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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T4574 |
Sacubitril
AHU 377,AHU377,沙库必曲,AHU-377 |
Neprilysin | Metabolism |
Sacubitril (AHU-377) 是一种有效的NEP 抑制剂,IC50=5 nM。它是研究心力衰竭药物 LCZ696 的组分之一。 | |||
T4200 |
Sacubitril hemicalcium salt
AHU-377 (hemicalcium salt),LCZ696中间体,AHU377 calcium salt |
Neprilysin | Metabolism |
Sacubitril hemicalcium salt (AHU377 calcium salt) 是一种有效的 NEP 抑制剂,IC50=5 nM。它是研究心力衰竭药物 LCZ696 的组分之一。 | |||
T4574L |
Sacubitril sodium
AHU377,AHU-377,LCZ696,AHU 377 |
Others | Others |
Sacubitril is an angiotensin receptor neprilysin inhibitor being studied for use in combination with valsartan for heart failure. Sacubitril is a prodrug that is activated to LBQ657 by de-ethylation via esterases. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TMIH-0076 |
AHU-377-d4
|
||
AHU-377-d4 是 AHU-377 的氘代化合物。 | |||
TMIH-0511 |
Sacubitril-d4 calcium salt
AHU-377-d4 calcium salt |
||
Sacubitril-d4 calcium salt 是 Sacubitril calcium salt 的氘代化合物。 |