacin
Cat.No: T0116
Synonym:
Target: DNA gyrase, Antibacterial, Antibiotic
Galocitabine
Cat.No: T27399
Synonym: RO 091390,RO-091390,RO091390,RO-09-1390,Neofrutulon
Target: Others
MGCD-265 analog
Cat.No: T6351
Synonym: MGCD-265,Glesatinib
Target: Apoptosis, VEGFR, c-Met/HGFR
Halopemide
Cat.No: T15461
Synonym:
Target: Others, Phospholipase, Dopamine Receptor
RR-11a analog
Cat.No: T12770
Synonym: aza-peptide Michael acceptor, 7a
Target: Parasite
Haloperidol decanoate
Cat.No: T25487
Synonym: KD 16,KD-136,KD 136,Neoperidole,Haldol
Target: Others
ALOX15-IN-2
Cat.No: T62606
Synonym:
Target: Lipoxygenase
Halobetasol propionate
Cat.No: T6529
Synonym: 卤贝他索丙酸酯,Halobetasol Propionate,Ulobetasol propionate,BMY-30056,卤倍他索丙酸酯,CGP-14458
Target: Phospholipase
Labetalol hydrochloride
Cat.No: T0348
Synonym: 盐酸拉贝洛尔,Sch-15719W,AH-5158 hydrochloride,Labetalol HCl,柳胺苄心定
Target: Adrenergic Receptor
BenzeneazoMalononitrile
Cat.No: T9436
Synonym:
Target: Others
6-Chloro-1-tetralone
Cat.No: T21355
Synonym: 6-Chloro-α-Tetralone,5-CHLORO-L-INDOMONE,6-chloro-3;5-CHLORO-1-INDOMONE,5-CHLORO-1-INDOMONE,6-chloro-3
Target: Others
Prucalopride
Cat.No: T2542
Synonym: R-93877,普芦卡必利,普卡必利
Target: 5-HT Receptor
Amosulalol
Cat.No: T30027
Synonym:
Target: Adrenergic Receptor
MK-8245 analog
Cat.No: T20950
Synonym: MK-8245-analog,MK 8245 analog
Target: Others
idalopirdine
Cat.No: T7103
Synonym: Lu AE58054
Target: 5-HT Receptor
palovarotene
Cat.No: T4538
Synonym: Ro 3300074,R 667,帕罗伐汀
Target: Retinoid Receptor, Autophagy
VPS34 inhibitor 1 (Compound 19, PIK-III analogue)
Cat.No: T7944
Synonym: PIK-III analogue
Target: PI3K
Arhalofenate
Cat.No: T16022
Synonym: JNJ 39659100,芳卤芬酯,4-氯-ALPHA-[3-(三氟甲基)苯氧基]苯乙酸 2-(乙酰基氨基)乙酯,MBX 102
Target: PPAR
Caloxin 2A1 acetate
Cat.No: T40437L
Synonym:
Target: Proton pump
Naloxegol oxalate
Cat.No: T3355
Synonym: NKTR-118,NKTR-118 oxalate,AZ 13337019,AZ-13337019 oxalate
Target: P450
rac Desmethyl Citalopram Hydrochloride
Cat.No: T67851
Synonym:
Target: 5-HT Receptor
Idalopirdine Hydrochloride
Cat.No: T22936
Synonym: Lu AE58054盐酸盐,Lu AE58054 Hydrochloride,Idalopirdine HCl
Target: 5-HT Receptor
Alogliptin Benzoate
Cat.No: T2401
Synonym: 苯甲酸阿格列汀,SYR 322,Alogliptin(SYR-322)benzoate
Target: Ferroptosis, Proteasome, DPP-4
Halofenozide
Cat.No: T4384
Synonym:
Target: Others
Tabernanthalog
Cat.No: T60221
Synonym: TBG
Target: 5-HT Receptor
Aloxistatin
Cat.No: T6040
Synonym: E64d,Loxistatin,阿洛司他丁,E64c ethyl ester
Target: SARS-CoV, Cysteine Protease
Cephalonium
Cat.No: T0141
Synonym: 头孢洛宁,Cefalonium
Target: Others
Valorphin TFA(144313-54-2(free base))
Cat.No: T7666
Synonym: Valorphin TFA(144313-54-2(free bas))
Target: Others
Abaloparatide acetate(247062-33-5 free base)
Cat.No: TP1215L
Synonym:
Target: Others
Labetalone hydrochloride
Cat.No: T35326
Synonym: Labetalone hydrochloride,Benzoic amide
Target: Others, Adrenergic Receptor
Halothane
Cat.No: T0954
Synonym: Narcotane,氟烷,Anestan
Target: Potassium Channel, Chloride channel, GABA Receptor, NMDAR
Haloperidol
Cat.No: T0025
Synonym: Aloperidin,氟哌啶醇,Serenace,Haldol
Target: Dopamine Receptor, 5-HT Receptor
ONO-4059 analog
Cat.No: T6921
Synonym: ONO-4059 analogue,ONO-WG-307,GS-4059 analog
Target: Apoptosis, BTK
Palosuran
Cat.No: T2058
Synonym: ACT-058362
Target: GPR
Faropenem daloxate
Cat.No: T11265
Synonym: 法罗培南酯,Faropenem medoxil
Target: Antibacterial, Antibiotic
ARRY-380 (analog )
Cat.No: T2518
Synonym: HER2-Inhibitor-1,ARRY380,ARRY-380 analog
Target: EGFR, HER
Apabetalone
Cat.No: T2480
Synonym: RVX-208,RVX000222,阿帕他隆
Target: Epigenetic Reader Domain, HIV Protease
Phosalone
Cat.No: T5839
Synonym:
Target: Parasite
Cat. No. Product Name Target Signaling Pathways
T4S0592 Toddalolactone

(+)-Toddalolactone,飞龙掌血内酯,毛两面针素

PAI-1 Metabolism
Toddalolactone ((+)-Toddalolactone) 是一种Toddalia asiatica 的主要成分,能够抑制重组人纤溶酶原激活物抑制物-1(PAI-1)的活性, IC50=37.31 μM。
T0176 Isobarbaloin

Aloin,Aloin-A,芦荟甙,Barbaloin-A

Tyrosinase Proteases/Proteasome
Isobarbaloin (Barbaloin-A) 是一种来自芦荟的天然蒽环类药物,是一种酪氨酸酶抑制剂。
T8179 Aloeresin D

芦荟新甙D,芦荟新苷 D

Beta-Secretase; BACE Neuroscience
Aloeresin D 是一种从芦荟中分离得到的色原酮苷,能够抑制 β-分泌酶活性,IC50=39 μM。
T6856 Halofuginone

卤夫酮,常山酮,Tempostatin,empostatin,RU-19110

Calcium Channel; DNA/RNA Synthesis; Sodium Channel; Parasite; TGF-beta/Smad Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Stem Cells
Halofuginone (RU-19110) 是Febrifugine 的衍生物,是一种竞争性脯氨酰-tRNA 合成酶抑制剂。它也是肺血管扩张剂,可激活Kv 通道并阻断电压门控、受体操作和存储操作的钙离子通道。它具有抗炎、抗癌、抗疟疾和抗纤维化作用。
T5291 Malonic acid

Carboxyacetic Acid,1,3-Propanedioic Acid,丙二酸,Propanedioic Acid

Others Others
Malonic acid (propanedioic acid) 是竞争性抑制剂的典型例子:它作用于呼吸电子传递链中的琥珀酸脱氢酶(复合物 II)。发现丙二酸与丙二酰辅酶A 脱羧酶缺乏有关,这是一种先天性代谢错误。
T6377 Aloperine

Apoptosis; Virus Protease; HIV Protease; Antibiotic; Autophagy Apoptosis; Autophagy; Microbiology/Virology; Proteases/Proteasome
Aloperine 是一种在苦参类植物中的生物碱,其具有抗癌,抗炎、抗肿瘤和抗病毒特性,可用于研究过敏性接触性皮炎湿疹和其他皮肤炎症。
T15716 Lasalocid sodium

拉沙洛西钠,拉沙里菌素,Ionophore X-537A sodium,Antibiotic X-537A sodium,Lasalocid-A sodium

Antibacterial; Antibiotic; Autophagy Autophagy; Microbiology/Virology
Lasalocid sodium (Lasalocid-A sodium) 是一种抗菌剂。
T5S1177 Aloin B

Isobarbaloin,芦荟苷B,芦荟素B

Others Others
Aloin B (Isobarbaloin) 是一种芦荟素的异构体。其中芦荟素是芦荟中的具生理活性蒽醌化合物。
TN7078 MALONIC ACID, (P-HYDROXYBENZYL)- (7CI)

对羟基苄基丙二酸,2-[(4-hydroxyphenyl)methyl]propanedioic acid

Others Others
MALONIC ACID, (P-HYDROXYBENZYL)- (7CI) (2-[(4-hydroxyphenyl)methyl]propanedioic acid) 是一种天然产物。
TN2256 Taccalonolide B

根薯酮内酯B,根薯酮内酯 B

Microtubule Associated Cytoskeletal Signaling
Taccalonolide B 是从广西裂果薯中分离得到的一种微管稳定剂,具有抗肿瘤活性。它抑制 SK-OV-3 细胞的生长,IC50 为 208 nM,在体外对过表达 P-糖蛋白 (Pgp) 和多药耐药蛋白 (MRP7) 的细胞系有效。
T5279 Ethylmalonic acid

alpha-Carboxybutyrate,2-Ethylmalonic acid,乙基丙二酸

Others; Endogenous Metabolite Metabolism; Others
Ethylmalonic acid 是潜在有毒物质,非致癌性,与神经性厌食和甲氧基脱羧酶缺乏症有关。
T8014 Epoxylinalool

氧化芳樟醇,2-(2-Hydroxy-2-Propyl)-5-Methyl-5-Vinyltetrahydrofuran

Others Others
Epoxylinalool (2-(2-Hydroxy-2-Propyl)-5-Methyl-5-Vinyltetrahydrofuran) 是一种天然存在的单萜醇,广泛用于香水和调味品的生产。
T5662 5-Hydroxy-1-tetralone

Others Others
5-hydroxy-1-tetralone 是一种荧光标记试剂,可用于生物样品中的鞘糖脂的测定。
T4082 Astragaloside

MMP; ERK; JNK MAPK; Proteases/Proteasome
Astragaloside 是黄芪中的主要活性成分之一。
TN6910 Aloinoside B

11-o-Rhamnosylaloin B

Aloinoside B (11-o-Rhamnosylaloin B) 是一种来自芦荟的糖苷。
T5S0833 Astragaloside III

Antioxidant oxidation-reduction
Astragaloside III 是一种分离自黄芪中的一种天然产物。
T7878 Halosulfuron-methyl

A841101,Sempra,A 841101,氯吡嘧磺隆,A-841101

Others Others
Halosulfuron-methyl (A841101) 是一种常见的除草剂。
T3924 Astragaloside II

黄芪皂苷 II,Astrasieversianin VIII

TGF-beta/Smad Stem Cells
Astragaloside II (Astrasieversianin VIII) 是一种分离自黄芪中的天然化合物。
TN7021 Ent-toddalolactone

Others Others
Ent-toddalolactone 是一种天然化合物,属于香豆素类,来源于两面针,具有抗炎、抗癌活性。
T5244 Aminomalonic acid

2-Aminopropanedioic Acid,氨基丙二酸,Aminomalonate

Others; Endogenous Metabolite Metabolism; Others
Aminomalonic acid 是氨基内源性代谢产物,在体外能作为来源 Leukemia 5178Y/AR 和小鼠胰腺的L- 天冬酰胺合成酶的高效抑制剂 (Leukemia 5178Y/AR:Ki= 0.0023 M,小鼠胰腺:Ki= 0.0015 M)。它有潜力用作区分黑素瘤转移的不同阶段生物标志物。
T0989 7-Aminocephalosporanic acid

7-氨基头孢烷酸,7-ACA

Others; HSP; Antibacterial; Antibiotic Cytoskeletal Signaling; Metabolism; Microbiology/Virology; Others
7-Aminocephalosporanic acid 是一种 HSP90β 抑制剂,用于合成头孢菌素类抗生素及其中间体。
T4817 Methylmalonic acid

NSC 25201,MMA,Isosuccinic acid,甲基丙二酸,Methylpropanedioic acid,Methylmalonate

Others; Dehydrogenase; Endogenous Metabolite Metabolism; Others
Methylmalonic acid 是癌症患者缺乏维生素 B-12的指标。Methylmalonic acid 是竞争性琥珀酸脱氢酶抑制剂。
T1353 DL-Mevalonolactone

甲瓦龙酸内酯,Mevalonolactone

Others; Endogenous Metabolite Metabolism; Others
DL-Mevalonolactone ,一种人内源性代谢物,是甲羟戊酸的 δ-lactone 形式,甲羟戊酸途径的一个前体。它能够降低大脑中线粒体膜电位 (∆Ψm),Ca2+的保留能力和NAD (P) H 的含量 , 而且还诱导线粒体肿胀。DL-Mevalonolactone 诱导炎症和氧化应激反应,降低线粒体膜电位。
T15717 Lasalocid

Lasalocid-A,Antibiotic X-537A,Ionophore X-537A

Antibacterial Microbiology/Virology
Lasalocid (Lasalocid-A) 是一种由链霉菌产生的离子载体抗生素,具有抗菌和寄生虫作用,常添加进饲料中。
T5616 Diethyl malonate

Others Others
Diethyl malonate 天然存在于葡萄和草莓中。
T5755 Aloesin

Tyrosinase Proteases/Proteasome
Aloesin 是芦荟的活性成分之一,能够通过 MAPK 信号通路发挥抗癌作用,并具有抗炎、紫外线保护和抗菌作用。
TN1773 Isoastragaloside IV

异黄芪皂苷 IV,异黄芪皂苷IV

Others Others
Isoastragaloside IV 是一种天然三萜糖苷类产物,来源于黄芪中。
T0185 Escitalopram

Seroplex,依他普仑,S-(+)-Citalopram,艾司西酞普兰,(S)-Citalopram

Dopamine Receptor; 5-HT Receptor; Serotonin Transporter; Adrenergic Receptor; AChR; Norepinephrine; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Escitalopram (Seroplex) 是一种外消旋 Citalopram 的 S-对映体,是一种选择性 5-羟色胺再摄取抑制剂,Ki=0.89 nM,比 R(-)-enantiomer 结合亲和力高 30 倍。它对多巴胺转运体和去甲肾上腺素转运体均有选择性,是一种研究抑郁症的抗抑郁药。
TN1724 Harmalol hydrochloride

Harmidol hydrochloride

P450; Antioxidant Metabolism; oxidation-reduction
Harmalol hydrochloride (Harmidol hydrochloride) 是一种可从Peganum harmala L.的种子中提取出来的β-咔啉生物碱。Harmalol hydrochloride 是Harmaline 的主要代谢产物,在转录和翻译后水平上显著抑制二恶英介导的 CYP1A1 诱导。Harmalol hydrochloride 在去氧肾上腺素或KCl 预先收缩的分离大鼠胸主动脉制剂中显示出血管松弛活性。 Harmalol hydrochloride 具有抗氧化活性.
TN2139 Regaloside B

鸦胆子苦醇,王百合苷 B

NOS; COX; NO Synthase Immunology/Inflammation; Neuroscience
Regaloside B 是从麝香百合中分离出来的一种苯丙烷,可抑制iNOS 和COX-2的表达,具有抗炎活性。
T3925 Astragaloside I

黄芪皂苷I,Cyclosieversioside B,Astrasieversianin IV

Wnt/beta-catenin Cytoskeletal Signaling; Stem Cells
Astragaloside I (Cyclosieversioside B) 是从黄芪中分离得到天然产物。它可通过 Wnt/β-catenin 信号通路刺激成骨细胞分化,可用于成骨活性研究。
T4S0290 Araloside A

Chikusetsusaponin IV,竹节参皂苷IV

RAAS; Fas/FasL Apoptosis; Endocrinology/Hormones
Araloside A (Chikusetsusaponin IV) 是竹节参中的一种成分,对肾素renin 具有低抑制活性(IC50:77.4 μM)。
T5S0836 Isoastragaloside II

黄芪甲苷VII,Astrasieversianin VII

Others Others
Isoastragaloside II (Astrasieversianin VII) 是一种是从黄芪毛状根培养分离得到的黄芪甲苷。
T2843 Aloe emodin

芦荟大黄素,NSC 38628,3-Hydroxymethylchrysazine,Rhabarberone,Aloe-emodin

Autophagy; HSV Autophagy; Microbiology/Virology
Aloe emodin (Rhabarberone) 是从芦荟叶中提取出的一种羟基蒽醌,在体内外有抗肿瘤活性。
T2217 Cephalomannine

Baccatin III,三尖杉宁碱

Microtubule Associated Cytoskeletal Signaling
Cephalomannine (Baccatin III) 是一种从云南红豆杉中提取的紫杉醇衍生物,具有抗肿瘤活性,可用于癌症研究。
TN2254 Taccalonolide A

根薯酮内酯A,根薯酮内酯 A

Apoptosis; Microtubule Associated Apoptosis; Cytoskeletal Signaling
Taccalonolide A 是从水田七根茎中分离得到的一种类固醇,具有细胞毒性和抗疟活性。它在体外对过表达 p 糖蛋白、多药耐药蛋白 7 细胞系有抑制作用,抑制 SK-OV-3 细胞生长的 IC50值为 622 nM。它是微管稳定剂,能引起 G2-M 期滞留、Bcl-2 磷酸化,并引发细胞凋亡。
T5695 Dimethyl malonate

Others Others
Dimethyl malonate 是一种琥珀酸脱氢酶抑制剂。
T1549 Raloxifene hydrochloride

LY156758 hydrochloride,盐酸雷洛昔芬,Raloxifene HCl,LY139481 hydrochloride,Keoxifene hydrochloride,LY156758 (Keoxifene) HCl

Estrogen Receptor/ERR; Others; MAO; Estrogen/progestogen Receptor; Autophagy Autophagy; Endocrinology/Hormones; Metabolism; Neuroscience; Others
Raloxifene hydrochloride (LY156758 hydrochloride) 是一种选择性且可口服的雌激素受体调节剂,用于预防绝经后妇女的骨质疏松症。它对骨骼和胆固醇代谢具有雌激素激动作用,但对乳腺和子宫组织具有完全的雌激素拮抗作用。
T3366 Cephalotaxine

ZINC19795976,三尖杉碱,(-)-Cephalotaxine,Cephalotaxlen

Antiviral; Influenza Virus Immunology/Inflammation; Microbiology/Virology
Cephalotaxine (ZINC19795976) 是从头孢紫杉中分离得到的一种生物碱,具有抗白血病和抗病毒活性,如抗 Zika 病毒。
Fr12275 7-Methoxy-1-tetralone

Others Others
7-Methoxy-1-tetralone 可能具有杀虫活性。
T2S1181 Aloenin

Aloenin A,Aloearbonaside,芦荟宁

Beta-Secretase; AChR Neuroscience
Aloenin (Aloenin A) A 是一种具有清除过氧自由基作用的天然产物,对 β-分泌酶 (BACE) 具有中等抑制活性。
T3145 D-(+)-Trehalose dihydrate

Trehalose dihydrate,α,α-Trehalose dihydrate,alpha,alpha-Trehalose dihydrate,D-Trehalose dihydrate,二水合海藻糖

Others Others
D-(+)-Trehalose dihydrate (α,α-Trehalose dihydrate) 是分离自 Saccharomyces cerevisiae 中,可用作食品成分和药物赋形剂。
T3524 Halofuginone hydrobromide

卤夫酮溴氢酸盐,Tempostatin,RU-19110 (hydrobromide),Stenorol,常山酮溴酸盐

Others; Calcium Channel; DNA/RNA Synthesis; Sodium Channel; Parasite; TGF-beta/Smad Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Others; Stem Cells
Halofuginone hydrobromid 是Febrifugine 的衍生物,是竞争性脯氨酰-tRNA 合成酶抑制剂。它是 I 型胶原合成的特异性抑制剂,并通过抑制TGF-β活性可减轻骨关节炎。它具有抗疟疾、抗炎、抗癌、抗纤维化作用。
TN6490 Regaloside C

Others Others
Regaloside C 是一种从百合属的中分离出来的甘油葡糖苷,具有抗炎作用。
T2O2798 D-(+)-Trehalose

Ergot Sugar,D-Trehalose,Mycose,D-(+)-Trehalose Anhydrous,D-海藻糖,Trehalose

Others; Endogenous Metabolite Metabolism; Others
D-(+)-Trehalose (Mycose) 来源于自Saccharomyces cerevisiae,常用作食品成分和药物赋形剂。
TN1053 Aloe-emodin-8-O-β-D-glucopyranoside

Aloe-emodin-8-O-beta-D-glucopyranoside,芦荟大黄素-8-O-β-D-葡萄糖苷

Phosphatase Metabolism
Aloe-emodin-8-O-β-D-glucopyranoside (Aloe-emodin-8-O-beta-D-glucopyranoside) 是一种分离自Saussrurea lappa 中的化合物,是一种温和的人类蛋白酪氨酸磷酸酶 1B 抑制剂,其IC50=26.6 μM。
TQ0171 Isoastragaloside I

Others Others
Isoastragaloside I 是一种中药黄芪的天然化合物,能够增强脂联素量活性。
TN7117 regaloside I

Others Others
Regaloside I 是百合中的单体成分,可能是保护人类皮肤成纤维细胞免受 UVA 诱导的形态变化的主要成分。
TN1082 Apigenin 7-O-malonylglucoside

Apigenin 7-O-(6''-O-malonylglucoside)

Apigenin 7-O-malonylglucoside (Apigenin 7-O-(6''-O-malonylglucoside)) 存在于菊花中,是一种黄酮,也是一种糖苷。
T19284 Dimethylmalonic acid

2,2-Dimethylmalonic acid

Endogenous Metabolite Metabolism
Dimethylmalonic acid(2,2-Dimethylmalonic acid) 是人血清中的短链二羧酸,可用于预防或延缓鱼肌动球蛋白在冷冻缓冲溶液(pH 7)中的变性。
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天然产物

Toddalolactone
Cat.No: T4S0592
Synonym: (+)-Toddalolactone,飞龙掌血内酯,毛两面针素
Target: PAI-1
Isobarbaloin
Cat.No: T0176
Synonym: Aloin,Aloin-A,芦荟甙,Barbaloin-A
Target: Tyrosinase
Aloeresin D
Cat.No: T8179
Synonym: 芦荟新甙D,芦荟新苷 D
Target: Beta-Secretase, BACE
Halofuginone
Cat.No: T6856
Synonym: 卤夫酮,常山酮,Tempostatin,empostatin,RU-19110
Target: Calcium Channel, DNA/RNA Synthesis, Sodium Channel, Parasite, TGF-beta/Smad
Malonic acid
Cat.No: T5291
Synonym: Carboxyacetic Acid,1,3-Propanedioic Acid,丙二酸,Propanedioic Acid
Target: Others
Aloperine
Cat.No: T6377
Synonym:
Target: Apoptosis, Virus Protease, HIV Protease, Antibiotic, Autophagy
Lasalocid sodium
Cat.No: T15716
Synonym: 拉沙洛西钠,拉沙里菌素,Ionophore X-537A sodium,Antibiotic X-537A sodium,Lasalocid-A sodium
Target: Antibacterial, Antibiotic, Autophagy
Aloin B
Cat.No: T5S1177
Synonym: Isobarbaloin,芦荟苷B,芦荟素B
Target: Others
MALONIC ACID, (P-HYDROXYBENZYL)- (7CI)
Cat.No: TN7078
Synonym: 对羟基苄基丙二酸,2-[(4-hydroxyphenyl)methyl]propanedioic acid
Target: Others
Taccalonolide B
Cat.No: TN2256
Synonym: 根薯酮内酯B,根薯酮内酯 B
Target: Microtubule Associated
Ethylmalonic acid
Cat.No: T5279
Synonym: alpha-Carboxybutyrate,2-Ethylmalonic acid,乙基丙二酸
Target: Others, Endogenous Metabolite
Epoxylinalool
Cat.No: T8014
Synonym: 氧化芳樟醇,2-(2-Hydroxy-2-Propyl)-5-Methyl-5-Vinyltetrahydrofuran
Target: Others
5-Hydroxy-1-tetralone
Cat.No: T5662
Synonym:
Target: Others
Astragaloside
Cat.No: T4082
Synonym:
Target: MMP, ERK, JNK
Aloinoside B
Cat.No: TN6910
Synonym: 11-o-Rhamnosylaloin B
Target:
Astragaloside III
Cat.No: T5S0833
Synonym:
Target: Antioxidant
Halosulfuron-methyl
Cat.No: T7878
Synonym: A841101,Sempra,A 841101,氯吡嘧磺隆,A-841101
Target: Others
Astragaloside II
Cat.No: T3924
Synonym: 黄芪皂苷 II,Astrasieversianin VIII
Target: TGF-beta/Smad
Ent-toddalolactone
Cat.No: TN7021
Synonym:
Target: Others
Aminomalonic acid
Cat.No: T5244
Synonym: 2-Aminopropanedioic Acid,氨基丙二酸,Aminomalonate
Target: Others, Endogenous Metabolite
7-Aminocephalosporanic acid
Cat.No: T0989
Synonym: 7-氨基头孢烷酸,7-ACA
Target: Others, HSP, Antibacterial, Antibiotic
Methylmalonic acid
Cat.No: T4817
Synonym: NSC 25201,MMA,Isosuccinic acid,甲基丙二酸,Methylpropanedioic acid,Methylmalonate
Target: Others, Dehydrogenase, Endogenous Metabolite
DL-Mevalonolactone
Cat.No: T1353
Synonym: 甲瓦龙酸内酯,Mevalonolactone
Target: Others, Endogenous Metabolite
Lasalocid
Cat.No: T15717
Synonym: Lasalocid-A,Antibiotic X-537A,Ionophore X-537A
Target: Antibacterial
Diethyl malonate
Cat.No: T5616
Synonym:
Target: Others
Aloesin
Cat.No: T5755
Synonym:
Target: Tyrosinase
Isoastragaloside IV
Cat.No: TN1773
Synonym: 异黄芪皂苷 IV,异黄芪皂苷IV
Target: Others
Escitalopram
Cat.No: T0185
Synonym: Seroplex,依他普仑,S-(+)-Citalopram,艾司西酞普兰,(S)-Citalopram
Target: Dopamine Receptor, 5-HT Receptor, Serotonin Transporter, Adrenergic Receptor, AChR, Norepinephrine, Histamine Receptor
Harmalol hydrochloride
Cat.No: TN1724
Synonym: Harmidol hydrochloride
Target: P450, Antioxidant
Regaloside B
Cat.No: TN2139
Synonym: 鸦胆子苦醇,王百合苷 B
Target: NOS, COX, NO Synthase
Astragaloside I
Cat.No: T3925
Synonym: 黄芪皂苷I,Cyclosieversioside B,Astrasieversianin IV
Target: Wnt/beta-catenin
Araloside A
Cat.No: T4S0290
Synonym: Chikusetsusaponin IV,竹节参皂苷IV
Target: RAAS, Fas/FasL
Isoastragaloside II
Cat.No: T5S0836
Synonym: 黄芪甲苷VII,Astrasieversianin VII
Target: Others
Aloe emodin
Cat.No: T2843
Synonym: 芦荟大黄素,NSC 38628,3-Hydroxymethylchrysazine,Rhabarberone,Aloe-emodin
Target: Autophagy, HSV
Cephalomannine
Cat.No: T2217
Synonym: Baccatin III,三尖杉宁碱
Target: Microtubule Associated
Taccalonolide A
Cat.No: TN2254
Synonym: 根薯酮内酯A,根薯酮内酯 A
Target: Apoptosis, Microtubule Associated
Dimethyl malonate
Cat.No: T5695
Synonym:
Target: Others
Raloxifene hydrochloride
Cat.No: T1549
Synonym: LY156758 hydrochloride,盐酸雷洛昔芬,Raloxifene HCl,LY139481 hydrochloride,Keoxifene hydrochloride,LY156758 (Keoxifene) HCl
Target: Estrogen Receptor/ERR, Others, MAO, Estrogen/progestogen Receptor, Autophagy
Cephalotaxine
Cat.No: T3366
Synonym: ZINC19795976,三尖杉碱,(-)-Cephalotaxine,Cephalotaxlen
Target: Antiviral, Influenza Virus
7-Methoxy-1-tetralone
Cat.No: Fr12275
Synonym:
Target: Others
Aloenin
Cat.No: T2S1181
Synonym: Aloenin A,Aloearbonaside,芦荟宁
Target: Beta-Secretase, AChR
D-(+)-Trehalose dihydrate
Cat.No: T3145
Synonym: Trehalose dihydrate,α,α-Trehalose dihydrate,alpha,alpha-Trehalose dihydrate,D-Trehalose dihydrate,二水合海藻糖
Target: Others
Halofuginone hydrobromide
Cat.No: T3524
Synonym: 卤夫酮溴氢酸盐,Tempostatin,RU-19110 (hydrobromide),Stenorol,常山酮溴酸盐
Target: Others, Calcium Channel, DNA/RNA Synthesis, Sodium Channel, Parasite, TGF-beta/Smad
Regaloside C
Cat.No: TN6490
Synonym:
Target: Others
D-(+)-Trehalose
Cat.No: T2O2798
Synonym: Ergot Sugar,D-Trehalose,Mycose,D-(+)-Trehalose Anhydrous,D-海藻糖,Trehalose
Target: Others, Endogenous Metabolite
Aloe-emodin-8-O-β-D-glucopyranoside
Cat.No: TN1053
Synonym: Aloe-emodin-8-O-beta-D-glucopyranoside,芦荟大黄素-8-O-β-D-葡萄糖苷
Target: Phosphatase
Isoastragaloside I
Cat.No: TQ0171
Synonym:
Target: Others
regaloside I
Cat.No: TN7117
Synonym:
Target: Others
Apigenin 7-O-malonylglucoside
Cat.No: TN1082
Synonym: Apigenin 7-O-(6''-O-malonylglucoside)
Target:
Dimethylmalonic acid
Cat.No: T19284
Synonym: 2,2-Dimethylmalonic acid
Target: Endogenous Metabolite
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Cat. No. Product Name Species Expression System
TMPY-01201 Human cytomegalovirus (HCMV) Glycoprotein B/gB Protein (His)

Human cytωlovirus (HCMV) Glycoprotein B/gB

CMV HEK293 Cells
Human cytomegalovirus (HCMV) Glycoprotein B/gB Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 93.2 kDa and the accession number is P13201.
TMPY-00811 Human cytomegalovirus (HCMV) Glycoprotein B/gB Protein

Human cytωlovirus (HCMV) Glycoprotein B/gB

CMV HEK293 Cells
Human cytomegalovirus (HCMV) Glycoprotein B/gB Protein is expressed in HEK293 mammalian cells. The predicted molecular weight is 92 kDa and the accession number is P13201.
TMPH-00955 ALOX12 Protein, Human, Recombinant (His)

Polyunsaturated fatty acid lipoxygenase ALOX12,LOG1...

Human E. coli
ALOX12 Protein, Human, Recombinant (His) is expressed in E. coli.
TMPH-00788 PYP Protein, Halochromatium salexigens, Recombinant (His)

pyp,Photoactive yellow protein

Halochromatium salexigens E. coli
Photoactive blue light protein. Probably functions as a photoreceptor for a negative phototaxis response.
TMPH-01194 Human cytomegalovirus (HCMV) (strain AD169) UL130 Protein (His & SUMO)

UL130,Uncharacterized protein UL130

HHV-5 E. coli
Plays a role in viral entry into host cells. Forms a pentameric complex at the surface of the viral envelope together with gH, gL, UL130 and UL131. This complex is required for entry in epithelial, endothelial and myeloid host cells. Mechanistically, engages host receptor(s) including neurophilin 2/NRP2 to mediate infection. Human cytomegalovirus (HCMV) (strain AD169) UL130 Protein (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 37....
TMPH-03406 Rhesus cytomegalovirus (RhCMV) (strain 68-1) Glycoprotein B/gB Protein (His & Myc)

gB,Envelope glycoprotein B

RhCMV E. coli
Rhesus cytomegalovirus (RhCMV) (strain 68-1) Glycoprotein B/gB Protein (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 18.0 kDa and the accession number is P89053.
TMPY-00810 Human cytomegalovirus (HCMV) Glycoprotein B/gB Protein (hFc)

Human cytωlovirus (HCMV) Glycoprotein B/gB

CMV HEK293 Cells
Human cytomegalovirus (HCMV) Glycoprotein B/gB Protein (hFc) is expressed in HEK293 mammalian cells with Fc tag. The predicted molecular weight is 118 kDa and the accession number is P13201.
TMPH-00785 Bacteriorhodopsin Protein, Halobacterium halobium, Recombinant (His & Myc & SUMO)

bop,Bacteriorhodopsin,BR

Halobacterium halobium E. coli
Light-driven proton pump.
TMPH-01195 Human cytomegalovirus (HCMV) (strain Merlin) Viral interleukin-10 homolog

UL111A,Viral interleukin-10 homolog

HCMV E. coli
Functional viral IL-10 homolog. Can bind to the human IL-10 receptor and compete with human IL-10 for binding sites. Requires both subunits of the human IL-10 receptor complex to induce signal transduction events and biological activities. IL-10 signaling pathway has several immunosuppressive activities that are exploited by the virus. Inhibits TLR-induced type I interferon production in host plasmacytoid dendritic cells. Human cytomegalovirus (HCMV) (strain Merlin) Viral interleukin-10 homolog ...
TMPH-01192 Human cytomegalovirus (HCMV) (strain AD169) Large structural phosphoprotein (Avi & His & MBP), Biotinylated

Phosphoprotein UL32,150 kDa matrix phosphoprotein,Tegument p...

HHV-5 E. coli
Human cytomegalovirus (HCMV) (strain AD169) Large structural phosphoprotein (Avi & His & MBP), Biotinylated is expressed in E. coli.
TMPH-00042 Haloalkane dehalogenase Protein, Agrobacterium tumefaciens, Recombinant (His & Myc)

Haloalkane dehalogenase,dhaA

Agrobacterium fabrum E. coli
Catalyzes hydrolytic cleavage of carbon-halogen bonds in halogenated aliphatic compounds, leading to the formation of the corresponding primary alcohols, halide ions and protons. Haloalkane dehalogenase Protein, Agrobacterium tumefaciens, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 41.8 kDa and the accession number is Q8U671.
TMPY-00812 Human cytomegalovirus (HCMV) Glycoprotein B/gB Protein (aa 1-700, hFc)

Human cytωlovirus (HCMV) Glycoprotein B/gB

CMV HEK293 Cells
Human cytomegalovirus (HCMV) Glycoprotein B/gB Protein (aa 1-700, hFc) is expressed in HEK293 mammalian cells with Fc tag. The predicted molecular weight is 104 kDa and the accession number is P13201.
TMPH-00787 BtuD Protein, Halobacterium salinarum, Recombinant

Vitamin B12-transporting ATPase,Cobalamin import ATP-binding...

Halobacterium salinarum E. coli
Required for corrinoid utilization. Probably part of the ABC transporter complex BtuCDF involved in cobalamin (vitamin B12) import. Probably responsible for energy coupling to the transport system.
TMPH-01190 Human cytomegalovirus (HCMV) (strain AD169) glycoprotein H/gH Protein (His & SUMO)

gH,Envelope glycoprotein H

HHV-5 E. coli
Human cytomegalovirus (HCMV) (strain AD169) glycoprotein H/gH Protein (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 35.8 kDa and the accession number is P12824.
TMPY-00054 Macaca fascicularis Cytomegalovirus (CyCMV) (strain OT-1) glycoprotein B/gB Protein (hFc)

Macaca fascicularis Cytωlovirus (CyCMV) (strain OT-1) glycop...

CyCMV HEK293 Cells
Macaca fascicularis Cytomegalovirus (CyCMV) (strain OT-1) glycoprotein B/gB Protein (hFc) is expressed in HEK293 mammalian cells with Fc tag. The predicted molecular weight is 102.5 kDa and the accession number is E7DB34.
TMPH-00786 BtuD Protein, Halobacterium salinarum, Recombinant (His)

Vitamin B12-transporting ATPase,btuD,Cobalamin import ATP-bi...

Halobacterium salinarum E. coli
Required for corrinoid utilization. Probably part of the ABC transporter complex BtuCDF involved in cobalamin (vitamin B12) import. Probably responsible for energy coupling to the transport system.
TMPH-00158 BH0637 Protein, Bacillus halodurans, Recombinant (His & Myc & SUMO)

Putative adenine deaminase BH0637,Adenase,Adenine aminase

Bacillus halodurans E. coli
N/A. BH0637 Protein, Bacillus halodurans, Recombinant (His & Myc & SUMO) is expressed in E. coli expression system with N-10xHis-SUMO and C-Myc tag. The predicted molecular weight is 57.7 kDa and the accession number is Q9KF49.
TMPH-01191 Human cytomegalovirus (HCMV) (strain Towne) glycoprotein UL132 Protein (Avi & His & MBP), Biotinylated

UL132,Envelope glycoprotein UL132

HHV-5 E. coli
Human cytomegalovirus (HCMV) (strain Towne) glycoprotein UL132 Protein (Avi & His & MBP), Biotinylated is expressed in E. coli.
TMPH-01193 Human cytomegalovirus (HCMV) (strain AD169) Uncharacterized protein UL128 (His)

Uncharacterized protein UL128,UL128

HHV-5 E. coli
Human cytomegalovirus (HCMV) (strain AD169) Uncharacterized protein UL128 (His) is expressed in E. coli.

重组蛋白

Human cytomegalovirus (HCMV) Glycoprotein B/gB Protein (His)
Cat.No: TMPY-01201
Species: CMV
Expression System: HEK293 Cells
Human cytomegalovirus (HCMV) Glycoprotein B/gB Protein
Cat.No: TMPY-00811
Species: CMV
Expression System: HEK293 Cells
ALOX12 Protein, Human, Recombinant (His)
Cat.No: TMPH-00955
Species: Human
Expression System: E. coli
PYP Protein, Halochromatium salexigens, Recombinant (His)
Cat.No: TMPH-00788
Species: Halochromatium salexigens
Expression System: E. coli
Human cytomegalovirus (HCMV) (strain AD169) UL130 Protein (His & SUMO)
Cat.No: TMPH-01194
Species: HHV-5
Expression System: E. coli
Rhesus cytomegalovirus (RhCMV) (strain 68-1) Glycoprotein B/gB Protein (His & Myc)
Cat.No: TMPH-03406
Species: RhCMV
Expression System: E. coli
Human cytomegalovirus (HCMV) Glycoprotein B/gB Protein (hFc)
Cat.No: TMPY-00810
Species: CMV
Expression System: HEK293 Cells
Bacteriorhodopsin Protein, Halobacterium halobium, Recombinant (His & Myc & SUMO)
Cat.No: TMPH-00785
Species: Halobacterium halobium
Expression System: E. coli
Human cytomegalovirus (HCMV) (strain Merlin) Viral interleukin-10 homolog
Cat.No: TMPH-01195
Species: HCMV
Expression System: E. coli
Human cytomegalovirus (HCMV) (strain AD169) Large structural phosphoprotein (Avi & His & MBP), Biotinylated
Cat.No: TMPH-01192
Species: HHV-5
Expression System: E. coli
Haloalkane dehalogenase Protein, Agrobacterium tumefaciens, Recombinant (His & Myc)
Cat.No: TMPH-00042
Species: Agrobacterium fabrum
Expression System: E. coli
Human cytomegalovirus (HCMV) Glycoprotein B/gB Protein (aa 1-700, hFc)
Cat.No: TMPY-00812
Species: CMV
Expression System: HEK293 Cells
BtuD Protein, Halobacterium salinarum, Recombinant
Cat.No: TMPH-00787
Species: Halobacterium salinarum
Expression System: E. coli
Human cytomegalovirus (HCMV) (strain AD169) glycoprotein H/gH Protein (His & SUMO)
Cat.No: TMPH-01190
Species: HHV-5
Expression System: E. coli
Macaca fascicularis Cytomegalovirus (CyCMV) (strain OT-1) glycoprotein B/gB Protein (hFc)
Cat.No: TMPY-00054
Species: CyCMV
Expression System: HEK293 Cells
BtuD Protein, Halobacterium salinarum, Recombinant (His)
Cat.No: TMPH-00786
Species: Halobacterium salinarum
Expression System: E. coli
BH0637 Protein, Bacillus halodurans, Recombinant (His & Myc & SUMO)
Cat.No: TMPH-00158
Species: Bacillus halodurans
Expression System: E. coli
Human cytomegalovirus (HCMV) (strain Towne) glycoprotein UL132 Protein (Avi & His & MBP), Biotinylated
Cat.No: TMPH-01191
Species: HHV-5
Expression System: E. coli
Human cytomegalovirus (HCMV) (strain AD169) Uncharacterized protein UL128 (His)
Cat.No: TMPH-01193
Species: HHV-5
Expression System: E. coli
Cat. No. Product Name Target Signaling Pathways
TMIJ-0066 Alosetron-13C-d3

Alosetron-13C-d3 是 Alosetron 的 13C 和氘代化合物。Alosetron 的 CAS 号为 122852-42-0。
T19191 Alosetron-d3

Alosetron D3,GR 68755 D3,GR 68755X D3

Others Others
Alosetron D3 (GR 68755 D3) is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.
TMIH-0034 2-Ethyl-2-phenylmalonamide-d5

2-Ethyl-2-phenylmalonamide-d5 是 2-Ethyl-2-phenylmalonamide 的氘代化合物。
TMIH-0364 Naloxone-d5

Naloxone-d5 是 Naloxone 的氘代化合物。
TMIH-0191 dimethyl 2-(methyl-d3)malonate

dimethyl 2-(methyl-d3)malonate 是 dimethyl 2-(methyl)malonate 的氘代化合物。dimethyl 2-(methyl)malonate 的 CAS 号为 516-05-2。Methylmalonic acid 是癌症患者缺乏维生素 B-12的指标。
TMIH-0159 Citalopram-d6

Citalopram-d6 是 Citalopram 的氘代化合物。Citalopram 的 CAS 号为 59729-33-8。Citalopram (Lu 10-171) 是一种具有口服活性的、选择性的血清素再摄取抑制剂 (SSRI),是一种选择性5-羟色胺再摄取抑制剂,是一种 S(+)-对映体 (Escitalopram) 和 R(-)-对映体的外消旋混合物。Citalopram 具有抗抑郁活性,可增强血清素能神经传递,可用于研究老年痴呆。
TMIJ-0144 Palonosetron-d3 HCl

Palonosetron-d3 HCl 是 Palonosetron HCl 的氘代化合物。Palonosetron HCl 的 CAS 号为 135729-62-3。Palonosetron hydrochloride 是一种 5-HT3 拮抗剂,用于预防和治疗化疗引起的恶心和呕吐。
TMID-0097 Ethyl-d5-malonic Acid

Ethyl-d5-malonic Acid 是 Ethyl-malonic Acid 的氘代化合物。Ethyl-malonic Acid 的 CAS 号为 601-75-2。Ethylmalonic acid 是潜在有毒物质,非致癌性,与神经性厌食和甲氧基脱羧酶缺乏症有关。
T71285 Metaxalone-d6

Metaxalone-d6 is intended for use as an internal standard for the quantification of metaxalone by GC-or LC-MS. Metaxalone is a skeletal muscle relaxant. It inhibits the proliferation of, and induces apoptosis in, RAW 264.7 cells in vitro when used at concentrations ranging from 1 to 100 µM. Metaxalone also reduces LPS-induced increases in COX-1, COX-2, and NF-kB levels and inhibits LPS-induced production of TNF-α, IL-6, and prostaglandin E2 in RAW 264.7 cells. Formulations containing metaxalone ...
T10288 Alogliptin (13CD3)

SYR-322 (13CD3)

Others Others
Alogliptin (SYR-322) 13CD3 is the deuterium-labeled Alogliptin. Alogliptin is a selective inhibitor of DPP-4.
T19190 Alosetron D3 Hydrochloride

GR-68755C D3

Others Others
Alosetron D3 (GR 68755 D3) Hydrochloride is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.
TMIH-0373 N-Desmethyl citalopram-d4 Oxalate

N-Desmethyl citalopram-d4 Oxalate 是 N-Desmethyl citalopram Oxalate 的氘代化合物。
TMIH-0488 Reduced Haloperidol-d4

Reduced Haloperidol-d4 是 Reduced Haloperidol 的氘代化合物。Reduced Haloperidol 的 CAS 号为 34104-67-1。
TMIH-0010 (S)-Alogliptin Benzoate Salt-13C-d3

(S)-Alogliptin Benzoate Salt-13C-d3 是 (S)-Alogliptin Benzoate Salt 的 13C 和氘代化合物。
TMIH-0105 Baloxavir-d4

Baloxavir-d4 是 Baloxavir 的氘代化合物。Baloxavir 的 CAS 号为 1985605-59-1。Baloxavir 是衍生自前药 Baloxavir marboxil,是流感病毒聚合酶 PA 亚基的一流帽依赖性核酸内切酶抑制剂。它抑制病毒 RNA 的转录和复制,具有强大的抗病毒活性。
TMIH-0158 Citalopram-d6 Oxalate

Citalopram-d6 Oxalate 是 Citalopram Oxalate 的氘代化合物。Citalopram Oxalate 的 CAS 号为 207559-01-1。
TMIH-0461 Prucalopride-13C-d3

Prucalopride-13C-d3 是 Prucalopride 的 13C 和氘代化合物。Prucalopride 的 CAS 号为 179474-81-8。Prucalopride 是一种选择性、高亲和力的 5-HT4A/4B 受体激动剂,Ki为2.5和 8 nM。它对 5-HT4A/4B 受体的选择性是其他 5-HT 受体亚型的 290 倍以上。
TMIH-0157 Citalopram-d4 Oxalate

Citalopram-d4 Oxalate 是 Citalopram Oxalate 的氘代化合物。Citalopram Oxalate 的 CAS 号为 207559-01-1。
T10181 6-beta-Naloxol D5 hydrochloride

6β-Naloxol D5 hydrochloride

Others Others
6-beta-Naloxol D5 hydrochloride is a deuterium-labeled opioid antagonist, closely related to naloxone, that serves as an effective compound in the field of chemical research.
T11535 Haloperidol D4

氟哌啶醇D4

Others Others
Haloperidol D4 is deuterium-labeled haloperidol.
TMID-0034 Haloperidol-d4 TFA

Haloperidol-d4 TFA 是 Haloperidol TFA 的氘代化合物。
T11536 Haloperidol (D4')

Haloperidol D4',氟哌啶醇 (D4')

Others Others
Haloperidol D4' is deuterium-labeled haloperidol. Haloperidol is a dopamine D2 receptor antagonist.
TMIJ-0213 Naloxone-d5 HCl

Naloxone-d5 HCl 是 Naloxone HCl 的氘代化合物。Naloxone HCl 的 CAS 号为 357-08-4。Naloxone hydrochloride 是一种特异性、没有激动剂活性的opiate拮抗剂。它是 mu、delta 和 kappa 阿片受体的竞争性拮抗剂。
TMID-0254 Linalool-d3

Linalool-d3 是 Linalool 的氘代化合物。Linalool 的 CAS 号为 78-70-6。Linalool 是存在芫荽等植物中的单萜类天然产物,是竞争性NMDA受体拮抗剂,具有抗肿瘤和抗心脏毒性的作用。它通过激活 Nrf2 诱导抗氧化防御和通过抑制 NF-κB 减少炎症反应来保护其免受 LPS/GalN 诱导的肝损伤,具有镇痛、抗菌和抗炎的特性。

同位素标记化合物

Alosetron-13C-d3
Cat.No: TMIJ-0066
Synonym:
Target:
Alosetron-d3
Cat.No: T19191
Synonym: Alosetron D3,GR 68755 D3,GR 68755X D3
Target: Others
2-Ethyl-2-phenylmalonamide-d5
Cat.No: TMIH-0034
Synonym:
Target:
Naloxone-d5
Cat.No: TMIH-0364
Synonym:
Target:
dimethyl 2-(methyl-d3)malonate
Cat.No: TMIH-0191
Synonym:
Target:
Citalopram-d6
Cat.No: TMIH-0159
Synonym:
Target:
Palonosetron-d3 HCl
Cat.No: TMIJ-0144
Synonym:
Target:
Ethyl-d5-malonic Acid
Cat.No: TMID-0097
Synonym:
Target:
Metaxalone-d6
Cat.No: T71285
Synonym:
Target:
Alogliptin (13CD3)
Cat.No: T10288
Synonym: SYR-322 (13CD3)
Target: Others
Alosetron D3 Hydrochloride
Cat.No: T19190
Synonym: GR-68755C D3
Target: Others
N-Desmethyl citalopram-d4 Oxalate
Cat.No: TMIH-0373
Synonym:
Target:
Reduced Haloperidol-d4
Cat.No: TMIH-0488
Synonym:
Target:
(S)-Alogliptin Benzoate Salt-13C-d3
Cat.No: TMIH-0010
Synonym:
Target:
Baloxavir-d4
Cat.No: TMIH-0105
Synonym:
Target:
Citalopram-d6 Oxalate
Cat.No: TMIH-0158
Synonym:
Target:
Prucalopride-13C-d3
Cat.No: TMIH-0461
Synonym:
Target:
Citalopram-d4 Oxalate
Cat.No: TMIH-0157
Synonym:
Target:
6-beta-Naloxol D5 hydrochloride
Cat.No: T10181
Synonym: 6β-Naloxol D5 hydrochloride
Target: Others
Haloperidol D4
Cat.No: T11535
Synonym: 氟哌啶醇D4
Target: Others
Haloperidol-d4 TFA
Cat.No: TMID-0034
Synonym:
Target:
Haloperidol (D4')
Cat.No: T11536
Synonym: Haloperidol D4',氟哌啶醇 (D4')
Target: Others
Naloxone-d5 HCl
Cat.No: TMIJ-0213
Synonym:
Target:
Linalool-d3
Cat.No: TMID-0254
Synonym:
Target:
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